| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.649 | 0.004 | 0.649 | Peroxidase inhibitor | 0.464 0.013 CHEMBL2111041 0.355 0.027 CHEMBL3544855 0.379 0.024 CHEMBL3544856 0.578 0.005 CHEMBL1203 0.4 0.02 CHEMBL1442231 0.607 0.004 CHEMBL3544636 0.113 0.108 CHEMBL3544637 0.624 0.004 CHEMBL3091859 0.631 0.004 CHEMBL1237174 0.52 0.008 CHEMBL3091852 | ||
| 0.606 | 0.001 | 0.919 | Maillard reaction inhibitor | 0.147 0.006 CHEMBL2111041 0.101 0.016 CHEMBL3544855 0.149 0.006 CHEMBL3544856 0.084 0.023 CHEMBL1203 0.058 0.036 CHEMBL1442231 0.741 0.001 CHEMBL3091859 0.919 0 CHEMBL1237174 0.1 0.017 CHEMBL3091852 | CHEMBL1237174 | |
| 0.583 | 0.058 | 0.688 | Alpha-glucosidase inhibitor | 0.546 0.067 CHEMBL2111041 0.253 0.186 CHEMBL3544855 0.688 0.036 CHEMBL3544856 0.221 0.205 CHEMBL1203 0.578 0.059 CHEMBL1442231 0.676 0.038 CHEMBL3544637 0.58 0.058 CHEMBL3091859 0.255 0.184 CHEMBL1237174 0.493 0.082 CHEMBL3091852 | CHEMBL3544856 | |
| 0.544 | 0.023 | 0.791 | Streptokinase A inhibitor | 0.454 0.035 CHEMBL2111041 0.309 0.075 CHEMBL3544855 0.246 0.106 CHEMBL3544856 0.779 0.005 CHEMBL1442231 0.655 0.012 CHEMBL3091859 0.18 0.146 CHEMBL1237174 0.791 0.005 CHEMBL3091852 | CHEMBL3091852 | |
| 0.503 | 0.004 | 0.905 | Alcohol oxidase inhibitor | 0.19 0.007 CHEMBL2111041 0.102 0.018 CHEMBL3544855 0.119 0.014 CHEMBL3544856 0.898 0.002 CHEMBL1203 0.192 0.007 CHEMBL1442231 0.158 0.009 CHEMBL3544636 0.111 0.016 CHEMBL3544637 0.905 0.002 CHEMBL3091859 0.786 0.003 CHEMBL1237174 0.811 0.003 CHEMBL3091852 | CHEMBL3091859 | |
| 0.524 | 0.068 | 0.574 | Transcription factor inhibitor | 0.392 0.113 CHEMBL2111041 0.244 0.19 CHEMBL3544855 0.574 0.054 CHEMBL1442231 0.459 0.088 CHEMBL3091859 0.217 0.212 CHEMBL1237174 0.438 0.095 CHEMBL3091852 | CHEMBL1442231 | |
| 0.477 | 0.045 | 0.59 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.368 0.132 CHEMBL2111041 0.285 0.233 CHEMBL3544855 0.59 0.008 CHEMBL1203 0.472 0.048 CHEMBL1442231 0.502 0.033 CHEMBL3544636 0.417 0.086 CHEMBL3091859 0.535 0.02 CHEMBL1237174 0.49 0.038 CHEMBL3091852 | CHEMBL1203 | |
| 0.457 | 0.026 | 0.486 | Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase inhibitor | 0.402 0.038 CHEMBL2111041 0.201 0.099 CHEMBL3544855 0.276 0.071 CHEMBL1203 0.195 0.103 CHEMBL1442231 0.486 0.022 CHEMBL3091859 0.344 0.052 CHEMBL1237174 0.25 0.078 CHEMBL3091852 | CHEMBL3091859 | |
| 0.42 | 0.005 | 0.779 | Cyclin-dependent kinase 5 inhibitor | 0.57 0.004 CHEMBL1442231 0.779 0.002 CHEMBL3091859 0.619 0.004 CHEMBL1237174 0.754 0.003 CHEMBL3091852 | CHEMBL3091859 | |
| 0.415 | 0.018 | 0.415 | Pyruvate kinase inhibitor | 0.318 0.043 CHEMBL2111041 0.281 0.053 CHEMBL3544855 0.335 0.039 CHEMBL3544856 0.331 0.04 CHEMBL1203 0.246 0.062 CHEMBL1442231 0.265 0.057 CHEMBL3091859 0.281 0.053 CHEMBL1237174 0.181 0.093 CHEMBL3091852 | ||
| 0.399 | 0.018 | 0.399 | Ca2+/calmodulin-dependent kinase II gamma inhibitor | 0.154 0.086 CHEMBL1442231 0.152 0.087 CHEMBL3091852 | ||
| 0.426 | 0.051 | 0.612 | GABA C receptor rho-3 antagonist | 0.334 0.095 CHEMBL2111041 0.258 0.147 CHEMBL3544855 0.546 0.015 CHEMBL1203 0.392 0.065 CHEMBL1442231 0.583 0.009 CHEMBL3544636 0.448 0.042 CHEMBL3091859 0.612 0.006 CHEMBL1237174 0.541 0.016 CHEMBL3091852 | CHEMBL1237174 | |
| 0.377 | 0.014 | 0.377 | Dual specificity tyrosine-phosphorylation regulated kinase 3 inhibitor | 0.242 0.049 CHEMBL1203 0.226 0.059 CHEMBL1442231 0.177 0.095 CHEMBL3091852 | ||
| 0.399 | 0.038 | 0.399 | Aryl hydrocarbon receptor agonist | 0.198 0.103 CHEMBL2111041 0.232 0.086 CHEMBL1203 0.275 0.069 CHEMBL1442231 0.265 0.073 CHEMBL3091859 0.311 0.058 CHEMBL1237174 0.254 0.077 CHEMBL3091852 | ||
| 0.362 | 0.006 | 0.362 | Histone acetyltransferase inhibitor | 0.189 0.087 CHEMBL2111041 0.167 0.117 CHEMBL3544855 0.218 0.046 CHEMBL1203 0.229 0.037 CHEMBL1442231 0.166 0.119 CHEMBL3544636 0.205 0.062 CHEMBL3091859 0.202 0.066 CHEMBL1237174 0.209 0.056 CHEMBL3091852 | ||
| 0.42 | 0.066 | 0.637 | 5 Hydroxytryptamine release inhibitor | 0.456 0.049 CHEMBL2111041 0.377 0.093 CHEMBL3544855 0.435 0.058 CHEMBL3544856 0.637 0.007 CHEMBL1203 0.431 0.06 CHEMBL1442231 0.47 0.043 CHEMBL3544636 0.527 0.025 CHEMBL3544637 0.453 0.05 CHEMBL3091859 0.495 0.034 CHEMBL1237174 0.56 0.017 CHEMBL3091852 | CHEMBL1203 | |
| 0.437 | 0.085 | 0.437 | MAP kinase 1 inhibitor | 0.244 0.241 CHEMBL1442231 | ||
| 0.368 | 0.02 | 0.368 | Ca2+/calmodulin-dependent kinase II beta inhibitor | 0.169 0.105 CHEMBL1442231 0.19 0.085 CHEMBL3091852 | ||
| 0.365 | 0.021 | 0.424 | Anesthetic general | 0.371 0.02 CHEMBL1203 0.144 0.12 CHEMBL1442231 0.424 0.014 CHEMBL3544637 0.38 0.019 CHEMBL3091859 0.396 0.017 CHEMBL1237174 0.278 0.039 CHEMBL3091852 | CHEMBL3544637 | |
| 0.343 | 0.003 | 0.425 | Glutamate decarboxylase inhibitor | 0.176 0.009 CHEMBL2111041 0.246 0.004 CHEMBL3544855 0.12 0.021 CHEMBL3544856 0.425 0.003 CHEMBL1203 0.128 0.018 CHEMBL1442231 0.223 0.005 CHEMBL3544636 0.071 0.054 CHEMBL3544637 0.264 0.004 CHEMBL3091859 0.264 0.004 CHEMBL1237174 0.193 0.007 CHEMBL3091852 | CHEMBL1203 | |
| 0.434 | 0.106 | 0.434 | DNA polymerase beta inhibitor | 0.269 0.181 CHEMBL2111041 0.222 0.209 CHEMBL1203 0.366 0.133 CHEMBL1442231 0.288 0.171 CHEMBL3091859 0.312 0.159 CHEMBL3091852 | ||
| 0.402 | 0.076 | 0.646 | Antibacterial | 0.427 0.065 CHEMBL2111041 0.365 0.094 CHEMBL3544855 0.53 0.033 CHEMBL3544856 0.415 0.07 CHEMBL1203 0.413 0.071 CHEMBL1442231 0.221 0.206 CHEMBL3544636 0.646 0.013 CHEMBL3544637 0.466 0.051 CHEMBL3091859 0.312 0.126 CHEMBL1237174 0.423 0.067 CHEMBL3091852 | CHEMBL3544637 | |
| 0.34 | 0.023 | 0.34 | MAP kinase kinase 2 inhibitor | 0.196 0.085 CHEMBL1203 0.163 0.11 CHEMBL3544636 0.203 0.08 CHEMBL3091859 0.269 0.046 CHEMBL1237174 0.163 0.109 CHEMBL3091852 | ||
| 0.329 | 0.023 | 0.329 | Interleukin-1 receptor-associated protein kinase 1 inhibitor | 0.127 0.119 CHEMBL1442231 | ||
| 0.301 | 0.011 | 0.445 | Nitric-oxide synthase stimulant | 0.257 0.028 CHEMBL2111041 0.211 0.072 CHEMBL3544855 0.236 0.043 CHEMBL3544856 0.335 0.006 CHEMBL1203 0.284 0.016 CHEMBL1442231 0.445 0.003 CHEMBL3544636 0.336 0.006 CHEMBL3544637 0.211 0.072 CHEMBL3091859 0.295 0.013 CHEMBL1237174 0.255 0.029 CHEMBL3091852 | CHEMBL3544636 | |
| 0.402 | 0.115 | 0.402 | DNA directed DNA polymerase inhibitor | 0.254 0.189 CHEMBL2111041 0.222 0.211 CHEMBL1203 0.334 0.145 CHEMBL1442231 0.251 0.191 CHEMBL3091859 0.294 0.165 CHEMBL3091852 | ||
| 0.286 | 0.011 | 0.286 | MAP kinase kinase 3 inhibitor | 0.235 0.049 CHEMBL2111041 0.216 0.083 CHEMBL3544855 0.203 0.113 CHEMBL3544856 0.261 0.023 CHEMBL1203 0.267 0.019 CHEMBL1442231 0.249 0.033 CHEMBL3544636 | ||
| 0.269 | 0.004 | 0.269 | Myeloperoxidase inhibitor | 0.085 0.058 CHEMBL2111041 0.077 0.073 CHEMBL3544855 0.102 0.032 CHEMBL1203 0.094 0.043 CHEMBL1442231 0.143 0.012 CHEMBL3091859 0.149 0.011 CHEMBL1237174 0.1 0.034 CHEMBL3091852 | ||
| 0.274 | 0.015 | 0.274 | Alkaline phosphatase inhibitor | 0.107 0.105 CHEMBL2111041 0.184 0.04 CHEMBL1203 0.142 0.065 CHEMBL3544636 0.171 0.047 CHEMBL3544637 0.169 0.048 CHEMBL3091859 0.174 0.045 CHEMBL1237174 0.119 0.088 CHEMBL3091852 | ||
| 0.258 | 0.011 | 0.392 | Xanthine oxidase inhibitor | 0.111 0.052 CHEMBL2111041 0.094 0.066 CHEMBL3544855 0.288 0.008 CHEMBL1203 0.084 0.082 CHEMBL1442231 0.098 0.061 CHEMBL3544636 0.392 0.005 CHEMBL3544637 0.133 0.041 CHEMBL3091859 0.145 0.036 CHEMBL1237174 0.087 0.076 CHEMBL3091852 | CHEMBL3544637 | |
| 0.249 | 0.015 | 0.362 | Cystathionine beta-synthase inhibitor | 0.14 0.045 CHEMBL2111041 0.117 0.06 CHEMBL3544855 0.362 0.006 CHEMBL1203 0.09 0.089 CHEMBL1442231 0.128 0.052 CHEMBL3544636 0.206 0.023 CHEMBL3544637 0.249 0.015 CHEMBL3091859 0.313 0.009 CHEMBL1237174 0.18 0.03 CHEMBL3091852 | CHEMBL1203 | |
| 0.289 | 0.059 | 0.311 | Transcription factor STAT3 inhibitor | 0.271 0.069 CHEMBL1203 0.196 0.14 CHEMBL1442231 0.183 0.159 CHEMBL3544636 0.311 0.048 CHEMBL3091859 0.252 0.082 CHEMBL1237174 0.238 0.094 CHEMBL3091852 | CHEMBL3091859 | |
| 0.258 | 0.029 | 0.258 | Ca2+/calmodulin-dependent kinase II delta inhibitor | |||
| 0.243 | 0.014 | 0.27 | Cathepsin H inhibitor | 0.121 0.074 CHEMBL2111041 0.108 0.093 CHEMBL3544855 0.119 0.076 CHEMBL3544856 0.173 0.033 CHEMBL1203 0.2 0.022 CHEMBL1442231 0.105 0.099 CHEMBL3544636 0.27 0.012 CHEMBL3091859 0.225 0.017 CHEMBL1237174 0.247 0.014 CHEMBL3091852 | CHEMBL3091859 | |
| 0.234 | 0.01 | 0.4 | Histidine decarboxylase inhibitor | 0.087 0.038 CHEMBL2111041 0.061 0.06 CHEMBL3544855 0.4 0.004 CHEMBL1203 0.253 0.009 CHEMBL3544636 0.326 0.005 CHEMBL3091859 0.353 0.005 CHEMBL1237174 0.201 0.013 CHEMBL3091852 | CHEMBL1203 | |
| 0.256 | 0.035 | 0.256 | LIM domain kinase 1 inhibitor | 0.185 0.071 CHEMBL1203 0.173 0.078 CHEMBL1442231 0.139 0.109 CHEMBL3091859 0.165 0.084 CHEMBL1237174 0.167 0.082 CHEMBL3091852 | ||
| 0.283 | 0.066 | 0.287 | Transcription factor STAT inhibitor | 0.28 0.068 CHEMBL1203 0.198 0.141 CHEMBL1442231 0.287 0.063 CHEMBL3091859 0.242 0.093 CHEMBL1237174 0.225 0.106 CHEMBL3091852 | CHEMBL3091859 | |
| 0.236 | 0.019 | 0.421 | Cell wall synthesis inhibitor | 0.22 0.023 CHEMBL2111041 0.198 0.03 CHEMBL3544855 0.162 0.055 CHEMBL3544856 0.273 0.012 CHEMBL1203 0.212 0.026 CHEMBL1442231 0.194 0.033 CHEMBL3544636 0.421 0.005 CHEMBL3544637 0.202 0.029 CHEMBL3091859 0.221 0.023 CHEMBL1237174 0.227 0.021 CHEMBL3091852 | CHEMBL3544637 | |
| 0.222 | 0.015 | 0.296 | Carbonic anhydrase XV inhibitor | 0.267 0.01 CHEMBL1203 0.089 0.086 CHEMBL1442231 0.296 0.008 CHEMBL3091859 0.281 0.009 CHEMBL1237174 0.197 0.019 CHEMBL3091852 | CHEMBL3091859 | |
| 0.214 | 0.009 | 0.214 | Urease inhibitor | 0.117 0.048 CHEMBL2111041 0.099 0.069 CHEMBL3544855 0.115 0.05 CHEMBL3544856 0.133 0.033 CHEMBL1203 0.191 0.011 CHEMBL1442231 0.124 0.041 CHEMBL3544636 0.211 0.009 CHEMBL3091859 0.149 0.024 CHEMBL1237174 0.162 0.018 CHEMBL3091852 | ||
| 0.229 | 0.024 | 0.341 | MAO A inhibitor | 0.149 0.041 CHEMBL1442231 0.341 0.012 CHEMBL3091859 0.121 0.052 CHEMBL1237174 0.181 0.033 CHEMBL3091852 | CHEMBL3091859 | |
| 0.206 | 0.002 | 0.206 | S-adenosyl-L-methionine decarboxylase inhibitor | 0.118 0.006 CHEMBL2111041 0.093 0.019 CHEMBL3544855 0.083 0.031 CHEMBL3544856 0.115 0.007 CHEMBL1203 0.107 0.009 CHEMBL1442231 0.098 0.015 CHEMBL3544636 0.068 0.065 CHEMBL3544637 0.136 0.004 CHEMBL3091859 0.144 0.004 CHEMBL1237174 0.113 0.008 CHEMBL3091852 | ||
| 0.213 | 0.011 | 0.354 | Uric acid excretion stimulant | 0.354 0.004 CHEMBL1203 0.088 0.067 CHEMBL3544636 0.241 0.008 CHEMBL3544637 | CHEMBL1203 | |
| 0.223 | 0.034 | 0.309 | MAO inhibitor | 0.135 0.067 CHEMBL1442231 0.309 0.019 CHEMBL3091859 0.136 0.067 CHEMBL1237174 0.176 0.049 CHEMBL3091852 | CHEMBL3091859 | |
| 0.234 | 0.051 | 0.234 | CDC-like kinase 2 inhibitor | 0.139 0.101 CHEMBL1203 0.124 0.115 CHEMBL1442231 | ||
| 0.232 | 0.051 | 0.313 | Glyceraldehyde-3-phosphate dehydrogenase inhibitor | 0.181 0.092 CHEMBL2111041 0.175 0.1 CHEMBL3544855 0.303 0.023 CHEMBL1203 0.241 0.047 CHEMBL1442231 0.199 0.073 CHEMBL3544636 0.197 0.074 CHEMBL3544637 0.262 0.037 CHEMBL3091859 0.313 0.02 CHEMBL1237174 0.291 0.027 CHEMBL3091852 | CHEMBL1237174 | |
| 0.251 | 0.074 | 0.633 | Superoxide dismutase inhibitor | 0.276 0.06 CHEMBL2111041 0.213 0.104 CHEMBL3544855 0.633 0.005 CHEMBL1203 0.275 0.061 CHEMBL1442231 0.444 0.02 CHEMBL3544636 0.304 0.049 CHEMBL3091859 0.375 0.031 CHEMBL1237174 0.451 0.019 CHEMBL3091852 | CHEMBL1203 | |
| 0.173 | 0.005 | 0.249 | Xanthine dehydrogenase inhibitor | 0.073 0.029 CHEMBL2111041 0.249 0.004 CHEMBL1203 0.071 0.031 CHEMBL3544636 0.123 0.01 CHEMBL3544637 0.058 0.039 CHEMBL3091859 0.076 0.027 CHEMBL1237174 | CHEMBL1203 | |
| 0.243 | 0.088 | 0.443 | 5 Hydroxytryptamine uptake stimulant | 0.206 0.14 CHEMBL2111041 0.228 0.107 CHEMBL3544855 0.443 0.008 CHEMBL1203 0.234 0.098 CHEMBL1442231 0.287 0.052 CHEMBL3544636 0.299 0.045 CHEMBL3091859 0.435 0.009 CHEMBL1237174 0.389 0.016 CHEMBL3091852 | CHEMBL1203 | |
| 0.179 | 0.025 | 0.259 | Falcipain 3 inhibitor | 0.126 0.05 CHEMBL2111041 0.096 0.075 CHEMBL3544855 0.163 0.031 CHEMBL1203 0.259 0.007 CHEMBL1442231 0.166 0.03 CHEMBL3544636 0.159 0.032 CHEMBL3091859 0.148 0.038 CHEMBL1237174 0.233 0.01 CHEMBL3091852 | CHEMBL1442231 | |
| 0.2 | 0.047 | 0.2 | Protein kinase C nu inhibitor | |||
| 0.166 | 0.014 | 0.227 | DOPA decarboxylase inhibitor | 0.111 0.056 CHEMBL2111041 0.1 0.075 CHEMBL3544855 0.202 0.006 CHEMBL1203 0.115 0.051 CHEMBL1442231 0.112 0.056 CHEMBL3544636 0.207 0.006 CHEMBL3091859 0.227 0.004 CHEMBL1237174 0.195 0.007 CHEMBL3091852 | CHEMBL1237174 | |
| 0.238 | 0.087 | 0.727 | Aldehyde oxidase inhibitor | 0.675 0.01 CHEMBL1203 0.3 0.066 CHEMBL3544636 0.519 0.03 CHEMBL3091859 0.727 0.006 CHEMBL1237174 0.458 0.039 CHEMBL3091852 | CHEMBL1237174 | |
| 0.172 | 0.021 | 0.221 | Protein kinase C gamma inhibitor | 0.221 0.01 CHEMBL1203 0.107 0.065 CHEMBL1442231 0.104 0.07 CHEMBL3544636 0.182 0.018 CHEMBL3544637 0.131 0.044 CHEMBL1237174 0.123 0.05 CHEMBL3091852 | CHEMBL1203 | |
| 0.166 | 0.017 | 0.771 | Porphobilinogen synthase inhibitor | 0.28 0.006 CHEMBL2111041 0.336 0.005 CHEMBL3544855 0.771 0.002 CHEMBL1203 0.185 0.014 CHEMBL1442231 0.346 0.004 CHEMBL3544636 0.068 0.057 CHEMBL3544637 0.234 0.009 CHEMBL3091859 0.266 0.007 CHEMBL1237174 0.378 0.004 CHEMBL3091852 | CHEMBL1203 | |
| 0.152 | 0.007 | 0.198 | GABA aminotransferase inhibitor | 0.119 0.016 CHEMBL2111041 0.155 0.007 CHEMBL3544855 0.073 0.056 CHEMBL3544856 0.161 0.006 CHEMBL1203 0.075 0.053 CHEMBL1442231 0.074 0.055 CHEMBL3544636 0.114 0.019 CHEMBL3544637 0.198 0.004 CHEMBL3091859 0.174 0.005 CHEMBL1237174 0.137 0.01 CHEMBL3091852 | CHEMBL3091859 | |
| 0.182 | 0.037 | 0.379 | Monophenol monooxygenase inhibitor | 0.228 0.027 CHEMBL2111041 0.167 0.041 CHEMBL3544855 0.099 0.077 CHEMBL3544856 0.179 0.038 CHEMBL1203 0.095 0.08 CHEMBL3544636 0.379 0.012 CHEMBL3544637 0.165 0.042 CHEMBL3091859 0.143 0.05 CHEMBL1237174 0.125 0.058 CHEMBL3091852 | CHEMBL3544637 | |
| 0.171 | 0.027 | 0.676 | GABA C receptor agonist | 0.181 0.024 CHEMBL2111041 0.329 0.008 CHEMBL3544855 0.676 0.002 CHEMBL1203 0.115 0.053 CHEMBL1442231 0.461 0.004 CHEMBL3544636 0.112 0.055 CHEMBL3544637 0.224 0.016 CHEMBL3091859 0.53 0.003 CHEMBL1237174 0.333 0.008 CHEMBL3091852 | CHEMBL1203 | |
| 0.166 | 0.027 | 0.284 | Check point kinase 2 inhibitor | 0.224 0.013 CHEMBL1442231 0.133 0.04 CHEMBL3091859 0.284 0.007 CHEMBL3091852 | CHEMBL3091852 | |
| 0.278 | 0.144 | 0.324 | 15-Lipoxygenase inhibitor | 0.317 0.12 CHEMBL2111041 0.25 0.164 CHEMBL1203 0.324 0.115 CHEMBL3091859 0.289 0.138 CHEMBL1237174 0.289 0.138 CHEMBL3091852 | CHEMBL3091859 | |
| 0.172 | 0.041 | 0.172 | Protein kinase (CK1) delta inhibitor | |||
| 0.133 | 0.005 | 0.133 | Fatty acid synthase inhibitor | 0.08 0.019 CHEMBL1203 0.074 0.023 CHEMBL1442231 0.074 0.022 CHEMBL3544637 0.07 0.026 CHEMBL3091859 0.076 0.021 CHEMBL1237174 0.071 0.025 CHEMBL3091852 | ||
| 0.156 | 0.032 | 0.157 | Death-associated protein kinase 1 inhibitor | 0.123 0.102 CHEMBL2111041 0.132 0.077 CHEMBL1203 0.157 0.03 CHEMBL1442231 0.132 0.076 CHEMBL3544636 | CHEMBL1442231 | |
| 0.125 | 0.004 | 0.125 | Diamine oxidase inhibitor | 0.046 0.018 CHEMBL2111041 0.061 0.009 CHEMBL1203 0.064 0.008 CHEMBL1442231 0.036 0.029 CHEMBL3544636 0.124 0.004 CHEMBL3091859 0.086 0.005 CHEMBL1237174 0.075 0.005 CHEMBL3091852 | ||
| 0.166 | 0.046 | 0.75 | Alpha-N-acetylglucosaminidase inhibitor | 0.219 0.029 CHEMBL2111041 0.131 0.068 CHEMBL3544855 0.392 0.009 CHEMBL3544856 0.75 0.003 CHEMBL1203 0.251 0.023 CHEMBL1442231 0.374 0.01 CHEMBL3544636 0.716 0.003 CHEMBL3544637 0.596 0.004 CHEMBL3091859 0.635 0.004 CHEMBL1237174 0.727 0.003 CHEMBL3091852 | CHEMBL1203 | |
| 0.131 | 0.011 | 0.163 | DNA gyrase inhibitor | 0.163 0.007 CHEMBL1203 0.063 0.045 CHEMBL3544636 0.076 0.03 CHEMBL3091859 0.072 0.034 CHEMBL1237174 | CHEMBL1203 | |
| 0.186 | 0.069 | 0.322 | Dual specificity phosphatase 3 inhibitor | 0.179 0.074 CHEMBL2111041 0.17 0.081 CHEMBL3544855 0.247 0.041 CHEMBL1203 0.147 0.099 CHEMBL1442231 0.322 0.025 CHEMBL1237174 | CHEMBL1237174 | |
| 0.148 | 0.037 | 0.148 | MAP kinase 13 inhibitor | |||
| 0.187 | 0.077 | 0.276 | Growth factor agonist | 0.276 0.022 CHEMBL3544856 0.271 0.024 CHEMBL1203 0.206 0.058 CHEMBL1442231 0.272 0.023 CHEMBL3544636 0.174 0.096 CHEMBL3544637 | CHEMBL3544856 | |
| 0.137 | 0.029 | 0.171 | Nitric-oxide synthase inhibitor | 0.09 0.078 CHEMBL1203 0.143 0.025 CHEMBL3091859 0.171 0.016 CHEMBL1237174 0.096 0.066 CHEMBL3091852 | CHEMBL1237174 | |
| 0.165 | 0.056 | 0.274 | GABA C receptor rho-2 antagonist | 0.141 0.086 CHEMBL2111041 0.264 0.009 CHEMBL1203 0.153 0.07 CHEMBL1442231 0.269 0.008 CHEMBL3544636 0.17 0.051 CHEMBL3091859 0.274 0.008 CHEMBL1237174 0.22 0.02 CHEMBL3091852 | CHEMBL1237174 | |
| 0.127 | 0.021 | 0.162 | Ornithine decarboxylase inhibitor | 0.104 0.04 CHEMBL2111041 0.09 0.056 CHEMBL3544855 0.162 0.008 CHEMBL1203 0.104 0.04 CHEMBL3544636 0.09 0.056 CHEMBL3544637 0.12 0.026 CHEMBL3091859 0.137 0.016 CHEMBL1237174 0.097 0.048 CHEMBL3091852 | CHEMBL1203 | |
| 0.125 | 0.02 | 0.151 | Carbonic anhydrase V inhibitor | 0.113 0.023 CHEMBL1203 0.131 0.019 CHEMBL3091859 0.151 0.014 CHEMBL1237174 0.086 0.033 CHEMBL3091852 | CHEMBL1237174 | |
| 0.11 | 0.004 | 0.11 | DNA gyrase subunit B inhibitor | 0.08 0.005 CHEMBL1203 0.065 0.007 CHEMBL3544636 0.044 0.018 CHEMBL3091859 0.042 0.02 CHEMBL1237174 | ||
| 0.121 | 0.018 | 0.139 | Carbonic anhydrase VA inhibitor | 0.109 0.021 CHEMBL1203 0.121 0.018 CHEMBL3091859 0.139 0.013 CHEMBL1237174 0.088 0.031 CHEMBL3091852 | CHEMBL1237174 | |
| 0.196 | 0.095 | 0.321 | Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor | 0.321 0.044 CHEMBL1203 | CHEMBL1203 | |
| 0.106 | 0.006 | 0.224 | CDK5/p25 inhibitor | 0.183 0.004 CHEMBL1442231 0.224 0.004 CHEMBL3091859 0.056 0.017 CHEMBL1237174 0.134 0.005 CHEMBL3091852 | CHEMBL3091859 | |
| 0.115 | 0.017 | 0.125 | Carbonic anhydrase IX inhibitor | 0.047 0.045 CHEMBL1442231 0.125 0.015 CHEMBL3091859 0.075 0.03 CHEMBL1237174 0.062 0.036 CHEMBL3091852 | CHEMBL3091859 | |
| 0.154 | 0.061 | 0.264 | Mannose-6-phosphate isomerase inhibitor | 0.178 0.044 CHEMBL2111041 0.136 0.078 CHEMBL3544855 0.264 0.009 CHEMBL3544856 0.26 0.01 CHEMBL1203 0.133 0.081 CHEMBL1442231 0.128 0.088 CHEMBL3544636 0.254 0.011 CHEMBL3544637 0.139 0.075 CHEMBL3091859 0.205 0.028 CHEMBL1237174 0.203 0.029 CHEMBL3091852 | CHEMBL3544856 | |
| 0.181 | 0.087 | 0.181 | Ca2+/calmodulin-dependent protein kinase inhibitor | 0.176 0.091 CHEMBL1203 | ||
| 0.118 | 0.025 | 0.118 | Rho-associated kinase II inhibitor | 0.081 0.044 CHEMBL1442231 0.071 0.055 CHEMBL3544636 | ||
| 0.193 | 0.103 | 0.309 | Dyrk kinase inhibitor | 0.309 0.05 CHEMBL1203 | CHEMBL1203 | |
| 0.168 | 0.079 | 0.2 | Tumour necrosis factor antagonist | 0.2 0.054 CHEMBL1203 0.17 0.077 CHEMBL1237174 | CHEMBL1203 | |
| 0.097 | 0.008 | 0.097 | Myc inhibitor | 0.056 0.034 CHEMBL2111041 0.053 0.04 CHEMBL3544855 0.082 0.012 CHEMBL1203 0.073 0.017 CHEMBL1442231 0.062 0.027 CHEMBL3091859 0.055 0.036 CHEMBL3091852 | ||
| 0.126 | 0.039 | 0.204 | Acetylcholine release stimulant | 0.183 0.005 CHEMBL1203 0.144 0.02 CHEMBL1442231 0.141 0.023 CHEMBL3544636 0.204 0.004 CHEMBL3544637 0.097 0.095 CHEMBL3091859 0.134 0.03 CHEMBL1237174 0.132 0.032 CHEMBL3091852 | CHEMBL3544637 | |
| 0.152 | 0.065 | 0.183 | Glycogen synthase kinase-3 alpha inhibitor | 0.183 0.047 CHEMBL1203 | CHEMBL1203 | |
| 0.145 | 0.059 | 0.476 | Cyclin-dependent kinase inhibitor | 0.253 0.027 CHEMBL1442231 0.476 0.008 CHEMBL3091859 0.444 0.009 CHEMBL3091852 | CHEMBL3091859 | |
| 0.086 | 0.005 | 0.091 | Vascular adhesion protein 1 inhibitor | 0.035 0.034 CHEMBL1203 0.035 0.034 CHEMBL1442231 0.091 0.004 CHEMBL3091859 0.082 0.005 CHEMBL1237174 0.053 0.013 CHEMBL3091852 | CHEMBL3091859 | |
| 0.163 | 0.081 | 0.244 | Dual specificity phosphatase inhibitor | 0.167 0.077 CHEMBL2111041 0.168 0.076 CHEMBL3544855 0.244 0.039 CHEMBL1203 0.145 0.1 CHEMBL1442231 0.207 0.051 CHEMBL1237174 | CHEMBL1203 | |
| 0.2 | 0.119 | 0.279 | Neuropeptide Y2 antagonist | 0.185 0.148 CHEMBL1203 0.211 0.101 CHEMBL1442231 0.279 0.031 CHEMBL3091859 0.269 0.039 CHEMBL1237174 0.276 0.033 CHEMBL3091852 | CHEMBL3091859 | |
| 0.101 | 0.022 | 0.104 | HIV-1 integrase (Strand Transfer) inhibitor | 0.095 0.024 CHEMBL1203 0.104 0.021 CHEMBL1237174 | CHEMBL1237174 | |
| 0.104 | 0.026 | 0.139 | Carbonic anhydrase inhibitor | 0.139 0.018 CHEMBL3091859 0.083 0.033 CHEMBL1237174 0.064 0.044 CHEMBL3091852 | CHEMBL3091859 | |
| 0.205 | 0.127 | 0.399 | Tyrosine 3 hydroxylase inhibitor | 0.277 0.046 CHEMBL2111041 0.242 0.076 CHEMBL3544855 0.283 0.042 CHEMBL1203 0.208 0.121 CHEMBL1442231 0.348 0.017 CHEMBL3544636 0.316 0.026 CHEMBL3091859 0.399 0.008 CHEMBL1237174 0.385 0.01 CHEMBL3091852 | CHEMBL1237174 | |
| 0.225 | 0.149 | 0.683 | Vasodilator, peripheral | 0.571 0.019 CHEMBL1203 0.272 0.112 CHEMBL3544636 0.683 0.007 CHEMBL3544637 0.283 0.106 CHEMBL3091859 0.462 0.037 CHEMBL1237174 0.267 0.115 CHEMBL3091852 | CHEMBL3544637 | |
| 0.09 | 0.014 | 0.09 | Enoyl-[acyl-carrier-protein] reductase inhibitor | 0.064 0.036 CHEMBL3091859 0.074 0.024 CHEMBL1237174 | ||
| 0.111 | 0.036 | 0.111 | Stem cell growth factor agonist | 0.1 0.045 CHEMBL1442231 0.079 0.067 CHEMBL3544636 | ||
| 0.238 | 0.163 | 0.365 | Beta lactamase inhibitor | 0.365 0.111 CHEMBL1442231 0.283 0.141 CHEMBL3091859 0.307 0.132 CHEMBL3091852 | CHEMBL1442231 | |
| 0.081 | 0.006 | 0.081 | Plasmepsin II inhibitor | 0.068 0.009 CHEMBL1442231 0.077 0.006 CHEMBL3091859 0.047 0.02 CHEMBL1237174 0.058 0.013 CHEMBL3091852 | ||
| 0.087 | 0.013 | 0.284 | Plasminogen activator inhibitor antagonist | 0.175 0.005 CHEMBL1203 0.06 0.024 CHEMBL3544636 0.284 0.004 CHEMBL3091859 0.248 0.004 CHEMBL1237174 | CHEMBL3091859 | |
| 0.213 | 0.138 | 0.373 | Insulysin inhibitor | 0.216 0.134 CHEMBL2111041 0.266 0.083 CHEMBL3544855 0.365 0.029 CHEMBL1203 0.243 0.103 CHEMBL1442231 0.373 0.027 CHEMBL3544636 0.246 0.1 CHEMBL3091859 0.294 0.062 CHEMBL1237174 0.314 0.05 CHEMBL3091852 | CHEMBL3544636 | |
| 0.094 | 0.02 | 0.094 | Carbonic anhydrase I inhibitor | 0.049 0.044 CHEMBL3544636 0.092 0.021 CHEMBL3091859 0.071 0.029 CHEMBL1237174 | ||
| 0.1 | 0.026 | 0.117 | HIV-1 integrase (3'-Processing) inhibitor | 0.095 0.028 CHEMBL1203 0.056 0.052 CHEMBL3091859 0.117 0.02 CHEMBL1237174 | CHEMBL1237174 | |
| 0.1 | 0.029 | 0.133 | D-Ala-D-Ala ligase inhibitor | 0.096 0.034 CHEMBL2111041 0.078 0.075 CHEMBL3544855 0.133 0.009 CHEMBL1203 0.105 0.024 CHEMBL1442231 0.082 0.062 CHEMBL3544636 0.101 0.028 CHEMBL3091859 0.116 0.016 CHEMBL1237174 0.123 0.012 CHEMBL3091852 | CHEMBL1203 | |
| 0.086 | 0.015 | 0.113 | Carbonic anhydrase XIV inhibitor | 0.092 0.013 CHEMBL1203 0.048 0.035 CHEMBL3544636 0.113 0.008 CHEMBL3544637 0.068 0.021 CHEMBL3091859 0.08 0.017 CHEMBL1237174 0.044 0.041 CHEMBL3091852 | CHEMBL3544637 | |
| 0.077 | 0.007 | 0.087 | Dihydropteroate synthase inhibitor | 0.071 0.008 CHEMBL1203 0.052 0.016 CHEMBL3544636 0.067 0.009 CHEMBL3091859 0.087 0.005 CHEMBL1237174 0.048 0.018 CHEMBL3091852 | CHEMBL1237174 | |
| 0.148 | 0.079 | 0.382 | Dual specificity tyrosine-phosphorylation-regulated kinase 4 inhibitor | 0.163 0.069 CHEMBL1203 0.323 0.021 CHEMBL1442231 0.382 0.01 CHEMBL3091852 | CHEMBL3091852 | |
| 0.087 | 0.018 | 0.148 | Exportin-1 inhibitor | 0.068 0.047 CHEMBL2111041 0.09 0.015 CHEMBL1203 0.116 0.005 CHEMBL1442231 0.068 0.047 CHEMBL3544636 0.095 0.011 CHEMBL3091859 0.109 0.006 CHEMBL1237174 0.148 0.004 CHEMBL3091852 | CHEMBL3091852 | |
| 0.088 | 0.019 | 0.161 | Carbonic anhydrase VB inhibitor | 0.12 0.012 CHEMBL1203 0.116 0.013 CHEMBL3091859 0.161 0.008 CHEMBL1237174 0.074 0.025 CHEMBL3091852 | CHEMBL1237174 | |
| 0.08 | 0.012 | 0.081 | Lysine-specific demethylase 1A inhibitor | 0.071 0.017 CHEMBL3091859 0.081 0.012 CHEMBL1237174 | CHEMBL1237174 | |
| 0.076 | 0.009 | 0.097 | Factor XIIIa inhibitor | 0.05 0.016 CHEMBL3544636 0.097 0.006 CHEMBL3091859 0.052 0.015 CHEMBL1237174 0.033 0.032 CHEMBL3091852 | CHEMBL3091859 | |
| 0.106 | 0.039 | 0.139 | Polo-like kinase-1 inhibitor | 0.089 0.063 CHEMBL1203 0.139 0.021 CHEMBL1442231 0.085 0.072 CHEMBL3544636 0.084 0.074 CHEMBL1237174 0.101 0.044 CHEMBL3091852 | CHEMBL1442231 | |
| 0.157 | 0.09 | 0.301 | 3C-like protease (Human coronavirus) inhibitor | 0.301 0.011 CHEMBL1203 0.2 0.051 CHEMBL1442231 0.184 0.062 CHEMBL3544636 0.183 0.062 CHEMBL3091859 0.207 0.048 CHEMBL1237174 0.269 0.02 CHEMBL3091852 | CHEMBL1203 | |
| 0.102 | 0.035 | 0.159 | Inducible nitric-oxide synthase inhibitor | 0.086 0.053 CHEMBL1203 0.106 0.032 CHEMBL3091859 0.159 0.014 CHEMBL1237174 0.075 0.072 CHEMBL3091852 | CHEMBL1237174 | |
| 0.138 | 0.074 | 0.138 | Ribosomal protein S6 kinase inhibitor | |||
| 0.095 | 0.032 | 0.122 | Estrogen-related receptor beta agonist | 0.105 0.02 CHEMBL2111041 0.102 0.022 CHEMBL3544855 0.084 0.054 CHEMBL3544856 0.089 0.043 CHEMBL1203 0.096 0.03 CHEMBL1442231 0.117 0.011 CHEMBL3544636 0.102 0.022 CHEMBL3091859 0.112 0.014 CHEMBL1237174 0.122 0.009 CHEMBL3091852 | CHEMBL3091852 | |
| 0.177 | 0.114 | 0.423 | Cyclic AMP phosphodiesterase inhibitor | 0.338 0.029 CHEMBL1203 0.423 0.014 CHEMBL3544637 0.236 0.071 CHEMBL3091859 0.313 0.037 CHEMBL1237174 0.255 0.061 CHEMBL3091852 | CHEMBL3544637 | |
| 0.12 | 0.058 | 0.142 | DNA intercalator | 0.142 0.046 CHEMBL3544637 | CHEMBL3544637 | |
| 0.115 | 0.053 | 0.161 | MAO B inhibitor | 0.161 0.034 CHEMBL3091859 0.091 0.065 CHEMBL1237174 | CHEMBL3091859 | |
| 0.176 | 0.116 | 0.283 | 5 Hydroxytryptamine 3E antagonist | 0.19 0.081 CHEMBL1203 0.184 0.096 CHEMBL1442231 0.218 0.038 CHEMBL3091859 0.283 0.007 CHEMBL1237174 0.253 0.015 CHEMBL3091852 | CHEMBL1237174 | |
| 0.205 | 0.146 | 0.375 | Hypoxia-inducible factor 1 alpha inhibitor | 0.31 0.061 CHEMBL1203 0.301 0.065 CHEMBL3544636 0.375 0.037 CHEMBL3544637 0.224 0.124 CHEMBL3091859 0.253 0.098 CHEMBL1237174 | CHEMBL3544637 | |
| 0.085 | 0.025 | 0.085 | MAP kinase kinase 10 inhibitor | |||
| 0.097 | 0.038 | 0.169 | CYP2A6 inhibitor | 0.169 0.012 CHEMBL1203 0.078 0.05 CHEMBL1442231 0.069 0.061 CHEMBL3544636 0.128 0.023 CHEMBL1237174 0.069 0.061 CHEMBL3091852 | CHEMBL1203 | |
| 0.083 | 0.024 | 0.083 | Carbonic anhydrase XII inhibitor | 0.047 0.04 CHEMBL3544637 0.076 0.027 CHEMBL3091859 0.058 0.034 CHEMBL1237174 | ||
| 0.138 | 0.082 | 0.174 | Thiol protease inhibitor | 0.146 0.073 CHEMBL2111041 0.129 0.098 CHEMBL3544855 0.122 0.112 CHEMBL3544856 0.169 0.055 CHEMBL1203 0.143 0.076 CHEMBL1442231 0.158 0.062 CHEMBL3544636 0.135 0.087 CHEMBL3091859 0.147 0.072 CHEMBL1237174 0.174 0.052 CHEMBL3091852 | CHEMBL3091852 | |
| 0.081 | 0.025 | 0.115 | Carbonic anhydrase II inhibitor | 0.115 0.015 CHEMBL3091859 0.071 0.029 CHEMBL1237174 0.058 0.037 CHEMBL3091852 | CHEMBL3091859 | |
| 0.153 | 0.099 | 0.153 | CDC-like kinase 4 inhibitor | |||
| 0.118 | 0.064 | 0.305 | Protein kinase (CK2) alpha inhibitor | 0.305 0.011 CHEMBL1203 0.136 0.051 CHEMBL3091859 0.107 0.071 CHEMBL1237174 0.104 0.073 CHEMBL3091852 | CHEMBL1203 | |
| 0.15 | 0.096 | 0.166 | Cyclin-dependent kinase 3 inhibitor | 0.166 0.066 CHEMBL3544856 0.157 0.08 CHEMBL1203 0.166 0.066 CHEMBL1442231 0.166 0.066 CHEMBL3544636 0.139 0.125 CHEMBL3091852 | CHEMBL3544636 | |
| 0.136 | 0.086 | 0.277 | Cytidine deaminase inhibitor | 0.277 0.023 CHEMBL1203 0.115 0.106 CHEMBL1442231 0.118 0.102 CHEMBL3544636 0.114 0.108 CHEMBL3091859 0.196 0.05 CHEMBL1237174 0.158 0.069 CHEMBL3091852 | CHEMBL1203 | |
| 0.132 | 0.082 | 0.132 | Protein kinase (CK1) inhibitor | 0.107 0.102 CHEMBL1203 | ||
| 0.073 | 0.024 | 0.161 | Cyclin D1 inhibitor | 0.161 0.004 CHEMBL1442231 0.077 0.02 CHEMBL3091859 0.065 0.035 CHEMBL1237174 0.132 0.004 CHEMBL3091852 | CHEMBL1442231 | |
| 0.093 | 0.044 | 0.197 | Carbonic anhydrase VI inhibitor | 0.148 0.021 CHEMBL1203 0.072 0.069 CHEMBL3544637 0.139 0.023 CHEMBL3091859 0.197 0.013 CHEMBL1237174 0.092 0.045 CHEMBL3091852 | CHEMBL1237174 | |
| 0.11 | 0.062 | 0.488 | Ferrochelatase inhibitor | 0.196 0.023 CHEMBL2111041 0.177 0.028 CHEMBL3544855 0.488 0.003 CHEMBL1203 0.13 0.047 CHEMBL1442231 0.229 0.016 CHEMBL3544636 0.303 0.007 CHEMBL3091859 0.388 0.004 CHEMBL1237174 0.391 0.004 CHEMBL3091852 | CHEMBL1203 | |
| 0.104 | 0.057 | 0.27 | GABA C receptor rho-1 antagonist | 0.099 0.063 CHEMBL2111041 0.27 0.004 CHEMBL1203 0.095 0.07 CHEMBL1442231 0.236 0.005 CHEMBL3544636 0.123 0.038 CHEMBL3091859 0.23 0.005 CHEMBL1237174 0.172 0.014 CHEMBL3091852 | CHEMBL1203 | |
| 0.053 | 0.006 | 0.102 | Methionyl aminopeptidase 2 inhibitor | 0.102 0.004 CHEMBL1203 0.061 0.005 CHEMBL1442231 0.026 0.017 CHEMBL1237174 0.045 0.008 CHEMBL3091852 | CHEMBL1203 | |
| 0.066 | 0.019 | 0.12 | Topoisomerase II beta inhibitor | 0.12 0.007 CHEMBL1203 0.06 0.022 CHEMBL1442231 0.08 0.013 CHEMBL3544636 0.054 0.028 CHEMBL3544637 0.068 0.017 CHEMBL3091859 0.099 0.009 CHEMBL1237174 0.093 0.01 CHEMBL3091852 | CHEMBL1203 | |
| 0.101 | 0.054 | 0.154 | Lanosterol 14 alpha demethylase inhibitor | 0.084 0.083 CHEMBL2111041 0.154 0.01 CHEMBL1203 0.099 0.057 CHEMBL1442231 0.151 0.011 CHEMBL3544636 0.084 0.083 CHEMBL3544637 0.131 0.021 CHEMBL1237174 0.105 0.048 CHEMBL3091852 | CHEMBL1203 | |
| 0.069 | 0.023 | 0.069 | Cyclin A1 inhibitor | 0.062 0.034 CHEMBL3091859 0.064 0.031 CHEMBL1237174 0.056 0.048 CHEMBL3091852 | ||
| 0.152 | 0.108 | 0.393 | Succinate dehydrogenase inhibitor | 0.191 0.057 CHEMBL2111041 0.196 0.052 CHEMBL3544855 0.138 0.136 CHEMBL3544856 0.393 0.004 CHEMBL1203 0.156 0.101 CHEMBL1442231 0.228 0.031 CHEMBL3544636 0.144 0.124 CHEMBL3544637 0.241 0.026 CHEMBL3091859 0.302 0.01 CHEMBL1237174 0.296 0.011 CHEMBL3091852 | CHEMBL1203 | |
| 0.223 | 0.18 | 0.417 | Calcium channel activator | 0.417 0.019 CHEMBL1203 0.267 0.127 CHEMBL3544636 0.228 0.174 CHEMBL3544637 0.241 0.158 CHEMBL3091859 0.381 0.032 CHEMBL1237174 0.327 0.067 CHEMBL3091852 | CHEMBL1203 | |
| 0.156 | 0.114 | 0.3 | I kappa B kinase epsilon inhibitor | 0.3 0.015 CHEMBL1203 0.158 0.111 CHEMBL1442231 0.201 0.07 CHEMBL3544636 0.179 0.09 CHEMBL1237174 0.169 0.1 CHEMBL3091852 | CHEMBL1203 | |
| 0.107 | 0.068 | 0.271 | GABA C receptor antagonist | 0.102 0.075 CHEMBL2111041 0.263 0.005 CHEMBL1203 0.098 0.082 CHEMBL1442231 0.22 0.009 CHEMBL3544636 0.148 0.031 CHEMBL3091859 0.271 0.005 CHEMBL1237174 0.209 0.011 CHEMBL3091852 | CHEMBL1237174 | |
| 0.153 | 0.115 | 0.348 | DNA methylase inhibitor | 0.158 0.11 CHEMBL3544855 0.278 0.035 CHEMBL1203 0.227 0.062 CHEMBL3544636 0.348 0.017 CHEMBL3544637 0.238 0.055 CHEMBL1237174 0.142 0.125 CHEMBL3091852 | CHEMBL3544637 | |
| 0.104 | 0.066 | 0.104 | Cyclin-dependent kinase 2 inhibitor | 0.096 0.074 CHEMBL1442231 0.092 0.08 CHEMBL3091859 | ||
| 0.066 | 0.029 | 0.209 | Mannitol-1-phosphate 5-dehydrogenase inhibitor | 0.063 0.031 CHEMBL2111041 0.139 0.009 CHEMBL3544856 0.148 0.009 CHEMBL1203 0.058 0.037 CHEMBL1442231 0.088 0.017 CHEMBL3544636 0.209 0.006 CHEMBL3544637 0.072 0.024 CHEMBL3091859 0.153 0.008 CHEMBL1237174 0.101 0.014 CHEMBL3091852 | CHEMBL3544637 | |
| 0.061 | 0.025 | 0.526 | Aconitate hydratase inhibitor | 0.071 0.018 CHEMBL2111041 0.114 0.006 CHEMBL3544855 0.048 0.043 CHEMBL3544856 0.526 0.001 CHEMBL1203 0.048 0.043 CHEMBL1442231 0.146 0.004 CHEMBL3544636 0.064 0.023 CHEMBL3544637 0.058 0.028 CHEMBL3091859 0.137 0.005 CHEMBL1237174 0.081 0.013 CHEMBL3091852 | CHEMBL1203 | |
| 0.081 | 0.046 | 0.081 | Rho-associated kinase inhibitor | |||
| 0.102 | 0.067 | 0.459 | Beta glucuronidase inhibitor | 0.103 0.065 CHEMBL2111041 0.103 0.065 CHEMBL3544856 0.119 0.047 CHEMBL1203 0.113 0.053 CHEMBL1442231 0.459 0.004 CHEMBL3544637 0.099 0.071 CHEMBL1237174 0.106 0.061 CHEMBL3091852 | CHEMBL3544637 | |
| 0.113 | 0.078 | 0.354 | Aldehyde dehydrogenase inhibitor | 0.354 0.007 CHEMBL1203 0.257 0.017 CHEMBL3544636 0.211 0.025 CHEMBL3544637 0.137 0.056 CHEMBL3091859 0.271 0.015 CHEMBL1237174 0.127 0.064 CHEMBL3091852 | CHEMBL1203 | |
| 0.175 | 0.141 | 0.265 | Calpain inhibitor | 0.174 0.143 CHEMBL1203 0.243 0.072 CHEMBL1442231 0.209 0.105 CHEMBL3544636 0.212 0.102 CHEMBL3091859 0.227 0.088 CHEMBL1237174 0.265 0.052 CHEMBL3091852 | CHEMBL3091852 | |
| 0.065 | 0.03 | 0.089 | Botulinum neurotoxin type A inhibitor | 0.076 0.02 CHEMBL1203 0.078 0.018 CHEMBL1442231 0.089 0.012 CHEMBL3544636 0.07 0.025 CHEMBL3091859 0.073 0.022 CHEMBL1237174 0.086 0.014 CHEMBL3091852 | CHEMBL3544636 | |
| 0.056 | 0.022 | 0.057 | Carbonic anhydrase VII inhibitor | 0.054 0.024 CHEMBL3091859 0.057 0.021 CHEMBL1237174 | CHEMBL1237174 | |
| 0.134 | 0.1 | 0.203 | Ca2+-transporting ATPase inhibitor | 0.129 0.124 CHEMBL2111041 0.13 0.119 CHEMBL3544855 0.203 0.003 CHEMBL1203 0.131 0.115 CHEMBL1442231 0.138 0.082 CHEMBL3544636 0.183 0.005 CHEMBL3544637 0.157 0.029 CHEMBL3091859 0.188 0.005 CHEMBL1237174 0.171 0.012 CHEMBL3091852 | CHEMBL1203 | |
| 0.092 | 0.06 | 0.144 | Protein kinase C delta inhibitor | 0.144 0.024 CHEMBL1203 0.117 0.039 CHEMBL3544637 | CHEMBL1203 | |
| 0.087 | 0.057 | 0.142 | Granulocyte macrophage colony stimulating factor agonist | 0.079 0.078 CHEMBL2111041 0.133 0.009 CHEMBL1203 0.085 0.063 CHEMBL1442231 0.114 0.02 CHEMBL3544636 0.096 0.04 CHEMBL3091859 0.142 0.007 CHEMBL1237174 0.12 0.016 CHEMBL3091852 | CHEMBL1237174 | |
| 0.236 | 0.209 | 0.332 | MAP kinase kinase 6 inhibitor | 0.332 0.107 CHEMBL1203 | CHEMBL1203 | |
| 0.134 | 0.108 | 0.218 | Arachidonic acid antagonist | 0.154 0.084 CHEMBL2111041 0.159 0.078 CHEMBL3544855 0.218 0.019 CHEMBL1203 0.13 0.113 CHEMBL1442231 0.173 0.062 CHEMBL3544636 0.16 0.077 CHEMBL3544637 0.178 0.056 CHEMBL3091859 0.215 0.021 CHEMBL1237174 0.204 0.03 CHEMBL3091852 | CHEMBL1203 | |
| 0.094 | 0.068 | 0.477 | UDP-glucose 4-epimerase inhibitor | 0.17 0.023 CHEMBL3544856 0.409 0.005 CHEMBL1203 0.105 0.055 CHEMBL1442231 0.103 0.057 CHEMBL3544636 0.477 0.003 CHEMBL3544637 0.201 0.018 CHEMBL3091859 0.316 0.009 CHEMBL1237174 0.301 0.01 CHEMBL3091852 | CHEMBL3544637 | |
| 0.062 | 0.037 | 0.12 | Glutamate (mGluR1) antagonist | 0.12 0.011 CHEMBL1203 0.077 0.025 CHEMBL3544636 0.075 0.027 CHEMBL1237174 | CHEMBL1203 | |
| 0.03 | 0.006 | 0.06 | ICAM 1 antagonist | 0.034 0.005 CHEMBL1203 0.06 0.004 CHEMBL3544636 0.026 0.01 CHEMBL1237174 | CHEMBL3544636 | |
| 0.038 | 0.014 | 0.11 | Methionyl aminopeptidase 1 inhibitor | 0.03 0.027 CHEMBL3544856 0.048 0.007 CHEMBL1203 0.11 0.004 CHEMBL1442231 0.033 0.02 CHEMBL1237174 0.065 0.004 CHEMBL3091852 | CHEMBL1442231 | |
| 0.139 | 0.119 | 0.535 | Platelet adhesion inhibitor | 0.247 0.05 CHEMBL2111041 0.215 0.063 CHEMBL3544855 0.535 0.005 CHEMBL3544637 | CHEMBL3544637 | |
| 0.126 | 0.107 | 0.233 | Phospholipase A2 inhibitor | 0.204 0.04 CHEMBL1203 0.137 0.09 CHEMBL3544636 0.132 0.097 CHEMBL3544637 0.233 0.028 CHEMBL3091859 0.176 0.056 CHEMBL1237174 0.138 0.088 CHEMBL3091852 | CHEMBL3091859 | |
| 0.198 | 0.179 | 0.773 | Antithrombotic | 0.205 0.171 CHEMBL3544855 0.412 0.046 CHEMBL1203 0.459 0.036 CHEMBL3544636 0.773 0.005 CHEMBL3544637 0.223 0.151 CHEMBL3091859 0.312 0.081 CHEMBL1237174 0.223 0.15 CHEMBL3091852 | CHEMBL3544637 | |
| 0.087 | 0.068 | 0.383 | Alcohol dehydrogenase inhibitor | 0.119 0.035 CHEMBL2111041 0.136 0.026 CHEMBL3544855 0.383 0.004 CHEMBL1203 0.098 0.054 CHEMBL1442231 0.221 0.01 CHEMBL3544636 0.156 0.019 CHEMBL3544637 0.089 0.066 CHEMBL3091859 0.108 0.044 CHEMBL1237174 0.139 0.024 CHEMBL3091852 | CHEMBL1203 | |
| 0.132 | 0.114 | 0.191 | CF transmembrane conductance regulator agonist | 0.163 0.055 CHEMBL1203 0.149 0.077 CHEMBL3544636 0.162 0.057 CHEMBL3544637 0.13 0.119 CHEMBL3091859 0.191 0.027 CHEMBL1237174 0.172 0.045 CHEMBL3091852 | CHEMBL1237174 | |
| 0.059 | 0.041 | 0.343 | Biliverdin reductase inhibitor | 0.075 0.029 CHEMBL2111041 0.069 0.033 CHEMBL3544855 0.068 0.034 CHEMBL3544856 0.343 0.003 CHEMBL1203 0.059 0.042 CHEMBL1442231 0.113 0.015 CHEMBL3544636 0.128 0.012 CHEMBL3544637 0.114 0.015 CHEMBL3091859 0.197 0.006 CHEMBL1237174 0.171 0.008 CHEMBL3091852 | CHEMBL1203 | |
| 0.062 | 0.045 | 0.082 | Histone deacetylase SIRT3 inhibitor | 0.062 0.043 CHEMBL1203 0.071 0.026 CHEMBL1442231 0.082 0.017 CHEMBL3544636 0.065 0.037 CHEMBL1237174 0.069 0.03 CHEMBL3091852 | CHEMBL3544636 | |
| 0.117 | 0.1 | 0.208 | Neurotrophic factor | 0.208 0.024 CHEMBL1203 0.123 0.09 CHEMBL3544637 | CHEMBL1203 | |
| 0.125 | 0.109 | 0.143 | Cyclin-dependent kinase 8 inhibitor | 0.143 0.087 CHEMBL1203 0.132 0.1 CHEMBL1442231 0.127 0.106 CHEMBL1237174 0.133 0.099 CHEMBL3091852 | CHEMBL1203 | |
| 0.06 | 0.044 | 0.06 | Cyclin A inhibitor | |||
| 0.058 | 0.043 | 0.118 | Carbonic anhydrase stimulant | 0.087 0.023 CHEMBL2111041 0.085 0.023 CHEMBL3544855 0.073 0.029 CHEMBL1203 0.062 0.038 CHEMBL1442231 0.118 0.015 CHEMBL3544636 0.055 0.047 CHEMBL3091859 0.077 0.027 CHEMBL1237174 0.081 0.025 CHEMBL3091852 | CHEMBL3544636 | |
| 0.208 | 0.193 | 0.662 | Histamine release inhibitor | 0.286 0.132 CHEMBL2111041 0.311 0.118 CHEMBL3544855 0.322 0.113 CHEMBL3544856 0.646 0.007 CHEMBL1203 0.267 0.143 CHEMBL1442231 0.497 0.03 CHEMBL3544636 0.662 0.006 CHEMBL3544637 0.305 0.121 CHEMBL3091859 0.404 0.073 CHEMBL1237174 0.447 0.051 CHEMBL3091852 | CHEMBL3544637 | |
| 0.055 | 0.041 | 0.077 | Cathepsin B inhibitor | 0.077 0.025 CHEMBL3091859 0.06 0.035 CHEMBL1237174 0.057 0.038 CHEMBL3091852 | CHEMBL3091859 | |
| 0.087 | 0.074 | 0.136 | Potassium channel (Voltage-sensitive) activator | 0.136 0.019 CHEMBL1442231 0.129 0.024 CHEMBL3091852 | CHEMBL1442231 | |
| 0.031 | 0.018 | 0.066 | Cyclin E2 inhibitor | 0.066 0.006 CHEMBL3091859 0.03 0.019 CHEMBL1237174 0.029 0.019 CHEMBL3091852 | CHEMBL3091859 | |
| 0.053 | 0.041 | 0.153 | Thromboxane synthase inhibitor | 0.062 0.025 CHEMBL2111041 0.099 0.007 CHEMBL3544855 0.153 0.004 CHEMBL1203 0.121 0.005 CHEMBL3544636 0.054 0.039 CHEMBL1237174 | CHEMBL1203 | |
| 0.07 | 0.058 | 0.151 | Carbonic anhydrase XIII inhibitor | 0.139 0.024 CHEMBL1203 0.069 0.06 CHEMBL3544637 0.115 0.031 CHEMBL3091859 0.151 0.021 CHEMBL1237174 0.083 0.048 CHEMBL3091852 | CHEMBL1237174 | |
| 0.19 | 0.179 | 0.71 | Transcription factor NF kappa B inhibitor | 0.304 0.092 CHEMBL1203 0.194 0.175 CHEMBL3544636 0.71 0.019 CHEMBL3544637 0.234 0.139 CHEMBL3091859 0.266 0.116 CHEMBL1237174 0.237 0.137 CHEMBL3091852 | CHEMBL3544637 | |
| 0.055 | 0.044 | 0.224 | Cyclin E inhibitor | 0.109 0.021 CHEMBL1442231 0.224 0.005 CHEMBL3091859 0.142 0.012 CHEMBL3091852 | CHEMBL3091859 | |
| 0.028 | 0.018 | 0.031 | Glucosylceramidase stimulant | 0.029 0.015 CHEMBL1203 0.027 0.022 CHEMBL1442231 0.03 0.012 CHEMBL3544636 0.031 0.011 CHEMBL1237174 | CHEMBL1237174 | |
| 0.092 | 0.082 | 0.332 | Adenylate kinase inhibitor | 0.11 0.054 CHEMBL2111041 0.116 0.047 CHEMBL3544855 0.332 0.005 CHEMBL1203 0.179 0.018 CHEMBL3544636 0.209 0.014 CHEMBL3544637 0.159 0.023 CHEMBL3091859 0.27 0.009 CHEMBL1237174 0.223 0.012 CHEMBL3091852 | CHEMBL1203 | |
| 0.064 | 0.055 | 0.13 | Glutamate (mGluR7) antagonist | 0.13 0.004 CHEMBL1203 0.07 0.042 CHEMBL3544636 0.062 0.06 CHEMBL3091859 0.106 0.008 CHEMBL1237174 0.084 0.023 CHEMBL3091852 | CHEMBL1203 | |
| 0.045 | 0.037 | 0.14 | AMPA receptor antagonist | 0.14 0.006 CHEMBL1203 0.058 0.026 CHEMBL3544636 0.043 0.04 CHEMBL1237174 0.052 0.03 CHEMBL3091852 | CHEMBL1203 | |
| 0.042 | 0.034 | 0.052 | Dihydrofolate reductase inhibitor | 0.04 0.039 CHEMBL1203 0.041 0.038 CHEMBL3544636 0.052 0.016 CHEMBL1237174 | CHEMBL1237174 | |
| 0.029 | 0.022 | 0.045 | Nicotinic alpha3beta4 receptor agonist | 0.037 0.012 CHEMBL1203 0.045 0.007 CHEMBL1237174 0.029 0.022 CHEMBL3091852 | CHEMBL1237174 | |
| 0.048 | 0.042 | 0.079 | Ribonucleoside-diphosphate reductase inhibitor | 0.06 0.034 CHEMBL2111041 0.071 0.028 CHEMBL3544855 0.076 0.026 CHEMBL3544856 0.048 0.042 CHEMBL1203 0.049 0.041 CHEMBL1442231 0.079 0.025 CHEMBL3544636 0.065 0.031 CHEMBL3091859 0.061 0.034 CHEMBL1237174 0.072 0.028 CHEMBL3091852 | CHEMBL3544636 | |
| 0.125 | 0.119 | 0.215 | Heat shock protein 90 alpha antagonist | 0.142 0.096 CHEMBL3544855 0.177 0.065 CHEMBL1203 0.215 0.041 CHEMBL1442231 0.124 0.121 CHEMBL1237174 0.172 0.068 CHEMBL3091852 | CHEMBL1442231 | |
| 0.063 | 0.058 | 0.138 | CDK2/cyclin E2 inhibitor | 0.138 0.019 CHEMBL3091859 | CHEMBL3091859 | |
| 0.081 | 0.075 | 0.409 | Triose-phosphate isomerase inhibitor | 0.091 0.058 CHEMBL2111041 0.11 0.039 CHEMBL3544855 0.165 0.016 CHEMBL3544856 0.399 0.003 CHEMBL1203 0.133 0.026 CHEMBL3544636 0.409 0.003 CHEMBL3544637 0.147 0.021 CHEMBL3091859 0.267 0.006 CHEMBL1237174 0.212 0.01 CHEMBL3091852 | CHEMBL3544637 | |
| 0.032 | 0.027 | 0.076 | 1-Alkyl-2-acetylglycerophosphocholine esterase inhibitor | 0.043 0.013 CHEMBL1203 0.076 0.005 CHEMBL3091859 0.043 0.014 CHEMBL1237174 0.034 0.024 CHEMBL3091852 | CHEMBL3091859 | |
| 0.125 | 0.12 | 0.165 | MAP kinase 3 inhibitor | 0.165 0.048 CHEMBL1203 0.139 0.087 CHEMBL3544636 0.137 0.09 CHEMBL1237174 0.124 0.123 CHEMBL3091852 | CHEMBL1203 | |
| 0.029 | 0.025 | 0.063 | Endothelial nitric-oxide synthase inhibitor | 0.03 0.023 CHEMBL3091859 0.063 0.007 CHEMBL1237174 | CHEMBL1237174 | |
| 0.108 | 0.105 | 0.118 | Toll-Like receptor antagonist | 0.112 0.099 CHEMBL1442231 0.118 0.088 CHEMBL3091852 | CHEMBL3091852 | |
| 0.047 | 0.044 | 0.081 | Ribonucleotide reductase inhibitor | 0.06 0.037 CHEMBL2111041 0.071 0.03 CHEMBL3544855 0.076 0.028 CHEMBL3544856 0.048 0.044 CHEMBL1203 0.048 0.043 CHEMBL1442231 0.081 0.026 CHEMBL3544636 0.067 0.033 CHEMBL3091859 0.062 0.035 CHEMBL1237174 0.074 0.029 CHEMBL3091852 | CHEMBL3544636 | |
| 0.039 | 0.036 | 0.073 | Histamine H2 receptor agonist | 0.045 0.027 CHEMBL1442231 0.039 0.037 CHEMBL3544636 0.051 0.021 CHEMBL3091859 0.072 0.009 CHEMBL1237174 0.073 0.009 CHEMBL3091852 | CHEMBL3091852 | |
| 0.149 | 0.147 | 0.639 | Free radical scavenger | 0.304 0.051 CHEMBL2111041 0.196 0.101 CHEMBL3544855 0.166 0.127 CHEMBL1203 0.639 0.007 CHEMBL3544637 0.239 0.073 CHEMBL3091859 0.211 0.089 CHEMBL1237174 | CHEMBL3544637 | |
| 0.027 | 0.026 | 0.068 | Peptide deformylase inhibitor | 0.032 0.019 CHEMBL3544636 0.068 0.005 CHEMBL3091859 0.052 0.009 CHEMBL1237174 0.04 0.014 CHEMBL3091852 | CHEMBL3091859 | |
| 0.052 | 0.051 | 0.124 | 3-Oxoacyl-[acyl-carrier-protein] synthase inhibitor | 0.081 0.024 CHEMBL2111041 0.083 0.023 CHEMBL3544855 0.124 0.011 CHEMBL1203 0.058 0.042 CHEMBL1442231 0.072 0.029 CHEMBL3544637 0.053 0.049 CHEMBL1237174 0.073 0.028 CHEMBL3091852 | CHEMBL1203 | |
| 0.133 | 0.133 | 0.3 | Psychostimulant | 0.173 0.098 CHEMBL1203 0.153 0.113 CHEMBL3544636 0.197 0.082 CHEMBL3544637 0.225 0.068 CHEMBL3091859 0.3 0.043 CHEMBL1237174 0.15 0.116 CHEMBL3091852 | CHEMBL1237174 | |
| 0.078 | 0.078 | 0.506 | NADH dehydrogenase inhibitor | 0.079 0.077 CHEMBL2111041 0.117 0.03 CHEMBL3544856 0.347 0.005 CHEMBL1203 0.139 0.02 CHEMBL3544636 0.506 0.003 CHEMBL3544637 0.123 0.027 CHEMBL3091859 0.247 0.008 CHEMBL1237174 0.164 0.015 CHEMBL3091852 | CHEMBL3544637 | |
| 0.049 | 0.049 | 0.073 | Sphingosine kinase 2 inhibitor | 0.053 0.043 CHEMBL3544856 0.051 0.045 CHEMBL1203 0.073 0.019 CHEMBL1237174 0.056 0.036 CHEMBL3091852 | CHEMBL1237174 | |
| 0.024 | 0.025 | 0.05 | Thymidine phosphorylase inhibitor | 0.025 0.021 CHEMBL1203 0.029 0.013 CHEMBL3091859 0.05 0.005 CHEMBL1237174 0.027 0.016 CHEMBL3091852 | CHEMBL1237174 | |
| 0.068 | 0.069 | 0.084 | Potassium channel (Tandem pore domain) blocker | 0.07 0.065 CHEMBL1203 0.08 0.034 CHEMBL1442231 0.082 0.031 CHEMBL3544636 0.084 0.027 CHEMBL1237174 0.082 0.029 CHEMBL3091852 | CHEMBL1237174 | |
| 0.08 | 0.083 | 0.28 | Protein kinase (CK2) inhibitor | 0.28 0.008 CHEMBL1203 0.089 0.073 CHEMBL3091859 0.088 0.074 CHEMBL1237174 | CHEMBL1203 | |
| 0.117 | 0.119 | 0.15 | Heat shock protein 90 antagonist | 0.132 0.094 CHEMBL1203 0.15 0.075 CHEMBL1442231 0.129 0.099 CHEMBL1237174 0.138 0.088 CHEMBL3091852 | CHEMBL1442231 | |
| 0.062 | 0.065 | 0.093 | Benzodiazepine agonist | 0.086 0.035 CHEMBL3091859 0.093 0.03 CHEMBL1237174 | CHEMBL1237174 | |
| 0.011 | 0.014 | 0.02 | 1-Deoxy-D-xylulose-5-phosphate reductoisomerase inhibitor | 0.014 0.008 CHEMBL1203 0.015 0.007 CHEMBL1442231 0.018 0.005 CHEMBL3544636 0.014 0.008 CHEMBL3091859 0.018 0.004 CHEMBL1237174 0.02 0.004 CHEMBL3091852 | CHEMBL3091852 | |
| 0.029 | 0.033 | 0.047 | Carnitine palmitoyltransferase 1 inhibitor | 0.047 0.01 CHEMBL1203 0.034 0.024 CHEMBL1237174 | CHEMBL1203 | |
| 0.04 | 0.044 | 0.23 | Cyclin E1 inhibitor | 0.095 0.02 CHEMBL1442231 0.23 0.005 CHEMBL3091859 0.133 0.011 CHEMBL3091852 | CHEMBL3091859 | |
| 0.035 | 0.039 | 0.062 | Carbonic anhydrase IV inhibitor | 0.059 0.02 CHEMBL3544636 0.052 0.023 CHEMBL3091859 0.062 0.018 CHEMBL1237174 0.04 0.033 CHEMBL3091852 | CHEMBL1237174 | |
| 0.096 | 0.1 | 0.144 | MAP kinase kinase inhibitor | 0.144 0.055 CHEMBL1203 0.117 0.077 CHEMBL1442231 0.1 0.095 CHEMBL1237174 0.128 0.067 CHEMBL3091852 | CHEMBL1203 | |
| 0.062 | 0.066 | 0.179 | Aminopeptidase I inhibitor | 0.076 0.046 CHEMBL2111041 0.075 0.048 CHEMBL3544855 0.179 0.009 CHEMBL1203 0.068 0.056 CHEMBL1442231 0.155 0.012 CHEMBL3544636 0.1 0.028 CHEMBL3091859 0.138 0.015 CHEMBL1237174 0.13 0.017 CHEMBL3091852 | CHEMBL1203 | |
| 0.084 | 0.088 | 0.318 | Electrolyte absorption antagonist | 0.09 0.074 CHEMBL2111041 0.088 0.078 CHEMBL3544855 0.318 0.004 CHEMBL1203 0.089 0.076 CHEMBL1442231 0.174 0.012 CHEMBL3544636 0.113 0.042 CHEMBL3091859 0.176 0.012 CHEMBL1237174 0.162 0.015 CHEMBL3091852 | CHEMBL1203 | |
| 0.042 | 0.046 | 0.114 | Glucose-6-phosphate isomerase inhibitor | 0.055 0.023 CHEMBL3544855 0.075 0.01 CHEMBL3544856 0.076 0.01 CHEMBL1203 0.054 0.024 CHEMBL3544636 0.114 0.004 CHEMBL3544637 0.065 0.015 CHEMBL3091859 0.107 0.004 CHEMBL1237174 0.081 0.008 CHEMBL3091852 | CHEMBL3544637 | |
| 0.069 | 0.074 | 0.172 | Protein kinase A inhibitor | 0.09 0.052 CHEMBL1203 0.172 0.019 CHEMBL3544637 | CHEMBL3544637 | |
| 0.009 | 0.015 | 0.021 | Thrombopoietin agonist | 0.013 0.007 CHEMBL2111041 0.021 0.004 CHEMBL1203 0.012 0.008 CHEMBL1442231 | CHEMBL1203 | |
| 0.002 | 0.009 | 0.004 | Reverse transcriptase (HBV) inhibitor | 0.004 0.003 CHEMBL3544636 | CHEMBL3544636 | |
| 0.021 | 0.028 | 0.032 | 11-Beta-hydroxysteroid dehydrogenase 2 inhibitor | 0.03 0.017 CHEMBL1203 0.032 0.015 CHEMBL1237174 | CHEMBL1237174 | |
| 0.028 | 0.035 | 0.047 | Carnitine palmitoyltransferase inhibitor | 0.047 0.01 CHEMBL1203 0.033 0.025 CHEMBL1237174 | CHEMBL1203 | |
| 0.063 | 0.07 | 0.144 | Phospholipase D inhibitor | 0.088 0.024 CHEMBL1203 0.144 0.004 CHEMBL3544636 0.108 0.01 CHEMBL1237174 0.087 0.025 CHEMBL3091852 | CHEMBL3544636 | |
| 0.127 | 0.134 | 0.26 | DNA methyltransferase I inhibitor | 0.136 0.121 CHEMBL3544855 0.253 0.045 CHEMBL1203 0.17 0.086 CHEMBL3544636 0.26 0.043 CHEMBL3544637 0.146 0.108 CHEMBL3091859 0.247 0.048 CHEMBL1237174 0.152 0.101 CHEMBL3091852 | CHEMBL3544637 | |
| 0.004 | 0.012 | 0.007 | CC chemokine 6 receptor agonist | 0.007 0.004 CHEMBL1237174 | CHEMBL1237174 | |
| 0.162 | 0.17 | 0.369 | RNA-directed DNA polymerase inhibitor | 0.369 0.022 CHEMBL1203 0.185 0.123 CHEMBL3544636 0.269 0.04 CHEMBL3544637 0.18 0.132 CHEMBL3091859 0.3 0.032 CHEMBL1237174 0.235 0.06 CHEMBL3091852 | CHEMBL1203 | |
| 0.049 | 0.057 | 0.208 | Carbamoyl phosphate synthetase inhibitor | 0.057 0.046 CHEMBL2111041 0.09 0.024 CHEMBL3544855 0.053 0.051 CHEMBL3544856 0.128 0.014 CHEMBL1203 0.095 0.022 CHEMBL3544636 0.072 0.033 CHEMBL3544637 0.103 0.02 CHEMBL3091859 0.208 0.007 CHEMBL1237174 0.142 0.012 CHEMBL3091852 | CHEMBL1237174 | |
| 0.031 | 0.04 | 0.081 | Alpha 1d adrenoreceptor agonist | 0.052 0.015 CHEMBL1203 0.081 0.005 CHEMBL1237174 0.048 0.018 CHEMBL3091852 | CHEMBL1237174 | |
| 0.015 | 0.024 | 0.023 | Estrogen-related receptor gamma agonist | 0.018 0.014 CHEMBL2111041 0.02 0.01 CHEMBL1442231 0.019 0.012 CHEMBL3544636 0.017 0.016 CHEMBL3091859 0.023 0.007 CHEMBL3091852 | CHEMBL3091852 | |
| 0.071 | 0.08 | 0.099 | MAP kinase kinase 7 inhibitor | 0.099 0.014 CHEMBL1203 0.08 0.047 CHEMBL3544636 0.098 0.015 CHEMBL1237174 0.086 0.031 CHEMBL3091852 | CHEMBL1203 | |
| 0.004 | 0.014 | 0.01 | Integrin alpha5beta6 antagonist | 0.006 0.005 CHEMBL3544855 0.007 0.004 CHEMBL1203 0.01 0.003 CHEMBL3544636 0.006 0.005 CHEMBL1237174 0.007 0.004 CHEMBL3091852 | CHEMBL3544636 | |
| 0.036 | 0.046 | 0.052 | CF transmembrane conductance regulator antagonist | 0.052 0.007 CHEMBL1203 0.04 0.026 CHEMBL1237174 0.043 0.019 CHEMBL3091852 | CHEMBL1203 | |
| 0.189 | 0.199 | 0.407 | Calpain 2 inhibitor | 0.221 0.171 CHEMBL1203 0.387 0.068 CHEMBL1442231 0.235 0.16 CHEMBL3544636 0.225 0.168 CHEMBL3091859 0.268 0.137 CHEMBL1237174 0.407 0.058 CHEMBL3091852 | CHEMBL3091852 | |
| 0.024 | 0.034 | 0.047 | Purinergic P2Y15 antagonist | 0.029 0.019 CHEMBL1203 0.026 0.025 CHEMBL1442231 0.03 0.018 CHEMBL3544636 0.037 0.009 CHEMBL3091859 0.047 0.004 CHEMBL1237174 0.046 0.005 CHEMBL3091852 | CHEMBL1237174 | |
| 0.055 | 0.066 | 0.363 | Phenylalanine 4-hydroxylase inhibitor | 0.071 0.045 CHEMBL2111041 0.067 0.05 CHEMBL3544855 0.082 0.036 CHEMBL3544856 0.363 0.003 CHEMBL1203 0.063 0.054 CHEMBL1442231 0.202 0.007 CHEMBL3544636 0.087 0.033 CHEMBL3091859 0.157 0.011 CHEMBL1237174 0.137 0.014 CHEMBL3091852 | CHEMBL1203 | |
| 0.032 | 0.043 | 0.088 | Glutamate (mGluR1a) antagonist | 0.088 0.007 CHEMBL1203 0.063 0.014 CHEMBL3544636 0.04 0.029 CHEMBL1237174 0.036 0.035 CHEMBL3091852 | CHEMBL1203 | |
| 0.021 | 0.034 | 0.039 | Nicotinic alpha4beta2 receptor agonist | 0.03 0.018 CHEMBL1203 0.039 0.008 CHEMBL1237174 | CHEMBL1237174 | |
| 0.129 | 0.143 | 0.254 | ATPase inhibitor | 0.141 0.118 CHEMBL2111041 0.143 0.113 CHEMBL3544856 0.167 0.075 CHEMBL1203 0.14 0.119 CHEMBL1442231 0.145 0.11 CHEMBL3544636 0.254 0.013 CHEMBL3544637 0.134 0.133 CHEMBL3091859 0.179 0.059 CHEMBL1237174 0.195 0.041 CHEMBL3091852 | CHEMBL3544637 | |
| 0.054 | 0.068 | 0.075 | CDC7 inhibitor | 0.075 0.039 CHEMBL1203 0.062 0.054 CHEMBL1442231 | CHEMBL1203 | |
| 0.02 | 0.034 | 0.144 | Glucagon receptor antagonist | 0.07 0.006 CHEMBL2111041 0.084 0.005 CHEMBL3544855 0.032 0.019 CHEMBL1442231 0.144 0.004 CHEMBL3544636 | CHEMBL3544636 | |
| 0.024 | 0.038 | 0.047 | Epoxide hydrolase 1 inhibitor | 0.047 0.007 CHEMBL1203 0.033 0.019 CHEMBL1442231 0.038 0.012 CHEMBL3544636 0.029 0.024 CHEMBL3091859 0.037 0.014 CHEMBL1237174 0.042 0.01 CHEMBL3091852 | CHEMBL1203 | |
| 0.099 | 0.114 | 0.157 | Toll-Like receptor 9 antagonist | 0.157 0.058 CHEMBL1237174 | CHEMBL1237174 | |
| 0.015 | 0.03 | 0.033 | Antibiotic Anthracycline-like | 0.033 0.003 CHEMBL3544637 0.027 0.004 CHEMBL3091859 0.029 0.004 CHEMBL1237174 0.02 0.011 CHEMBL3091852 | CHEMBL3544637 | |
| 0.134 | 0.149 | 0.251 | Death-associated protein kinase 3 inhibitor | 0.228 0.061 CHEMBL1203 0.233 0.059 CHEMBL1442231 0.251 0.052 CHEMBL3091852 | CHEMBL3091852 | |
| 0.034 | 0.05 | 0.087 | Geranyltranstransferase inhibitor | 0.087 0.004 CHEMBL1203 0.066 0.009 CHEMBL3544636 0.064 0.011 CHEMBL1237174 0.045 0.028 CHEMBL3091852 | CHEMBL1203 | |
| 0.017 | 0.033 | 0.083 | AMPA 1 receptor antagonist | 0.083 0.007 CHEMBL1203 0.055 0.01 CHEMBL3544636 | CHEMBL1203 | |
| 0.023 | 0.04 | 0.036 | Hedgehog signaling activator | 0.029 0.014 CHEMBL1203 0.036 0.006 CHEMBL1237174 0.028 0.017 CHEMBL3091852 | CHEMBL1237174 | |
| 0.026 | 0.042 | 0.033 | Calcium release-activated channel blocker | 0.033 0.022 CHEMBL1203 | CHEMBL1203 | |
| 0.007 | 0.026 | 0.113 | Egl nine homolog 3 inhibitor | 0.046 0.003 CHEMBL1203 0.113 0.002 CHEMBL3544636 0.011 0.009 CHEMBL1237174 | CHEMBL3544636 | |
| 0.055 | 0.075 | 0.077 | Transcription factor RelA inhibitor | 0.063 0.047 CHEMBL1203 0.061 0.053 CHEMBL3091859 0.077 0.02 CHEMBL1237174 0.073 0.026 CHEMBL3091852 | CHEMBL1237174 | |
| 0.036 | 0.056 | 0.061 | Histamine H1 receptor agonist | 0.061 0.008 CHEMBL1237174 0.048 0.021 CHEMBL3091852 | CHEMBL1237174 | |
| 0.072 | 0.092 | 0.185 | HIV-1 integrase (Overall Integration) inhibitor | 0.08 0.078 CHEMBL2111041 0.185 0.015 CHEMBL1203 0.117 0.041 CHEMBL1442231 0.154 0.024 CHEMBL3544636 0.159 0.022 CHEMBL1237174 0.163 0.021 CHEMBL3091852 | CHEMBL1203 | |
| 0.155 | 0.175 | 0.568 | 5 Hydroxytryptamine release stimulant | 0.395 0.047 CHEMBL1203 0.216 0.109 CHEMBL3544636 0.342 0.058 CHEMBL3544637 0.203 0.119 CHEMBL3091859 0.568 0.018 CHEMBL1237174 0.357 0.055 CHEMBL3091852 | CHEMBL1237174 | |
| 0.03 | 0.051 | 0.047 | Potassium channel Kv1.1 blocker | 0.047 0.015 CHEMBL1237174 0.037 0.028 CHEMBL3091852 | CHEMBL1237174 | |
| 0.01 | 0.031 | 0.025 | Steroid 17-alpha-hydroxylase/17,20 lyase inhibitor | 0.025 0.011 CHEMBL1203 | CHEMBL1203 | |
| 0.012 | 0.034 | 0.022 | CC chemokine 9 receptor antagonist | 0.022 0.005 CHEMBL1203 0.016 0.015 CHEMBL1237174 | CHEMBL1203 | |
| 0.032 | 0.055 | 0.1 | Stearoyl-CoA desaturase inhibitor | 0.1 0.007 CHEMBL3544636 | CHEMBL3544636 | |
| 0.058 | 0.081 | 0.321 | Glutamate dehydrogenase inhibitor | 0.07 0.057 CHEMBL2111041 0.094 0.034 CHEMBL3544855 0.321 0.005 CHEMBL1203 0.149 0.016 CHEMBL3544636 0.114 0.025 CHEMBL3544637 0.124 0.021 CHEMBL3091859 0.182 0.012 CHEMBL1237174 0.177 0.012 CHEMBL3091852 | CHEMBL1203 | |
| 0.035 | 0.058 | 0.229 | Glutamate (mGluR4) antagonist | 0.041 0.035 CHEMBL3544855 0.229 0.003 CHEMBL1203 0.071 0.01 CHEMBL3544636 0.053 0.018 CHEMBL1237174 | CHEMBL1203 | |
| 0.027 | 0.051 | 0.111 | Protein kinase (CK2) beta inhibitor | 0.111 0.003 CHEMBL1203 0.037 0.016 CHEMBL1237174 0.031 0.03 CHEMBL3091852 | CHEMBL1203 | |
| 0.055 | 0.079 | 0.144 | Histone deacetylase stimulant | 0.085 0.039 CHEMBL3544856 0.087 0.037 CHEMBL1203 0.144 0.01 CHEMBL3544637 | CHEMBL3544637 | |
| 0.055 | 0.079 | 0.144 | Histone deacetylase SIRT1 stimulant | 0.085 0.039 CHEMBL3544856 0.087 0.037 CHEMBL1203 0.144 0.01 CHEMBL3544637 | CHEMBL3544637 | |
| 0.025 | 0.051 | 0.039 | Delayed rectifier potassium channel activator | 0.039 0.023 CHEMBL3091852 | CHEMBL3091852 | |
| 0.025 | 0.051 | 0.039 | Potassium channel KCNQ activator | 0.039 0.023 CHEMBL3091852 | CHEMBL3091852 | |
| 0.07 | 0.097 | 0.161 | Potassium channel activator | 0.091 0.059 CHEMBL1203 0.152 0.019 CHEMBL1442231 0.091 0.059 CHEMBL3091859 0.161 0.016 CHEMBL3091852 | CHEMBL3091852 | |
| 0.037 | 0.064 | 0.21 | Acyl-CoA dehydrogenase inhibitor | 0.21 0.005 CHEMBL1203 0.083 0.021 CHEMBL3544636 0.069 0.027 CHEMBL3544637 0.123 0.012 CHEMBL3091859 0.185 0.006 CHEMBL1237174 0.177 0.007 CHEMBL3091852 | CHEMBL1203 | |
| 0.043 | 0.071 | 0.072 | Epithelial sodium channel blocker | 0.055 0.038 CHEMBL3544856 0.072 0.017 CHEMBL3544636 0.064 0.024 CHEMBL1237174 0.057 0.033 CHEMBL3091852 | CHEMBL3544636 | |
| 0.08 | 0.108 | 0.2 | Phosphodiesterase 6D inhibitor | 0.129 0.019 CHEMBL1203 0.2 0.005 CHEMBL3544637 0.099 0.055 CHEMBL1237174 | CHEMBL3544637 | |
| 0.031 | 0.059 | 0.113 | Thymidylate synthase inhibitor | 0.048 0.03 CHEMBL3544855 0.061 0.017 CHEMBL1203 0.113 0.004 CHEMBL3544636 0.054 0.023 CHEMBL1237174 | CHEMBL3544636 | |
| 0.009 | 0.038 | 0.017 | Adenosine A2 receptor agonist | 0.015 0.013 CHEMBL3544856 0.017 0.01 CHEMBL1237174 | CHEMBL1237174 | |
| 0.05 | 0.079 | 0.066 | Aryl hydrocarbon receptor antagonist | 0.059 0.056 CHEMBL1203 0.066 0.044 CHEMBL1237174 | CHEMBL1237174 | |
| 0.021 | 0.05 | 0.031 | Thymidine kinase (Herpes simplex virus 1) inhibitor | 0.027 0.016 CHEMBL1203 0.026 0.02 CHEMBL3544637 0.031 0.01 CHEMBL1237174 0.027 0.016 CHEMBL3091852 | CHEMBL1237174 | |
| 0.009 | 0.039 | 0.024 | Cyclin T1 inhibitor | 0.018 0.013 CHEMBL1203 0.024 0.008 CHEMBL1237174 | CHEMBL1237174 | |
| 0.058 | 0.088 | 0.078 | Adenosine A3 receptor antagonist | 0.078 0.046 CHEMBL1237174 | CHEMBL1237174 | |
| 0.013 | 0.044 | 0.051 | Glutamate (mGluR1a) agonist | 0.049 0.005 CHEMBL1203 0.03 0.009 CHEMBL3544636 0.051 0.005 CHEMBL1237174 0.029 0.009 CHEMBL3091852 | CHEMBL1237174 | |
| 0.009 | 0.04 | 0.021 | Thromboxane A2 agonist | 0.017 0.008 CHEMBL3544855 0.014 0.013 CHEMBL3091859 0.021 0.005 CHEMBL1237174 0.02 0.005 CHEMBL3091852 | CHEMBL1237174 | |
| 0.01 | 0.041 | 0.018 | Nicotinic alpha4 receptor agonist | 0.018 0.009 CHEMBL1237174 | CHEMBL1237174 | |
| 0.033 | 0.064 | 0.062 | Glutamate (mGluR5) agonist | 0.062 0.017 CHEMBL1203 | CHEMBL1203 | |
| 0.038 | 0.069 | 0.078 | Dopamine beta hydroxylase inhibitor | 0.078 0.005 CHEMBL1203 0.045 0.043 CHEMBL3544636 0.067 0.01 CHEMBL1237174 0.048 0.034 CHEMBL3091852 | CHEMBL1203 | |
| 0.029 | 0.061 | 0.061 | Angiotensin AT1 receptor antagonist | 0.061 0.005 CHEMBL1203 0.048 0.021 CHEMBL1237174 0.048 0.02 CHEMBL3091852 | CHEMBL1203 | |
| 0.07 | 0.102 | 0.084 | Pim-3 kinase inhibitor | 0.084 0.069 CHEMBL1203 | CHEMBL1203 | |
| 0.006 | 0.038 | 0.03 | Carbonic anhydrase XI inhibitor | 0.012 0.009 CHEMBL1203 0.02 0.004 CHEMBL3091859 0.018 0.005 CHEMBL1237174 0.03 0.003 CHEMBL3091852 | CHEMBL3091852 | |
| 0.02 | 0.052 | 0.034 | Complement factor 1s inhibitor | 0.029 0.009 CHEMBL1203 0.034 0.005 CHEMBL1237174 0.025 0.019 CHEMBL3091852 | CHEMBL1237174 | |
| 0.006 | 0.038 | 0.013 | Purinergic P2Y2 agonist | 0.013 0.004 CHEMBL3544637 0.01 0.008 CHEMBL1237174 | CHEMBL3544637 | |
| 0.043 | 0.075 | 0.1 | Dihydroorotate oxidase inhibitor | 0.1 0.005 CHEMBL1203 0.064 0.024 CHEMBL3091859 0.08 0.01 CHEMBL1237174 0.084 0.009 CHEMBL3091852 | CHEMBL1203 | |
| 0.013 | 0.046 | 0.039 | NMDA receptor glycine site antagonist | 0.039 0.009 CHEMBL1203 0.023 0.019 CHEMBL1237174 | CHEMBL1203 | |
| 0.037 | 0.071 | 0.09 | Cathepsin D inhibitor | 0.09 0.021 CHEMBL3091859 | CHEMBL3091859 | |
| 0.009 | 0.045 | 0.044 | Nicotinic acid receptor 1 antagonist | 0.044 0.003 CHEMBL1203 0.022 0.007 CHEMBL1237174 0.022 0.007 CHEMBL3091852 | CHEMBL1203 | |
| 0.031 | 0.066 | 0.092 | Nerve growth factor antagonist | 0.092 0.003 CHEMBL1203 0.057 0.011 CHEMBL1237174 0.047 0.023 CHEMBL3091852 | CHEMBL1203 | |
| 0.134 | 0.17 | 0.532 | Immunostimulant | 0.203 0.119 CHEMBL1203 0.273 0.088 CHEMBL3544636 0.532 0.025 CHEMBL3544637 0.223 0.108 CHEMBL3091859 0.255 0.094 CHEMBL1237174 0.205 0.117 CHEMBL3091852 | CHEMBL3544637 | |
| 0.006 | 0.042 | 0.011 | Purine nucleoside phosphorylase inhibitor | 0.011 0.01 CHEMBL1237174 | CHEMBL1237174 | |
| 0.006 | 0.042 | 0.017 | Adenosine A2a receptor agonist | 0.017 0.009 CHEMBL1237174 | CHEMBL1237174 | |
| 0.021 | 0.057 | 0.033 | MAP3K8 inhibitor | 0.031 0.017 CHEMBL1203 0.033 0.013 CHEMBL1237174 | CHEMBL1237174 | |
| 0.032 | 0.068 | 0.111 | 3-Hydroxyanthranilate 3,4-dioxygenase inhibitor | 0.111 0.003 CHEMBL1203 0.046 0.02 CHEMBL3091859 0.072 0.004 CHEMBL1237174 0.058 0.008 CHEMBL3091852 | CHEMBL1203 | |
| 0.02 | 0.056 | 0.116 | Fumarate hydratase inhibitor | 0.035 0.023 CHEMBL3544855 0.116 0.005 CHEMBL1203 0.039 0.019 CHEMBL3544636 0.039 0.02 CHEMBL3544637 0.046 0.015 CHEMBL3091859 0.083 0.007 CHEMBL1237174 0.07 0.008 CHEMBL3091852 | CHEMBL1203 | |
| 0.013 | 0.049 | 0.021 | Caspase 8 inhibitor | 0.018 0.017 CHEMBL1442231 0.021 0.011 CHEMBL3544636 0.019 0.015 CHEMBL3091852 | CHEMBL3544636 | |
| 0.043 | 0.08 | 0.287 | Phosphofructokinase-1 inhibitor | 0.086 0.038 CHEMBL3544855 0.093 0.035 CHEMBL3544856 0.227 0.009 CHEMBL1203 0.092 0.035 CHEMBL3544636 0.287 0.006 CHEMBL3544637 0.094 0.034 CHEMBL3091859 0.205 0.011 CHEMBL1237174 0.138 0.02 CHEMBL3091852 | CHEMBL3544637 | |
| 0.069 | 0.106 | 0.146 | Sphingomyelinase inhibitor | 0.146 0.026 CHEMBL3544856 0.102 0.057 CHEMBL1203 0.084 0.081 CHEMBL1442231 0.094 0.067 CHEMBL3544636 0.101 0.058 CHEMBL3544637 0.128 0.035 CHEMBL1237174 0.118 0.043 CHEMBL3091852 | CHEMBL3544856 | |
| 0.021 | 0.059 | 0.142 | Kainate receptor antagonist | 0.142 0.005 CHEMBL1203 0.039 0.03 CHEMBL3544636 0.044 0.026 CHEMBL1237174 0.041 0.028 CHEMBL3091852 | CHEMBL1203 | |
| 0.006 | 0.044 | 0.017 | Human herpes virus 5 capsid protein P40 inhibitor | 0.016 0.005 CHEMBL1203 0.017 0.005 CHEMBL1237174 | CHEMBL1237174 | |
| 0.065 | 0.102 | 0.144 | Falcipain inhibitor | 0.114 0.047 CHEMBL1442231 0.144 0.034 CHEMBL3091852 | CHEMBL3091852 | |
| 0.107 | 0.146 | 0.174 | Protein kinase (CK1) gamma 3 inhibitor | 0.146 0.095 CHEMBL1203 0.174 0.066 CHEMBL1442231 0.161 0.078 CHEMBL3091852 | CHEMBL1442231 | |
| 0.069 | 0.108 | 0.284 | Creatine kinase inhibitor | 0.09 0.072 CHEMBL2111041 0.284 0.004 CHEMBL1203 0.1 0.06 CHEMBL3544636 0.136 0.031 CHEMBL3091859 0.21 0.009 CHEMBL1237174 0.187 0.013 CHEMBL3091852 | CHEMBL1203 | |
| 0.041 | 0.08 | 0.072 | Glucosylceramidase inhibitor | 0.065 0.026 CHEMBL3544856 0.055 0.037 CHEMBL1203 0.061 0.03 CHEMBL3544637 0.072 0.02 CHEMBL1237174 | CHEMBL1237174 | |
| 0.075 | 0.114 | 0.206 | 5 Hydroxytryptamine 3A agonist | 0.206 0.013 CHEMBL1237174 0.143 0.039 CHEMBL3091852 | CHEMBL1237174 | |
| 0.026 | 0.065 | 0.04 | Delayed rectifier potassium channel blocker | 0.035 0.03 CHEMBL3544636 0.04 0.021 CHEMBL1237174 0.034 0.033 CHEMBL3091852 | CHEMBL1237174 | |
| 0.047 | 0.087 | 0.065 | Leukotriene C antagonist | 0.065 0.019 CHEMBL1203 0.055 0.044 CHEMBL3544636 0.061 0.026 CHEMBL3091859 0.064 0.021 CHEMBL1237174 0.054 0.049 CHEMBL3091852 | CHEMBL1203 | |
| 0.024 | 0.064 | 0.067 | Glutamate (mGluR4) agonist | 0.067 0.007 CHEMBL1203 0.032 0.027 CHEMBL1237174 | CHEMBL1203 | |
| 0.045 | 0.086 | 0.101 | Pregnane X receptor antagonist | 0.101 0.004 CHEMBL1203 0.053 0.05 CHEMBL3544637 0.076 0.009 CHEMBL1237174 0.065 0.022 CHEMBL3091852 | CHEMBL1203 | |
| 0.009 | 0.049 | 0.014 | Cyclin D2 inhibitor | 0.014 0.007 CHEMBL1237174 | CHEMBL1237174 | |
| 0.072 | 0.113 | 0.12 | Protein kinase C zeta inhibitor | 0.12 0.032 CHEMBL1203 0.088 0.068 CHEMBL3544637 0.084 0.078 CHEMBL1237174 | CHEMBL1203 | |
| 0.014 | 0.055 | 0.025 | Thymidine kinase (Herpes simplex virus 2) inhibitor | 0.025 0.007 CHEMBL1237174 0.023 0.009 CHEMBL3091852 | CHEMBL1237174 | |
| 0.233 | 0.275 | 0.515 | Caspase 9 stimulant | 0.385 0.12 CHEMBL1203 0.276 0.222 CHEMBL1442231 0.318 0.175 CHEMBL3544636 0.515 0.054 CHEMBL3544637 0.337 0.157 CHEMBL3091859 0.458 0.079 CHEMBL1237174 0.469 0.074 CHEMBL3091852 | CHEMBL3544637 | |
| 0.007 | 0.049 | 0.043 | Carbonic anhydrase X inhibitor | 0.03 0.004 CHEMBL1203 0.03 0.004 CHEMBL3091859 0.037 0.004 CHEMBL1237174 0.043 0.003 CHEMBL3091852 | CHEMBL3091852 | |
| 0.007 | 0.049 | 0.043 | Carbonic anhydrase VIII inhibitor | 0.03 0.004 CHEMBL1203 0.03 0.004 CHEMBL3091859 0.037 0.004 CHEMBL1237174 0.043 0.003 CHEMBL3091852 | CHEMBL3091852 | |
| 0.032 | 0.075 | 0.061 | Adenosine A1 receptor antagonist | 0.061 0.039 CHEMBL1237174 | CHEMBL1237174 | |
| 0.027 | 0.071 | 0.083 | Glutamate (mGluR8) agonist | 0.037 0.027 CHEMBL3544855 0.083 0.004 CHEMBL1203 0.036 0.03 CHEMBL3544636 0.043 0.018 CHEMBL3091859 0.073 0.005 CHEMBL1237174 0.056 0.009 CHEMBL3091852 | CHEMBL1203 | |
| 0.044 | 0.088 | 0.07 | Heat shock protein 90 beta antagonist | 0.056 0.047 CHEMBL3544636 0.07 0.029 CHEMBL1237174 | CHEMBL1237174 | |
| 0.06 | 0.104 | 0.163 | Potassium channel (Ca-activated) activator | 0.163 0.024 CHEMBL1203 0.133 0.034 CHEMBL1237174 | CHEMBL1203 | |
| 0.022 | 0.067 | 0.038 | Histone deacetylase class I inhibitor | 0.038 0.029 CHEMBL1442231 | CHEMBL1442231 | |
| 0.003 | 0.048 | 0.01 | DNA topoisomerase III inhibitor | 0.01 0.004 CHEMBL1237174 0.007 0.006 CHEMBL3091852 | CHEMBL1237174 | |
| 0.029 | 0.075 | 0.047 | Vanilloid 3 antagonist | 0.047 0.011 CHEMBL1203 0.044 0.015 CHEMBL1237174 0.036 0.033 CHEMBL3091852 | CHEMBL1203 | |
| 0.027 | 0.073 | 0.039 | Histone deacetylase 9 inhibitor | 0.038 0.029 CHEMBL1442231 0.036 0.034 CHEMBL3544636 0.039 0.028 CHEMBL3091852 | CHEMBL3091852 | |
| 0.018 | 0.064 | 0.049 | Calcitonin receptor agonist | 0.049 0.017 CHEMBL3544636 0.033 0.024 CHEMBL1237174 0.03 0.027 CHEMBL3091852 | CHEMBL3544636 | |
| 0.152 | 0.199 | 0.524 | DNA synthesis inhibitor | 0.233 0.08 CHEMBL2111041 0.214 0.103 CHEMBL3544855 0.307 0.041 CHEMBL3544856 0.395 0.022 CHEMBL1203 0.299 0.044 CHEMBL3544636 0.524 0.012 CHEMBL3544637 0.201 0.121 CHEMBL3091859 0.287 0.048 CHEMBL1237174 0.264 0.058 CHEMBL3091852 | CHEMBL3544637 | |
| 0.015 | 0.062 | 0.059 | Nicotinic acid receptor 2 antagonist | 0.059 0.003 CHEMBL1203 0.026 0.019 CHEMBL3091859 0.037 0.006 CHEMBL1237174 0.037 0.006 CHEMBL3091852 | CHEMBL1203 | |
| 0.013 | 0.06 | 0.024 | Methylmalonyl-CoA mutase inhibitor | 0.024 0.004 CHEMBL1203 0.017 0.015 CHEMBL3544636 0.019 0.011 CHEMBL3091859 0.023 0.005 CHEMBL1237174 0.022 0.006 CHEMBL3091852 | CHEMBL1203 | |
| 0.06 | 0.107 | 0.136 | Falcipain 2 inhibitor | 0.104 0.05 CHEMBL1442231 0.136 0.035 CHEMBL3091852 | CHEMBL3091852 | |
| 0.009 | 0.057 | 0.053 | Hypoxanthine phosphoribosyltransferase inhibitor | 0.032 0.016 CHEMBL1203 0.027 0.02 CHEMBL3544636 0.053 0.008 CHEMBL1237174 0.036 0.014 CHEMBL3091852 | CHEMBL1237174 | |
| 0.033 | 0.082 | 0.245 | Argininosuccinate synthase inhibitor | 0.245 0.005 CHEMBL1203 0.081 0.025 CHEMBL3544636 0.088 0.022 CHEMBL3544637 0.074 0.028 CHEMBL3091859 0.165 0.01 CHEMBL1237174 0.118 0.015 CHEMBL3091852 | CHEMBL1203 | |
| 0.055 | 0.103 | 0.088 | Bcr-Abl kinase inhibitor | 0.088 0.054 CHEMBL1203 | CHEMBL1203 | |
| 0.021 | 0.07 | 0.054 | Angiotensin II receptor antagonist | 0.054 0.005 CHEMBL1203 0.035 0.023 CHEMBL1237174 0.035 0.023 CHEMBL3091852 | CHEMBL1203 | |
| 0.062 | 0.111 | 0.104 | Vascular endothelial growth factor 1 antagonist | 0.104 0.063 CHEMBL1203 | CHEMBL1203 | |
| 0.032 | 0.081 | 0.092 | Lysophosphatidic acid 3 receptor antagonist | 0.045 0.044 CHEMBL3544855 0.092 0.006 CHEMBL1203 0.056 0.027 CHEMBL3544636 0.047 0.041 CHEMBL3091859 0.068 0.016 CHEMBL1237174 0.063 0.019 CHEMBL3091852 | CHEMBL1203 | |
| 0.035 | 0.084 | 0.048 | Heme oxygenase inhibitor | 0.043 0.028 CHEMBL1203 0.048 0.015 CHEMBL1237174 | CHEMBL1237174 | |
| 0.07 | 0.12 | 0.092 | Glycogen synthase kinase-3 beta inhibitor | 0.092 0.088 CHEMBL1442231 | CHEMBL1442231 | |
| 0.038 | 0.088 | 0.061 | Dipeptidyl peptidase inhibitor | 0.061 0.025 CHEMBL1237174 | CHEMBL1237174 | |
| 0.071 | 0.121 | 0.144 | Anabolic | 0.144 0.021 CHEMBL1203 0.103 0.059 CHEMBL3544636 0.102 0.06 CHEMBL3544637 0.116 0.043 CHEMBL3091859 0.143 0.022 CHEMBL1237174 0.14 0.024 CHEMBL3091852 | CHEMBL1203 | |
| 0.019 | 0.07 | 0.035 | Estrogen-related receptor gamma antagonist | 0.035 0.008 CHEMBL1237174 0.033 0.011 CHEMBL3091852 | CHEMBL1237174 | |
| 0.042 | 0.092 | 0.066 | Sphingosine kinase inhibitor | 0.059 0.041 CHEMBL3544856 0.063 0.034 CHEMBL1237174 0.066 0.03 CHEMBL3091852 | CHEMBL3091852 | |
| 0.034 | 0.084 | 0.051 | Dipeptidyl peptidase IV inhibitor | 0.051 0.019 CHEMBL1237174 | CHEMBL1237174 | |
| 0.015 | 0.066 | 0.109 | Kainate receptor 2 antagonist | 0.109 0.004 CHEMBL1203 0.037 0.024 CHEMBL1442231 0.043 0.02 CHEMBL3544636 0.033 0.028 CHEMBL1237174 0.054 0.014 CHEMBL3091852 | CHEMBL1203 | |
| 0.013 | 0.064 | 0.093 | Lysine carboxypeptidase inhibitor | 0.031 0.015 CHEMBL1203 0.093 0.004 CHEMBL3544636 0.033 0.013 CHEMBL1237174 | CHEMBL3544636 | |
| 0.146 | 0.197 | 0.261 | 5 Hydroxytryptamine 1E antagonist | 0.184 0.15 CHEMBL3091859 0.261 0.063 CHEMBL1237174 0.256 0.068 CHEMBL3091852 | CHEMBL1237174 | |
| 0.006 | 0.058 | 0.021 | Integrin alphaVbeta6 antagonist | 0.021 0.005 CHEMBL3544636 | CHEMBL3544636 | |
| 0.025 | 0.077 | 0.08 | Tryptophan 5 hydroxylase inhibitor | 0.05 0.005 CHEMBL1203 0.08 0.003 CHEMBL3544636 0.041 0.013 CHEMBL1237174 | CHEMBL3544636 | |
| 0.022 | 0.074 | 0.06 | Oxytocin agonist | 0.038 0.034 CHEMBL3091859 0.058 0.018 CHEMBL1237174 0.06 0.017 CHEMBL3091852 | CHEMBL3091852 | |
| 0.096 | 0.148 | 0.203 | DNA repair enzyme inhibitor | 0.132 0.052 CHEMBL1203 0.203 0.008 CHEMBL3544637 0.111 0.094 CHEMBL3091859 0.158 0.025 CHEMBL1237174 0.132 0.052 CHEMBL3091852 | CHEMBL3544637 | |
| 0.024 | 0.077 | 0.037 | MAP3K5 inhibitor | 0.037 0.031 CHEMBL1237174 | CHEMBL1237174 | |
| 0.126 | 0.179 | 0.229 | Neurotrophic factor enhancer | 0.219 0.06 CHEMBL1203 0.225 0.055 CHEMBL3544636 0.211 0.067 CHEMBL3544637 0.161 0.122 CHEMBL3091859 0.229 0.052 CHEMBL1237174 0.22 0.059 CHEMBL3091852 | CHEMBL1237174 | |
| 0.011 | 0.065 | 0.061 | Uridine phosphorylase inhibitor | 0.061 0.005 CHEMBL1203 0.053 0.007 CHEMBL3544637 0.049 0.008 CHEMBL1237174 0.033 0.016 CHEMBL3091852 | CHEMBL1203 | |
| 0.011 | 0.065 | 0.02 | Alpha 2b adrenoreceptor agonist | 0.02 0.01 CHEMBL1237174 | CHEMBL1237174 | |
| 0.041 | 0.095 | 0.162 | Purinergic P2X1 antagonist | 0.162 0.006 CHEMBL1203 0.083 0.024 CHEMBL3544637 0.118 0.012 CHEMBL1237174 0.075 0.028 CHEMBL3091852 | CHEMBL1203 | |
| 0.031 | 0.086 | 0.206 | Glutamate (mGluR group III) antagonist | 0.206 0.003 CHEMBL1203 0.051 0.019 CHEMBL3544636 0.049 0.022 CHEMBL1237174 | CHEMBL1203 | |
| 0.03 | 0.084 | 0.067 | Kainate receptor agonist | 0.066 0.005 CHEMBL1203 0.043 0.025 CHEMBL3544636 0.043 0.024 CHEMBL3091859 0.067 0.005 CHEMBL1237174 0.055 0.01 CHEMBL3091852 | CHEMBL1237174 | |
| 0.004 | 0.059 | 0.019 | Glutamate (mGluR6) agonist | 0.019 0.004 CHEMBL1203 0.019 0.004 CHEMBL1237174 0.013 0.007 CHEMBL3091852 | CHEMBL1237174 | |
| 0.055 | 0.11 | 0.29 | Keratolytic | 0.29 0.004 CHEMBL1203 0.097 0.032 CHEMBL3544636 0.071 0.062 CHEMBL3544637 0.102 0.029 CHEMBL1237174 0.08 0.049 CHEMBL3091852 | CHEMBL1203 | |
| 0.014 | 0.069 | 0.031 | Carnitine palmitoyltransferase 1A inhibitor | 0.031 0.017 CHEMBL1203 | CHEMBL1203 | |
| 0.045 | 0.1 | 0.111 | Protein kinase C beta inhibitor | 0.108 0.01 CHEMBL1203 0.111 0.009 CHEMBL3544637 0.071 0.046 CHEMBL1237174 | CHEMBL3544637 | |
| 0.024 | 0.079 | 0.078 | Glutamate (mGluR group I) agonist | 0.078 0.013 CHEMBL1203 0.043 0.039 CHEMBL3544636 | CHEMBL1203 | |
| 0.045 | 0.101 | 0.107 | Protease 3C (Human rhinovirus) inhibitor | 0.065 0.044 CHEMBL1442231 0.072 0.034 CHEMBL3091859 0.081 0.026 CHEMBL1237174 0.107 0.013 CHEMBL3091852 | CHEMBL3091852 | |
| 0.002 | 0.059 | 0.015 | KiSS-1 receptor agonist | 0.015 0.004 CHEMBL3091852 | CHEMBL3091852 | |
| 0.044 | 0.101 | 0.103 | Elastase 1 inhibitor | 0.065 0.054 CHEMBL2111041 0.069 0.048 CHEMBL3544855 0.103 0.019 CHEMBL3544856 0.063 0.056 CHEMBL1442231 | CHEMBL3544856 | |
| 0.012 | 0.069 | 0.028 | Acetylcholine M4 receptor agonist | 0.028 0.023 CHEMBL1237174 | CHEMBL1237174 | |
| 0.036 | 0.094 | 0.066 | Cyclin-dependent kinase 6 inhibitor | 0.053 0.05 CHEMBL1203 0.066 0.035 CHEMBL1237174 | CHEMBL1237174 | |
| 0.003 | 0.062 | 0.009 | Thyroid hormone beta agonist | 0.009 0.006 CHEMBL3091859 | CHEMBL3091859 | |
| 0.008 | 0.068 | 0.025 | Telomerase stimulant | 0.016 0.015 CHEMBL1203 0.023 0.005 CHEMBL3544637 0.016 0.015 CHEMBL3091859 0.025 0.004 CHEMBL1237174 0.02 0.008 CHEMBL3091852 | CHEMBL1237174 | |
| 0.027 | 0.087 | 0.073 | AICAR transformylase inhibitor | 0.043 0.033 CHEMBL3544855 0.064 0.012 CHEMBL1203 0.073 0.009 CHEMBL3544636 0.054 0.018 CHEMBL1237174 0.047 0.026 CHEMBL3091852 | CHEMBL3544636 | |
| 0.025 | 0.085 | 0.15 | Ornithine carbamoyltransferase inhibitor | 0.15 0.01 CHEMBL1203 0.091 0.018 CHEMBL3544636 0.052 0.038 CHEMBL3544637 0.061 0.031 CHEMBL3091859 0.11 0.014 CHEMBL1237174 0.087 0.019 CHEMBL3091852 | CHEMBL1203 | |
| 0.023 | 0.084 | 0.096 | Antimetabolite | 0.048 0.033 CHEMBL3544855 0.043 0.037 CHEMBL1203 0.096 0.017 CHEMBL3544636 0.05 0.032 CHEMBL3544637 0.041 0.039 CHEMBL1237174 0.041 0.039 CHEMBL3091852 | CHEMBL3544636 | |
| 0.12 | 0.182 | 0.199 | Focal adhesion kinase 2 inhibitor | 0.156 0.12 CHEMBL1203 0.182 0.085 CHEMBL1442231 0.154 0.124 CHEMBL1237174 0.199 0.07 CHEMBL3091852 | CHEMBL3091852 | |
| 0.047 | 0.109 | 0.111 | Nicotinic alpha4beta2 receptor antagonist | 0.111 0.023 CHEMBL1203 0.096 0.035 CHEMBL1237174 | CHEMBL1203 | |
| 0.028 | 0.091 | 0.088 | Adenylate cyclase 1 inhibitor | 0.088 0.005 CHEMBL1237174 0.062 0.017 CHEMBL3091852 | CHEMBL1237174 | |
| 0.007 | 0.071 | 0.059 | Prostaglandin H2 antagonist | 0.03 0.013 CHEMBL3544855 0.059 0.003 CHEMBL1203 0.038 0.007 CHEMBL3544636 | CHEMBL1203 | |
| 0.015 | 0.079 | 0.036 | Thyroid hormone agonist | 0.025 0.02 CHEMBL3544636 0.036 0.008 CHEMBL3091859 0.029 0.013 CHEMBL1237174 0.025 0.02 CHEMBL3091852 | CHEMBL3091859 | |
| 0.032 | 0.097 | 0.06 | Potassium channel (ATP-sensitive) activator | 0.044 0.042 CHEMBL1203 0.06 0.016 CHEMBL1237174 0.052 0.027 CHEMBL3091852 | CHEMBL1237174 | |
| 0.026 | 0.091 | 0.05 | Thymidine kinase inhibitor | 0.041 0.029 CHEMBL1203 0.041 0.028 CHEMBL3544636 0.05 0.019 CHEMBL1237174 0.04 0.03 CHEMBL3091852 | CHEMBL1237174 | |
| 0.013 | 0.078 | 0.023 | Factor XIII inhibitor | 0.023 0.01 CHEMBL1237174 0.02 0.016 CHEMBL3091852 | CHEMBL1237174 | |
| 0.032 | 0.097 | 0.441 | Selectin antagonist | 0.091 0.031 CHEMBL1203 0.097 0.029 CHEMBL3544636 0.441 0.003 CHEMBL3544637 | CHEMBL3544637 | |
| 0.033 | 0.099 | 0.063 | Potassium channel (Inward rectifier) activator | 0.046 0.044 CHEMBL1203 0.063 0.016 CHEMBL1237174 0.054 0.028 CHEMBL3091852 | CHEMBL1237174 | |
| 0.026 | 0.092 | 0.117 | Glutamate (mGluR group III) agonist | 0.117 0.008 CHEMBL1203 0.039 0.036 CHEMBL3544636 0.042 0.031 CHEMBL1237174 | CHEMBL1203 | |
| 0.019 | 0.086 | 0.034 | Histone deacetylase 7 inhibitor | 0.034 0.028 CHEMBL3091852 | CHEMBL3091852 | |
| 0.122 | 0.189 | 0.188 | Neurotensin receptor agonist | 0.162 0.076 CHEMBL2111041 0.139 0.133 CHEMBL3544855 0.188 0.043 CHEMBL1203 0.14 0.128 CHEMBL1442231 0.186 0.044 CHEMBL3544636 0.152 0.097 CHEMBL3091859 0.179 0.05 CHEMBL1237174 0.185 0.045 CHEMBL3091852 | CHEMBL1203 | |
| 0.057 | 0.125 | 0.086 | Bronchodilator | 0.086 0.079 CHEMBL1203 | CHEMBL1203 | |
| 0.035 | 0.104 | 0.072 | Alpha 2 adrenoreceptor agonist | 0.072 0.03 CHEMBL1237174 | CHEMBL1237174 | |
| 0.062 | 0.131 | 0.372 | UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor | 0.372 0.004 CHEMBL1203 0.103 0.051 CHEMBL3544636 0.339 0.005 CHEMBL3544637 0.176 0.02 CHEMBL3091859 0.257 0.009 CHEMBL1237174 0.263 0.009 CHEMBL3091852 | CHEMBL1203 | |
| 0.022 | 0.092 | 0.066 | Membrane dipeptidase inhibitor | 0.036 0.034 CHEMBL2111041 0.04 0.027 CHEMBL3544855 0.054 0.013 CHEMBL1203 0.066 0.008 CHEMBL3544636 0.042 0.023 CHEMBL3091859 0.055 0.013 CHEMBL1237174 0.056 0.012 CHEMBL3091852 | CHEMBL3544636 | |
| 0.008 | 0.079 | 0.02 | Purinergic P2Y1 agonist | 0.02 0.007 CHEMBL1237174 | CHEMBL1237174 | |
| 0.007 | 0.078 | 0.025 | Alpha 2a adrenoreceptor agonist | 0.025 0.007 CHEMBL1237174 | CHEMBL1237174 | |
| 0.025 | 0.096 | 0.044 | Sphingosine kinase 1 inhibitor | 0.041 0.029 CHEMBL1237174 0.044 0.024 CHEMBL3091852 | CHEMBL3091852 | |
| 0.054 | 0.125 | 0.222 | Aminopeptidase B inhibitor | 0.222 0.017 CHEMBL1203 0.199 0.022 CHEMBL3544636 0.123 0.051 CHEMBL3091859 0.18 0.027 CHEMBL1237174 0.165 0.032 CHEMBL3091852 | CHEMBL1203 | |
| 0.054 | 0.126 | 0.081 | Interleukin-1 receptor-associated protein kinase 4 inhibitor | 0.081 0.069 CHEMBL3544636 | CHEMBL3544636 | |
| 0.035 | 0.109 | 0.076 | 5 Hydroxytryptamine 3A antagonist | 0.076 0.035 CHEMBL1237174 | CHEMBL1237174 | |
| 0.015 | 0.088 | 0.057 | Glutamate (mGluR1) agonist | 0.057 0.004 CHEMBL1203 0.027 0.013 CHEMBL3544636 0.03 0.009 CHEMBL1237174 0.026 0.015 CHEMBL3091852 | CHEMBL1203 | |
| 0.014 | 0.088 | 0.044 | Cathepsin L1 inhibitor | 0.044 0.024 CHEMBL3091852 | CHEMBL3091852 | |
| 0.079 | 0.153 | 0.199 | Toll-Like receptor 2 antagonist | 0.106 0.095 CHEMBL3544855 0.17 0.04 CHEMBL1203 0.128 0.069 CHEMBL1442231 0.199 0.024 CHEMBL3544636 0.151 0.052 CHEMBL3091859 0.153 0.051 CHEMBL1237174 0.198 0.024 CHEMBL3091852 | CHEMBL3544636 | |
| 0.048 | 0.122 | 0.08 | Acetylcholine nicotinic agonist | 0.08 0.056 CHEMBL1203 | CHEMBL1203 | |
| 0.049 | 0.124 | 0.134 | Glutamate (mGluR6) antagonist | 0.134 0.004 CHEMBL1203 0.064 0.054 CHEMBL3544636 0.074 0.032 CHEMBL3091859 0.114 0.007 CHEMBL1237174 0.092 0.014 CHEMBL3091852 | CHEMBL1203 | |
| 0.008 | 0.083 | 0.019 | Complement factor D inhibitor | 0.018 0.013 CHEMBL1203 0.019 0.012 CHEMBL1237174 | CHEMBL1237174 | |
| 0.018 | 0.094 | 0.072 | Toll-Like receptor 2 agonist | 0.038 0.031 CHEMBL1203 0.072 0.018 CHEMBL3544636 0.046 0.025 CHEMBL3544637 0.044 0.027 CHEMBL1237174 0.049 0.024 CHEMBL3091852 | CHEMBL3544636 | |
| 0.119 | 0.195 | 0.207 | Heat shock protein 70 antagonist | 0.207 0.005 CHEMBL1203 0.141 0.073 CHEMBL3544636 0.166 0.021 CHEMBL3544637 0.156 0.034 CHEMBL1237174 0.148 0.051 CHEMBL3091852 | CHEMBL1203 | |
| 0.031 | 0.107 | 0.13 | Alpha-mannosidase inhibitor | 0.056 0.033 CHEMBL3544856 0.063 0.023 CHEMBL1203 0.071 0.016 CHEMBL3544636 0.13 0.004 CHEMBL3544637 0.064 0.022 CHEMBL3091859 0.101 0.006 CHEMBL1237174 0.071 0.016 CHEMBL3091852 | CHEMBL3544637 | |
| 0.038 | 0.115 | 0.075 | Histone deacetylase inhibitor | 0.075 0.035 CHEMBL1442231 0.063 0.049 CHEMBL3091852 | CHEMBL1442231 | |
| 0.102 | 0.18 | 0.249 | Melanin inhibitor | 0.157 0.073 CHEMBL1203 0.249 0.029 CHEMBL3544637 0.13 0.113 CHEMBL3091859 0.16 0.069 CHEMBL1237174 0.162 0.067 CHEMBL3091852 | CHEMBL3544637 | |
| 0.021 | 0.099 | 0.052 | Glutamate (mGluR3) agonist | 0.052 0.004 CHEMBL1203 0.031 0.027 CHEMBL3091859 0.042 0.008 CHEMBL1237174 0.038 0.011 CHEMBL3091852 | CHEMBL1203 | |
| 0.066 | 0.145 | 0.104 | CC chemokine 5 receptor agonist | 0.104 0.018 CHEMBL1237174 0.089 0.038 CHEMBL3091852 | CHEMBL1237174 | |
| 0.085 | 0.166 | 0.18 | Antibacterial (Helicobacter pylori) | 0.121 0.08 CHEMBL3544856 0.18 0.028 CHEMBL1203 0.126 0.073 CHEMBL1442231 0.136 0.06 CHEMBL3544636 0.126 0.072 CHEMBL3544637 0.138 0.058 CHEMBL3091852 | CHEMBL1203 | |
| 0.063 | 0.144 | 0.376 | Chelator | 0.134 0.043 CHEMBL2111041 0.135 0.042 CHEMBL3544855 0.325 0.009 CHEMBL3544856 0.208 0.023 CHEMBL1203 0.107 0.068 CHEMBL1442231 0.376 0.007 CHEMBL3544636 0.105 0.07 CHEMBL3091852 | CHEMBL3544636 | |
| 0.003 | 0.084 | 0.011 | Thromboxane agonist | 0.011 0.007 CHEMBL3091852 | CHEMBL3091852 | |
| 0.008 | 0.09 | 0.019 | Integrin beta6 antagonist | 0.014 0.009 CHEMBL3544855 0.019 0.005 CHEMBL3544636 | CHEMBL3544636 | |
| 0.004 | 0.086 | 0.114 | Egl nine homolog 1 inhibitor | 0.042 0.004 CHEMBL1203 0.114 0.002 CHEMBL3544636 | CHEMBL3544636 | |
| 0.003 | 0.085 | 0.021 | Lysophosphatidic acid receptor 3 agonist | 0.021 0.005 CHEMBL1237174 0.017 0.007 CHEMBL3091852 | CHEMBL1237174 | |
| 0.025 | 0.108 | 0.065 | Cathepsin L inhibitor | 0.065 0.034 CHEMBL3091852 | CHEMBL3091852 | |
| 0.015 | 0.099 | 0.03 | 5 Hydroxytryptamine 6 agonist | 0.03 0.017 CHEMBL1237174 | CHEMBL1237174 | |
| 0.077 | 0.161 | 0.18 | NADPH oxidase inhibitor | 0.18 0.041 CHEMBL1203 0.105 0.104 CHEMBL1237174 0.137 0.065 CHEMBL3091852 | CHEMBL1203 | |
| 0.013 | 0.098 | 0.039 | Vanilloid 2 agonist | 0.036 0.005 CHEMBL1203 0.039 0.004 CHEMBL3544637 0.036 0.005 CHEMBL1237174 0.028 0.012 CHEMBL3091852 | CHEMBL3544637 | |
| 0.063 | 0.148 | 0.232 | M18 aspartyl aminopeptidase inhibitor | 0.1 0.092 CHEMBL1203 0.153 0.051 CHEMBL1442231 0.232 0.025 CHEMBL3091852 | CHEMBL3091852 | |
| 0.005 | 0.09 | 0.031 | KiSS-1 receptor antagonist | 0.031 0.005 CHEMBL3091852 | CHEMBL3091852 | |
| 0.035 | 0.121 | 0.205 | Catalase inhibitor | 0.071 0.054 CHEMBL3544855 0.205 0.014 CHEMBL1203 0.15 0.026 CHEMBL3544636 0.13 0.031 CHEMBL3091859 0.161 0.024 CHEMBL1237174 0.199 0.015 CHEMBL3091852 | CHEMBL1203 | |
| 0.005 | 0.091 | 0.017 | Aminopeptidase A inhibitor | 0.017 0.013 CHEMBL1203 | CHEMBL1203 | |
| 0.016 | 0.102 | 0.027 | Thrombin receptor antagonist | 0.027 0.022 CHEMBL3091852 | CHEMBL3091852 | |
| 0.019 | 0.107 | 0.079 | Adenosine deaminase inhibitor | 0.079 0.009 CHEMBL1203 0.055 0.025 CHEMBL3544636 0.069 0.014 CHEMBL3544637 0.061 0.02 CHEMBL1237174 0.047 0.033 CHEMBL3091852 | CHEMBL1203 | |
| 0.045 | 0.135 | 0.093 | CDK/cyclin complex inhibitor | 0.092 0.058 CHEMBL3091859 0.093 0.057 CHEMBL3091852 | CHEMBL3091852 | |
| 0.021 | 0.111 | 0.152 | Mannosidase inhibitor | 0.044 0.034 CHEMBL3544856 0.063 0.015 CHEMBL1203 0.059 0.017 CHEMBL3544636 0.152 0.004 CHEMBL3544637 0.048 0.028 CHEMBL3091859 0.09 0.007 CHEMBL1237174 0.056 0.019 CHEMBL3091852 | CHEMBL3544637 | |
| 0.03 | 0.121 | 0.069 | Cytokine production stimulant | 0.069 0.008 CHEMBL3544637 0.058 0.015 CHEMBL1237174 0.056 0.018 CHEMBL3091852 | CHEMBL3544637 | |
| 0.018 | 0.11 | 0.089 | Dopamine D5 agonist | 0.036 0.034 CHEMBL1203 0.089 0.005 CHEMBL1237174 0.049 0.018 CHEMBL3091852 | CHEMBL1237174 | |
| 0.018 | 0.11 | 0.183 | Phosphorylase inhibitor | 0.078 0.017 CHEMBL1203 0.135 0.009 CHEMBL3544636 0.183 0.005 CHEMBL3544637 | CHEMBL3544637 | |
| 0.054 | 0.147 | 0.129 | Glutathione S-transferase inhibitor | 0.098 0.039 CHEMBL1203 0.076 0.069 CHEMBL1442231 0.121 0.022 CHEMBL3544636 0.088 0.05 CHEMBL3091859 0.085 0.054 CHEMBL1237174 0.129 0.019 CHEMBL3091852 | CHEMBL3091852 | |
| 0.016 | 0.109 | 0.026 | Baculoviral IAP repeat-containing protein 4 inhibitor | 0.026 0.022 CHEMBL3091852 | CHEMBL3091852 | |
| 0.084 | 0.177 | 0.219 | Mcl-1 antagonist | 0.13 0.111 CHEMBL2111041 0.219 0.047 CHEMBL1203 | CHEMBL1203 | |
| 0.024 | 0.117 | 0.075 | Protein kinase C epsilon inhibitor | 0.075 0.022 CHEMBL1203 0.056 0.034 CHEMBL3544636 | CHEMBL1203 | |
| 0.046 | 0.14 | 0.082 | I kappa B kinase inhibitor | 0.082 0.058 CHEMBL1203 | CHEMBL1203 | |
| 0.01 | 0.103 | 0.026 | Isoleucine-tRNA ligase inhibitor | 0.021 0.019 CHEMBL1203 0.026 0.009 CHEMBL1237174 0.025 0.011 CHEMBL3091852 | CHEMBL1237174 | |
| 0.006 | 0.1 | 0.019 | Alpha 2c adrenoreceptor agonist | 0.019 0.013 CHEMBL1237174 | CHEMBL1237174 | |
| 0.097 | 0.191 | 0.196 | Adenylate cyclase stimulant | 0.157 0.051 CHEMBL1203 0.156 0.054 CHEMBL3544636 0.148 0.066 CHEMBL3544637 0.143 0.075 CHEMBL3091859 0.196 0.015 CHEMBL1237174 0.171 0.034 CHEMBL3091852 | CHEMBL1237174 | |
| 0.133 | 0.227 | 0.296 | Lipoxygenase inhibitor | 0.296 0.073 CHEMBL2111041 0.217 0.124 CHEMBL3544855 0.22 0.122 CHEMBL1203 0.22 0.121 CHEMBL3091859 0.204 0.137 CHEMBL3091852 | CHEMBL2111041 | |
| 0.028 | 0.122 | 0.065 | Aldosterone antagonist | 0.065 0.017 CHEMBL1203 0.054 0.024 CHEMBL1237174 | CHEMBL1203 | |
| 0.012 | 0.106 | 0.048 | Potassium channel small-conductance Ca-activated activator | 0.048 0.012 CHEMBL1237174 | CHEMBL1237174 | |
| 0.089 | 0.184 | 0.304 | Hexokinase inhibitor | 0.138 0.093 CHEMBL3544856 0.302 0.011 CHEMBL1203 0.141 0.09 CHEMBL1442231 0.133 0.1 CHEMBL3544636 0.304 0.01 CHEMBL3544637 0.161 0.066 CHEMBL1237174 0.199 0.036 CHEMBL3091852 | CHEMBL3544637 | |
| 0.028 | 0.124 | 0.055 | Nicotinic receptor alpha7 subunit antagonist | 0.055 0.035 CHEMBL1203 | CHEMBL1203 | |
| 0.011 | 0.107 | 0.031 | Neuraminidase (Influenza B) inhibitor | 0.031 0.004 CHEMBL1203 0.023 0.01 CHEMBL3091859 0.025 0.008 CHEMBL1237174 0.03 0.004 CHEMBL3091852 | CHEMBL1203 | |
| 0.006 | 0.103 | 0.02 | Adenosine kinase inhibitor | 0.02 0.017 CHEMBL1237174 | CHEMBL1237174 | |
| 0.027 | 0.124 | 0.048 | Purinergic P2X4 antagonist | 0.048 0.029 CHEMBL1203 0.047 0.03 CHEMBL1237174 | CHEMBL1203 | |
| 0.04 | 0.138 | 0.089 | Thrombin inhibitor | 0.089 0.033 CHEMBL1237174 | CHEMBL1237174 | |
| 0.052 | 0.15 | 0.109 | Vanilloid 4 agonist | 0.081 0.038 CHEMBL3091859 0.109 0.011 CHEMBL1237174 0.101 0.016 CHEMBL3091852 | CHEMBL1237174 | |
| 0.062 | 0.161 | 0.139 | MAP kinase kinase 1 inhibitor | 0.134 0.024 CHEMBL1203 0.118 0.037 CHEMBL1442231 0.104 0.052 CHEMBL1237174 0.139 0.021 CHEMBL3091852 | CHEMBL3091852 | |
| 0.018 | 0.117 | 0.068 | RNA-directed RNA polymerase inhibitor | 0.068 0.008 CHEMBL1203 0.041 0.017 CHEMBL3544636 0.031 0.03 CHEMBL1237174 | CHEMBL1203 | |
| 0.135 | 0.234 | 0.264 | 12-Lipoxygenase inhibitor | 0.243 0.113 CHEMBL2111041 0.231 0.121 CHEMBL1203 0.221 0.13 CHEMBL1442231 0.264 0.101 CHEMBL3091852 | CHEMBL3091852 | |
| 0.012 | 0.112 | 0.085 | Plasmepsin I inhibitor | 0.053 0.007 CHEMBL3544856 0.053 0.006 CHEMBL1442231 0.085 0.004 CHEMBL3091852 | CHEMBL3091852 | |
| 0.101 | 0.202 | 0.152 | Pregnane X receptor agonist | 0.139 0.077 CHEMBL1203 0.152 0.049 CHEMBL1237174 0.139 0.075 CHEMBL3091852 | CHEMBL1237174 | |
| 0.003 | 0.105 | 0.012 | Imidazoline I2 receptor antagonist | 0.012 0.006 CHEMBL1237174 | CHEMBL1237174 | |
| 0.044 | 0.146 | 0.154 | Histamine N-methyltransferase inhibitor | 0.154 0.013 CHEMBL1203 0.131 0.023 CHEMBL1237174 0.075 0.073 CHEMBL3091852 | CHEMBL1203 | |
| 0.083 | 0.186 | 0.21 | Diuretic | 0.21 0.041 CHEMBL1203 0.209 0.041 CHEMBL3544636 0.175 0.057 CHEMBL3544637 0.16 0.069 CHEMBL1237174 | CHEMBL1203 | |
| 0.012 | 0.116 | 0.034 | Lysophosphatidic acid receptor 1 agonist | 0.025 0.017 CHEMBL1203 0.025 0.018 CHEMBL3091859 0.034 0.008 CHEMBL1237174 0.032 0.009 CHEMBL3091852 | CHEMBL1237174 | |
| 0.002 | 0.106 | 0.015 | Integrin alphaVbeta5 antagonist | 0.015 0.005 CHEMBL3544636 | CHEMBL3544636 | |
| 0.067 | 0.172 | 0.132 | Glutamate (mGluR7) agonist | 0.094 0.074 CHEMBL1203 0.098 0.065 CHEMBL3544636 0.097 0.067 CHEMBL3091859 0.132 0.02 CHEMBL1237174 0.126 0.025 CHEMBL3091852 | CHEMBL1237174 | |
| 0.012 | 0.116 | 0.059 | Phosphoglycerate kinase inhibitor | 0.059 0.011 CHEMBL1203 0.046 0.016 CHEMBL1237174 | CHEMBL1203 | |
| 0.018 | 0.122 | 0.038 | Ceramide glucosyltransferase inhibitor | 0.038 0.021 CHEMBL3544636 0.038 0.019 CHEMBL3544637 0.038 0.021 CHEMBL1237174 | CHEMBL1237174 | |
| 0.027 | 0.132 | 0.084 | 3(or 17)beta-hydroxysteroid dehydrogenase inhibitor | 0.084 0.014 CHEMBL1203 0.074 0.019 CHEMBL1237174 0.059 0.031 CHEMBL3091852 | CHEMBL1203 | |
| 0.114 | 0.219 | 0.163 | Death-associated protein kinase 2 inhibitor | 0.152 0.102 CHEMBL1442231 0.163 0.079 CHEMBL3091852 | CHEMBL3091852 | |
| 0.019 | 0.124 | 0.057 | Integrin alpha2 antagonist | 0.045 0.015 CHEMBL1203 0.057 0.008 CHEMBL3544636 0.039 0.022 CHEMBL1237174 | CHEMBL3544636 | |
| 0.03 | 0.135 | 0.073 | Neuronal nicotinic receptor antagonist | 0.073 0.042 CHEMBL1203 | CHEMBL1203 | |
| 0.009 | 0.114 | 0.02 | CXC chemokine 5 receptor antagonist | 0.02 0.009 CHEMBL1203 | CHEMBL1203 | |
| 0.042 | 0.148 | 0.085 | HIV-1 integrase inhibitor | 0.085 0.035 CHEMBL1203 0.072 0.046 CHEMBL3544636 | CHEMBL1203 | |
| 0.06 | 0.166 | 0.162 | Interleukin 1 beta converting enzyme inhibitor | 0.086 0.079 CHEMBL3544855 0.109 0.046 CHEMBL1203 0.104 0.053 CHEMBL1442231 0.162 0.013 CHEMBL3544636 0.088 0.076 CHEMBL1237174 0.107 0.049 CHEMBL3091852 | CHEMBL3544636 | |
| 0.035 | 0.141 | 0.083 | 5 Hydroxytryptamine 3 agonist | 0.083 0.025 CHEMBL1237174 | CHEMBL1237174 | |
| 0.036 | 0.143 | 0.099 | Cathepsin G inhibitor | 0.064 0.062 CHEMBL1203 0.069 0.055 CHEMBL3091859 0.099 0.034 CHEMBL1237174 | CHEMBL1237174 | |
| 0.033 | 0.141 | 0.056 | 5 Hydroxytryptamine 7 agonist | 0.056 0.038 CHEMBL1237174 | CHEMBL1237174 | |
| 0.07 | 0.178 | 0.192 | Folate antagonist | 0.097 0.07 CHEMBL2111041 0.159 0.019 CHEMBL3544855 0.121 0.038 CHEMBL1203 0.192 0.011 CHEMBL3544636 | CHEMBL3544636 | |
| 0.051 | 0.16 | 0.165 | Prolactin inhibitor | 0.116 0.041 CHEMBL1203 0.088 0.069 CHEMBL3091859 0.165 0.017 CHEMBL1237174 0.132 0.031 CHEMBL3091852 | CHEMBL1237174 | |
| 0.033 | 0.143 | 0.115 | Na+ K+ transporting ATPase inhibitor | 0.082 0.048 CHEMBL1203 0.115 0.02 CHEMBL3544637 0.105 0.027 CHEMBL1237174 0.088 0.043 CHEMBL3091852 | CHEMBL3544637 | |
| 0.106 | 0.215 | 0.175 | MAP kinase kinase 4 inhibitor | 0.131 0.11 CHEMBL3544856 0.175 0.029 CHEMBL1203 | CHEMBL1203 | |
| 0.052 | 0.162 | 0.133 | GABA B receptor agonist | 0.071 0.066 CHEMBL2111041 0.075 0.053 CHEMBL3544855 0.133 0.005 CHEMBL1203 0.095 0.021 CHEMBL3544636 0.07 0.068 CHEMBL3091859 0.102 0.015 CHEMBL1237174 0.091 0.025 CHEMBL3091852 | CHEMBL1203 | |
| 0.017 | 0.127 | 0.035 | Carboxypeptidase B inhibitor | 0.034 0.021 CHEMBL1203 0.035 0.019 CHEMBL3544636 0.031 0.027 CHEMBL1237174 | CHEMBL3544636 | |
| 0.011 | 0.121 | 0.196 | Nicotinic acid receptor agonist | 0.196 0.003 CHEMBL1203 0.032 0.031 CHEMBL1237174 0.035 0.026 CHEMBL3091852 | CHEMBL1203 | |
| 0.057 | 0.167 | 0.111 | mTOR complex 2 inhibitor | 0.082 0.063 CHEMBL1203 0.111 0.023 CHEMBL1237174 0.085 0.056 CHEMBL3091852 | CHEMBL1237174 | |
| 0.018 | 0.129 | 0.057 | Retinoid X alpha receptor antagonist | 0.057 0.004 CHEMBL1203 0.036 0.021 CHEMBL1237174 0.031 0.03 CHEMBL3091852 | CHEMBL1203 | |
| 0.05 | 0.161 | 0.083 | MDM2 inhibitor | 0.083 0.016 CHEMBL1203 0.073 0.032 CHEMBL3091859 0.083 0.016 CHEMBL1237174 0.068 0.044 CHEMBL3091852 | CHEMBL1237174 | |
| 0.04 | 0.152 | 0.069 | Immunoglobulin Fc receptor antagonist | 0.057 0.032 CHEMBL1203 0.053 0.047 CHEMBL3091859 0.069 0.012 CHEMBL1237174 0.064 0.018 CHEMBL3091852 | CHEMBL1237174 | |
| 0.009 | 0.121 | 0.044 | Lysophosphatidic acid 1 receptor antagonist | 0.044 0.004 CHEMBL1203 | CHEMBL1203 | |
| 0.029 | 0.142 | 0.169 | Heparanase inhibitor | 0.073 0.01 CHEMBL1203 0.062 0.02 CHEMBL3544636 0.169 0.003 CHEMBL3544637 0.055 0.033 CHEMBL1237174 0.05 0.045 CHEMBL3091852 | CHEMBL3544637 | |
| 0.016 | 0.129 | 0.054 | CDK2/cyclin E inhibitor | 0.054 0.049 CHEMBL3091859 | CHEMBL3091859 | |
| 0.013 | 0.128 | 0.034 | Integrin alpha2beta1 antagonist | 0.034 0.009 CHEMBL1203 0.029 0.013 CHEMBL3544636 0.028 0.015 CHEMBL1237174 | CHEMBL1203 | |
| 0.041 | 0.156 | 0.074 | Ryanodine receptor antagonist | 0.074 0.013 CHEMBL1203 0.055 0.054 CHEMBL3544636 0.073 0.014 CHEMBL1237174 0.058 0.042 CHEMBL3091852 | CHEMBL1203 | |
| 0.036 | 0.152 | 0.076 | Corticotropin releasing factor 2 receptor antagonist | 0.076 0.02 CHEMBL1237174 0.064 0.038 CHEMBL3091852 | CHEMBL1237174 | |
| 0.01 | 0.126 | 0.04 | Retinoid X beta receptor antagonist | 0.04 0.003 CHEMBL1203 0.022 0.011 CHEMBL1237174 | CHEMBL1203 | |
| 0.02 | 0.137 | 0.104 | Dihydroorotase inhibitor | 0.104 0.005 CHEMBL1203 0.049 0.026 CHEMBL1237174 0.04 0.039 CHEMBL3091852 | CHEMBL1203 | |
| 0.009 | 0.126 | 0.058 | HCV NS5B polymerase inhibitor | 0.058 0.008 CHEMBL1203 0.032 0.021 CHEMBL3544636 | CHEMBL1203 | |
| 0.02 | 0.138 | 0.066 | Retinoid X receptor antagonist | 0.066 0.004 CHEMBL1203 0.04 0.023 CHEMBL1237174 0.035 0.033 CHEMBL3091852 | CHEMBL1203 | |
| 0.011 | 0.129 | 0.161 | Urate transporter 1 inhibitor | 0.161 0.004 CHEMBL1203 | CHEMBL1203 | |
| 0.087 | 0.207 | 0.168 | Sphingosine 1-phosphate receptor 2 antagonist | 0.158 0.031 CHEMBL1203 0.114 0.112 CHEMBL3544636 0.133 0.068 CHEMBL3091859 0.157 0.032 CHEMBL1237174 0.168 0.023 CHEMBL3091852 | CHEMBL3091852 | |
| 0.022 | 0.142 | 0.06 | Prolyl endopeptidase inhibitor | 0.056 0.028 CHEMBL1203 0.06 0.024 CHEMBL3544636 0.049 0.038 CHEMBL1237174 | CHEMBL3544636 | |
| 0.044 | 0.164 | 0.125 | Glycine receptor agonist | 0.125 0.011 CHEMBL1203 0.071 0.053 CHEMBL3544636 0.085 0.033 CHEMBL3544637 0.074 0.047 CHEMBL3091859 0.122 0.012 CHEMBL1237174 0.102 0.02 CHEMBL3091852 | CHEMBL1203 | |
| 0.031 | 0.152 | 0.064 | Nicotinic alpha3beta2 receptor antagonist | 0.058 0.029 CHEMBL1203 0.064 0.022 CHEMBL1237174 0.049 0.047 CHEMBL3091852 | CHEMBL1237174 | |
| 0.161 | 0.284 | 0.203 | Ca(v)3.3 blocker | 0.203 0.185 CHEMBL3544636 | CHEMBL3544636 | |
| 0.008 | 0.132 | 0.033 | Integrin alphaVbeta3 antagonist | 0.024 0.013 CHEMBL3544855 0.022 0.015 CHEMBL1442231 0.033 0.007 CHEMBL3544636 | CHEMBL3544636 | |
| 0.054 | 0.178 | 0.266 | Cholesterol synthesis inhibitor | 0.266 0.015 CHEMBL1203 0.152 0.043 CHEMBL3544636 0.171 0.035 CHEMBL3544637 0.129 0.057 CHEMBL1237174 | CHEMBL1203 | |
| 0.017 | 0.142 | 0.046 | Melatonin receptor 1A agonist | 0.033 0.024 CHEMBL3091859 0.037 0.017 CHEMBL1237174 0.046 0.009 CHEMBL3091852 | CHEMBL3091852 | |
| 0.016 | 0.141 | 0.131 | Glutamate (mGluR3) antagonist | 0.131 0.004 CHEMBL1203 0.047 0.014 CHEMBL1237174 0.034 0.03 CHEMBL3091852 | CHEMBL1203 | |
| 0.029 | 0.155 | 0.053 | Bombesin 2 receptor antagonist | 0.047 0.039 CHEMBL1203 0.053 0.029 CHEMBL3544636 0.05 0.034 CHEMBL1237174 | CHEMBL3544636 | |
| 0.007 | 0.133 | 0.106 | Kynurenine 3 monooxygenase inhibitor | 0.106 0.004 CHEMBL1203 | CHEMBL1203 | |
| 0.026 | 0.152 | 0.064 | HCV NS3/NS4A protease inhibitor | 0.045 0.044 CHEMBL3544636 0.047 0.039 CHEMBL3091859 0.05 0.032 CHEMBL1237174 0.064 0.018 CHEMBL3091852 | CHEMBL3091852 | |
| 0.011 | 0.14 | 0.025 | Myristoyl transferase inhibitor | 0.025 0.024 CHEMBL1237174 | CHEMBL1237174 | |
| 0.018 | 0.147 | 0.067 | Neutrophil collagenase inhibitor | 0.062 0.048 CHEMBL3544636 0.067 0.042 CHEMBL1237174 | CHEMBL1237174 | |
| 0.042 | 0.173 | 0.097 | Phosphodiesterase VI inhibitor | 0.08 0.041 CHEMBL1203 0.097 0.022 CHEMBL3544637 | CHEMBL3544637 | |
| 0.008 | 0.139 | 0.028 | Protease (Human cytomegalovirus) inhibitor | 0.023 0.014 CHEMBL1203 0.025 0.012 CHEMBL1237174 0.028 0.009 CHEMBL3091852 | CHEMBL3091852 | |
| 0.033 | 0.165 | 0.091 | Potassium channel intermediate-conductance Ca-activated blocker | 0.091 0.012 CHEMBL1203 0.074 0.023 CHEMBL1237174 0.056 0.05 CHEMBL3091852 | CHEMBL1203 | |
| 0.022 | 0.155 | 0.05 | Benzodiazepine antagonist | 0.05 0.027 CHEMBL3091852 | CHEMBL3091852 | |
| 0.007 | 0.14 | 0.028 | Imidazoline I1 receptor antagonist | 0.028 0.008 CHEMBL1237174 | CHEMBL1237174 | |
| 0.03 | 0.164 | 0.127 | CD45 antagonist | 0.081 0.012 CHEMBL1203 0.127 0.007 CHEMBL3544636 | CHEMBL3544636 | |
| 0.005 | 0.138 | 0.058 | Arginase inhibitor | 0.056 0.012 CHEMBL1203 0.041 0.021 CHEMBL3544636 0.058 0.011 CHEMBL3544637 0.051 0.015 CHEMBL1237174 0.044 0.019 CHEMBL3091852 | CHEMBL3544637 | |
| 0.053 | 0.188 | 0.1 | Bromodomain-containing protein 2 inhibitor | 0.089 0.058 CHEMBL1203 0.1 0.04 CHEMBL1237174 0.095 0.047 CHEMBL3091852 | CHEMBL1237174 | |
| 0.029 | 0.164 | 0.058 | Bombesin 3 receptor antagonist | 0.058 0.035 CHEMBL1203 | CHEMBL1203 | |
| 0.056 | 0.191 | 0.151 | Proteasome inhibitor | 0.096 0.093 CHEMBL1442231 0.118 0.067 CHEMBL3544636 0.1 0.088 CHEMBL1237174 0.151 0.046 CHEMBL3091852 | CHEMBL3091852 | |
| 0.012 | 0.147 | 0.031 | Acid ceramidase inhibitor | 0.031 0.008 CHEMBL1237174 0.024 0.021 CHEMBL3091852 | CHEMBL1237174 | |
| 0.015 | 0.151 | 0.076 | Aromatase inhibitor | 0.076 0.03 CHEMBL1203 | CHEMBL1203 | |
| 0.06 | 0.197 | 0.247 | Microtubule formation inhibitor | 0.149 0.038 CHEMBL1203 0.119 0.061 CHEMBL3544636 0.247 0.009 CHEMBL3544637 0.142 0.042 CHEMBL1237174 0.116 0.065 CHEMBL3091852 | CHEMBL3544637 | |
| 0.027 | 0.165 | 0.077 | Squalene epoxidase inhibitor | 0.06 0.021 CHEMBL1203 0.077 0.01 CHEMBL3544637 0.061 0.019 CHEMBL1237174 0.047 0.039 CHEMBL3091852 | CHEMBL3544637 | |
| 0.015 | 0.153 | 0.031 | Dipeptidyl peptidase II inhibitor | 0.031 0.026 CHEMBL1237174 | CHEMBL1237174 | |
| 0.025 | 0.164 | 0.082 | Sphingosine 1-phosphate receptor 3 antagonist | 0.082 0.015 CHEMBL1203 0.07 0.026 CHEMBL3544636 0.059 0.04 CHEMBL1237174 | CHEMBL1203 | |
| 0.027 | 0.167 | 0.078 | Syk tyrosine kinase inhibitor | 0.078 0.042 CHEMBL1203 | CHEMBL1203 | |
| 0.055 | 0.194 | 0.237 | Alkylator | 0.108 0.08 CHEMBL1203 0.127 0.061 CHEMBL3544636 0.237 0.018 CHEMBL3544637 0.131 0.058 CHEMBL1237174 0.124 0.064 CHEMBL3091852 | CHEMBL3544637 | |
| 0.003 | 0.142 | 0.023 | Angiotensin AT1B receptor antagonist | 0.023 0.005 CHEMBL1203 | CHEMBL1203 | |
| 0.021 | 0.161 | 0.083 | Diacylglycerol O-acyltransferase inhibitor | 0.069 0.02 CHEMBL1203 0.083 0.013 CHEMBL3544636 | CHEMBL3544636 | |
| 0.091 | 0.232 | 0.334 | Interferon gamma antagonist | 0.256 0.027 CHEMBL1203 0.334 0.016 CHEMBL3544637 0.179 0.051 CHEMBL1237174 0.155 0.071 CHEMBL3091852 | CHEMBL3544637 | |
| 0.037 | 0.177 | 0.068 | Metalloproteinase-9 inhibitor | 0.068 0.059 CHEMBL1237174 | CHEMBL1237174 | |
| 0.031 | 0.172 | 0.123 | Phosphodiesterase IV inhibitor | 0.123 0.032 CHEMBL1203 | CHEMBL1203 | |
| 0.043 | 0.187 | 0.101 | GABA A receptor agonist | 0.101 0.037 CHEMBL1203 | CHEMBL1203 | |
| 0.063 | 0.207 | 0.207 | Photosensitizer | 0.164 0.024 CHEMBL1203 0.117 0.061 CHEMBL3544636 0.207 0.011 CHEMBL3544637 0.099 0.091 CHEMBL3091859 0.152 0.03 CHEMBL1237174 0.134 0.043 CHEMBL3091852 | CHEMBL3544637 | |
| 0.034 | 0.179 | 0.059 | Phosphodiesterase 1A inhibitor | 0.056 0.053 CHEMBL1203 0.059 0.044 CHEMBL1237174 | CHEMBL1237174 | |
| 0.003 | 0.15 | 0.019 | G-protein-coupled receptor 120 agonist | 0.019 0.01 CHEMBL1203 | CHEMBL1203 | |
| 0.02 | 0.167 | 0.099 | Acetylcholine M5 receptor agonist | 0.099 0.021 CHEMBL1237174 0.08 0.034 CHEMBL3091852 | CHEMBL1237174 | |
| 0.009 | 0.156 | 0.053 | Free fatty acid receptor 1 antagonist | 0.053 0.008 CHEMBL1203 0.033 0.025 CHEMBL1237174 | CHEMBL1203 | |
| 0.009 | 0.158 | 0.474 | Protocollagen prolyl hydroxylase inhibitor | 0.056 0.005 CHEMBL1203 0.474 0.002 CHEMBL3544636 | CHEMBL3544636 | |
| 0.074 | 0.223 | 0.124 | Transcription factor STAT6 inhibitor | 0.117 0.065 CHEMBL1203 0.124 0.053 CHEMBL1237174 0.124 0.054 CHEMBL3091852 | CHEMBL3091852 | |
| 0.021 | 0.171 | 0.049 | Matrix metalloproteinase (membrane-type) inhibitor | 0.049 0.048 CHEMBL1237174 | CHEMBL1237174 | |
| 0.03 | 0.182 | 0.084 | Acetylcholine nicotinic antagonist | 0.084 0.05 CHEMBL1203 | CHEMBL1203 | |
| 0.003 | 0.156 | 0.027 | Integrin beta2 antagonist | 0.011 0.01 CHEMBL1203 0.027 0.004 CHEMBL3544636 | CHEMBL3544636 | |
| 0.02 | 0.173 | 0.066 | Beta 1 adrenoreceptor antagonist | 0.052 0.043 CHEMBL1203 0.06 0.036 CHEMBL3544636 0.066 0.03 CHEMBL1237174 | CHEMBL1237174 | |
| 0.092 | 0.247 | 0.455 | Spasmolytic | 0.251 0.09 CHEMBL1203 0.455 0.03 CHEMBL3544637 0.185 0.133 CHEMBL3091859 0.241 0.095 CHEMBL1237174 | CHEMBL3544637 | |
| 0.091 | 0.247 | 0.249 | Ca2+/calmodulin-dependent protein kinase kinase B inhibitor | 0.249 0.006 CHEMBL1203 0.132 0.112 CHEMBL3544636 | CHEMBL1203 | |
| 0.008 | 0.166 | 0.024 | Prostaglandin F2 alpha agonist | 0.024 0.013 CHEMBL1237174 | CHEMBL1237174 | |
| 0.02 | 0.178 | 0.056 | TRPA1 antagonist | 0.056 0.05 CHEMBL1203 | CHEMBL1203 | |
| 0.042 | 0.2 | 0.086 | Neuropeptide Y antagonist | 0.086 0.051 CHEMBL1442231 0.083 0.055 CHEMBL3091852 | CHEMBL1442231 | |
| 0.019 | 0.177 | 0.043 | 5 Hydroxytryptamine 2B agonist | 0.043 0.02 CHEMBL1237174 | CHEMBL1237174 | |
| 0.003 | 0.163 | 0.012 | Melatonin 2 antagonist | 0.012 0.009 CHEMBL3091852 | CHEMBL3091852 | |
| 0.024 | 0.184 | 0.061 | Alpha adrenoreceptor agonist | 0.061 0.054 CHEMBL1237174 | CHEMBL1237174 | |
| 0.032 | 0.193 | 0.074 | Metalloproteinase-2 inhibitor | 0.074 0.059 CHEMBL3544636 | CHEMBL3544636 | |
| 0.014 | 0.176 | 0.066 | Fructose-1,6-bisphosphatase inhibitor | 0.048 0.027 CHEMBL1203 0.066 0.014 CHEMBL1237174 | CHEMBL1237174 | |
| 0.037 | 0.199 | 0.07 | Phosphodiesterase 1C inhibitor | 0.07 0.029 CHEMBL1203 0.059 0.052 CHEMBL1237174 0.058 0.055 CHEMBL3091852 | CHEMBL1203 | |
| 0.011 | 0.175 | 0.034 | Lysophosphatidic acid 2 receptor antagonist | 0.034 0.017 CHEMBL1237174 0.03 0.022 CHEMBL3091852 | CHEMBL1237174 | |
| 0.119 | 0.284 | 0.795 | Cholesterol antagonist | 0.188 0.176 CHEMBL3544855 0.634 0.014 CHEMBL1203 0.355 0.062 CHEMBL3544636 0.795 0.004 CHEMBL3544637 0.319 0.079 CHEMBL1237174 0.252 0.124 CHEMBL3091852 | CHEMBL3544637 | |
| 0.023 | 0.188 | 0.043 | Leukotriene C4 antagonist | 0.043 0.019 CHEMBL1203 0.037 0.034 CHEMBL1237174 | CHEMBL1203 | |
| 0.016 | 0.181 | 0.095 | Thromboxane antagonist | 0.095 0.013 CHEMBL1203 0.055 0.037 CHEMBL3544636 | CHEMBL1203 | |
| 0.021 | 0.187 | 0.067 | Collagenase 3 inhibitor | 0.067 0.034 CHEMBL1203 0.058 0.045 CHEMBL3544636 | CHEMBL1203 | |
| 0.007 | 0.173 | 0.083 | Sodium/glucose cotransporter 2 inhibitor | 0.083 0.004 CHEMBL3544637 0.025 0.021 CHEMBL1237174 | CHEMBL3544637 | |
| 0.011 | 0.177 | 0.069 | Guanylate cyclase inhibitor | 0.069 0.005 CHEMBL1203 0.058 0.014 CHEMBL3544637 0.066 0.007 CHEMBL1237174 0.042 0.03 CHEMBL3091852 | CHEMBL1203 | |
| 0.059 | 0.226 | 0.152 | Glutamate release inhibitor | 0.119 0.023 CHEMBL1203 0.152 0.009 CHEMBL3544637 0.14 0.012 CHEMBL1237174 0.103 0.038 CHEMBL3091852 | CHEMBL3544637 | |
| 0.021 | 0.189 | 0.079 | Leukotriene antagonist | 0.079 0.033 CHEMBL1203 | CHEMBL1203 | |
| 0.103 | 0.274 | 0.644 | Hypoglycemic | 0.551 0.011 CHEMBL2111041 0.19 0.123 CHEMBL3544855 0.282 0.059 CHEMBL3544856 0.243 0.081 CHEMBL1203 0.204 0.109 CHEMBL3544636 0.644 0.006 CHEMBL3544637 | CHEMBL3544637 | |
| 0.034 | 0.205 | 0.067 | Secretase beta inhibitor | 0.064 0.062 CHEMBL1203 0.067 0.054 CHEMBL1237174 | CHEMBL1237174 | |
| 0.015 | 0.187 | 0.125 | Dihydroorotate dehydrogenase inhibitor | 0.125 0.007 CHEMBL1203 | CHEMBL1203 | |
| 0.007 | 0.18 | 0.053 | AMPA 3 receptor antagonist | 0.053 0.008 CHEMBL1203 0.041 0.013 CHEMBL3544636 | CHEMBL1203 | |
| 0.004 | 0.177 | 0.015 | 5-Alpha-reductase 1 inhibitor | 0.015 0.013 CHEMBL1203 | CHEMBL1203 | |
| 0.016 | 0.189 | 0.072 | AMPA 4 receptor antagonist | 0.072 0.008 CHEMBL1203 0.039 0.028 CHEMBL1237174 0.036 0.035 CHEMBL3091852 | CHEMBL1203 | |
| 0.007 | 0.18 | 0.02 | 5-Alpha-reductase 2 inhibitor | 0.02 0.013 CHEMBL1203 | CHEMBL1203 | |
| 0.002 | 0.175 | 0.009 | Progesterone receptor A antagonist | 0.009 0.008 CHEMBL1237174 | CHEMBL1237174 | |
| 0.006 | 0.18 | 0.042 | Glutamate (mGluR2) antagonist | 0.042 0.011 CHEMBL1203 | CHEMBL1203 | |
| 0.075 | 0.249 | 0.17 | Neuropeptide Y1 antagonist | 0.146 0.072 CHEMBL3091859 0.164 0.046 CHEMBL1237174 0.17 0.039 CHEMBL3091852 | CHEMBL3091852 | |
| 0.003 | 0.178 | 0.055 | Kainate receptor 1 antagonist | 0.055 0.005 CHEMBL1203 | CHEMBL1203 | |
| 0.021 | 0.197 | 0.061 | GABA B receptor antagonist | 0.061 0.012 CHEMBL1203 0.043 0.03 CHEMBL1237174 | CHEMBL1203 | |
| 0.049 | 0.225 | 0.23 | Carbonic anhydrase III inhibitor | 0.23 0.012 CHEMBL1203 0.089 0.076 CHEMBL3544636 0.101 0.061 CHEMBL3544637 0.133 0.036 CHEMBL1237174 0.125 0.041 CHEMBL3091852 | CHEMBL1203 | |
| 0.06 | 0.237 | 0.168 | TRPA1 agonist | 0.168 0.02 CHEMBL1203 0.109 0.073 CHEMBL3544636 0.125 0.053 CHEMBL1237174 0.098 0.091 CHEMBL3091852 | CHEMBL1203 | |
| 0.01 | 0.188 | 0.063 | Oleamide hydrolase inhibitor | 0.063 0.019 CHEMBL1203 | CHEMBL1203 | |
| 0.04 | 0.217 | 0.131 | Gastric antisecretory | 0.131 0.036 CHEMBL1203 0.094 0.073 CHEMBL3544636 0.093 0.075 CHEMBL1237174 | CHEMBL1203 | |
| 0.017 | 0.196 | 0.062 | Phosphodiesterase 4C inhibitor | 0.062 0.033 CHEMBL1203 0.06 0.034 CHEMBL1442231 | CHEMBL1203 | |
| 0.009 | 0.19 | 0.111 | Retinoid X alpha receptor agonist | 0.111 0.004 CHEMBL1203 0.034 0.025 CHEMBL1237174 | CHEMBL1203 | |
| 0.061 | 0.243 | 0.149 | CDK3/cyclin E inhibitor | 0.103 0.082 CHEMBL1442231 0.12 0.055 CHEMBL3544636 0.149 0.027 CHEMBL3091852 | CHEMBL3091852 | |
| 0.094 | 0.276 | 0.18 | Prostaglandin dehydrogenase inhibitor | 0.18 0.172 CHEMBL1237174 | CHEMBL1237174 | |
| 0.019 | 0.202 | 0.063 | 5 Hydroxytryptamine 2A agonist | 0.063 0.044 CHEMBL1237174 | CHEMBL1237174 | |
| 0.016 | 0.201 | 0.039 | DNA topoisomerase IV inhibitor | 0.039 0.009 CHEMBL1203 | CHEMBL1203 | |
| 0.094 | 0.279 | 0.209 | Phospholipase C inhibitor | 0.209 0.038 CHEMBL1203 0.193 0.049 CHEMBL3544636 0.153 0.1 CHEMBL3544637 0.144 0.12 CHEMBL3091859 0.194 0.048 CHEMBL1237174 0.183 0.058 CHEMBL3091852 | CHEMBL1203 | |
| 0.047 | 0.232 | 0.462 | Amylase inhibitor | 0.223 0.036 CHEMBL3544856 0.196 0.046 CHEMBL1203 0.462 0.007 CHEMBL3544637 0.185 0.05 CHEMBL1237174 0.139 0.07 CHEMBL3091852 | CHEMBL3544637 | |
| 0.048 | 0.234 | 0.187 | Mucolytic | 0.168 0.024 CHEMBL1203 0.187 0.017 CHEMBL3544636 0.185 0.017 CHEMBL3544637 0.109 0.066 CHEMBL3091859 0.141 0.038 CHEMBL1237174 0.153 0.031 CHEMBL3091852 | CHEMBL3544636 | |
| 0.039 | 0.225 | 0.084 | Histamine H2 receptor antagonist | 0.08 0.064 CHEMBL1203 0.084 0.057 CHEMBL1237174 | CHEMBL1237174 | |
| 0.008 | 0.195 | 0.056 | LFA antagonist | 0.042 0.007 CHEMBL1203 0.056 0.005 CHEMBL3544636 | CHEMBL3544636 | |
| 0.037 | 0.224 | 0.405 | Mediator release inhibitor | 0.178 0.019 CHEMBL1203 0.101 0.069 CHEMBL3544636 0.405 0.005 CHEMBL3544637 0.094 0.077 CHEMBL3091852 | CHEMBL3544637 | |
| 0.028 | 0.215 | 0.089 | Epoxide hydrolase inhibitor | 0.065 0.061 CHEMBL1203 0.089 0.033 CHEMBL3544636 | CHEMBL3544636 | |
| 0.033 | 0.221 | 0.08 | Potassium channel large-conductance Ca-activated activator | 0.08 0.035 CHEMBL1203 | CHEMBL1203 | |
| 0.012 | 0.201 | 0.086 | Thromboxane A2 antagonist | 0.086 0.012 CHEMBL1203 0.052 0.034 CHEMBL3544636 | CHEMBL1203 | |
| 0.009 | 0.198 | 0.065 | Glutamate (mGluR group II) antagonist | 0.065 0.009 CHEMBL1203 | CHEMBL1203 | |
| 0.054 | 0.244 | 0.18 | Cytokine production inhibitor | 0.18 0.043 CHEMBL1203 | CHEMBL1203 | |
| 0.006 | 0.198 | 0.018 | O6-alkylguanine-DNA alkyltransferase inhibitor | 0.018 0.009 CHEMBL3544637 | CHEMBL3544637 | |
| 0.088 | 0.28 | 0.685 | Antioxidant | 0.277 0.071 CHEMBL2111041 0.36 0.044 CHEMBL3544855 0.158 0.156 CHEMBL1203 0.685 0.006 CHEMBL3544637 | CHEMBL3544637 | |
| 0.02 | 0.212 | 0.052 | VCAM-1 antagonist | 0.04 0.025 CHEMBL1203 0.052 0.008 CHEMBL3544636 | CHEMBL3544636 | |
| 0.031 | 0.224 | 0.152 | Macrophage migration inhibitory factor inhibitor | 0.152 0.015 CHEMBL1203 | CHEMBL1203 | |
| 0.008 | 0.201 | 0.073 | Sodium/glucose cotransporter inhibitor | 0.073 0.004 CHEMBL3544637 0.024 0.023 CHEMBL1237174 | CHEMBL3544637 | |
| 0.02 | 0.213 | 0.052 | VCAM antagonist | 0.04 0.025 CHEMBL1203 0.052 0.008 CHEMBL3544636 | CHEMBL3544636 | |
| 0.056 | 0.25 | 0.243 | Interleukin 1 antagonist | 0.243 0.02 CHEMBL1203 0.128 0.078 CHEMBL3544637 | CHEMBL1203 | |
| 0.067 | 0.262 | 0.158 | Sphingosine 1-phosphate receptor 4 antagonist | 0.158 0.027 CHEMBL1203 0.137 0.046 CHEMBL1237174 0.132 0.054 CHEMBL3091852 | CHEMBL1203 | |
| 0.107 | 0.303 | 0.329 | Gastrin inhibitor | 0.311 0.026 CHEMBL1203 0.329 0.017 CHEMBL3544636 0.208 0.136 CHEMBL3544637 0.275 0.053 CHEMBL1237174 0.255 0.074 CHEMBL3091852 | CHEMBL3544636 | |
| 0.061 | 0.257 | 0.186 | Interleukin 8 antagonist | 0.186 0.017 CHEMBL1203 0.122 0.059 CHEMBL3544636 0.11 0.076 CHEMBL1237174 | CHEMBL1203 | |
| 0.005 | 0.202 | 0.024 | Fructose-1,6-bisphosphatase 1 inhibitor | 0.024 0.015 CHEMBL1237174 | CHEMBL1237174 | |
| 0.085 | 0.285 | 0.194 | Sphingosine 1-phosphate receptor 5 antagonist | 0.194 0.014 CHEMBL1203 0.128 0.106 CHEMBL3091859 0.17 0.034 CHEMBL1237174 0.167 0.037 CHEMBL3091852 | CHEMBL1203 | |
| 0.061 | 0.261 | 0.267 | Protein kinase stimulant | 0.176 0.052 CHEMBL1203 0.267 0.022 CHEMBL3544637 0.144 0.072 CHEMBL1237174 0.134 0.08 CHEMBL3091852 | CHEMBL3544637 | |
| 0.003 | 0.204 | 0.048 | Egl nine homolog 2 inhibitor | 0.013 0.008 CHEMBL1203 0.048 0.004 CHEMBL3544636 | CHEMBL3544636 | |
| 0.006 | 0.207 | 0.095 | Retinoid X receptor agonist | 0.095 0.005 CHEMBL1203 | CHEMBL1203 | |
| 0.01 | 0.211 | 0.032 | ATP citrate lysase inhibitor | 0.032 0.021 CHEMBL1203 0.031 0.023 CHEMBL1237174 | CHEMBL1203 | |
| 0.025 | 0.228 | 0.116 | NMDA receptor agonist | 0.116 0.014 CHEMBL1203 0.084 0.026 CHEMBL3544636 0.087 0.025 CHEMBL1237174 0.088 0.024 CHEMBL3091852 | CHEMBL1203 | |
| 0.003 | 0.206 | 0.014 | NMDA receptor phencyclidine site antagonist | 0.014 0.012 CHEMBL1237174 | CHEMBL1237174 | |
| 0.007 | 0.21 | 0.119 | TRPM8 blocker | 0.119 0.005 CHEMBL1203 | CHEMBL1203 | |
| 0.015 | 0.22 | 0.097 | NMDA receptor glycine site agonist | 0.097 0.018 CHEMBL1203 0.067 0.039 CHEMBL3544636 0.058 0.048 CHEMBL3091859 0.092 0.021 CHEMBL1237174 0.096 0.019 CHEMBL3091852 | CHEMBL1203 | |
| 0.067 | 0.273 | 0.207 | Anticonvulsant | 0.149 0.131 CHEMBL1203 0.163 0.114 CHEMBL3544636 0.181 0.098 CHEMBL3091859 0.207 0.077 CHEMBL3091852 | CHEMBL3091852 | |
| 0.075 | 0.282 | 0.138 | Vanilloid 1 agonist | 0.122 0.082 CHEMBL1203 0.138 0.052 CHEMBL3544636 0.124 0.078 CHEMBL3544637 0.136 0.056 CHEMBL1237174 0.128 0.07 CHEMBL3091852 | CHEMBL3544636 | |
| 0.004 | 0.211 | 0.045 | Prostaglandin EP2 agonist | 0.045 0.007 CHEMBL1203 | CHEMBL1203 | |
| 0.019 | 0.228 | 0.21 | Glutamate receptor agonist | 0.21 0.009 CHEMBL1203 | CHEMBL1203 | |
| 0.077 | 0.286 | 0.524 | Non-steroidal antiinflammatory agent | 0.269 0.036 CHEMBL1203 0.139 0.131 CHEMBL1442231 0.172 0.093 CHEMBL3544636 0.524 0.006 CHEMBL3544637 0.153 0.112 CHEMBL1237174 0.228 0.053 CHEMBL3091852 | CHEMBL3544637 | |
| 0.04 | 0.252 | 0.148 | GABA receptor agonist | 0.148 0.037 CHEMBL1203 0.103 0.074 CHEMBL3544636 | CHEMBL1203 | |
| 0.068 | 0.28 | 0.416 | Interleukin agonist | 0.318 0.04 CHEMBL1203 0.251 0.078 CHEMBL3544636 0.416 0.017 CHEMBL3544637 0.238 0.088 CHEMBL3091859 0.287 0.055 CHEMBL1237174 0.32 0.039 CHEMBL3091852 | CHEMBL3544637 | |
| 0.02 | 0.231 | 0.061 | Leukotriene B4 antagonist | 0.061 0.027 CHEMBL1203 0.055 0.034 CHEMBL3544637 | CHEMBL1203 | |
| 0.042 | 0.254 | 0.124 | Bile acid receptor antagonist | 0.124 0.016 CHEMBL1203 0.101 0.046 CHEMBL3544636 0.097 0.056 CHEMBL1237174 | CHEMBL1203 | |
| 0.007 | 0.22 | 0.044 | Liver X receptor beta antagonist | 0.044 0.01 CHEMBL1203 | CHEMBL1203 | |
| 0.029 | 0.241 | 0.055 | 5 Hydroxytryptamine 5A antagonist | 0.055 0.054 CHEMBL1237174 | CHEMBL1237174 | |
| 0.091 | 0.303 | 0.365 | DNA damaging | 0.195 0.12 CHEMBL3544855 0.245 0.083 CHEMBL1203 0.25 0.08 CHEMBL3544636 0.365 0.037 CHEMBL3544637 | CHEMBL3544637 | |
| 0.018 | 0.231 | 0.067 | Amidase inhibitor | 0.064 0.059 CHEMBL1203 0.067 0.053 CHEMBL3544636 | CHEMBL3544636 | |
| 0.063 | 0.276 | 0.203 | Amyloid beta precursor protein antagonist | 0.179 0.073 CHEMBL2111041 0.139 0.115 CHEMBL1203 0.203 0.055 CHEMBL3091859 | CHEMBL3091859 | |
| 0.035 | 0.249 | 0.085 | Caspase 7 inhibitor | 0.085 0.05 CHEMBL1203 0.085 0.05 CHEMBL3544636 0.084 0.053 CHEMBL1237174 0.076 0.072 CHEMBL3091852 | CHEMBL3544636 | |
| 0.011 | 0.226 | 0.071 | GABA uptake inhibitor | 0.071 0.007 CHEMBL1203 0.052 0.014 CHEMBL1237174 | CHEMBL1203 | |
| 0.044 | 0.262 | 0.137 | Caspase 3 inhibitor | 0.112 0.072 CHEMBL3544855 0.129 0.047 CHEMBL1203 0.137 0.039 CHEMBL3544636 0.101 0.09 CHEMBL1237174 0.132 0.044 CHEMBL3091852 | CHEMBL3544636 | |
| 0.036 | 0.254 | 0.133 | Protein kinase C mu inhibitor | 0.089 0.068 CHEMBL3544636 0.133 0.034 CHEMBL3544637 | CHEMBL3544637 | |
| 0.037 | 0.257 | 0.092 | Aminoacyl-tRNA synthetase inhibitor | 0.092 0.056 CHEMBL1203 0.091 0.057 CHEMBL3544636 | CHEMBL1203 | |
| 0.024 | 0.246 | 0.069 | Beta adrenoreceptor antagonist | 0.067 0.043 CHEMBL3544636 0.069 0.04 CHEMBL1237174 | CHEMBL1237174 | |
| 0.002 | 0.228 | 0.018 | Ileal bile acid transport inhibitor | 0.018 0.011 CHEMBL3544637 | CHEMBL3544637 | |
| 0.023 | 0.249 | 0.127 | NAD(P)H dehydrogenase (quinone) inhibitor | 0.127 0.027 CHEMBL1203 0.082 0.049 CHEMBL1237174 | CHEMBL1203 | |
| 0.024 | 0.25 | 0.064 | Potassium channel (ATP-sensitive) blocker | 0.064 0.052 CHEMBL1237174 | CHEMBL1237174 | |
| 0.11 | 0.336 | 0.552 | Vasodilator, coronary | 0.354 0.053 CHEMBL1203 0.27 0.114 CHEMBL3544636 0.552 0.01 CHEMBL3544637 0.276 0.108 CHEMBL1237174 0.276 0.109 CHEMBL3091852 | CHEMBL3544637 | |
| 0.017 | 0.245 | 0.037 | Adenosine uptake inhibitor | 0.037 0.019 CHEMBL1237174 0.033 0.031 CHEMBL3091852 | CHEMBL1237174 | |
| 0.011 | 0.239 | 0.042 | Leukocyte elastase inhibitor | 0.042 0.031 CHEMBL1203 0.041 0.032 CHEMBL3091852 | CHEMBL1203 | |
| 0.033 | 0.262 | 0.086 | Peroxisome proliferator-activated receptor gamma antagonist | 0.086 0.027 CHEMBL1203 0.078 0.037 CHEMBL3544636 | CHEMBL1203 | |
| 0.017 | 0.246 | 0.078 | Phosphodiesterase 4B inhibitor | 0.078 0.038 CHEMBL1203 | CHEMBL1203 | |
| 0.002 | 0.235 | 0.017 | Integrin alpha4beta1 antagonist | 0.017 0.01 CHEMBL3544636 | CHEMBL3544636 | |
| 0.006 | 0.24 | 0.078 | Farnesoid X receptor agonist | 0.078 0.005 CHEMBL1203 | CHEMBL1203 | |
| 0.005 | 0.242 | 0.041 | 5-Alpha-reductase inhibitor | 0.041 0.023 CHEMBL1203 | CHEMBL1203 | |
| 0.028 | 0.266 | 0.1 | Interferon inducer | 0.064 0.045 CHEMBL1203 0.1 0.013 CHEMBL3544637 0.078 0.025 CHEMBL1237174 0.065 0.042 CHEMBL3091852 | CHEMBL3544637 | |
| 0.002 | 0.241 | 0.018 | Prostaglandin EP4 agonist | 0.018 0.009 CHEMBL1203 | CHEMBL1203 | |
| 0.014 | 0.254 | 0.074 | Prostaglandin-E synthase inhibitor | 0.074 0.044 CHEMBL1203 | CHEMBL1203 | |
| 0.027 | 0.267 | 0.137 | Glycine receptor antagonist | 0.092 0.04 CHEMBL1203 0.137 0.011 CHEMBL3544637 0.096 0.037 CHEMBL3091859 0.126 0.015 CHEMBL1237174 0.128 0.014 CHEMBL3091852 | CHEMBL3544637 | |
| 0.028 | 0.27 | 0.085 | DNA helicase inhibitor | 0.054 0.038 CHEMBL2111041 0.062 0.025 CHEMBL1203 0.085 0.009 CHEMBL3544636 | CHEMBL3544636 | |
| 0.003 | 0.246 | 0.031 | Prostaglandin E2 agonist | 0.031 0.01 CHEMBL1203 | CHEMBL1203 | |
| 0.051 | 0.296 | 0.108 | Nav1.2 sodium channel blocker | 0.108 0.099 CHEMBL3544636 | CHEMBL3544636 | |
| 0.018 | 0.263 | 0.05 | CC chemokine 4 receptor antagonist | 0.05 0.027 CHEMBL1237174 0.043 0.039 CHEMBL3091852 | CHEMBL1237174 | |
| 0.021 | 0.267 | 0.047 | Beta adrenoreceptor agonist | 0.047 0.026 CHEMBL1203 | CHEMBL1203 | |
| 0.017 | 0.263 | 0.079 | Androgen agonist | 0.064 0.036 CHEMBL1237174 0.079 0.024 CHEMBL3091852 | CHEMBL3091852 | |
| 0.067 | 0.314 | 0.451 | Hemostatic | 0.219 0.027 CHEMBL1203 0.232 0.024 CHEMBL3544636 0.451 0.005 CHEMBL3544637 0.137 0.085 CHEMBL3091852 | CHEMBL3544637 | |
| 0.017 | 0.267 | 0.134 | Sphingosine 1-phosphate receptor 4 agonist | 0.081 0.036 CHEMBL1203 0.134 0.012 CHEMBL3544636 0.087 0.032 CHEMBL1237174 | CHEMBL3544636 | |
| 0.049 | 0.299 | 0.291 | Cyclooxygenase 3 inhibitor | 0.171 0.033 CHEMBL1203 0.291 0.006 CHEMBL3544637 0.12 0.078 CHEMBL3091859 0.154 0.045 CHEMBL1237174 0.166 0.036 CHEMBL3091852 | CHEMBL3544637 | |
| 0.073 | 0.324 | 0.393 | Ca2+/calmodulin-dependent kinase I alpha inhibitor | 0.215 0.08 CHEMBL1442231 0.393 0.016 CHEMBL3091852 | CHEMBL3091852 | |
| 0.077 | 0.331 | 0.148 | Papain-like protease (SARS coronavirus) inhibitor | 0.119 0.083 CHEMBL1442231 0.115 0.094 CHEMBL3544636 0.148 0.036 CHEMBL3091852 | CHEMBL3091852 | |
| 0.042 | 0.297 | 0.148 | Adenylate cyclase inhibitor | 0.104 0.081 CHEMBL1203 0.148 0.047 CHEMBL3544636 0.124 0.064 CHEMBL1237174 0.102 0.082 CHEMBL3091852 | CHEMBL3544636 | |
| 0.043 | 0.302 | 0.127 | Dual specificity tyrosine-phosphorylation regulated kinase 1B inhibitor | 0.127 0.098 CHEMBL1203 | CHEMBL1203 | |
| 0.005 | 0.265 | 0.041 | Prostaglandin agonist | 0.041 0.013 CHEMBL1203 | CHEMBL1203 | |
| 0.026 | 0.289 | 0.365 | Expectorant | 0.149 0.036 CHEMBL1203 0.15 0.035 CHEMBL3544636 0.365 0.005 CHEMBL3544637 0.112 0.056 CHEMBL1237174 0.119 0.051 CHEMBL3091852 | CHEMBL3544637 | |
| 0.093 | 0.356 | 0.157 | CC chemokine 6 receptor antagonist | 0.148 0.025 CHEMBL1203 0.157 0.015 CHEMBL3544637 | CHEMBL3544637 | |
| 0.016 | 0.279 | 0.056 | Beta 2 adrenoreceptor antagonist | 0.056 0.028 CHEMBL3544636 | CHEMBL3544636 | |
| 0.004 | 0.271 | 0.033 | Vitronectin receptor antagonist | 0.033 0.01 CHEMBL3544636 | CHEMBL3544636 | |
| 0.005 | 0.274 | 0.069 | Glycine transporter inhibitor | 0.069 0.021 CHEMBL3544636 | CHEMBL3544636 | |
| 0.005 | 0.274 | 0.023 | Beta 1 adrenoreceptor agonist | 0.023 0.016 CHEMBL1203 | CHEMBL1203 | |
| 0.034 | 0.305 | 0.124 | Cyclooxygenase 1 inhibitor | 0.124 0.076 CHEMBL2111041 | CHEMBL2111041 | |
| 0.023 | 0.295 | 0.124 | Pim-1 kinase inhibitor | 0.124 0.04 CHEMBL1203 | CHEMBL1203 | |
| 0.005 | 0.282 | 0.038 | Prostaglandin EP4 antagonist | 0.038 0.012 CHEMBL1203 | CHEMBL1203 | |
| 0.009 | 0.286 | 0.117 | Glycine transporter 2 inhibitor | 0.117 0.01 CHEMBL3544636 | CHEMBL3544636 | |
| 0.061 | 0.338 | 0.12 | Interleukin 2 antagonist | 0.12 0.045 CHEMBL1203 | CHEMBL1203 | |
| 0.017 | 0.295 | 0.093 | NMDA receptor antagonist | 0.093 0.052 CHEMBL1203 | CHEMBL1203 | |
| 0.088 | 0.367 | 0.246 | MAP-kinase-activated kinase 5 inhibitor | 0.169 0.151 CHEMBL1442231 0.246 0.062 CHEMBL3091852 | CHEMBL3091852 | |
| 0.022 | 0.301 | 0.071 | Glutamate (mGluR) antagonist | 0.071 0.059 CHEMBL1203 | CHEMBL1203 | |
| 0.016 | 0.299 | 0.044 | Aggrecanase 1 inhibitor | 0.037 0.033 CHEMBL1442231 0.044 0.019 CHEMBL3091852 | CHEMBL3091852 | |
| 0.033 | 0.316 | 0.535 | AMP-activated protein kinase stimulant | 0.184 0.014 CHEMBL1203 0.115 0.053 CHEMBL3544636 0.535 0.003 CHEMBL3544637 | CHEMBL3544637 | |
| 0.023 | 0.307 | 0.097 | Adrenaline agonist | 0.097 0.039 CHEMBL1203 0.074 0.066 CHEMBL3544636 | CHEMBL1203 | |
| 0.008 | 0.294 | 0.259 | Purinergic P2Y14 antagonist | 0.259 0.003 CHEMBL1203 | CHEMBL1203 | |
| 0.074 | 0.359 | 0.2 | Thyroid hormone antagonist | 0.2 0.162 CHEMBL3544636 0.196 0.165 CHEMBL3091852 | CHEMBL3544636 | |
| 0.024 | 0.313 | 0.119 | Interferon agonist | 0.076 0.059 CHEMBL1203 0.119 0.018 CHEMBL3544637 0.093 0.035 CHEMBL1237174 0.078 0.056 CHEMBL3091852 | CHEMBL3544637 | |
| 0.034 | 0.326 | 0.081 | Phosphodiesterase I inhibitor | 0.081 0.075 CHEMBL1203 | CHEMBL1203 | |
| 0.004 | 0.3 | 0.05 | Aggrecanase 2 inhibitor | 0.02 0.017 CHEMBL1442231 0.05 0.005 CHEMBL3091852 | CHEMBL3091852 | |
| 0.006 | 0.303 | 0.028 | Integrin alphaVbeta1 antagonist | 0.028 0.007 CHEMBL3544636 | CHEMBL3544636 | |
| 0.006 | 0.306 | 0.05 | Purinergic P2Y antagonist | 0.05 0.027 CHEMBL1203 | CHEMBL1203 | |
| 0.025 | 0.328 | 0.062 | Beta 3 adrenoreceptor antagonist | 0.062 0.05 CHEMBL1237174 | CHEMBL1237174 | |
| 0.008 | 0.312 | 0.072 | NMDA 2C receptor antagonist | 0.072 0.031 CHEMBL1203 0.056 0.051 CHEMBL1237174 | CHEMBL1203 | |
| 0.036 | 0.343 | 0.226 | Beta amyloid protein antagonist | 0.12 0.067 CHEMBL1203 0.108 0.08 CHEMBL3544636 0.226 0.011 CHEMBL3544637 0.099 0.091 CHEMBL1237174 | CHEMBL3544637 | |
| 0.037 | 0.344 | 0.073 | Calcium channel P-type blocker | 0.073 0.023 CHEMBL1237174 | CHEMBL1237174 | |
| 0.019 | 0.328 | 0.06 | Sphingosine 1-phosphate receptor 1 antagonist | 0.055 0.039 CHEMBL1203 0.06 0.03 CHEMBL3544636 | CHEMBL3544636 | |
| 0.057 | 0.367 | 0.125 | Polo-like kinase-3 inhibitor | 0.125 0.117 CHEMBL3091852 | CHEMBL3091852 | |
| 0.059 | 0.37 | 0.536 | Vasodilator | 0.19 0.113 CHEMBL1203 0.536 0.009 CHEMBL3544637 0.467 0.014 CHEMBL3091859 0.519 0.01 CHEMBL1237174 0.456 0.015 CHEMBL3091852 | CHEMBL3544637 | |
| 0.004 | 0.316 | 0.082 | GP IIb/IIIa receptor antagonist | 0.082 0.021 CHEMBL3544636 | CHEMBL3544636 | |
| 0.026 | 0.339 | 0.085 | Sphingosine 1-phosphate receptor antagonist | 0.08 0.045 CHEMBL1203 0.085 0.037 CHEMBL3544636 | CHEMBL3544636 | |
| 0.01 | 0.328 | 0.039 | Liver X receptor alpha agonist | 0.039 0.032 CHEMBL1203 | CHEMBL1203 | |
| 0.032 | 0.351 | 0.149 | Nav1.6 sodium channel blocker | 0.118 0.099 CHEMBL1203 0.149 0.056 CHEMBL1237174 | CHEMBL1237174 | |
| 0.005 | 0.328 | 0.042 | Peroxisome proliferator-activated receptor alpha agonist | 0.042 0.039 CHEMBL1203 | CHEMBL1203 | |
| 0.043 | 0.367 | 0.128 | MAP3K9 inhibitor | 0.12 0.114 CHEMBL3544856 0.128 0.098 CHEMBL1203 | CHEMBL1203 | |
| 0.005 | 0.331 | 0.072 | NMDA 2 receptor antagonist | 0.072 0.05 CHEMBL1203 | CHEMBL1203 | |
| 0.013 | 0.342 | 0.088 | Histamine H1 receptor antagonist | 0.088 0.05 CHEMBL1203 | CHEMBL1203 | |
| 0.006 | 0.336 | 0.027 | Calcium-sensing receptor agonist | 0.027 0.018 CHEMBL1203 0.026 0.019 CHEMBL3544636 | CHEMBL1203 | |
| 0.008 | 0.339 | 0.063 | Phosphodiesterase 4A inhibitor | 0.063 0.028 CHEMBL1203 | CHEMBL1203 | |
| 0.007 | 0.341 | 0.047 | Neuropeptide Y5 antagonist | 0.047 0.04 CHEMBL1442231 | CHEMBL1442231 | |
| 0.035 | 0.371 | 0.199 | Interleukin 1b antagonist | 0.199 0.019 CHEMBL1203 0.151 0.04 CHEMBL3544637 | CHEMBL1203 | |
| 0.007 | 0.344 | 0.056 | NMDA receptor subunit 3B antagonist | 0.056 0.021 CHEMBL1203 | CHEMBL1203 | |
| 0.081 | 0.419 | 0.21 | Catenin beta inhibitor | 0.152 0.102 CHEMBL2111041 0.21 0.025 CHEMBL3544855 0.164 0.076 CHEMBL1203 | CHEMBL3544855 | |
| 0.014 | 0.355 | 0.076 | Androgen antagonist | 0.076 0.071 CHEMBL1237174 | CHEMBL1237174 | |
| 0.005 | 0.349 | 0.046 | NMDA receptor subunit 3A antagonist | 0.046 0.022 CHEMBL1203 | CHEMBL1203 | |
| 0.059 | 0.409 | 0.188 | Thyroid hormone beta antagonist | 0.184 0.17 CHEMBL3544636 0.188 0.165 CHEMBL3091852 | CHEMBL3091852 | |
| 0.013 | 0.364 | 0.226 | Neuraminidase (influenza) inhibitor | 0.088 0.02 CHEMBL3544856 0.128 0.01 CHEMBL1203 0.063 0.048 CHEMBL1442231 0.157 0.007 CHEMBL3544637 0.186 0.005 CHEMBL3091859 0.226 0.004 CHEMBL3091852 | CHEMBL3091852 | |
| 0.035 | 0.39 | 0.143 | Acetylcholine M1 receptor antagonist | 0.143 0.082 CHEMBL1237174 0.12 0.108 CHEMBL3091852 | CHEMBL1237174 | |
| 0.004 | 0.359 | 0.039 | Sphingosine 1-phosphate receptor 1 agonist | 0.039 0.035 CHEMBL1203 | CHEMBL1203 | |
| 0.017 | 0.373 | 0.213 | 5-Lipoxygenase inhibitor | 0.213 0.022 CHEMBL2111041 0.12 0.05 CHEMBL3544855 | CHEMBL2111041 | |
| 0.018 | 0.374 | 0.098 | Autotaxin inhibitor | 0.098 0.013 CHEMBL1203 | CHEMBL1203 | |
| 0.053 | 0.409 | 0.426 | NOS3 expression enhancer | 0.285 0.02 CHEMBL1203 0.426 0.007 CHEMBL3544637 | CHEMBL3544637 | |
| 0.022 | 0.381 | 0.263 | Topoisomerase II inhibitor | 0.152 0.048 CHEMBL1203 0.263 0.023 CHEMBL3544637 | CHEMBL3544637 | |
| 0.014 | 0.374 | 0.074 | Protein kinase C alpha inhibitor | 0.064 0.053 CHEMBL1203 0.074 0.039 CHEMBL3544637 | CHEMBL3544637 | |
| 0.007 | 0.369 | 0.052 | Sphingosine 1-phosphate receptor agonist | 0.052 0.023 CHEMBL1203 0.047 0.028 CHEMBL3544636 | CHEMBL1203 | |
| 0.043 | 0.412 | 0.166 | Histone deacetylase SIRT1 inhibitor | 0.112 0.101 CHEMBL1203 0.119 0.093 CHEMBL1442231 0.166 0.049 CHEMBL3544636 0.127 0.084 CHEMBL3091852 | CHEMBL3544636 | |
| 0.02 | 0.391 | 0.06 | Beta 2 adrenoreceptor agonist | 0.06 0.051 CHEMBL1237174 | CHEMBL1237174 | |
| 0.021 | 0.397 | 0.07 | Factor III inhibitor | 0.07 0.011 CHEMBL1203 0.058 0.019 CHEMBL3544636 0.052 0.03 CHEMBL3544637 | CHEMBL1203 | |
| 0 | 0.378 | 0.117 | Mannitol 2-dehydrogenase inhibitor | 0.117 0 CHEMBL3544856 0.017 0.003 CHEMBL1203 | CHEMBL3544856 | |
| 0.016 | 0.396 | 0.101 | Calcium antagonist | 0.101 0.047 CHEMBL1237174 | CHEMBL1237174 | |
| 0.014 | 0.405 | 0.085 | Nitric oxide donor | 0.085 0.018 CHEMBL3544637 | CHEMBL3544637 | |
| 0.034 | 0.427 | 0.226 | Insulin sensitizer | 0.226 0.05 CHEMBL1203 0.216 0.058 CHEMBL3544636 0.151 0.132 CHEMBL3544637 0.168 0.11 CHEMBL1237174 0.158 0.122 CHEMBL3091852 | CHEMBL1203 | |
| 0.004 | 0.4 | 0.024 | Bombesin agonist | 0.024 0.013 CHEMBL1203 | CHEMBL1203 | |
| 0.006 | 0.408 | 0.125 | NMDA 2D receptor antagonist | 0.125 0.003 CHEMBL1203 | CHEMBL1203 | |
| 0.004 | 0.407 | 0.02 | Bombesin 3 receptor agonist | 0.02 0.012 CHEMBL1203 | CHEMBL1203 | |
| 0.01 | 0.42 | 0.175 | Protein kinase C eta inhibitor | 0.12 0.012 CHEMBL1203 0.175 0.005 CHEMBL3544637 | CHEMBL3544637 | |
| 0.023 | 0.434 | 0.139 | Histone deacetylase class III inhibitor | 0.096 0.094 CHEMBL1203 0.139 0.053 CHEMBL3544636 | CHEMBL3544636 | |
| 0.017 | 0.429 | 0.045 | Integrin alpha1beta1 antagonist | 0.045 0.012 CHEMBL3544636 | CHEMBL3544636 | |
| 0.015 | 0.43 | 0.083 | Guanylate cyclase stimulant | 0.083 0.008 CHEMBL1203 | CHEMBL1203 | |
| 0.055 | 0.471 | 0.424 | Angiogenesis inhibitor | 0.193 0.178 CHEMBL1203 0.424 0.047 CHEMBL3544637 | CHEMBL3544637 | |
| 0.011 | 0.43 | 0.092 | Anesthetic local | 0.092 0.091 CHEMBL1237174 | CHEMBL1237174 | |
| 0.013 | 0.435 | 0.066 | Carnitine palmitoyltransferase 1B inhibitor | 0.066 0.013 CHEMBL1203 | CHEMBL1203 | |
| 0.016 | 0.437 | 0.062 | Transcription factor AP-1 inhibitor | 0.056 0.053 CHEMBL1203 0.062 0.041 CHEMBL3544637 | CHEMBL3544637 | |
| 0.006 | 0.43 | 0.027 | Cathepsin K inhibitor | 0.027 0.018 CHEMBL3091852 | CHEMBL3091852 | |
| 0.005 | 0.431 | 0.186 | Nicotinic acid receptor 2 agonist | 0.186 0.004 CHEMBL1203 | CHEMBL1203 | |
| 0.089 | 0.52 | 0.409 | Peptidyltransferase inhibitor | 0.173 0.141 CHEMBL3544856 0.196 0.105 CHEMBL1203 0.185 0.12 CHEMBL1442231 0.321 0.018 CHEMBL3544636 0.409 0.006 CHEMBL3544637 0.19 0.112 CHEMBL3091859 0.27 0.038 CHEMBL3091852 | CHEMBL3544637 | |
| 0.015 | 0.455 | 0.298 | Topoisomerase I inhibitor | 0.298 0.011 CHEMBL3544637 | CHEMBL3544637 | |
| 0.014 | 0.457 | 0.049 | DNA gyrase subunit A inhibitor | 0.049 0.018 CHEMBL1203 0.045 0.024 CHEMBL1237174 | CHEMBL1203 | |
| 0.006 | 0.453 | 0.035 | Protein kinase C beta II inhibitor | 0.035 0.017 CHEMBL1203 0.032 0.025 CHEMBL3544637 | CHEMBL1203 | |
| 0.009 | 0.464 | 0.041 | Protein kinase C beta I inhibitor | 0.039 0.01 CHEMBL1203 0.041 0.008 CHEMBL3544637 | CHEMBL3544637 | |
| 0.007 | 0.465 | 0.063 | Integrin alpha5beta1 antagonist | 0.063 0.011 CHEMBL3544636 | CHEMBL3544636 | |
| 0.032 | 0.495 | 0.437 | Antiamyloidogenic | 0.22 0.086 CHEMBL1203 0.159 0.135 CHEMBL3544636 0.437 0.023 CHEMBL3544637 | CHEMBL3544637 | |
| 0.077 | 0.543 | 0.796 | Cyclophilin D inhibitor | 0.396 0.093 CHEMBL2111041 0.409 0.086 CHEMBL1203 0.362 0.114 CHEMBL3544636 0.796 0.007 CHEMBL3544637 | CHEMBL3544637 | |
| 0.007 | 0.483 | 0.02 | Tryptophan hydroxylase 1 inhibitor | 0.02 0.006 CHEMBL3544636 | CHEMBL3544636 | |
| 0.006 | 0.485 | 0.114 | Glutamate (mGluR) agonist | 0.114 0.02 CHEMBL1203 | CHEMBL1203 | |
| 0.012 | 0.497 | 0.078 | Nav1.8 sodium channel blocker | 0.078 0.045 CHEMBL1203 | CHEMBL1203 | |
| 0.006 | 0.495 | 0.193 | Neuraminidase inhibitor | 0.077 0.028 CHEMBL3544856 0.117 0.01 CHEMBL1203 0.117 0.01 CHEMBL3544637 0.144 0.006 CHEMBL3091859 0.193 0.004 CHEMBL3091852 | CHEMBL3091852 | |
| 0.01 | 0.508 | 0.037 | Purinergic P2Y2 antagonist | 0.037 0.019 CHEMBL1203 | CHEMBL1203 | |
| 0.002 | 0.507 | 0.088 | Retinoic acid beta receptor antagonist | 0.088 0.003 CHEMBL1203 | CHEMBL1203 | |
| 0.005 | 0.514 | 0.125 | Phosphodiesterase 4D inhibitor | 0.125 0.026 CHEMBL1203 | CHEMBL1203 | |
| 0.019 | 0.53 | 0.373 | Thrombolytic | 0.185 0.059 CHEMBL1203 0.244 0.035 CHEMBL3544636 0.373 0.014 CHEMBL3544637 | CHEMBL3544637 | |
| 0.033 | 0.552 | 0.211 | Interleukin 4 antagonist | 0.211 0.019 CHEMBL1203 0.123 0.081 CHEMBL3544636 0.192 0.025 CHEMBL3544637 | CHEMBL1203 | |
| 0.01 | 0.53 | 0.201 | M17 leucyl aminopeptidase inhibitor | 0.161 0.049 CHEMBL1203 0.201 0.032 CHEMBL3091852 | CHEMBL3091852 | |
| 0.011 | 0.532 | 0.055 | Acetyl-CoA transferase 2 inhibitor | 0.055 0.042 CHEMBL1203 0.054 0.045 CHEMBL3544637 | CHEMBL1203 | |
| 0.013 | 0.534 | 0.113 | Glucose-6-phosphate translocase inhibitor | 0.063 0.021 CHEMBL1203 0.113 0.005 CHEMBL3544637 | CHEMBL3544637 | |
| 0.032 | 0.554 | 0.174 | Antipruritic | 0.174 0.07 CHEMBL1203 | CHEMBL1203 | |
| 0.022 | 0.564 | 0.066 | Caspase 9 inhibitor | 0.058 0.053 CHEMBL3544855 0.066 0.037 CHEMBL3544636 | CHEMBL3544636 | |
| 0.004 | 0.561 | 0.066 | Glutamate (mGluR2) agonist | 0.066 0.01 CHEMBL1203 | CHEMBL1203 | |
| 0.002 | 0.56 | 0.076 | Retinoic acid receptor gamma antagonist | 0.076 0.003 CHEMBL1203 | CHEMBL1203 | |
| 0.004 | 0.565 | 0.041 | Factor XI inhibitor | 0.041 0.015 CHEMBL1203 | CHEMBL1203 | |
| 0.005 | 0.571 | 0.018 | Guanylate cyclase 1 stimulant | 0.018 0.017 CHEMBL1203 | CHEMBL1203 | |
| 0.004 | 0.573 | 0.085 | Aldose reductase inhibitor | 0.059 0.032 CHEMBL3544636 0.085 0.021 CHEMBL3544637 | CHEMBL3544637 | |
| 0.005 | 0.578 | 0.075 | Glutamate (mGluR group II) agonist | 0.075 0.009 CHEMBL1203 | CHEMBL1203 | |
| 0.02 | 0.599 | 0.26 | Platelet aggregation inhibitor | 0.145 0.134 CHEMBL3544855 0.206 0.077 CHEMBL1203 0.26 0.047 CHEMBL3544636 | CHEMBL3544636 | |
| 0.009 | 0.589 | 0.188 | Glutamate receptor antagonist | 0.188 0.03 CHEMBL1203 | CHEMBL1203 | |
| 0.003 | 0.584 | 0.046 | VLA-4 antagonist | 0.046 0.014 CHEMBL3544636 | CHEMBL3544636 | |
| 0.031 | 0.615 | 0.114 | Hematopoietic | 0.106 0.03 CHEMBL3544856 0.093 0.045 CHEMBL1203 0.114 0.025 CHEMBL3544636 | CHEMBL3544636 | |
| 0.014 | 0.612 | 0.045 | Glucagon-like peptide 1 receptor antagonist | 0.045 0.018 CHEMBL3544636 | CHEMBL3544636 | |
| 0.004 | 0.602 | 0.024 | Kainate receptor 4 antagonist | 0.024 0.018 CHEMBL1203 | CHEMBL1203 | |
| 0.011 | 0.613 | 0.179 | Topoisomerase II alpha inhibitor | 0.179 0.018 CHEMBL3544637 | CHEMBL3544637 | |
| 0.003 | 0.608 | 0.02 | Kainate receptor 3 antagonist | 0.02 0.009 CHEMBL1203 | CHEMBL1203 | |
| 0.003 | 0.609 | 0.026 | Integrin alpha4beta7 antagonist | 0.026 0.01 CHEMBL3544636 | CHEMBL3544636 | |
| 0.013 | 0.626 | 0.106 | ATPase (Vacuolar H+) inhibitor | 0.086 0.064 CHEMBL3544856 0.106 0.032 CHEMBL3544637 | CHEMBL3544637 | |
| 0.004 | 0.617 | 0.021 | Dopamine D1 agonist | 0.021 0.02 CHEMBL3544637 | CHEMBL3544637 | |
| 0.007 | 0.622 | 0.083 | Leukotriene synthesis inhibitor | 0.07 0.044 CHEMBL3544855 0.083 0.035 CHEMBL1203 | CHEMBL1203 | |
| 0.004 | 0.62 | 0.026 | Diacylglycerol O-acyltransferase 1 inhibitor | 0.026 0.023 CHEMBL3544636 | CHEMBL3544636 | |
| 0.006 | 0.623 | 0.091 | Lipase inhibitor | 0.091 0.033 CHEMBL3544637 | CHEMBL3544637 | |
| 0.027 | 0.649 | 0.089 | 3C-Like protease (SARS coronavirus) inhibitor | 0.089 0.048 CHEMBL1203 | CHEMBL1203 | |
| 0.004 | 0.63 | 0.115 | Integrin antagonist | 0.115 0.014 CHEMBL3544636 | CHEMBL3544636 | |
| 0.003 | 0.636 | 0.078 | Retinoic acid receptor antagonist | 0.078 0.003 CHEMBL1203 | CHEMBL1203 | |
| 0.005 | 0.643 | 0.065 | Factor XIa inhibitor | 0.065 0.011 CHEMBL1203 | CHEMBL1203 | |
| 0.013 | 0.662 | 0.146 | Dual specificity tyrosine-phosphorylation regulated kinase 2 inhibitor | 0.146 0.015 CHEMBL1203 | CHEMBL1203 | |
| 0.004 | 0.658 | 0.065 | Microtubule stabilization | 0.065 0.009 CHEMBL3544637 | CHEMBL3544637 | |
| 0.02 | 0.674 | 0.186 | P-glycoprotein inhibitor | 0.186 0.074 CHEMBL3544637 | CHEMBL3544637 | |
| 0.011 | 0.667 | 0.306 | Anticoagulant | 0.242 0.04 CHEMBL3544636 0.306 0.027 CHEMBL3544637 | CHEMBL3544637 | |
| 0.043 | 0.701 | 0.46 | Sodium/bile acid cotransporter inhibitor | 0.253 0.125 CHEMBL2111041 0.305 0.074 CHEMBL3544855 0.352 0.038 CHEMBL1203 0.46 0.006 CHEMBL3544636 | CHEMBL3544636 | |
| 0.004 | 0.667 | 0.033 | Prostacyclin antagonist | 0.033 0.023 CHEMBL3544855 0.029 0.026 CHEMBL3544636 | CHEMBL3544855 | |
| 0.003 | 0.67 | 0.042 | Kainate receptor 5 antagonist | 0.042 0.006 CHEMBL1203 | CHEMBL1203 | |
| 0.022 | 0.693 | 0.071 | Lipocortins synthesis agonist | 0.071 0.02 CHEMBL3544637 | CHEMBL3544637 | |
| 0.004 | 0.68 | 0.059 | Protein 30S ribosomal subunit inhibitor | 0.059 0.006 CHEMBL3544637 | CHEMBL3544637 | |
| 0.003 | 0.68 | 0.013 | Integrin alphaLbeta2 antagonist | 0.013 0.009 CHEMBL3544636 | CHEMBL3544636 | |
| 0.013 | 0.705 | 0.851 | Angiogenesis stimulant | 0.219 0.085 CHEMBL1203 0.261 0.065 CHEMBL3544636 0.851 0.003 CHEMBL3544637 | CHEMBL3544637 | |
| 0.015 | 0.709 | 0.106 | Thioredoxin inhibitor | 0.106 0.042 CHEMBL3544637 | CHEMBL3544637 | |
| 0.005 | 0.716 | 0.115 | Retinoic acid alpha receptor agonist | 0.115 0.004 CHEMBL1203 | CHEMBL1203 | |
| 0.008 | 0.721 | 0.062 | Nicotinic acid receptor 1 agonist | 0.062 0.015 CHEMBL1203 | CHEMBL1203 | |
| 0.016 | 0.737 | 0.166 | Cardiotonic | 0.166 0.156 CHEMBL3544636 | CHEMBL3544636 | |
| 0.009 | 0.734 | 0.421 | Platelet antagonist | 0.156 0.138 CHEMBL2111041 0.323 0.045 CHEMBL3544855 0.252 0.071 CHEMBL1203 0.331 0.043 CHEMBL3544636 0.421 0.023 CHEMBL3544637 | CHEMBL3544637 | |
| 0.003 | 0.73 | 0.033 | Integrin alpha4 antagonist | 0.033 0.015 CHEMBL3544636 | CHEMBL3544636 | |
| 0.008 | 0.738 | 0.091 | Protease inhibitor | 0.091 0.073 CHEMBL3091852 | CHEMBL3091852 | |
| 0.007 | 0.737 | 0.277 | Cell adhesion molecule inhibitor | 0.138 0.018 CHEMBL1203 0.173 0.012 CHEMBL3544636 0.277 0.005 CHEMBL3544637 | CHEMBL3544637 | |
| 0.012 | 0.745 | 0.232 | Interleukin antagonist | 0.232 0.069 CHEMBL1203 0.152 0.116 CHEMBL3544636 | CHEMBL1203 | |
| 0.019 | 0.755 | 0.541 | Immunosuppressant | 0.273 0.133 CHEMBL1203 0.217 0.179 CHEMBL3544636 0.541 0.023 CHEMBL3544637 | CHEMBL3544637 | |
| 0.007 | 0.745 | 0.361 | Lipid peroxidase inhibitor | 0.361 0.012 CHEMBL3544637 | CHEMBL3544637 | |
| 0.014 | 0.753 | 0.592 | Tumour necrosis factor alpha release inhibitor | 0.185 0.122 CHEMBL1203 0.592 0.008 CHEMBL3544637 | CHEMBL3544637 | |
| 0.022 | 0.763 | 0.159 | ABCA1 expression enhancer | 0.159 0.015 CHEMBL1203 | CHEMBL1203 | |
| 0.018 | 0.766 | 0.134 | Interleukin 5 antagonist | 0.134 0.016 CHEMBL1203 | CHEMBL1203 | |
| 0.012 | 0.766 | 0.189 | Interleukin 6 antagonist | 0.189 0.048 CHEMBL3544856 0.13 0.126 CHEMBL1203 0.166 0.068 CHEMBL3544636 0.182 0.053 CHEMBL3544637 | CHEMBL3544856 | |
| 0.004 | 0.759 | 0.034 | AMPA 2 receptor antagonist | 0.034 0.018 CHEMBL1203 | CHEMBL1203 | |
| 0.02 | 0.786 | 0.098 | T cell inhibitor | 0.098 0.026 CHEMBL3544636 | CHEMBL3544636 | |
| 0.067 | 0.834 | 0.404 | Calcium channel L-type activator | 0.404 0.079 CHEMBL1203 0.231 0.228 CHEMBL3544636 | CHEMBL1203 | |
| 0.006 | 0.776 | 0.184 | Erythropoietin receptor agonist | 0.184 0.007 CHEMBL3544636 | CHEMBL3544636 | |
| 0.01 | 0.784 | 0.079 | Thioredoxin reductase inhibitor | 0.079 0.065 CHEMBL1203 | CHEMBL1203 | |
| 0.031 | 0.823 | 0.101 | Factor V inhibitor | 0.101 0.068 CHEMBL1203 | CHEMBL1203 | |
| 0.002 | 0.794 | 0.021 | Angiotensin AT1A receptor antagonist | 0.021 0.017 CHEMBL1203 | CHEMBL1203 | |
| 0.021 | 0.816 | 0.25 | Transcription factor NF kappa B stimulant | 0.091 0.049 CHEMBL1203 0.25 0.006 CHEMBL3544637 | CHEMBL3544637 | |
| 0.003 | 0.799 | 0.203 | Antineoplastic antibiotic | 0.203 0.021 CHEMBL3544637 | CHEMBL3544637 | |
| 0.009 | 0.807 | 0.15 | Multidrug resistance-associated protein 1 inhibitor | 0.104 0.072 CHEMBL1203 0.093 0.092 CHEMBL3544636 0.15 0.025 CHEMBL3544637 | CHEMBL3544637 | |
| 0.004 | 0.804 | 0.144 | Prostaglandin EP2 antagonist | 0.144 0.01 CHEMBL1203 0.065 0.037 CHEMBL3544636 | CHEMBL1203 | |
| 0.029 | 0.835 | 0.419 | Caspase 3 stimulant | 0.419 0.039 CHEMBL3544637 0.208 0.158 CHEMBL3091852 | CHEMBL3544637 | |
| 0.011 | 0.821 | 0.107 | Factor IXa inhibitor | 0.05 0.038 CHEMBL1203 0.107 0.008 CHEMBL3544637 | CHEMBL3544637 | |
| 0.009 | 0.823 | 0.038 | Calcium-independent phospholipase A2 inhibitor | 0.038 0.014 CHEMBL1203 | CHEMBL1203 | |
| 0.003 | 0.821 | 0.054 | Somatostatin 5 antagonist | 0.054 0.011 CHEMBL1203 | CHEMBL1203 | |
| 0.004 | 0.826 | 0.045 | Acetyl-CoA carboxylase inhibitor | 0.045 0.024 CHEMBL3091852 | CHEMBL3091852 | |
| 0.007 | 0.831 | 0.094 | Prostaglandin F2 alpha antagonist | 0.057 0.053 CHEMBL3544855 0.094 0.014 CHEMBL1203 | CHEMBL1203 | |
| 0.002 | 0.828 | 0.062 | Retinoic acid alpha receptor antagonist | 0.062 0.004 CHEMBL1203 | CHEMBL1203 | |
| 0.003 | 0.83 | 0.055 | Angiotensin-converting enzyme inhibitor | 0.055 0.037 CHEMBL3544636 | CHEMBL3544636 | |
| 0.029 | 0.858 | 0.166 | Growth hormone agonist | 0.166 0.075 CHEMBL3544855 | CHEMBL3544855 | |
| 0.003 | 0.836 | 0.048 | Retinoic acid gamma receptor agonist | 0.048 0.004 CHEMBL1203 | CHEMBL1203 | |
| 0.008 | 0.842 | 0.397 | Cell adhesion inhibitor | 0.195 0.026 CHEMBL1203 0.249 0.015 CHEMBL3544636 0.397 0.005 CHEMBL3544637 | CHEMBL3544637 | |
| 0.031 | 0.868 | 0.278 | Lipocortins synthesis antagonist | 0.142 0.117 CHEMBL3544855 0.278 0.026 CHEMBL1203 0.15 0.105 CHEMBL3544637 | CHEMBL1203 | |
| 0 | 0.84 | 0.015 | Antibiotic Macrolide-like | 0.015 0.009 CHEMBL3544637 | CHEMBL3544637 | |
| 0.003 | 0.846 | 0.028 | Melatonin antagonist | 0.028 0.02 CHEMBL3091852 | CHEMBL3091852 | |
| 0.002 | 0.849 | 0.017 | Melatonin 1 antagonist | 0.017 0.016 CHEMBL3091852 | CHEMBL3091852 | |
| 0.003 | 0.858 | 0.086 | Retinoic acid beta receptor agonist | 0.086 0.003 CHEMBL1203 | CHEMBL1203 | |
| 0.003 | 0.861 | 0.042 | Melatonin agonist | 0.042 0.014 CHEMBL3091852 | CHEMBL3091852 | |
| 0.008 | 0.867 | 0.28 | Toll-Like receptor 7 agonist | 0.28 0.123 CHEMBL1203 0.228 0.169 CHEMBL3544636 | CHEMBL1203 | |
| 0.002 | 0.861 | 0.067 | Prostaglandin EP1 antagonist | 0.067 0.005 CHEMBL1203 | CHEMBL1203 | |
| 0.012 | 0.872 | 0.696 | Apoptosis agonist | 0.289 0.181 CHEMBL3544855 0.696 0.031 CHEMBL3544637 | CHEMBL3544637 | |
| 0.003 | 0.865 | 0.101 | Retinoic acid receptor agonist | 0.101 0.004 CHEMBL1203 | CHEMBL1203 | |
| 0.004 | 0.866 | 0.213 | Prostaglandin E2 antagonist | 0.213 0.005 CHEMBL1203 | CHEMBL1203 | |
| 0.003 | 0.867 | 0.069 | Peroxisome proliferator-activated receptor gamma agonist | 0.069 0.049 CHEMBL1203 | CHEMBL1203 | |
| 0.002 | 0.867 | 0.032 | Leukotriene B4 receptor 1 antagonist | 0.032 0.016 CHEMBL1203 | CHEMBL1203 | |
| 0.003 | 0.869 | 0.058 | Melatonin 2 agonist | 0.058 0.008 CHEMBL3091852 | CHEMBL3091852 | |
| 0.003 | 0.87 | 0.042 | Retinoid X gamma receptor antagonist | 0.042 0.004 CHEMBL1203 | CHEMBL1203 | |
| 0.007 | 0.876 | 0.273 | Toll-Like receptor agonist | 0.273 0.129 CHEMBL1203 0.236 0.162 CHEMBL3544636 | CHEMBL1203 | |
| 0.005 | 0.873 | 0.238 | Protein-tyrosine phosphatase inhibitor | 0.238 0.034 CHEMBL1203 0.235 0.035 CHEMBL3544637 | CHEMBL1203 | |
| 0.006 | 0.875 | 0.54 | Nitric oxide antagonist | 0.54 0.013 CHEMBL3544637 | CHEMBL3544637 | |
| 0.013 | 0.883 | 0.24 | DNA polymerase I inhibitor | 0.137 0.057 CHEMBL1203 0.24 0.019 CHEMBL3544637 | CHEMBL3544637 | |
| 0.002 | 0.873 | 0.1 | Retinoid X gamma receptor agonist | 0.1 0.004 CHEMBL1203 | CHEMBL1203 | |
| 0.002 | 0.88 | 0.063 | Leukotriene A4 hydrolase inhibitor | 0.063 0.014 CHEMBL1203 | CHEMBL1203 | |
| 0.004 | 0.882 | 0.079 | CDC25B inhibitor | 0.079 0.029 CHEMBL1203 | CHEMBL1203 | |
| 0.004 | 0.888 | 0.071 | Neuraminidase (Influenza A) inhibitor | 0.041 0.04 CHEMBL3544856 0.068 0.008 CHEMBL1203 0.071 0.007 CHEMBL3544637 0.043 0.036 CHEMBL3091859 0.069 0.008 CHEMBL3091852 | CHEMBL3544637 | |
| 0.002 | 0.887 | 0.096 | Retinoid X beta receptor agonist | 0.096 0.004 CHEMBL1203 | CHEMBL1203 | |
| 0.009 | 0.894 | 0.144 | Farnesoid X receptor antagonist | 0.144 0.06 CHEMBL1203 0.119 0.106 CHEMBL3544636 | CHEMBL1203 | |
| 0.003 | 0.893 | 0.05 | Melatonin 1 agonist | 0.05 0.009 CHEMBL3091852 | CHEMBL3091852 | |
| 0.007 | 0.899 | 0.151 | Bone formation stimulant | 0.151 0.058 CHEMBL3544636 | CHEMBL3544636 | |
| 0.005 | 0.907 | 0.119 | Protein 50S ribosomal subunit inhibitor | 0.119 0.009 CHEMBL3544637 0.062 0.03 CHEMBL3091852 | CHEMBL3544637 | |
| 0.003 | 0.909 | 0.063 | Glucagon-like peptide 1 agonist | 0.063 0.046 CHEMBL3544636 | CHEMBL3544636 | |
| 0.009 | 0.916 | 0.572 | Immunomodulator | 0.572 0.014 CHEMBL3544637 | CHEMBL3544637 | |
| 0.008 | 0.917 | 0.857 | Antiinflammatory | 0.39 0.145 CHEMBL1203 0.857 0.009 CHEMBL3544637 | CHEMBL3544637 | |
| 0.007 | 0.923 | 0.048 | Glutamate (mGluR8) antagonist | 0.048 0.01 CHEMBL1203 | CHEMBL1203 | |
| 0.003 | 0.926 | 0.141 | Prostaglandin antagonist | 0.141 0.011 CHEMBL1203 | CHEMBL1203 | |
| 0.001 | 0.925 | 0.023 | Corticosteroid-like | 0.023 0.013 CHEMBL3544637 | CHEMBL3544637 | |
| 0.005 | 0.935 | 0.214 | Antiobesity | 0.214 0.193 CHEMBL3544637 | CHEMBL3544637 | |
| 0.005 | 0.937 | 0.034 | Toll-Like receptor 4 agonist | 0.034 0.008 CHEMBL3544637 | CHEMBL3544637 | |
| 0.029 | 0.967 | 0.508 | Interleukin 2 agonist | 0.224 0.151 CHEMBL3544855 0.203 0.184 CHEMBL1203 0.22 0.157 CHEMBL3544636 0.508 0.007 CHEMBL3544637 0.206 0.178 CHEMBL3091859 0.307 0.069 CHEMBL3091852 | CHEMBL3544637 | |
| 0.009 | 0.954 | 0.1 | Adenine nucleotide translocase inhibitor | 0.1 0.005 CHEMBL1203 0.089 0.006 CHEMBL3544637 | CHEMBL1203 | |
| 0.01 | 0.957 | 0.602 | Hepatoprotectant | 0.165 0.095 CHEMBL1203 0.164 0.096 CHEMBL3544636 0.602 0.005 CHEMBL3544637 | CHEMBL3544637 | |
| 0.004 | 0.954 | 0.079 | Antibiotic Aminoglycoside-like | 0.079 0.004 CHEMBL3544637 | CHEMBL3544637 | |
| 0.008 | 0.968 | 0.615 | Apoptosis antagonist | 0.245 0.132 CHEMBL1203 0.276 0.103 CHEMBL3544636 0.615 0.008 CHEMBL3544637 | CHEMBL3544637 | |
| 0.001 | 0.966 | 0.042 | Squalene synthetase inhibitor | 0.042 0.017 CHEMBL3544637 | CHEMBL3544637 | |
| 0.003 | 0.974 | 0.06 | Sphingosine 1-phosphate receptor 5 agonist | 0.06 0.025 CHEMBL3544636 | CHEMBL3544636 | |
| 0.008 | 0.982 | 0.185 | Toll-Like receptor 4 antagonist | 0.185 0.009 CHEMBL3544637 | CHEMBL3544637 | |
| 0.004 | 0.979 | 0.326 | Hypolipemic | 0.15 0.136 CHEMBL1203 0.326 0.042 CHEMBL3544637 | CHEMBL3544637 | |
| 0.005 | 0.982 | 0.431 | Insulin secretagoues | 0.212 0.03 CHEMBL1203 0.177 0.05 CHEMBL3544636 0.431 0.005 CHEMBL3544637 | CHEMBL3544637 | |
| 0.003 | 0.985 | 0.216 | Protein-tyrosine phosphatase 1B inhibitor | 0.152 0.045 CHEMBL1203 0.216 0.025 CHEMBL3544637 | CHEMBL3544637 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |