Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.6490.0040.649Peroxidase inhibitor

0.464 0.013 CHEMBL2111041

0.355 0.027 CHEMBL3544855

0.379 0.024 CHEMBL3544856

0.578 0.005 CHEMBL1203

0.4 0.02 CHEMBL1442231

0.607 0.004 CHEMBL3544636

0.113 0.108 CHEMBL3544637

0.624 0.004 CHEMBL3091859

0.631 0.004 CHEMBL1237174

0.52 0.008 CHEMBL3091852

0.6060.0010.919Maillard reaction inhibitor

0.147 0.006 CHEMBL2111041

0.101 0.016 CHEMBL3544855

0.149 0.006 CHEMBL3544856

0.084 0.023 CHEMBL1203

0.058 0.036 CHEMBL1442231

0.741 0.001 CHEMBL3091859

0.919 0 CHEMBL1237174

0.1 0.017 CHEMBL3091852

CHEMBL1237174
0.5830.0580.688Alpha-glucosidase inhibitor

0.546 0.067 CHEMBL2111041

0.253 0.186 CHEMBL3544855

0.688 0.036 CHEMBL3544856

0.221 0.205 CHEMBL1203

0.578 0.059 CHEMBL1442231

0.676 0.038 CHEMBL3544637

0.58 0.058 CHEMBL3091859

0.255 0.184 CHEMBL1237174

0.493 0.082 CHEMBL3091852

CHEMBL3544856
0.5440.0230.791Streptokinase A inhibitor

0.454 0.035 CHEMBL2111041

0.309 0.075 CHEMBL3544855

0.246 0.106 CHEMBL3544856

0.779 0.005 CHEMBL1442231

0.655 0.012 CHEMBL3091859

0.18 0.146 CHEMBL1237174

0.791 0.005 CHEMBL3091852

CHEMBL3091852
0.5030.0040.905Alcohol oxidase inhibitor

0.19 0.007 CHEMBL2111041

0.102 0.018 CHEMBL3544855

0.119 0.014 CHEMBL3544856

0.898 0.002 CHEMBL1203

0.192 0.007 CHEMBL1442231

0.158 0.009 CHEMBL3544636

0.111 0.016 CHEMBL3544637

0.905 0.002 CHEMBL3091859

0.786 0.003 CHEMBL1237174

0.811 0.003 CHEMBL3091852

CHEMBL3091859
0.5240.0680.574Transcription factor inhibitor

0.392 0.113 CHEMBL2111041

0.244 0.19 CHEMBL3544855

0.574 0.054 CHEMBL1442231

0.459 0.088 CHEMBL3091859

0.217 0.212 CHEMBL1237174

0.438 0.095 CHEMBL3091852

CHEMBL1442231
0.4770.0450.59Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.368 0.132 CHEMBL2111041

0.285 0.233 CHEMBL3544855

0.59 0.008 CHEMBL1203

0.472 0.048 CHEMBL1442231

0.502 0.033 CHEMBL3544636

0.417 0.086 CHEMBL3091859

0.535 0.02 CHEMBL1237174

0.49 0.038 CHEMBL3091852

CHEMBL1203
0.4570.0260.486Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase inhibitor

0.402 0.038 CHEMBL2111041

0.201 0.099 CHEMBL3544855

0.276 0.071 CHEMBL1203

0.195 0.103 CHEMBL1442231

0.486 0.022 CHEMBL3091859

0.344 0.052 CHEMBL1237174

0.25 0.078 CHEMBL3091852

CHEMBL3091859
0.420.0050.779Cyclin-dependent kinase 5 inhibitor

0.57 0.004 CHEMBL1442231

0.779 0.002 CHEMBL3091859

0.619 0.004 CHEMBL1237174

0.754 0.003 CHEMBL3091852

CHEMBL3091859
0.4150.0180.415Pyruvate kinase inhibitor

0.318 0.043 CHEMBL2111041

0.281 0.053 CHEMBL3544855

0.335 0.039 CHEMBL3544856

0.331 0.04 CHEMBL1203

0.246 0.062 CHEMBL1442231

0.265 0.057 CHEMBL3091859

0.281 0.053 CHEMBL1237174

0.181 0.093 CHEMBL3091852

0.3990.0180.399Ca2+/calmodulin-dependent kinase II gamma inhibitor

0.154 0.086 CHEMBL1442231

0.152 0.087 CHEMBL3091852

0.4260.0510.612GABA C receptor rho-3 antagonist

0.334 0.095 CHEMBL2111041

0.258 0.147 CHEMBL3544855

0.546 0.015 CHEMBL1203

0.392 0.065 CHEMBL1442231

0.583 0.009 CHEMBL3544636

0.448 0.042 CHEMBL3091859

0.612 0.006 CHEMBL1237174

0.541 0.016 CHEMBL3091852

CHEMBL1237174
0.3770.0140.377Dual specificity tyrosine-phosphorylation regulated kinase 3 inhibitor

0.242 0.049 CHEMBL1203

0.226 0.059 CHEMBL1442231

0.177 0.095 CHEMBL3091852

0.3990.0380.399Aryl hydrocarbon receptor agonist

0.198 0.103 CHEMBL2111041

0.232 0.086 CHEMBL1203

0.275 0.069 CHEMBL1442231

0.265 0.073 CHEMBL3091859

0.311 0.058 CHEMBL1237174

0.254 0.077 CHEMBL3091852

0.3620.0060.362Histone acetyltransferase inhibitor

0.189 0.087 CHEMBL2111041

0.167 0.117 CHEMBL3544855

0.218 0.046 CHEMBL1203

0.229 0.037 CHEMBL1442231

0.166 0.119 CHEMBL3544636

0.205 0.062 CHEMBL3091859

0.202 0.066 CHEMBL1237174

0.209 0.056 CHEMBL3091852

0.420.0660.6375 Hydroxytryptamine release inhibitor

0.456 0.049 CHEMBL2111041

0.377 0.093 CHEMBL3544855

0.435 0.058 CHEMBL3544856

0.637 0.007 CHEMBL1203

0.431 0.06 CHEMBL1442231

0.47 0.043 CHEMBL3544636

0.527 0.025 CHEMBL3544637

0.453 0.05 CHEMBL3091859

0.495 0.034 CHEMBL1237174

0.56 0.017 CHEMBL3091852

CHEMBL1203
0.4370.0850.437MAP kinase 1 inhibitor

0.244 0.241 CHEMBL1442231

0.3680.020.368Ca2+/calmodulin-dependent kinase II beta inhibitor

0.169 0.105 CHEMBL1442231

0.19 0.085 CHEMBL3091852

0.3650.0210.424Anesthetic general

0.371 0.02 CHEMBL1203

0.144 0.12 CHEMBL1442231

0.424 0.014 CHEMBL3544637

0.38 0.019 CHEMBL3091859

0.396 0.017 CHEMBL1237174

0.278 0.039 CHEMBL3091852

CHEMBL3544637
0.3430.0030.425Glutamate decarboxylase inhibitor

0.176 0.009 CHEMBL2111041

0.246 0.004 CHEMBL3544855

0.12 0.021 CHEMBL3544856

0.425 0.003 CHEMBL1203

0.128 0.018 CHEMBL1442231

0.223 0.005 CHEMBL3544636

0.071 0.054 CHEMBL3544637

0.264 0.004 CHEMBL3091859

0.264 0.004 CHEMBL1237174

0.193 0.007 CHEMBL3091852

CHEMBL1203
0.4340.1060.434DNA polymerase beta inhibitor

0.269 0.181 CHEMBL2111041

0.222 0.209 CHEMBL1203

0.366 0.133 CHEMBL1442231

0.288 0.171 CHEMBL3091859

0.312 0.159 CHEMBL3091852

0.4020.0760.646Antibacterial

0.427 0.065 CHEMBL2111041

0.365 0.094 CHEMBL3544855

0.53 0.033 CHEMBL3544856

0.415 0.07 CHEMBL1203

0.413 0.071 CHEMBL1442231

0.221 0.206 CHEMBL3544636

0.646 0.013 CHEMBL3544637

0.466 0.051 CHEMBL3091859

0.312 0.126 CHEMBL1237174

0.423 0.067 CHEMBL3091852

CHEMBL3544637
0.340.0230.34MAP kinase kinase 2 inhibitor

0.196 0.085 CHEMBL1203

0.163 0.11 CHEMBL3544636

0.203 0.08 CHEMBL3091859

0.269 0.046 CHEMBL1237174

0.163 0.109 CHEMBL3091852

0.3290.0230.329Interleukin-1 receptor-associated protein kinase 1 inhibitor

0.127 0.119 CHEMBL1442231

0.3010.0110.445Nitric-oxide synthase stimulant

0.257 0.028 CHEMBL2111041

0.211 0.072 CHEMBL3544855

0.236 0.043 CHEMBL3544856

0.335 0.006 CHEMBL1203

0.284 0.016 CHEMBL1442231

0.445 0.003 CHEMBL3544636

0.336 0.006 CHEMBL3544637

0.211 0.072 CHEMBL3091859

0.295 0.013 CHEMBL1237174

0.255 0.029 CHEMBL3091852

CHEMBL3544636
0.4020.1150.402DNA directed DNA polymerase inhibitor

0.254 0.189 CHEMBL2111041

0.222 0.211 CHEMBL1203

0.334 0.145 CHEMBL1442231

0.251 0.191 CHEMBL3091859

0.294 0.165 CHEMBL3091852

0.2860.0110.286MAP kinase kinase 3 inhibitor

0.235 0.049 CHEMBL2111041

0.216 0.083 CHEMBL3544855

0.203 0.113 CHEMBL3544856

0.261 0.023 CHEMBL1203

0.267 0.019 CHEMBL1442231

0.249 0.033 CHEMBL3544636

0.2690.0040.269Myeloperoxidase inhibitor

0.085 0.058 CHEMBL2111041

0.077 0.073 CHEMBL3544855

0.102 0.032 CHEMBL1203

0.094 0.043 CHEMBL1442231

0.143 0.012 CHEMBL3091859

0.149 0.011 CHEMBL1237174

0.1 0.034 CHEMBL3091852

0.2740.0150.274Alkaline phosphatase inhibitor

0.107 0.105 CHEMBL2111041

0.184 0.04 CHEMBL1203

0.142 0.065 CHEMBL3544636

0.171 0.047 CHEMBL3544637

0.169 0.048 CHEMBL3091859

0.174 0.045 CHEMBL1237174

0.119 0.088 CHEMBL3091852

0.2580.0110.392Xanthine oxidase inhibitor

0.111 0.052 CHEMBL2111041

0.094 0.066 CHEMBL3544855

0.288 0.008 CHEMBL1203

0.084 0.082 CHEMBL1442231

0.098 0.061 CHEMBL3544636

0.392 0.005 CHEMBL3544637

0.133 0.041 CHEMBL3091859

0.145 0.036 CHEMBL1237174

0.087 0.076 CHEMBL3091852

CHEMBL3544637
0.2490.0150.362Cystathionine beta-synthase inhibitor

0.14 0.045 CHEMBL2111041

0.117 0.06 CHEMBL3544855

0.362 0.006 CHEMBL1203

0.09 0.089 CHEMBL1442231

0.128 0.052 CHEMBL3544636

0.206 0.023 CHEMBL3544637

0.249 0.015 CHEMBL3091859

0.313 0.009 CHEMBL1237174

0.18 0.03 CHEMBL3091852

CHEMBL1203
0.2890.0590.311Transcription factor STAT3 inhibitor

0.271 0.069 CHEMBL1203

0.196 0.14 CHEMBL1442231

0.183 0.159 CHEMBL3544636

0.311 0.048 CHEMBL3091859

0.252 0.082 CHEMBL1237174

0.238 0.094 CHEMBL3091852

CHEMBL3091859
0.2580.0290.258Ca2+/calmodulin-dependent kinase II delta inhibitor
0.2430.0140.27Cathepsin H inhibitor

0.121 0.074 CHEMBL2111041

0.108 0.093 CHEMBL3544855

0.119 0.076 CHEMBL3544856

0.173 0.033 CHEMBL1203

0.2 0.022 CHEMBL1442231

0.105 0.099 CHEMBL3544636

0.27 0.012 CHEMBL3091859

0.225 0.017 CHEMBL1237174

0.247 0.014 CHEMBL3091852

CHEMBL3091859
0.2340.010.4Histidine decarboxylase inhibitor

0.087 0.038 CHEMBL2111041

0.061 0.06 CHEMBL3544855

0.4 0.004 CHEMBL1203

0.253 0.009 CHEMBL3544636

0.326 0.005 CHEMBL3091859

0.353 0.005 CHEMBL1237174

0.201 0.013 CHEMBL3091852

CHEMBL1203
0.2560.0350.256LIM domain kinase 1 inhibitor

0.185 0.071 CHEMBL1203

0.173 0.078 CHEMBL1442231

0.139 0.109 CHEMBL3091859

0.165 0.084 CHEMBL1237174

0.167 0.082 CHEMBL3091852

0.2830.0660.287Transcription factor STAT inhibitor

0.28 0.068 CHEMBL1203

0.198 0.141 CHEMBL1442231

0.287 0.063 CHEMBL3091859

0.242 0.093 CHEMBL1237174

0.225 0.106 CHEMBL3091852

CHEMBL3091859
0.2360.0190.421Cell wall synthesis inhibitor

0.22 0.023 CHEMBL2111041

0.198 0.03 CHEMBL3544855

0.162 0.055 CHEMBL3544856

0.273 0.012 CHEMBL1203

0.212 0.026 CHEMBL1442231

0.194 0.033 CHEMBL3544636

0.421 0.005 CHEMBL3544637

0.202 0.029 CHEMBL3091859

0.221 0.023 CHEMBL1237174

0.227 0.021 CHEMBL3091852

CHEMBL3544637
0.2220.0150.296Carbonic anhydrase XV inhibitor

0.267 0.01 CHEMBL1203

0.089 0.086 CHEMBL1442231

0.296 0.008 CHEMBL3091859

0.281 0.009 CHEMBL1237174

0.197 0.019 CHEMBL3091852

CHEMBL3091859
0.2140.0090.214Urease inhibitor

0.117 0.048 CHEMBL2111041

0.099 0.069 CHEMBL3544855

0.115 0.05 CHEMBL3544856

0.133 0.033 CHEMBL1203

0.191 0.011 CHEMBL1442231

0.124 0.041 CHEMBL3544636

0.211 0.009 CHEMBL3091859

0.149 0.024 CHEMBL1237174

0.162 0.018 CHEMBL3091852

0.2290.0240.341MAO A inhibitor

0.149 0.041 CHEMBL1442231

0.341 0.012 CHEMBL3091859

0.121 0.052 CHEMBL1237174

0.181 0.033 CHEMBL3091852

CHEMBL3091859
0.2060.0020.206S-adenosyl-L-methionine decarboxylase inhibitor

0.118 0.006 CHEMBL2111041

0.093 0.019 CHEMBL3544855

0.083 0.031 CHEMBL3544856

0.115 0.007 CHEMBL1203

0.107 0.009 CHEMBL1442231

0.098 0.015 CHEMBL3544636

0.068 0.065 CHEMBL3544637

0.136 0.004 CHEMBL3091859

0.144 0.004 CHEMBL1237174

0.113 0.008 CHEMBL3091852

0.2130.0110.354Uric acid excretion stimulant

0.354 0.004 CHEMBL1203

0.088 0.067 CHEMBL3544636

0.241 0.008 CHEMBL3544637

CHEMBL1203
0.2230.0340.309MAO inhibitor

0.135 0.067 CHEMBL1442231

0.309 0.019 CHEMBL3091859

0.136 0.067 CHEMBL1237174

0.176 0.049 CHEMBL3091852

CHEMBL3091859
0.2340.0510.234CDC-like kinase 2 inhibitor

0.139 0.101 CHEMBL1203

0.124 0.115 CHEMBL1442231

0.2320.0510.313Glyceraldehyde-3-phosphate dehydrogenase inhibitor

0.181 0.092 CHEMBL2111041

0.175 0.1 CHEMBL3544855

0.303 0.023 CHEMBL1203

0.241 0.047 CHEMBL1442231

0.199 0.073 CHEMBL3544636

0.197 0.074 CHEMBL3544637

0.262 0.037 CHEMBL3091859

0.313 0.02 CHEMBL1237174

0.291 0.027 CHEMBL3091852

CHEMBL1237174
0.2510.0740.633Superoxide dismutase inhibitor

0.276 0.06 CHEMBL2111041

0.213 0.104 CHEMBL3544855

0.633 0.005 CHEMBL1203

0.275 0.061 CHEMBL1442231

0.444 0.02 CHEMBL3544636

0.304 0.049 CHEMBL3091859

0.375 0.031 CHEMBL1237174

0.451 0.019 CHEMBL3091852

CHEMBL1203
0.1730.0050.249Xanthine dehydrogenase inhibitor

0.073 0.029 CHEMBL2111041

0.249 0.004 CHEMBL1203

0.071 0.031 CHEMBL3544636

0.123 0.01 CHEMBL3544637

0.058 0.039 CHEMBL3091859

0.076 0.027 CHEMBL1237174

CHEMBL1203
0.2430.0880.4435 Hydroxytryptamine uptake stimulant

0.206 0.14 CHEMBL2111041

0.228 0.107 CHEMBL3544855

0.443 0.008 CHEMBL1203

0.234 0.098 CHEMBL1442231

0.287 0.052 CHEMBL3544636

0.299 0.045 CHEMBL3091859

0.435 0.009 CHEMBL1237174

0.389 0.016 CHEMBL3091852

CHEMBL1203
0.1790.0250.259Falcipain 3 inhibitor

0.126 0.05 CHEMBL2111041

0.096 0.075 CHEMBL3544855

0.163 0.031 CHEMBL1203

0.259 0.007 CHEMBL1442231

0.166 0.03 CHEMBL3544636

0.159 0.032 CHEMBL3091859

0.148 0.038 CHEMBL1237174

0.233 0.01 CHEMBL3091852

CHEMBL1442231
0.20.0470.2Protein kinase C nu inhibitor
0.1660.0140.227DOPA decarboxylase inhibitor

0.111 0.056 CHEMBL2111041

0.1 0.075 CHEMBL3544855

0.202 0.006 CHEMBL1203

0.115 0.051 CHEMBL1442231

0.112 0.056 CHEMBL3544636

0.207 0.006 CHEMBL3091859

0.227 0.004 CHEMBL1237174

0.195 0.007 CHEMBL3091852

CHEMBL1237174
0.2380.0870.727Aldehyde oxidase inhibitor

0.675 0.01 CHEMBL1203

0.3 0.066 CHEMBL3544636

0.519 0.03 CHEMBL3091859

0.727 0.006 CHEMBL1237174

0.458 0.039 CHEMBL3091852

CHEMBL1237174
0.1720.0210.221Protein kinase C gamma inhibitor

0.221 0.01 CHEMBL1203

0.107 0.065 CHEMBL1442231

0.104 0.07 CHEMBL3544636

0.182 0.018 CHEMBL3544637

0.131 0.044 CHEMBL1237174

0.123 0.05 CHEMBL3091852

CHEMBL1203
0.1660.0170.771Porphobilinogen synthase inhibitor

0.28 0.006 CHEMBL2111041

0.336 0.005 CHEMBL3544855

0.771 0.002 CHEMBL1203

0.185 0.014 CHEMBL1442231

0.346 0.004 CHEMBL3544636

0.068 0.057 CHEMBL3544637

0.234 0.009 CHEMBL3091859

0.266 0.007 CHEMBL1237174

0.378 0.004 CHEMBL3091852

CHEMBL1203
0.1520.0070.198GABA aminotransferase inhibitor

0.119 0.016 CHEMBL2111041

0.155 0.007 CHEMBL3544855

0.073 0.056 CHEMBL3544856

0.161 0.006 CHEMBL1203

0.075 0.053 CHEMBL1442231

0.074 0.055 CHEMBL3544636

0.114 0.019 CHEMBL3544637

0.198 0.004 CHEMBL3091859

0.174 0.005 CHEMBL1237174

0.137 0.01 CHEMBL3091852

CHEMBL3091859
0.1820.0370.379Monophenol monooxygenase inhibitor

0.228 0.027 CHEMBL2111041

0.167 0.041 CHEMBL3544855

0.099 0.077 CHEMBL3544856

0.179 0.038 CHEMBL1203

0.095 0.08 CHEMBL3544636

0.379 0.012 CHEMBL3544637

0.165 0.042 CHEMBL3091859

0.143 0.05 CHEMBL1237174

0.125 0.058 CHEMBL3091852

CHEMBL3544637
0.1710.0270.676GABA C receptor agonist

0.181 0.024 CHEMBL2111041

0.329 0.008 CHEMBL3544855

0.676 0.002 CHEMBL1203

0.115 0.053 CHEMBL1442231

0.461 0.004 CHEMBL3544636

0.112 0.055 CHEMBL3544637

0.224 0.016 CHEMBL3091859

0.53 0.003 CHEMBL1237174

0.333 0.008 CHEMBL3091852

CHEMBL1203
0.1660.0270.284Check point kinase 2 inhibitor

0.224 0.013 CHEMBL1442231

0.133 0.04 CHEMBL3091859

0.284 0.007 CHEMBL3091852

CHEMBL3091852
0.2780.1440.32415-Lipoxygenase inhibitor

0.317 0.12 CHEMBL2111041

0.25 0.164 CHEMBL1203

0.324 0.115 CHEMBL3091859

0.289 0.138 CHEMBL1237174

0.289 0.138 CHEMBL3091852

CHEMBL3091859
0.1720.0410.172Protein kinase (CK1) delta inhibitor
0.1330.0050.133Fatty acid synthase inhibitor

0.08 0.019 CHEMBL1203

0.074 0.023 CHEMBL1442231

0.074 0.022 CHEMBL3544637

0.07 0.026 CHEMBL3091859

0.076 0.021 CHEMBL1237174

0.071 0.025 CHEMBL3091852

0.1560.0320.157Death-associated protein kinase 1 inhibitor

0.123 0.102 CHEMBL2111041

0.132 0.077 CHEMBL1203

0.157 0.03 CHEMBL1442231

0.132 0.076 CHEMBL3544636

CHEMBL1442231
0.1250.0040.125Diamine oxidase inhibitor

0.046 0.018 CHEMBL2111041

0.061 0.009 CHEMBL1203

0.064 0.008 CHEMBL1442231

0.036 0.029 CHEMBL3544636

0.124 0.004 CHEMBL3091859

0.086 0.005 CHEMBL1237174

0.075 0.005 CHEMBL3091852

0.1660.0460.75Alpha-N-acetylglucosaminidase inhibitor

0.219 0.029 CHEMBL2111041

0.131 0.068 CHEMBL3544855

0.392 0.009 CHEMBL3544856

0.75 0.003 CHEMBL1203

0.251 0.023 CHEMBL1442231

0.374 0.01 CHEMBL3544636

0.716 0.003 CHEMBL3544637

0.596 0.004 CHEMBL3091859

0.635 0.004 CHEMBL1237174

0.727 0.003 CHEMBL3091852

CHEMBL1203
0.1310.0110.163DNA gyrase inhibitor

0.163 0.007 CHEMBL1203

0.063 0.045 CHEMBL3544636

0.076 0.03 CHEMBL3091859

0.072 0.034 CHEMBL1237174

CHEMBL1203
0.1860.0690.322Dual specificity phosphatase 3 inhibitor

0.179 0.074 CHEMBL2111041

0.17 0.081 CHEMBL3544855

0.247 0.041 CHEMBL1203

0.147 0.099 CHEMBL1442231

0.322 0.025 CHEMBL1237174

CHEMBL1237174
0.1480.0370.148MAP kinase 13 inhibitor
0.1870.0770.276Growth factor agonist

0.276 0.022 CHEMBL3544856

0.271 0.024 CHEMBL1203

0.206 0.058 CHEMBL1442231

0.272 0.023 CHEMBL3544636

0.174 0.096 CHEMBL3544637

CHEMBL3544856
0.1370.0290.171Nitric-oxide synthase inhibitor

0.09 0.078 CHEMBL1203

0.143 0.025 CHEMBL3091859

0.171 0.016 CHEMBL1237174

0.096 0.066 CHEMBL3091852

CHEMBL1237174
0.1650.0560.274GABA C receptor rho-2 antagonist

0.141 0.086 CHEMBL2111041

0.264 0.009 CHEMBL1203

0.153 0.07 CHEMBL1442231

0.269 0.008 CHEMBL3544636

0.17 0.051 CHEMBL3091859

0.274 0.008 CHEMBL1237174

0.22 0.02 CHEMBL3091852

CHEMBL1237174
0.1270.0210.162Ornithine decarboxylase inhibitor

0.104 0.04 CHEMBL2111041

0.09 0.056 CHEMBL3544855

0.162 0.008 CHEMBL1203

0.104 0.04 CHEMBL3544636

0.09 0.056 CHEMBL3544637

0.12 0.026 CHEMBL3091859

0.137 0.016 CHEMBL1237174

0.097 0.048 CHEMBL3091852

CHEMBL1203
0.1250.020.151Carbonic anhydrase V inhibitor

0.113 0.023 CHEMBL1203

0.131 0.019 CHEMBL3091859

0.151 0.014 CHEMBL1237174

0.086 0.033 CHEMBL3091852

CHEMBL1237174
0.110.0040.11DNA gyrase subunit B inhibitor

0.08 0.005 CHEMBL1203

0.065 0.007 CHEMBL3544636

0.044 0.018 CHEMBL3091859

0.042 0.02 CHEMBL1237174

0.1210.0180.139Carbonic anhydrase VA inhibitor

0.109 0.021 CHEMBL1203

0.121 0.018 CHEMBL3091859

0.139 0.013 CHEMBL1237174

0.088 0.031 CHEMBL3091852

CHEMBL1237174
0.1960.0950.321Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor

0.321 0.044 CHEMBL1203

CHEMBL1203
0.1060.0060.224CDK5/p25 inhibitor

0.183 0.004 CHEMBL1442231

0.224 0.004 CHEMBL3091859

0.056 0.017 CHEMBL1237174

0.134 0.005 CHEMBL3091852

CHEMBL3091859
0.1150.0170.125Carbonic anhydrase IX inhibitor

0.047 0.045 CHEMBL1442231

0.125 0.015 CHEMBL3091859

0.075 0.03 CHEMBL1237174

0.062 0.036 CHEMBL3091852

CHEMBL3091859
0.1540.0610.264Mannose-6-phosphate isomerase inhibitor

0.178 0.044 CHEMBL2111041

0.136 0.078 CHEMBL3544855

0.264 0.009 CHEMBL3544856

0.26 0.01 CHEMBL1203

0.133 0.081 CHEMBL1442231

0.128 0.088 CHEMBL3544636

0.254 0.011 CHEMBL3544637

0.139 0.075 CHEMBL3091859

0.205 0.028 CHEMBL1237174

0.203 0.029 CHEMBL3091852

CHEMBL3544856
0.1810.0870.181Ca2+/calmodulin-dependent protein kinase inhibitor

0.176 0.091 CHEMBL1203

0.1180.0250.118Rho-associated kinase II inhibitor

0.081 0.044 CHEMBL1442231

0.071 0.055 CHEMBL3544636

0.1930.1030.309Dyrk kinase inhibitor

0.309 0.05 CHEMBL1203

CHEMBL1203
0.1680.0790.2Tumour necrosis factor antagonist

0.2 0.054 CHEMBL1203

0.17 0.077 CHEMBL1237174

CHEMBL1203
0.0970.0080.097Myc inhibitor

0.056 0.034 CHEMBL2111041

0.053 0.04 CHEMBL3544855

0.082 0.012 CHEMBL1203

0.073 0.017 CHEMBL1442231

0.062 0.027 CHEMBL3091859

0.055 0.036 CHEMBL3091852

0.1260.0390.204Acetylcholine release stimulant

0.183 0.005 CHEMBL1203

0.144 0.02 CHEMBL1442231

0.141 0.023 CHEMBL3544636

0.204 0.004 CHEMBL3544637

0.097 0.095 CHEMBL3091859

0.134 0.03 CHEMBL1237174

0.132 0.032 CHEMBL3091852

CHEMBL3544637
0.1520.0650.183Glycogen synthase kinase-3 alpha inhibitor

0.183 0.047 CHEMBL1203

CHEMBL1203
0.1450.0590.476Cyclin-dependent kinase inhibitor

0.253 0.027 CHEMBL1442231

0.476 0.008 CHEMBL3091859

0.444 0.009 CHEMBL3091852

CHEMBL3091859
0.0860.0050.091Vascular adhesion protein 1 inhibitor

0.035 0.034 CHEMBL1203

0.035 0.034 CHEMBL1442231

0.091 0.004 CHEMBL3091859

0.082 0.005 CHEMBL1237174

0.053 0.013 CHEMBL3091852

CHEMBL3091859
0.1630.0810.244Dual specificity phosphatase inhibitor

0.167 0.077 CHEMBL2111041

0.168 0.076 CHEMBL3544855

0.244 0.039 CHEMBL1203

0.145 0.1 CHEMBL1442231

0.207 0.051 CHEMBL1237174

CHEMBL1203
0.20.1190.279Neuropeptide Y2 antagonist

0.185 0.148 CHEMBL1203

0.211 0.101 CHEMBL1442231

0.279 0.031 CHEMBL3091859

0.269 0.039 CHEMBL1237174

0.276 0.033 CHEMBL3091852

CHEMBL3091859
0.1010.0220.104HIV-1 integrase (Strand Transfer) inhibitor

0.095 0.024 CHEMBL1203

0.104 0.021 CHEMBL1237174

CHEMBL1237174
0.1040.0260.139Carbonic anhydrase inhibitor

0.139 0.018 CHEMBL3091859

0.083 0.033 CHEMBL1237174

0.064 0.044 CHEMBL3091852

CHEMBL3091859
0.2050.1270.399Tyrosine 3 hydroxylase inhibitor

0.277 0.046 CHEMBL2111041

0.242 0.076 CHEMBL3544855

0.283 0.042 CHEMBL1203

0.208 0.121 CHEMBL1442231

0.348 0.017 CHEMBL3544636

0.316 0.026 CHEMBL3091859

0.399 0.008 CHEMBL1237174

0.385 0.01 CHEMBL3091852

CHEMBL1237174
0.2250.1490.683Vasodilator, peripheral

0.571 0.019 CHEMBL1203

0.272 0.112 CHEMBL3544636

0.683 0.007 CHEMBL3544637

0.283 0.106 CHEMBL3091859

0.462 0.037 CHEMBL1237174

0.267 0.115 CHEMBL3091852

CHEMBL3544637
0.090.0140.09Enoyl-[acyl-carrier-protein] reductase inhibitor

0.064 0.036 CHEMBL3091859

0.074 0.024 CHEMBL1237174

0.1110.0360.111Stem cell growth factor agonist

0.1 0.045 CHEMBL1442231

0.079 0.067 CHEMBL3544636

0.2380.1630.365Beta lactamase inhibitor

0.365 0.111 CHEMBL1442231

0.283 0.141 CHEMBL3091859

0.307 0.132 CHEMBL3091852

CHEMBL1442231
0.0810.0060.081Plasmepsin II inhibitor

0.068 0.009 CHEMBL1442231

0.077 0.006 CHEMBL3091859

0.047 0.02 CHEMBL1237174

0.058 0.013 CHEMBL3091852

0.0870.0130.284Plasminogen activator inhibitor antagonist

0.175 0.005 CHEMBL1203

0.06 0.024 CHEMBL3544636

0.284 0.004 CHEMBL3091859

0.248 0.004 CHEMBL1237174

CHEMBL3091859
0.2130.1380.373Insulysin inhibitor

0.216 0.134 CHEMBL2111041

0.266 0.083 CHEMBL3544855

0.365 0.029 CHEMBL1203

0.243 0.103 CHEMBL1442231

0.373 0.027 CHEMBL3544636

0.246 0.1 CHEMBL3091859

0.294 0.062 CHEMBL1237174

0.314 0.05 CHEMBL3091852

CHEMBL3544636
0.0940.020.094Carbonic anhydrase I inhibitor

0.049 0.044 CHEMBL3544636

0.092 0.021 CHEMBL3091859

0.071 0.029 CHEMBL1237174

0.10.0260.117HIV-1 integrase (3'-Processing) inhibitor

0.095 0.028 CHEMBL1203

0.056 0.052 CHEMBL3091859

0.117 0.02 CHEMBL1237174

CHEMBL1237174
0.10.0290.133D-Ala-D-Ala ligase inhibitor

0.096 0.034 CHEMBL2111041

0.078 0.075 CHEMBL3544855

0.133 0.009 CHEMBL1203

0.105 0.024 CHEMBL1442231

0.082 0.062 CHEMBL3544636

0.101 0.028 CHEMBL3091859

0.116 0.016 CHEMBL1237174

0.123 0.012 CHEMBL3091852

CHEMBL1203
0.0860.0150.113Carbonic anhydrase XIV inhibitor

0.092 0.013 CHEMBL1203

0.048 0.035 CHEMBL3544636

0.113 0.008 CHEMBL3544637

0.068 0.021 CHEMBL3091859

0.08 0.017 CHEMBL1237174

0.044 0.041 CHEMBL3091852

CHEMBL3544637
0.0770.0070.087Dihydropteroate synthase inhibitor

0.071 0.008 CHEMBL1203

0.052 0.016 CHEMBL3544636

0.067 0.009 CHEMBL3091859

0.087 0.005 CHEMBL1237174

0.048 0.018 CHEMBL3091852

CHEMBL1237174
0.1480.0790.382Dual specificity tyrosine-phosphorylation-regulated kinase 4 inhibitor

0.163 0.069 CHEMBL1203

0.323 0.021 CHEMBL1442231

0.382 0.01 CHEMBL3091852

CHEMBL3091852
0.0870.0180.148Exportin-1 inhibitor

0.068 0.047 CHEMBL2111041

0.09 0.015 CHEMBL1203

0.116 0.005 CHEMBL1442231

0.068 0.047 CHEMBL3544636

0.095 0.011 CHEMBL3091859

0.109 0.006 CHEMBL1237174

0.148 0.004 CHEMBL3091852

CHEMBL3091852
0.0880.0190.161Carbonic anhydrase VB inhibitor

0.12 0.012 CHEMBL1203

0.116 0.013 CHEMBL3091859

0.161 0.008 CHEMBL1237174

0.074 0.025 CHEMBL3091852

CHEMBL1237174
0.080.0120.081Lysine-specific demethylase 1A inhibitor

0.071 0.017 CHEMBL3091859

0.081 0.012 CHEMBL1237174

CHEMBL1237174
0.0760.0090.097Factor XIIIa inhibitor

0.05 0.016 CHEMBL3544636

0.097 0.006 CHEMBL3091859

0.052 0.015 CHEMBL1237174

0.033 0.032 CHEMBL3091852

CHEMBL3091859
0.1060.0390.139Polo-like kinase-1 inhibitor

0.089 0.063 CHEMBL1203

0.139 0.021 CHEMBL1442231

0.085 0.072 CHEMBL3544636

0.084 0.074 CHEMBL1237174

0.101 0.044 CHEMBL3091852

CHEMBL1442231
0.1570.090.3013C-like protease (Human coronavirus) inhibitor

0.301 0.011 CHEMBL1203

0.2 0.051 CHEMBL1442231

0.184 0.062 CHEMBL3544636

0.183 0.062 CHEMBL3091859

0.207 0.048 CHEMBL1237174

0.269 0.02 CHEMBL3091852

CHEMBL1203
0.1020.0350.159Inducible nitric-oxide synthase inhibitor

0.086 0.053 CHEMBL1203

0.106 0.032 CHEMBL3091859

0.159 0.014 CHEMBL1237174

0.075 0.072 CHEMBL3091852

CHEMBL1237174
0.1380.0740.138Ribosomal protein S6 kinase inhibitor
0.0950.0320.122Estrogen-related receptor beta agonist

0.105 0.02 CHEMBL2111041

0.102 0.022 CHEMBL3544855

0.084 0.054 CHEMBL3544856

0.089 0.043 CHEMBL1203

0.096 0.03 CHEMBL1442231

0.117 0.011 CHEMBL3544636

0.102 0.022 CHEMBL3091859

0.112 0.014 CHEMBL1237174

0.122 0.009 CHEMBL3091852

CHEMBL3091852
0.1770.1140.423Cyclic AMP phosphodiesterase inhibitor

0.338 0.029 CHEMBL1203

0.423 0.014 CHEMBL3544637

0.236 0.071 CHEMBL3091859

0.313 0.037 CHEMBL1237174

0.255 0.061 CHEMBL3091852

CHEMBL3544637
0.120.0580.142DNA intercalator

0.142 0.046 CHEMBL3544637

CHEMBL3544637
0.1150.0530.161MAO B inhibitor

0.161 0.034 CHEMBL3091859

0.091 0.065 CHEMBL1237174

CHEMBL3091859
0.1760.1160.2835 Hydroxytryptamine 3E antagonist

0.19 0.081 CHEMBL1203

0.184 0.096 CHEMBL1442231

0.218 0.038 CHEMBL3091859

0.283 0.007 CHEMBL1237174

0.253 0.015 CHEMBL3091852

CHEMBL1237174
0.2050.1460.375Hypoxia-inducible factor 1 alpha inhibitor

0.31 0.061 CHEMBL1203

0.301 0.065 CHEMBL3544636

0.375 0.037 CHEMBL3544637

0.224 0.124 CHEMBL3091859

0.253 0.098 CHEMBL1237174

CHEMBL3544637
0.0850.0250.085MAP kinase kinase 10 inhibitor
0.0970.0380.169CYP2A6 inhibitor

0.169 0.012 CHEMBL1203

0.078 0.05 CHEMBL1442231

0.069 0.061 CHEMBL3544636

0.128 0.023 CHEMBL1237174

0.069 0.061 CHEMBL3091852

CHEMBL1203
0.0830.0240.083Carbonic anhydrase XII inhibitor

0.047 0.04 CHEMBL3544637

0.076 0.027 CHEMBL3091859

0.058 0.034 CHEMBL1237174

0.1380.0820.174Thiol protease inhibitor

0.146 0.073 CHEMBL2111041

0.129 0.098 CHEMBL3544855

0.122 0.112 CHEMBL3544856

0.169 0.055 CHEMBL1203

0.143 0.076 CHEMBL1442231

0.158 0.062 CHEMBL3544636

0.135 0.087 CHEMBL3091859

0.147 0.072 CHEMBL1237174

0.174 0.052 CHEMBL3091852

CHEMBL3091852
0.0810.0250.115Carbonic anhydrase II inhibitor

0.115 0.015 CHEMBL3091859

0.071 0.029 CHEMBL1237174

0.058 0.037 CHEMBL3091852

CHEMBL3091859
0.1530.0990.153CDC-like kinase 4 inhibitor
0.1180.0640.305Protein kinase (CK2) alpha inhibitor

0.305 0.011 CHEMBL1203

0.136 0.051 CHEMBL3091859

0.107 0.071 CHEMBL1237174

0.104 0.073 CHEMBL3091852

CHEMBL1203
0.150.0960.166Cyclin-dependent kinase 3 inhibitor

0.166 0.066 CHEMBL3544856

0.157 0.08 CHEMBL1203

0.166 0.066 CHEMBL1442231

0.166 0.066 CHEMBL3544636

0.139 0.125 CHEMBL3091852

CHEMBL3544636
0.1360.0860.277Cytidine deaminase inhibitor

0.277 0.023 CHEMBL1203

0.115 0.106 CHEMBL1442231

0.118 0.102 CHEMBL3544636

0.114 0.108 CHEMBL3091859

0.196 0.05 CHEMBL1237174

0.158 0.069 CHEMBL3091852

CHEMBL1203
0.1320.0820.132Protein kinase (CK1) inhibitor

0.107 0.102 CHEMBL1203

0.0730.0240.161Cyclin D1 inhibitor

0.161 0.004 CHEMBL1442231

0.077 0.02 CHEMBL3091859

0.065 0.035 CHEMBL1237174

0.132 0.004 CHEMBL3091852

CHEMBL1442231
0.0930.0440.197Carbonic anhydrase VI inhibitor

0.148 0.021 CHEMBL1203

0.072 0.069 CHEMBL3544637

0.139 0.023 CHEMBL3091859

0.197 0.013 CHEMBL1237174

0.092 0.045 CHEMBL3091852

CHEMBL1237174
0.110.0620.488Ferrochelatase inhibitor

0.196 0.023 CHEMBL2111041

0.177 0.028 CHEMBL3544855

0.488 0.003 CHEMBL1203

0.13 0.047 CHEMBL1442231

0.229 0.016 CHEMBL3544636

0.303 0.007 CHEMBL3091859

0.388 0.004 CHEMBL1237174

0.391 0.004 CHEMBL3091852

CHEMBL1203
0.1040.0570.27GABA C receptor rho-1 antagonist

0.099 0.063 CHEMBL2111041

0.27 0.004 CHEMBL1203

0.095 0.07 CHEMBL1442231

0.236 0.005 CHEMBL3544636

0.123 0.038 CHEMBL3091859

0.23 0.005 CHEMBL1237174

0.172 0.014 CHEMBL3091852

CHEMBL1203
0.0530.0060.102Methionyl aminopeptidase 2 inhibitor

0.102 0.004 CHEMBL1203

0.061 0.005 CHEMBL1442231

0.026 0.017 CHEMBL1237174

0.045 0.008 CHEMBL3091852

CHEMBL1203
0.0660.0190.12Topoisomerase II beta inhibitor

0.12 0.007 CHEMBL1203

0.06 0.022 CHEMBL1442231

0.08 0.013 CHEMBL3544636

0.054 0.028 CHEMBL3544637

0.068 0.017 CHEMBL3091859

0.099 0.009 CHEMBL1237174

0.093 0.01 CHEMBL3091852

CHEMBL1203
0.1010.0540.154Lanosterol 14 alpha demethylase inhibitor

0.084 0.083 CHEMBL2111041

0.154 0.01 CHEMBL1203

0.099 0.057 CHEMBL1442231

0.151 0.011 CHEMBL3544636

0.084 0.083 CHEMBL3544637

0.131 0.021 CHEMBL1237174

0.105 0.048 CHEMBL3091852

CHEMBL1203
0.0690.0230.069Cyclin A1 inhibitor

0.062 0.034 CHEMBL3091859

0.064 0.031 CHEMBL1237174

0.056 0.048 CHEMBL3091852

0.1520.1080.393Succinate dehydrogenase inhibitor

0.191 0.057 CHEMBL2111041

0.196 0.052 CHEMBL3544855

0.138 0.136 CHEMBL3544856

0.393 0.004 CHEMBL1203

0.156 0.101 CHEMBL1442231

0.228 0.031 CHEMBL3544636

0.144 0.124 CHEMBL3544637

0.241 0.026 CHEMBL3091859

0.302 0.01 CHEMBL1237174

0.296 0.011 CHEMBL3091852

CHEMBL1203
0.2230.180.417Calcium channel activator

0.417 0.019 CHEMBL1203

0.267 0.127 CHEMBL3544636

0.228 0.174 CHEMBL3544637

0.241 0.158 CHEMBL3091859

0.381 0.032 CHEMBL1237174

0.327 0.067 CHEMBL3091852

CHEMBL1203
0.1560.1140.3I kappa B kinase epsilon inhibitor

0.3 0.015 CHEMBL1203

0.158 0.111 CHEMBL1442231

0.201 0.07 CHEMBL3544636

0.179 0.09 CHEMBL1237174

0.169 0.1 CHEMBL3091852

CHEMBL1203
0.1070.0680.271GABA C receptor antagonist

0.102 0.075 CHEMBL2111041

0.263 0.005 CHEMBL1203

0.098 0.082 CHEMBL1442231

0.22 0.009 CHEMBL3544636

0.148 0.031 CHEMBL3091859

0.271 0.005 CHEMBL1237174

0.209 0.011 CHEMBL3091852

CHEMBL1237174
0.1530.1150.348DNA methylase inhibitor

0.158 0.11 CHEMBL3544855

0.278 0.035 CHEMBL1203

0.227 0.062 CHEMBL3544636

0.348 0.017 CHEMBL3544637

0.238 0.055 CHEMBL1237174

0.142 0.125 CHEMBL3091852

CHEMBL3544637
0.1040.0660.104Cyclin-dependent kinase 2 inhibitor

0.096 0.074 CHEMBL1442231

0.092 0.08 CHEMBL3091859

0.0660.0290.209Mannitol-1-phosphate 5-dehydrogenase inhibitor

0.063 0.031 CHEMBL2111041

0.139 0.009 CHEMBL3544856

0.148 0.009 CHEMBL1203

0.058 0.037 CHEMBL1442231

0.088 0.017 CHEMBL3544636

0.209 0.006 CHEMBL3544637

0.072 0.024 CHEMBL3091859

0.153 0.008 CHEMBL1237174

0.101 0.014 CHEMBL3091852

CHEMBL3544637
0.0610.0250.526Aconitate hydratase inhibitor

0.071 0.018 CHEMBL2111041

0.114 0.006 CHEMBL3544855

0.048 0.043 CHEMBL3544856

0.526 0.001 CHEMBL1203

0.048 0.043 CHEMBL1442231

0.146 0.004 CHEMBL3544636

0.064 0.023 CHEMBL3544637

0.058 0.028 CHEMBL3091859

0.137 0.005 CHEMBL1237174

0.081 0.013 CHEMBL3091852

CHEMBL1203
0.0810.0460.081Rho-associated kinase inhibitor
0.1020.0670.459Beta glucuronidase inhibitor

0.103 0.065 CHEMBL2111041

0.103 0.065 CHEMBL3544856

0.119 0.047 CHEMBL1203

0.113 0.053 CHEMBL1442231

0.459 0.004 CHEMBL3544637

0.099 0.071 CHEMBL1237174

0.106 0.061 CHEMBL3091852

CHEMBL3544637
0.1130.0780.354Aldehyde dehydrogenase inhibitor

0.354 0.007 CHEMBL1203

0.257 0.017 CHEMBL3544636

0.211 0.025 CHEMBL3544637

0.137 0.056 CHEMBL3091859

0.271 0.015 CHEMBL1237174

0.127 0.064 CHEMBL3091852

CHEMBL1203
0.1750.1410.265Calpain inhibitor

0.174 0.143 CHEMBL1203

0.243 0.072 CHEMBL1442231

0.209 0.105 CHEMBL3544636

0.212 0.102 CHEMBL3091859

0.227 0.088 CHEMBL1237174

0.265 0.052 CHEMBL3091852

CHEMBL3091852
0.0650.030.089Botulinum neurotoxin type A inhibitor

0.076 0.02 CHEMBL1203

0.078 0.018 CHEMBL1442231

0.089 0.012 CHEMBL3544636

0.07 0.025 CHEMBL3091859

0.073 0.022 CHEMBL1237174

0.086 0.014 CHEMBL3091852

CHEMBL3544636
0.0560.0220.057Carbonic anhydrase VII inhibitor

0.054 0.024 CHEMBL3091859

0.057 0.021 CHEMBL1237174

CHEMBL1237174
0.1340.10.203Ca2+-transporting ATPase inhibitor

0.129 0.124 CHEMBL2111041

0.13 0.119 CHEMBL3544855

0.203 0.003 CHEMBL1203

0.131 0.115 CHEMBL1442231

0.138 0.082 CHEMBL3544636

0.183 0.005 CHEMBL3544637

0.157 0.029 CHEMBL3091859

0.188 0.005 CHEMBL1237174

0.171 0.012 CHEMBL3091852

CHEMBL1203
0.0920.060.144Protein kinase C delta inhibitor

0.144 0.024 CHEMBL1203

0.117 0.039 CHEMBL3544637

CHEMBL1203
0.0870.0570.142Granulocyte macrophage colony stimulating factor agonist

0.079 0.078 CHEMBL2111041

0.133 0.009 CHEMBL1203

0.085 0.063 CHEMBL1442231

0.114 0.02 CHEMBL3544636

0.096 0.04 CHEMBL3091859

0.142 0.007 CHEMBL1237174

0.12 0.016 CHEMBL3091852

CHEMBL1237174
0.2360.2090.332MAP kinase kinase 6 inhibitor

0.332 0.107 CHEMBL1203

CHEMBL1203
0.1340.1080.218Arachidonic acid antagonist

0.154 0.084 CHEMBL2111041

0.159 0.078 CHEMBL3544855

0.218 0.019 CHEMBL1203

0.13 0.113 CHEMBL1442231

0.173 0.062 CHEMBL3544636

0.16 0.077 CHEMBL3544637

0.178 0.056 CHEMBL3091859

0.215 0.021 CHEMBL1237174

0.204 0.03 CHEMBL3091852

CHEMBL1203
0.0940.0680.477UDP-glucose 4-epimerase inhibitor

0.17 0.023 CHEMBL3544856

0.409 0.005 CHEMBL1203

0.105 0.055 CHEMBL1442231

0.103 0.057 CHEMBL3544636

0.477 0.003 CHEMBL3544637

0.201 0.018 CHEMBL3091859

0.316 0.009 CHEMBL1237174

0.301 0.01 CHEMBL3091852

CHEMBL3544637
0.0620.0370.12Glutamate (mGluR1) antagonist

0.12 0.011 CHEMBL1203

0.077 0.025 CHEMBL3544636

0.075 0.027 CHEMBL1237174

CHEMBL1203
0.030.0060.06ICAM 1 antagonist

0.034 0.005 CHEMBL1203

0.06 0.004 CHEMBL3544636

0.026 0.01 CHEMBL1237174

CHEMBL3544636
0.0380.0140.11Methionyl aminopeptidase 1 inhibitor

0.03 0.027 CHEMBL3544856

0.048 0.007 CHEMBL1203

0.11 0.004 CHEMBL1442231

0.033 0.02 CHEMBL1237174

0.065 0.004 CHEMBL3091852

CHEMBL1442231
0.1390.1190.535Platelet adhesion inhibitor

0.247 0.05 CHEMBL2111041

0.215 0.063 CHEMBL3544855

0.535 0.005 CHEMBL3544637

CHEMBL3544637
0.1260.1070.233Phospholipase A2 inhibitor

0.204 0.04 CHEMBL1203

0.137 0.09 CHEMBL3544636

0.132 0.097 CHEMBL3544637

0.233 0.028 CHEMBL3091859

0.176 0.056 CHEMBL1237174

0.138 0.088 CHEMBL3091852

CHEMBL3091859
0.1980.1790.773Antithrombotic

0.205 0.171 CHEMBL3544855

0.412 0.046 CHEMBL1203

0.459 0.036 CHEMBL3544636

0.773 0.005 CHEMBL3544637

0.223 0.151 CHEMBL3091859

0.312 0.081 CHEMBL1237174

0.223 0.15 CHEMBL3091852

CHEMBL3544637
0.0870.0680.383Alcohol dehydrogenase inhibitor

0.119 0.035 CHEMBL2111041

0.136 0.026 CHEMBL3544855

0.383 0.004 CHEMBL1203

0.098 0.054 CHEMBL1442231

0.221 0.01 CHEMBL3544636

0.156 0.019 CHEMBL3544637

0.089 0.066 CHEMBL3091859

0.108 0.044 CHEMBL1237174

0.139 0.024 CHEMBL3091852

CHEMBL1203
0.1320.1140.191CF transmembrane conductance regulator agonist

0.163 0.055 CHEMBL1203

0.149 0.077 CHEMBL3544636

0.162 0.057 CHEMBL3544637

0.13 0.119 CHEMBL3091859

0.191 0.027 CHEMBL1237174

0.172 0.045 CHEMBL3091852

CHEMBL1237174
0.0590.0410.343Biliverdin reductase inhibitor

0.075 0.029 CHEMBL2111041

0.069 0.033 CHEMBL3544855

0.068 0.034 CHEMBL3544856

0.343 0.003 CHEMBL1203

0.059 0.042 CHEMBL1442231

0.113 0.015 CHEMBL3544636

0.128 0.012 CHEMBL3544637

0.114 0.015 CHEMBL3091859

0.197 0.006 CHEMBL1237174

0.171 0.008 CHEMBL3091852

CHEMBL1203
0.0620.0450.082Histone deacetylase SIRT3 inhibitor

0.062 0.043 CHEMBL1203

0.071 0.026 CHEMBL1442231

0.082 0.017 CHEMBL3544636

0.065 0.037 CHEMBL1237174

0.069 0.03 CHEMBL3091852

CHEMBL3544636
0.1170.10.208Neurotrophic factor

0.208 0.024 CHEMBL1203

0.123 0.09 CHEMBL3544637

CHEMBL1203
0.1250.1090.143Cyclin-dependent kinase 8 inhibitor

0.143 0.087 CHEMBL1203

0.132 0.1 CHEMBL1442231

0.127 0.106 CHEMBL1237174

0.133 0.099 CHEMBL3091852

CHEMBL1203
0.060.0440.06Cyclin A inhibitor
0.0580.0430.118Carbonic anhydrase stimulant

0.087 0.023 CHEMBL2111041

0.085 0.023 CHEMBL3544855

0.073 0.029 CHEMBL1203

0.062 0.038 CHEMBL1442231

0.118 0.015 CHEMBL3544636

0.055 0.047 CHEMBL3091859

0.077 0.027 CHEMBL1237174

0.081 0.025 CHEMBL3091852

CHEMBL3544636
0.2080.1930.662Histamine release inhibitor

0.286 0.132 CHEMBL2111041

0.311 0.118 CHEMBL3544855

0.322 0.113 CHEMBL3544856

0.646 0.007 CHEMBL1203

0.267 0.143 CHEMBL1442231

0.497 0.03 CHEMBL3544636

0.662 0.006 CHEMBL3544637

0.305 0.121 CHEMBL3091859

0.404 0.073 CHEMBL1237174

0.447 0.051 CHEMBL3091852

CHEMBL3544637
0.0550.0410.077Cathepsin B inhibitor

0.077 0.025 CHEMBL3091859

0.06 0.035 CHEMBL1237174

0.057 0.038 CHEMBL3091852

CHEMBL3091859
0.0870.0740.136Potassium channel (Voltage-sensitive) activator

0.136 0.019 CHEMBL1442231

0.129 0.024 CHEMBL3091852

CHEMBL1442231
0.0310.0180.066Cyclin E2 inhibitor

0.066 0.006 CHEMBL3091859

0.03 0.019 CHEMBL1237174

0.029 0.019 CHEMBL3091852

CHEMBL3091859
0.0530.0410.153Thromboxane synthase inhibitor

0.062 0.025 CHEMBL2111041

0.099 0.007 CHEMBL3544855

0.153 0.004 CHEMBL1203

0.121 0.005 CHEMBL3544636

0.054 0.039 CHEMBL1237174

CHEMBL1203
0.070.0580.151Carbonic anhydrase XIII inhibitor

0.139 0.024 CHEMBL1203

0.069 0.06 CHEMBL3544637

0.115 0.031 CHEMBL3091859

0.151 0.021 CHEMBL1237174

0.083 0.048 CHEMBL3091852

CHEMBL1237174
0.190.1790.71Transcription factor NF kappa B inhibitor

0.304 0.092 CHEMBL1203

0.194 0.175 CHEMBL3544636

0.71 0.019 CHEMBL3544637

0.234 0.139 CHEMBL3091859

0.266 0.116 CHEMBL1237174

0.237 0.137 CHEMBL3091852

CHEMBL3544637
0.0550.0440.224Cyclin E inhibitor

0.109 0.021 CHEMBL1442231

0.224 0.005 CHEMBL3091859

0.142 0.012 CHEMBL3091852

CHEMBL3091859
0.0280.0180.031Glucosylceramidase stimulant

0.029 0.015 CHEMBL1203

0.027 0.022 CHEMBL1442231

0.03 0.012 CHEMBL3544636

0.031 0.011 CHEMBL1237174

CHEMBL1237174
0.0920.0820.332Adenylate kinase inhibitor

0.11 0.054 CHEMBL2111041

0.116 0.047 CHEMBL3544855

0.332 0.005 CHEMBL1203

0.179 0.018 CHEMBL3544636

0.209 0.014 CHEMBL3544637

0.159 0.023 CHEMBL3091859

0.27 0.009 CHEMBL1237174

0.223 0.012 CHEMBL3091852

CHEMBL1203
0.0640.0550.13Glutamate (mGluR7) antagonist

0.13 0.004 CHEMBL1203

0.07 0.042 CHEMBL3544636

0.062 0.06 CHEMBL3091859

0.106 0.008 CHEMBL1237174

0.084 0.023 CHEMBL3091852

CHEMBL1203
0.0450.0370.14AMPA receptor antagonist

0.14 0.006 CHEMBL1203

0.058 0.026 CHEMBL3544636

0.043 0.04 CHEMBL1237174

0.052 0.03 CHEMBL3091852

CHEMBL1203
0.0420.0340.052Dihydrofolate reductase inhibitor

0.04 0.039 CHEMBL1203

0.041 0.038 CHEMBL3544636

0.052 0.016 CHEMBL1237174

CHEMBL1237174
0.0290.0220.045Nicotinic alpha3beta4 receptor agonist

0.037 0.012 CHEMBL1203

0.045 0.007 CHEMBL1237174

0.029 0.022 CHEMBL3091852

CHEMBL1237174
0.0480.0420.079Ribonucleoside-diphosphate reductase inhibitor

0.06 0.034 CHEMBL2111041

0.071 0.028 CHEMBL3544855

0.076 0.026 CHEMBL3544856

0.048 0.042 CHEMBL1203

0.049 0.041 CHEMBL1442231

0.079 0.025 CHEMBL3544636

0.065 0.031 CHEMBL3091859

0.061 0.034 CHEMBL1237174

0.072 0.028 CHEMBL3091852

CHEMBL3544636
0.1250.1190.215Heat shock protein 90 alpha antagonist

0.142 0.096 CHEMBL3544855

0.177 0.065 CHEMBL1203

0.215 0.041 CHEMBL1442231

0.124 0.121 CHEMBL1237174

0.172 0.068 CHEMBL3091852

CHEMBL1442231
0.0630.0580.138CDK2/cyclin E2 inhibitor

0.138 0.019 CHEMBL3091859

CHEMBL3091859
0.0810.0750.409Triose-phosphate isomerase inhibitor

0.091 0.058 CHEMBL2111041

0.11 0.039 CHEMBL3544855

0.165 0.016 CHEMBL3544856

0.399 0.003 CHEMBL1203

0.133 0.026 CHEMBL3544636

0.409 0.003 CHEMBL3544637

0.147 0.021 CHEMBL3091859

0.267 0.006 CHEMBL1237174

0.212 0.01 CHEMBL3091852

CHEMBL3544637
0.0320.0270.0761-Alkyl-2-acetylglycerophosphocholine esterase inhibitor

0.043 0.013 CHEMBL1203

0.076 0.005 CHEMBL3091859

0.043 0.014 CHEMBL1237174

0.034 0.024 CHEMBL3091852

CHEMBL3091859
0.1250.120.165MAP kinase 3 inhibitor

0.165 0.048 CHEMBL1203

0.139 0.087 CHEMBL3544636

0.137 0.09 CHEMBL1237174

0.124 0.123 CHEMBL3091852

CHEMBL1203
0.0290.0250.063Endothelial nitric-oxide synthase inhibitor

0.03 0.023 CHEMBL3091859

0.063 0.007 CHEMBL1237174

CHEMBL1237174
0.1080.1050.118Toll-Like receptor antagonist

0.112 0.099 CHEMBL1442231

0.118 0.088 CHEMBL3091852

CHEMBL3091852
0.0470.0440.081Ribonucleotide reductase inhibitor

0.06 0.037 CHEMBL2111041

0.071 0.03 CHEMBL3544855

0.076 0.028 CHEMBL3544856

0.048 0.044 CHEMBL1203

0.048 0.043 CHEMBL1442231

0.081 0.026 CHEMBL3544636

0.067 0.033 CHEMBL3091859

0.062 0.035 CHEMBL1237174

0.074 0.029 CHEMBL3091852

CHEMBL3544636
0.0390.0360.073Histamine H2 receptor agonist

0.045 0.027 CHEMBL1442231

0.039 0.037 CHEMBL3544636

0.051 0.021 CHEMBL3091859

0.072 0.009 CHEMBL1237174

0.073 0.009 CHEMBL3091852

CHEMBL3091852
0.1490.1470.639Free radical scavenger

0.304 0.051 CHEMBL2111041

0.196 0.101 CHEMBL3544855

0.166 0.127 CHEMBL1203

0.639 0.007 CHEMBL3544637

0.239 0.073 CHEMBL3091859

0.211 0.089 CHEMBL1237174

CHEMBL3544637
0.0270.0260.068Peptide deformylase inhibitor

0.032 0.019 CHEMBL3544636

0.068 0.005 CHEMBL3091859

0.052 0.009 CHEMBL1237174

0.04 0.014 CHEMBL3091852

CHEMBL3091859
0.0520.0510.1243-Oxoacyl-[acyl-carrier-protein] synthase inhibitor

0.081 0.024 CHEMBL2111041

0.083 0.023 CHEMBL3544855

0.124 0.011 CHEMBL1203

0.058 0.042 CHEMBL1442231

0.072 0.029 CHEMBL3544637

0.053 0.049 CHEMBL1237174

0.073 0.028 CHEMBL3091852

CHEMBL1203
0.1330.1330.3Psychostimulant

0.173 0.098 CHEMBL1203

0.153 0.113 CHEMBL3544636

0.197 0.082 CHEMBL3544637

0.225 0.068 CHEMBL3091859

0.3 0.043 CHEMBL1237174

0.15 0.116 CHEMBL3091852

CHEMBL1237174
0.0780.0780.506NADH dehydrogenase inhibitor

0.079 0.077 CHEMBL2111041

0.117 0.03 CHEMBL3544856

0.347 0.005 CHEMBL1203

0.139 0.02 CHEMBL3544636

0.506 0.003 CHEMBL3544637

0.123 0.027 CHEMBL3091859

0.247 0.008 CHEMBL1237174

0.164 0.015 CHEMBL3091852

CHEMBL3544637
0.0490.0490.073Sphingosine kinase 2 inhibitor

0.053 0.043 CHEMBL3544856

0.051 0.045 CHEMBL1203

0.073 0.019 CHEMBL1237174

0.056 0.036 CHEMBL3091852

CHEMBL1237174
0.0240.0250.05Thymidine phosphorylase inhibitor

0.025 0.021 CHEMBL1203

0.029 0.013 CHEMBL3091859

0.05 0.005 CHEMBL1237174

0.027 0.016 CHEMBL3091852

CHEMBL1237174
0.0680.0690.084Potassium channel (Tandem pore domain) blocker

0.07 0.065 CHEMBL1203

0.08 0.034 CHEMBL1442231

0.082 0.031 CHEMBL3544636

0.084 0.027 CHEMBL1237174

0.082 0.029 CHEMBL3091852

CHEMBL1237174
0.080.0830.28Protein kinase (CK2) inhibitor

0.28 0.008 CHEMBL1203

0.089 0.073 CHEMBL3091859

0.088 0.074 CHEMBL1237174

CHEMBL1203
0.1170.1190.15Heat shock protein 90 antagonist

0.132 0.094 CHEMBL1203

0.15 0.075 CHEMBL1442231

0.129 0.099 CHEMBL1237174

0.138 0.088 CHEMBL3091852

CHEMBL1442231
0.0620.0650.093Benzodiazepine agonist

0.086 0.035 CHEMBL3091859

0.093 0.03 CHEMBL1237174

CHEMBL1237174
0.0110.0140.021-Deoxy-D-xylulose-5-phosphate reductoisomerase inhibitor

0.014 0.008 CHEMBL1203

0.015 0.007 CHEMBL1442231

0.018 0.005 CHEMBL3544636

0.014 0.008 CHEMBL3091859

0.018 0.004 CHEMBL1237174

0.02 0.004 CHEMBL3091852

CHEMBL3091852
0.0290.0330.047Carnitine palmitoyltransferase 1 inhibitor

0.047 0.01 CHEMBL1203

0.034 0.024 CHEMBL1237174

CHEMBL1203
0.040.0440.23Cyclin E1 inhibitor

0.095 0.02 CHEMBL1442231

0.23 0.005 CHEMBL3091859

0.133 0.011 CHEMBL3091852

CHEMBL3091859
0.0350.0390.062Carbonic anhydrase IV inhibitor

0.059 0.02 CHEMBL3544636

0.052 0.023 CHEMBL3091859

0.062 0.018 CHEMBL1237174

0.04 0.033 CHEMBL3091852

CHEMBL1237174
0.0960.10.144MAP kinase kinase inhibitor

0.144 0.055 CHEMBL1203

0.117 0.077 CHEMBL1442231

0.1 0.095 CHEMBL1237174

0.128 0.067 CHEMBL3091852

CHEMBL1203
0.0620.0660.179Aminopeptidase I inhibitor

0.076 0.046 CHEMBL2111041

0.075 0.048 CHEMBL3544855

0.179 0.009 CHEMBL1203

0.068 0.056 CHEMBL1442231

0.155 0.012 CHEMBL3544636

0.1 0.028 CHEMBL3091859

0.138 0.015 CHEMBL1237174

0.13 0.017 CHEMBL3091852

CHEMBL1203
0.0840.0880.318Electrolyte absorption antagonist

0.09 0.074 CHEMBL2111041

0.088 0.078 CHEMBL3544855

0.318 0.004 CHEMBL1203

0.089 0.076 CHEMBL1442231

0.174 0.012 CHEMBL3544636

0.113 0.042 CHEMBL3091859

0.176 0.012 CHEMBL1237174

0.162 0.015 CHEMBL3091852

CHEMBL1203
0.0420.0460.114Glucose-6-phosphate isomerase inhibitor

0.055 0.023 CHEMBL3544855

0.075 0.01 CHEMBL3544856

0.076 0.01 CHEMBL1203

0.054 0.024 CHEMBL3544636

0.114 0.004 CHEMBL3544637

0.065 0.015 CHEMBL3091859

0.107 0.004 CHEMBL1237174

0.081 0.008 CHEMBL3091852

CHEMBL3544637
0.0690.0740.172Protein kinase A inhibitor

0.09 0.052 CHEMBL1203

0.172 0.019 CHEMBL3544637

CHEMBL3544637
0.0090.0150.021Thrombopoietin agonist

0.013 0.007 CHEMBL2111041

0.021 0.004 CHEMBL1203

0.012 0.008 CHEMBL1442231

CHEMBL1203
0.0020.0090.004Reverse transcriptase (HBV) inhibitor

0.004 0.003 CHEMBL3544636

CHEMBL3544636
0.0210.0280.03211-Beta-hydroxysteroid dehydrogenase 2 inhibitor

0.03 0.017 CHEMBL1203

0.032 0.015 CHEMBL1237174

CHEMBL1237174
0.0280.0350.047Carnitine palmitoyltransferase inhibitor

0.047 0.01 CHEMBL1203

0.033 0.025 CHEMBL1237174

CHEMBL1203
0.0630.070.144Phospholipase D inhibitor

0.088 0.024 CHEMBL1203

0.144 0.004 CHEMBL3544636

0.108 0.01 CHEMBL1237174

0.087 0.025 CHEMBL3091852

CHEMBL3544636
0.1270.1340.26DNA methyltransferase I inhibitor

0.136 0.121 CHEMBL3544855

0.253 0.045 CHEMBL1203

0.17 0.086 CHEMBL3544636

0.26 0.043 CHEMBL3544637

0.146 0.108 CHEMBL3091859

0.247 0.048 CHEMBL1237174

0.152 0.101 CHEMBL3091852

CHEMBL3544637
0.0040.0120.007CC chemokine 6 receptor agonist

0.007 0.004 CHEMBL1237174

CHEMBL1237174
0.1620.170.369RNA-directed DNA polymerase inhibitor

0.369 0.022 CHEMBL1203

0.185 0.123 CHEMBL3544636

0.269 0.04 CHEMBL3544637

0.18 0.132 CHEMBL3091859

0.3 0.032 CHEMBL1237174

0.235 0.06 CHEMBL3091852

CHEMBL1203
0.0490.0570.208Carbamoyl phosphate synthetase inhibitor

0.057 0.046 CHEMBL2111041

0.09 0.024 CHEMBL3544855

0.053 0.051 CHEMBL3544856

0.128 0.014 CHEMBL1203

0.095 0.022 CHEMBL3544636

0.072 0.033 CHEMBL3544637

0.103 0.02 CHEMBL3091859

0.208 0.007 CHEMBL1237174

0.142 0.012 CHEMBL3091852

CHEMBL1237174
0.0310.040.081Alpha 1d adrenoreceptor agonist

0.052 0.015 CHEMBL1203

0.081 0.005 CHEMBL1237174

0.048 0.018 CHEMBL3091852

CHEMBL1237174
0.0150.0240.023Estrogen-related receptor gamma agonist

0.018 0.014 CHEMBL2111041

0.02 0.01 CHEMBL1442231

0.019 0.012 CHEMBL3544636

0.017 0.016 CHEMBL3091859

0.023 0.007 CHEMBL3091852

CHEMBL3091852
0.0710.080.099MAP kinase kinase 7 inhibitor

0.099 0.014 CHEMBL1203

0.08 0.047 CHEMBL3544636

0.098 0.015 CHEMBL1237174

0.086 0.031 CHEMBL3091852

CHEMBL1203
0.0040.0140.01Integrin alpha5beta6 antagonist

0.006 0.005 CHEMBL3544855

0.007 0.004 CHEMBL1203

0.01 0.003 CHEMBL3544636

0.006 0.005 CHEMBL1237174

0.007 0.004 CHEMBL3091852

CHEMBL3544636
0.0360.0460.052CF transmembrane conductance regulator antagonist

0.052 0.007 CHEMBL1203

0.04 0.026 CHEMBL1237174

0.043 0.019 CHEMBL3091852

CHEMBL1203
0.1890.1990.407Calpain 2 inhibitor

0.221 0.171 CHEMBL1203

0.387 0.068 CHEMBL1442231

0.235 0.16 CHEMBL3544636

0.225 0.168 CHEMBL3091859

0.268 0.137 CHEMBL1237174

0.407 0.058 CHEMBL3091852

CHEMBL3091852
0.0240.0340.047Purinergic P2Y15 antagonist

0.029 0.019 CHEMBL1203

0.026 0.025 CHEMBL1442231

0.03 0.018 CHEMBL3544636

0.037 0.009 CHEMBL3091859

0.047 0.004 CHEMBL1237174

0.046 0.005 CHEMBL3091852

CHEMBL1237174
0.0550.0660.363Phenylalanine 4-hydroxylase inhibitor

0.071 0.045 CHEMBL2111041

0.067 0.05 CHEMBL3544855

0.082 0.036 CHEMBL3544856

0.363 0.003 CHEMBL1203

0.063 0.054 CHEMBL1442231

0.202 0.007 CHEMBL3544636

0.087 0.033 CHEMBL3091859

0.157 0.011 CHEMBL1237174

0.137 0.014 CHEMBL3091852

CHEMBL1203
0.0320.0430.088Glutamate (mGluR1a) antagonist

0.088 0.007 CHEMBL1203

0.063 0.014 CHEMBL3544636

0.04 0.029 CHEMBL1237174

0.036 0.035 CHEMBL3091852

CHEMBL1203
0.0210.0340.039Nicotinic alpha4beta2 receptor agonist

0.03 0.018 CHEMBL1203

0.039 0.008 CHEMBL1237174

CHEMBL1237174
0.1290.1430.254ATPase inhibitor

0.141 0.118 CHEMBL2111041

0.143 0.113 CHEMBL3544856

0.167 0.075 CHEMBL1203

0.14 0.119 CHEMBL1442231

0.145 0.11 CHEMBL3544636

0.254 0.013 CHEMBL3544637

0.134 0.133 CHEMBL3091859

0.179 0.059 CHEMBL1237174

0.195 0.041 CHEMBL3091852

CHEMBL3544637
0.0540.0680.075CDC7 inhibitor

0.075 0.039 CHEMBL1203

0.062 0.054 CHEMBL1442231

CHEMBL1203
0.020.0340.144Glucagon receptor antagonist

0.07 0.006 CHEMBL2111041

0.084 0.005 CHEMBL3544855

0.032 0.019 CHEMBL1442231

0.144 0.004 CHEMBL3544636

CHEMBL3544636
0.0240.0380.047Epoxide hydrolase 1 inhibitor

0.047 0.007 CHEMBL1203

0.033 0.019 CHEMBL1442231

0.038 0.012 CHEMBL3544636

0.029 0.024 CHEMBL3091859

0.037 0.014 CHEMBL1237174

0.042 0.01 CHEMBL3091852

CHEMBL1203
0.0990.1140.157Toll-Like receptor 9 antagonist

0.157 0.058 CHEMBL1237174

CHEMBL1237174
0.0150.030.033Antibiotic Anthracycline-like

0.033 0.003 CHEMBL3544637

0.027 0.004 CHEMBL3091859

0.029 0.004 CHEMBL1237174

0.02 0.011 CHEMBL3091852

CHEMBL3544637
0.1340.1490.251Death-associated protein kinase 3 inhibitor

0.228 0.061 CHEMBL1203

0.233 0.059 CHEMBL1442231

0.251 0.052 CHEMBL3091852

CHEMBL3091852
0.0340.050.087Geranyltranstransferase inhibitor

0.087 0.004 CHEMBL1203

0.066 0.009 CHEMBL3544636

0.064 0.011 CHEMBL1237174

0.045 0.028 CHEMBL3091852

CHEMBL1203
0.0170.0330.083AMPA 1 receptor antagonist

0.083 0.007 CHEMBL1203

0.055 0.01 CHEMBL3544636

CHEMBL1203
0.0230.040.036Hedgehog signaling activator

0.029 0.014 CHEMBL1203

0.036 0.006 CHEMBL1237174

0.028 0.017 CHEMBL3091852

CHEMBL1237174
0.0260.0420.033Calcium release-activated channel blocker

0.033 0.022 CHEMBL1203

CHEMBL1203
0.0070.0260.113Egl nine homolog 3 inhibitor

0.046 0.003 CHEMBL1203

0.113 0.002 CHEMBL3544636

0.011 0.009 CHEMBL1237174

CHEMBL3544636
0.0550.0750.077Transcription factor RelA inhibitor

0.063 0.047 CHEMBL1203

0.061 0.053 CHEMBL3091859

0.077 0.02 CHEMBL1237174

0.073 0.026 CHEMBL3091852

CHEMBL1237174
0.0360.0560.061Histamine H1 receptor agonist

0.061 0.008 CHEMBL1237174

0.048 0.021 CHEMBL3091852

CHEMBL1237174
0.0720.0920.185HIV-1 integrase (Overall Integration) inhibitor

0.08 0.078 CHEMBL2111041

0.185 0.015 CHEMBL1203

0.117 0.041 CHEMBL1442231

0.154 0.024 CHEMBL3544636

0.159 0.022 CHEMBL1237174

0.163 0.021 CHEMBL3091852

CHEMBL1203
0.1550.1750.5685 Hydroxytryptamine release stimulant

0.395 0.047 CHEMBL1203

0.216 0.109 CHEMBL3544636

0.342 0.058 CHEMBL3544637

0.203 0.119 CHEMBL3091859

0.568 0.018 CHEMBL1237174

0.357 0.055 CHEMBL3091852

CHEMBL1237174
0.030.0510.047Potassium channel Kv1.1 blocker

0.047 0.015 CHEMBL1237174

0.037 0.028 CHEMBL3091852

CHEMBL1237174
0.010.0310.025Steroid 17-alpha-hydroxylase/17,20 lyase inhibitor

0.025 0.011 CHEMBL1203

CHEMBL1203
0.0120.0340.022CC chemokine 9 receptor antagonist

0.022 0.005 CHEMBL1203

0.016 0.015 CHEMBL1237174

CHEMBL1203
0.0320.0550.1Stearoyl-CoA desaturase inhibitor

0.1 0.007 CHEMBL3544636

CHEMBL3544636
0.0580.0810.321Glutamate dehydrogenase inhibitor

0.07 0.057 CHEMBL2111041

0.094 0.034 CHEMBL3544855

0.321 0.005 CHEMBL1203

0.149 0.016 CHEMBL3544636

0.114 0.025 CHEMBL3544637

0.124 0.021 CHEMBL3091859

0.182 0.012 CHEMBL1237174

0.177 0.012 CHEMBL3091852

CHEMBL1203
0.0350.0580.229Glutamate (mGluR4) antagonist

0.041 0.035 CHEMBL3544855

0.229 0.003 CHEMBL1203

0.071 0.01 CHEMBL3544636

0.053 0.018 CHEMBL1237174

CHEMBL1203
0.0270.0510.111Protein kinase (CK2) beta inhibitor

0.111 0.003 CHEMBL1203

0.037 0.016 CHEMBL1237174

0.031 0.03 CHEMBL3091852

CHEMBL1203
0.0550.0790.144Histone deacetylase stimulant

0.085 0.039 CHEMBL3544856

0.087 0.037 CHEMBL1203

0.144 0.01 CHEMBL3544637

CHEMBL3544637
0.0550.0790.144Histone deacetylase SIRT1 stimulant

0.085 0.039 CHEMBL3544856

0.087 0.037 CHEMBL1203

0.144 0.01 CHEMBL3544637

CHEMBL3544637
0.0250.0510.039Delayed rectifier potassium channel activator

0.039 0.023 CHEMBL3091852

CHEMBL3091852
0.0250.0510.039Potassium channel KCNQ activator

0.039 0.023 CHEMBL3091852

CHEMBL3091852
0.070.0970.161Potassium channel activator

0.091 0.059 CHEMBL1203

0.152 0.019 CHEMBL1442231

0.091 0.059 CHEMBL3091859

0.161 0.016 CHEMBL3091852

CHEMBL3091852
0.0370.0640.21Acyl-CoA dehydrogenase inhibitor

0.21 0.005 CHEMBL1203

0.083 0.021 CHEMBL3544636

0.069 0.027 CHEMBL3544637

0.123 0.012 CHEMBL3091859

0.185 0.006 CHEMBL1237174

0.177 0.007 CHEMBL3091852

CHEMBL1203
0.0430.0710.072Epithelial sodium channel blocker

0.055 0.038 CHEMBL3544856

0.072 0.017 CHEMBL3544636

0.064 0.024 CHEMBL1237174

0.057 0.033 CHEMBL3091852

CHEMBL3544636
0.080.1080.2Phosphodiesterase 6D inhibitor

0.129 0.019 CHEMBL1203

0.2 0.005 CHEMBL3544637

0.099 0.055 CHEMBL1237174

CHEMBL3544637
0.0310.0590.113Thymidylate synthase inhibitor

0.048 0.03 CHEMBL3544855

0.061 0.017 CHEMBL1203

0.113 0.004 CHEMBL3544636

0.054 0.023 CHEMBL1237174

CHEMBL3544636
0.0090.0380.017Adenosine A2 receptor agonist

0.015 0.013 CHEMBL3544856

0.017 0.01 CHEMBL1237174

CHEMBL1237174
0.050.0790.066Aryl hydrocarbon receptor antagonist

0.059 0.056 CHEMBL1203

0.066 0.044 CHEMBL1237174

CHEMBL1237174
0.0210.050.031Thymidine kinase (Herpes simplex virus 1) inhibitor

0.027 0.016 CHEMBL1203

0.026 0.02 CHEMBL3544637

0.031 0.01 CHEMBL1237174

0.027 0.016 CHEMBL3091852

CHEMBL1237174
0.0090.0390.024Cyclin T1 inhibitor

0.018 0.013 CHEMBL1203

0.024 0.008 CHEMBL1237174

CHEMBL1237174
0.0580.0880.078Adenosine A3 receptor antagonist

0.078 0.046 CHEMBL1237174

CHEMBL1237174
0.0130.0440.051Glutamate (mGluR1a) agonist

0.049 0.005 CHEMBL1203

0.03 0.009 CHEMBL3544636

0.051 0.005 CHEMBL1237174

0.029 0.009 CHEMBL3091852

CHEMBL1237174
0.0090.040.021Thromboxane A2 agonist

0.017 0.008 CHEMBL3544855

0.014 0.013 CHEMBL3091859

0.021 0.005 CHEMBL1237174

0.02 0.005 CHEMBL3091852

CHEMBL1237174
0.010.0410.018Nicotinic alpha4 receptor agonist

0.018 0.009 CHEMBL1237174

CHEMBL1237174
0.0330.0640.062Glutamate (mGluR5) agonist

0.062 0.017 CHEMBL1203

CHEMBL1203
0.0380.0690.078Dopamine beta hydroxylase inhibitor

0.078 0.005 CHEMBL1203

0.045 0.043 CHEMBL3544636

0.067 0.01 CHEMBL1237174

0.048 0.034 CHEMBL3091852

CHEMBL1203
0.0290.0610.061Angiotensin AT1 receptor antagonist

0.061 0.005 CHEMBL1203

0.048 0.021 CHEMBL1237174

0.048 0.02 CHEMBL3091852

CHEMBL1203
0.070.1020.084Pim-3 kinase inhibitor

0.084 0.069 CHEMBL1203

CHEMBL1203
0.0060.0380.03Carbonic anhydrase XI inhibitor

0.012 0.009 CHEMBL1203

0.02 0.004 CHEMBL3091859

0.018 0.005 CHEMBL1237174

0.03 0.003 CHEMBL3091852

CHEMBL3091852
0.020.0520.034Complement factor 1s inhibitor

0.029 0.009 CHEMBL1203

0.034 0.005 CHEMBL1237174

0.025 0.019 CHEMBL3091852

CHEMBL1237174
0.0060.0380.013Purinergic P2Y2 agonist

0.013 0.004 CHEMBL3544637

0.01 0.008 CHEMBL1237174

CHEMBL3544637
0.0430.0750.1Dihydroorotate oxidase inhibitor

0.1 0.005 CHEMBL1203

0.064 0.024 CHEMBL3091859

0.08 0.01 CHEMBL1237174

0.084 0.009 CHEMBL3091852

CHEMBL1203
0.0130.0460.039NMDA receptor glycine site antagonist

0.039 0.009 CHEMBL1203

0.023 0.019 CHEMBL1237174

CHEMBL1203
0.0370.0710.09Cathepsin D inhibitor

0.09 0.021 CHEMBL3091859

CHEMBL3091859
0.0090.0450.044Nicotinic acid receptor 1 antagonist

0.044 0.003 CHEMBL1203

0.022 0.007 CHEMBL1237174

0.022 0.007 CHEMBL3091852

CHEMBL1203
0.0310.0660.092Nerve growth factor antagonist

0.092 0.003 CHEMBL1203

0.057 0.011 CHEMBL1237174

0.047 0.023 CHEMBL3091852

CHEMBL1203
0.1340.170.532Immunostimulant

0.203 0.119 CHEMBL1203

0.273 0.088 CHEMBL3544636

0.532 0.025 CHEMBL3544637

0.223 0.108 CHEMBL3091859

0.255 0.094 CHEMBL1237174

0.205 0.117 CHEMBL3091852

CHEMBL3544637
0.0060.0420.011Purine nucleoside phosphorylase inhibitor

0.011 0.01 CHEMBL1237174

CHEMBL1237174
0.0060.0420.017Adenosine A2a receptor agonist

0.017 0.009 CHEMBL1237174

CHEMBL1237174
0.0210.0570.033MAP3K8 inhibitor

0.031 0.017 CHEMBL1203

0.033 0.013 CHEMBL1237174

CHEMBL1237174
0.0320.0680.1113-Hydroxyanthranilate 3,4-dioxygenase inhibitor

0.111 0.003 CHEMBL1203

0.046 0.02 CHEMBL3091859

0.072 0.004 CHEMBL1237174

0.058 0.008 CHEMBL3091852

CHEMBL1203
0.020.0560.116Fumarate hydratase inhibitor

0.035 0.023 CHEMBL3544855

0.116 0.005 CHEMBL1203

0.039 0.019 CHEMBL3544636

0.039 0.02 CHEMBL3544637

0.046 0.015 CHEMBL3091859

0.083 0.007 CHEMBL1237174

0.07 0.008 CHEMBL3091852

CHEMBL1203
0.0130.0490.021Caspase 8 inhibitor

0.018 0.017 CHEMBL1442231

0.021 0.011 CHEMBL3544636

0.019 0.015 CHEMBL3091852

CHEMBL3544636
0.0430.080.287Phosphofructokinase-1 inhibitor

0.086 0.038 CHEMBL3544855

0.093 0.035 CHEMBL3544856

0.227 0.009 CHEMBL1203

0.092 0.035 CHEMBL3544636

0.287 0.006 CHEMBL3544637

0.094 0.034 CHEMBL3091859

0.205 0.011 CHEMBL1237174

0.138 0.02 CHEMBL3091852

CHEMBL3544637
0.0690.1060.146Sphingomyelinase inhibitor

0.146 0.026 CHEMBL3544856

0.102 0.057 CHEMBL1203

0.084 0.081 CHEMBL1442231

0.094 0.067 CHEMBL3544636

0.101 0.058 CHEMBL3544637

0.128 0.035 CHEMBL1237174

0.118 0.043 CHEMBL3091852

CHEMBL3544856
0.0210.0590.142Kainate receptor antagonist

0.142 0.005 CHEMBL1203

0.039 0.03 CHEMBL3544636

0.044 0.026 CHEMBL1237174

0.041 0.028 CHEMBL3091852

CHEMBL1203
0.0060.0440.017Human herpes virus 5 capsid protein P40 inhibitor

0.016 0.005 CHEMBL1203

0.017 0.005 CHEMBL1237174

CHEMBL1237174
0.0650.1020.144Falcipain inhibitor

0.114 0.047 CHEMBL1442231

0.144 0.034 CHEMBL3091852

CHEMBL3091852
0.1070.1460.174Protein kinase (CK1) gamma 3 inhibitor

0.146 0.095 CHEMBL1203

0.174 0.066 CHEMBL1442231

0.161 0.078 CHEMBL3091852

CHEMBL1442231
0.0690.1080.284Creatine kinase inhibitor

0.09 0.072 CHEMBL2111041

0.284 0.004 CHEMBL1203

0.1 0.06 CHEMBL3544636

0.136 0.031 CHEMBL3091859

0.21 0.009 CHEMBL1237174

0.187 0.013 CHEMBL3091852

CHEMBL1203
0.0410.080.072Glucosylceramidase inhibitor

0.065 0.026 CHEMBL3544856

0.055 0.037 CHEMBL1203

0.061 0.03 CHEMBL3544637

0.072 0.02 CHEMBL1237174

CHEMBL1237174
0.0750.1140.2065 Hydroxytryptamine 3A agonist

0.206 0.013 CHEMBL1237174

0.143 0.039 CHEMBL3091852

CHEMBL1237174
0.0260.0650.04Delayed rectifier potassium channel blocker

0.035 0.03 CHEMBL3544636

0.04 0.021 CHEMBL1237174

0.034 0.033 CHEMBL3091852

CHEMBL1237174
0.0470.0870.065Leukotriene C antagonist

0.065 0.019 CHEMBL1203

0.055 0.044 CHEMBL3544636

0.061 0.026 CHEMBL3091859

0.064 0.021 CHEMBL1237174

0.054 0.049 CHEMBL3091852

CHEMBL1203
0.0240.0640.067Glutamate (mGluR4) agonist

0.067 0.007 CHEMBL1203

0.032 0.027 CHEMBL1237174

CHEMBL1203
0.0450.0860.101Pregnane X receptor antagonist

0.101 0.004 CHEMBL1203

0.053 0.05 CHEMBL3544637

0.076 0.009 CHEMBL1237174

0.065 0.022 CHEMBL3091852

CHEMBL1203
0.0090.0490.014Cyclin D2 inhibitor

0.014 0.007 CHEMBL1237174

CHEMBL1237174
0.0720.1130.12Protein kinase C zeta inhibitor

0.12 0.032 CHEMBL1203

0.088 0.068 CHEMBL3544637

0.084 0.078 CHEMBL1237174

CHEMBL1203
0.0140.0550.025Thymidine kinase (Herpes simplex virus 2) inhibitor

0.025 0.007 CHEMBL1237174

0.023 0.009 CHEMBL3091852

CHEMBL1237174
0.2330.2750.515Caspase 9 stimulant

0.385 0.12 CHEMBL1203

0.276 0.222 CHEMBL1442231

0.318 0.175 CHEMBL3544636

0.515 0.054 CHEMBL3544637

0.337 0.157 CHEMBL3091859

0.458 0.079 CHEMBL1237174

0.469 0.074 CHEMBL3091852

CHEMBL3544637
0.0070.0490.043Carbonic anhydrase X inhibitor

0.03 0.004 CHEMBL1203

0.03 0.004 CHEMBL3091859

0.037 0.004 CHEMBL1237174

0.043 0.003 CHEMBL3091852

CHEMBL3091852
0.0070.0490.043Carbonic anhydrase VIII inhibitor

0.03 0.004 CHEMBL1203

0.03 0.004 CHEMBL3091859

0.037 0.004 CHEMBL1237174

0.043 0.003 CHEMBL3091852

CHEMBL3091852
0.0320.0750.061Adenosine A1 receptor antagonist

0.061 0.039 CHEMBL1237174

CHEMBL1237174
0.0270.0710.083Glutamate (mGluR8) agonist

0.037 0.027 CHEMBL3544855

0.083 0.004 CHEMBL1203

0.036 0.03 CHEMBL3544636

0.043 0.018 CHEMBL3091859

0.073 0.005 CHEMBL1237174

0.056 0.009 CHEMBL3091852

CHEMBL1203
0.0440.0880.07Heat shock protein 90 beta antagonist

0.056 0.047 CHEMBL3544636

0.07 0.029 CHEMBL1237174

CHEMBL1237174
0.060.1040.163Potassium channel (Ca-activated) activator

0.163 0.024 CHEMBL1203

0.133 0.034 CHEMBL1237174

CHEMBL1203
0.0220.0670.038Histone deacetylase class I inhibitor

0.038 0.029 CHEMBL1442231

CHEMBL1442231
0.0030.0480.01DNA topoisomerase III inhibitor

0.01 0.004 CHEMBL1237174

0.007 0.006 CHEMBL3091852

CHEMBL1237174
0.0290.0750.047Vanilloid 3 antagonist

0.047 0.011 CHEMBL1203

0.044 0.015 CHEMBL1237174

0.036 0.033 CHEMBL3091852

CHEMBL1203
0.0270.0730.039Histone deacetylase 9 inhibitor

0.038 0.029 CHEMBL1442231

0.036 0.034 CHEMBL3544636

0.039 0.028 CHEMBL3091852

CHEMBL3091852
0.0180.0640.049Calcitonin receptor agonist

0.049 0.017 CHEMBL3544636

0.033 0.024 CHEMBL1237174

0.03 0.027 CHEMBL3091852

CHEMBL3544636
0.1520.1990.524DNA synthesis inhibitor

0.233 0.08 CHEMBL2111041

0.214 0.103 CHEMBL3544855

0.307 0.041 CHEMBL3544856

0.395 0.022 CHEMBL1203

0.299 0.044 CHEMBL3544636

0.524 0.012 CHEMBL3544637

0.201 0.121 CHEMBL3091859

0.287 0.048 CHEMBL1237174

0.264 0.058 CHEMBL3091852

CHEMBL3544637
0.0150.0620.059Nicotinic acid receptor 2 antagonist

0.059 0.003 CHEMBL1203

0.026 0.019 CHEMBL3091859

0.037 0.006 CHEMBL1237174

0.037 0.006 CHEMBL3091852

CHEMBL1203
0.0130.060.024Methylmalonyl-CoA mutase inhibitor

0.024 0.004 CHEMBL1203

0.017 0.015 CHEMBL3544636

0.019 0.011 CHEMBL3091859

0.023 0.005 CHEMBL1237174

0.022 0.006 CHEMBL3091852

CHEMBL1203
0.060.1070.136Falcipain 2 inhibitor

0.104 0.05 CHEMBL1442231

0.136 0.035 CHEMBL3091852

CHEMBL3091852
0.0090.0570.053Hypoxanthine phosphoribosyltransferase inhibitor

0.032 0.016 CHEMBL1203

0.027 0.02 CHEMBL3544636

0.053 0.008 CHEMBL1237174

0.036 0.014 CHEMBL3091852

CHEMBL1237174
0.0330.0820.245Argininosuccinate synthase inhibitor

0.245 0.005 CHEMBL1203

0.081 0.025 CHEMBL3544636

0.088 0.022 CHEMBL3544637

0.074 0.028 CHEMBL3091859

0.165 0.01 CHEMBL1237174

0.118 0.015 CHEMBL3091852

CHEMBL1203
0.0550.1030.088Bcr-Abl kinase inhibitor

0.088 0.054 CHEMBL1203

CHEMBL1203
0.0210.070.054Angiotensin II receptor antagonist

0.054 0.005 CHEMBL1203

0.035 0.023 CHEMBL1237174

0.035 0.023 CHEMBL3091852

CHEMBL1203
0.0620.1110.104Vascular endothelial growth factor 1 antagonist

0.104 0.063 CHEMBL1203

CHEMBL1203
0.0320.0810.092Lysophosphatidic acid 3 receptor antagonist

0.045 0.044 CHEMBL3544855

0.092 0.006 CHEMBL1203

0.056 0.027 CHEMBL3544636

0.047 0.041 CHEMBL3091859

0.068 0.016 CHEMBL1237174

0.063 0.019 CHEMBL3091852

CHEMBL1203
0.0350.0840.048Heme oxygenase inhibitor

0.043 0.028 CHEMBL1203

0.048 0.015 CHEMBL1237174

CHEMBL1237174
0.070.120.092Glycogen synthase kinase-3 beta inhibitor

0.092 0.088 CHEMBL1442231

CHEMBL1442231
0.0380.0880.061Dipeptidyl peptidase inhibitor

0.061 0.025 CHEMBL1237174

CHEMBL1237174
0.0710.1210.144Anabolic

0.144 0.021 CHEMBL1203

0.103 0.059 CHEMBL3544636

0.102 0.06 CHEMBL3544637

0.116 0.043 CHEMBL3091859

0.143 0.022 CHEMBL1237174

0.14 0.024 CHEMBL3091852

CHEMBL1203
0.0190.070.035Estrogen-related receptor gamma antagonist

0.035 0.008 CHEMBL1237174

0.033 0.011 CHEMBL3091852

CHEMBL1237174
0.0420.0920.066Sphingosine kinase inhibitor

0.059 0.041 CHEMBL3544856

0.063 0.034 CHEMBL1237174

0.066 0.03 CHEMBL3091852

CHEMBL3091852
0.0340.0840.051Dipeptidyl peptidase IV inhibitor

0.051 0.019 CHEMBL1237174

CHEMBL1237174
0.0150.0660.109Kainate receptor 2 antagonist

0.109 0.004 CHEMBL1203

0.037 0.024 CHEMBL1442231

0.043 0.02 CHEMBL3544636

0.033 0.028 CHEMBL1237174

0.054 0.014 CHEMBL3091852

CHEMBL1203
0.0130.0640.093Lysine carboxypeptidase inhibitor

0.031 0.015 CHEMBL1203

0.093 0.004 CHEMBL3544636

0.033 0.013 CHEMBL1237174

CHEMBL3544636
0.1460.1970.2615 Hydroxytryptamine 1E antagonist

0.184 0.15 CHEMBL3091859

0.261 0.063 CHEMBL1237174

0.256 0.068 CHEMBL3091852

CHEMBL1237174
0.0060.0580.021Integrin alphaVbeta6 antagonist

0.021 0.005 CHEMBL3544636

CHEMBL3544636
0.0250.0770.08Tryptophan 5 hydroxylase inhibitor

0.05 0.005 CHEMBL1203

0.08 0.003 CHEMBL3544636

0.041 0.013 CHEMBL1237174

CHEMBL3544636
0.0220.0740.06Oxytocin agonist

0.038 0.034 CHEMBL3091859

0.058 0.018 CHEMBL1237174

0.06 0.017 CHEMBL3091852

CHEMBL3091852
0.0960.1480.203DNA repair enzyme inhibitor

0.132 0.052 CHEMBL1203

0.203 0.008 CHEMBL3544637

0.111 0.094 CHEMBL3091859

0.158 0.025 CHEMBL1237174

0.132 0.052 CHEMBL3091852

CHEMBL3544637
0.0240.0770.037MAP3K5 inhibitor

0.037 0.031 CHEMBL1237174

CHEMBL1237174
0.1260.1790.229Neurotrophic factor enhancer

0.219 0.06 CHEMBL1203

0.225 0.055 CHEMBL3544636

0.211 0.067 CHEMBL3544637

0.161 0.122 CHEMBL3091859

0.229 0.052 CHEMBL1237174

0.22 0.059 CHEMBL3091852

CHEMBL1237174
0.0110.0650.061Uridine phosphorylase inhibitor

0.061 0.005 CHEMBL1203

0.053 0.007 CHEMBL3544637

0.049 0.008 CHEMBL1237174

0.033 0.016 CHEMBL3091852

CHEMBL1203
0.0110.0650.02Alpha 2b adrenoreceptor agonist

0.02 0.01 CHEMBL1237174

CHEMBL1237174
0.0410.0950.162Purinergic P2X1 antagonist

0.162 0.006 CHEMBL1203

0.083 0.024 CHEMBL3544637

0.118 0.012 CHEMBL1237174

0.075 0.028 CHEMBL3091852

CHEMBL1203
0.0310.0860.206Glutamate (mGluR group III) antagonist

0.206 0.003 CHEMBL1203

0.051 0.019 CHEMBL3544636

0.049 0.022 CHEMBL1237174

CHEMBL1203
0.030.0840.067Kainate receptor agonist

0.066 0.005 CHEMBL1203

0.043 0.025 CHEMBL3544636

0.043 0.024 CHEMBL3091859

0.067 0.005 CHEMBL1237174

0.055 0.01 CHEMBL3091852

CHEMBL1237174
0.0040.0590.019Glutamate (mGluR6) agonist

0.019 0.004 CHEMBL1203

0.019 0.004 CHEMBL1237174

0.013 0.007 CHEMBL3091852

CHEMBL1237174
0.0550.110.29Keratolytic

0.29 0.004 CHEMBL1203

0.097 0.032 CHEMBL3544636

0.071 0.062 CHEMBL3544637

0.102 0.029 CHEMBL1237174

0.08 0.049 CHEMBL3091852

CHEMBL1203
0.0140.0690.031Carnitine palmitoyltransferase 1A inhibitor

0.031 0.017 CHEMBL1203

CHEMBL1203
0.0450.10.111Protein kinase C beta inhibitor

0.108 0.01 CHEMBL1203

0.111 0.009 CHEMBL3544637

0.071 0.046 CHEMBL1237174

CHEMBL3544637
0.0240.0790.078Glutamate (mGluR group I) agonist

0.078 0.013 CHEMBL1203

0.043 0.039 CHEMBL3544636

CHEMBL1203
0.0450.1010.107Protease 3C (Human rhinovirus) inhibitor

0.065 0.044 CHEMBL1442231

0.072 0.034 CHEMBL3091859

0.081 0.026 CHEMBL1237174

0.107 0.013 CHEMBL3091852

CHEMBL3091852
0.0020.0590.015KiSS-1 receptor agonist

0.015 0.004 CHEMBL3091852

CHEMBL3091852
0.0440.1010.103Elastase 1 inhibitor

0.065 0.054 CHEMBL2111041

0.069 0.048 CHEMBL3544855

0.103 0.019 CHEMBL3544856

0.063 0.056 CHEMBL1442231

CHEMBL3544856
0.0120.0690.028Acetylcholine M4 receptor agonist

0.028 0.023 CHEMBL1237174

CHEMBL1237174
0.0360.0940.066Cyclin-dependent kinase 6 inhibitor

0.053 0.05 CHEMBL1203

0.066 0.035 CHEMBL1237174

CHEMBL1237174
0.0030.0620.009Thyroid hormone beta agonist

0.009 0.006 CHEMBL3091859

CHEMBL3091859
0.0080.0680.025Telomerase stimulant

0.016 0.015 CHEMBL1203

0.023 0.005 CHEMBL3544637

0.016 0.015 CHEMBL3091859

0.025 0.004 CHEMBL1237174

0.02 0.008 CHEMBL3091852

CHEMBL1237174
0.0270.0870.073AICAR transformylase inhibitor

0.043 0.033 CHEMBL3544855

0.064 0.012 CHEMBL1203

0.073 0.009 CHEMBL3544636

0.054 0.018 CHEMBL1237174

0.047 0.026 CHEMBL3091852

CHEMBL3544636
0.0250.0850.15Ornithine carbamoyltransferase inhibitor

0.15 0.01 CHEMBL1203

0.091 0.018 CHEMBL3544636

0.052 0.038 CHEMBL3544637

0.061 0.031 CHEMBL3091859

0.11 0.014 CHEMBL1237174

0.087 0.019 CHEMBL3091852

CHEMBL1203
0.0230.0840.096Antimetabolite

0.048 0.033 CHEMBL3544855

0.043 0.037 CHEMBL1203

0.096 0.017 CHEMBL3544636

0.05 0.032 CHEMBL3544637

0.041 0.039 CHEMBL1237174

0.041 0.039 CHEMBL3091852

CHEMBL3544636
0.120.1820.199Focal adhesion kinase 2 inhibitor

0.156 0.12 CHEMBL1203

0.182 0.085 CHEMBL1442231

0.154 0.124 CHEMBL1237174

0.199 0.07 CHEMBL3091852

CHEMBL3091852
0.0470.1090.111Nicotinic alpha4beta2 receptor antagonist

0.111 0.023 CHEMBL1203

0.096 0.035 CHEMBL1237174

CHEMBL1203
0.0280.0910.088Adenylate cyclase 1 inhibitor

0.088 0.005 CHEMBL1237174

0.062 0.017 CHEMBL3091852

CHEMBL1237174
0.0070.0710.059Prostaglandin H2 antagonist

0.03 0.013 CHEMBL3544855

0.059 0.003 CHEMBL1203

0.038 0.007 CHEMBL3544636

CHEMBL1203
0.0150.0790.036Thyroid hormone agonist

0.025 0.02 CHEMBL3544636

0.036 0.008 CHEMBL3091859

0.029 0.013 CHEMBL1237174

0.025 0.02 CHEMBL3091852

CHEMBL3091859
0.0320.0970.06Potassium channel (ATP-sensitive) activator

0.044 0.042 CHEMBL1203

0.06 0.016 CHEMBL1237174

0.052 0.027 CHEMBL3091852

CHEMBL1237174
0.0260.0910.05Thymidine kinase inhibitor

0.041 0.029 CHEMBL1203

0.041 0.028 CHEMBL3544636

0.05 0.019 CHEMBL1237174

0.04 0.03 CHEMBL3091852

CHEMBL1237174
0.0130.0780.023Factor XIII inhibitor

0.023 0.01 CHEMBL1237174

0.02 0.016 CHEMBL3091852

CHEMBL1237174
0.0320.0970.441Selectin antagonist

0.091 0.031 CHEMBL1203

0.097 0.029 CHEMBL3544636

0.441 0.003 CHEMBL3544637

CHEMBL3544637
0.0330.0990.063Potassium channel (Inward rectifier) activator

0.046 0.044 CHEMBL1203

0.063 0.016 CHEMBL1237174

0.054 0.028 CHEMBL3091852

CHEMBL1237174
0.0260.0920.117Glutamate (mGluR group III) agonist

0.117 0.008 CHEMBL1203

0.039 0.036 CHEMBL3544636

0.042 0.031 CHEMBL1237174

CHEMBL1203
0.0190.0860.034Histone deacetylase 7 inhibitor

0.034 0.028 CHEMBL3091852

CHEMBL3091852
0.1220.1890.188Neurotensin receptor agonist

0.162 0.076 CHEMBL2111041

0.139 0.133 CHEMBL3544855

0.188 0.043 CHEMBL1203

0.14 0.128 CHEMBL1442231

0.186 0.044 CHEMBL3544636

0.152 0.097 CHEMBL3091859

0.179 0.05 CHEMBL1237174

0.185 0.045 CHEMBL3091852

CHEMBL1203
0.0570.1250.086Bronchodilator

0.086 0.079 CHEMBL1203

CHEMBL1203
0.0350.1040.072Alpha 2 adrenoreceptor agonist

0.072 0.03 CHEMBL1237174

CHEMBL1237174
0.0620.1310.372UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor

0.372 0.004 CHEMBL1203

0.103 0.051 CHEMBL3544636

0.339 0.005 CHEMBL3544637

0.176 0.02 CHEMBL3091859

0.257 0.009 CHEMBL1237174

0.263 0.009 CHEMBL3091852

CHEMBL1203
0.0220.0920.066Membrane dipeptidase inhibitor

0.036 0.034 CHEMBL2111041

0.04 0.027 CHEMBL3544855

0.054 0.013 CHEMBL1203

0.066 0.008 CHEMBL3544636

0.042 0.023 CHEMBL3091859

0.055 0.013 CHEMBL1237174

0.056 0.012 CHEMBL3091852

CHEMBL3544636
0.0080.0790.02Purinergic P2Y1 agonist

0.02 0.007 CHEMBL1237174

CHEMBL1237174
0.0070.0780.025Alpha 2a adrenoreceptor agonist

0.025 0.007 CHEMBL1237174

CHEMBL1237174
0.0250.0960.044Sphingosine kinase 1 inhibitor

0.041 0.029 CHEMBL1237174

0.044 0.024 CHEMBL3091852

CHEMBL3091852
0.0540.1250.222Aminopeptidase B inhibitor

0.222 0.017 CHEMBL1203

0.199 0.022 CHEMBL3544636

0.123 0.051 CHEMBL3091859

0.18 0.027 CHEMBL1237174

0.165 0.032 CHEMBL3091852

CHEMBL1203
0.0540.1260.081Interleukin-1 receptor-associated protein kinase 4 inhibitor

0.081 0.069 CHEMBL3544636

CHEMBL3544636
0.0350.1090.0765 Hydroxytryptamine 3A antagonist

0.076 0.035 CHEMBL1237174

CHEMBL1237174
0.0150.0880.057Glutamate (mGluR1) agonist

0.057 0.004 CHEMBL1203

0.027 0.013 CHEMBL3544636

0.03 0.009 CHEMBL1237174

0.026 0.015 CHEMBL3091852

CHEMBL1203
0.0140.0880.044Cathepsin L1 inhibitor

0.044 0.024 CHEMBL3091852

CHEMBL3091852
0.0790.1530.199Toll-Like receptor 2 antagonist

0.106 0.095 CHEMBL3544855

0.17 0.04 CHEMBL1203

0.128 0.069 CHEMBL1442231

0.199 0.024 CHEMBL3544636

0.151 0.052 CHEMBL3091859

0.153 0.051 CHEMBL1237174

0.198 0.024 CHEMBL3091852

CHEMBL3544636
0.0480.1220.08Acetylcholine nicotinic agonist

0.08 0.056 CHEMBL1203

CHEMBL1203
0.0490.1240.134Glutamate (mGluR6) antagonist

0.134 0.004 CHEMBL1203

0.064 0.054 CHEMBL3544636

0.074 0.032 CHEMBL3091859

0.114 0.007 CHEMBL1237174

0.092 0.014 CHEMBL3091852

CHEMBL1203
0.0080.0830.019Complement factor D inhibitor

0.018 0.013 CHEMBL1203

0.019 0.012 CHEMBL1237174

CHEMBL1237174
0.0180.0940.072Toll-Like receptor 2 agonist

0.038 0.031 CHEMBL1203

0.072 0.018 CHEMBL3544636

0.046 0.025 CHEMBL3544637

0.044 0.027 CHEMBL1237174

0.049 0.024 CHEMBL3091852

CHEMBL3544636
0.1190.1950.207Heat shock protein 70 antagonist

0.207 0.005 CHEMBL1203

0.141 0.073 CHEMBL3544636

0.166 0.021 CHEMBL3544637

0.156 0.034 CHEMBL1237174

0.148 0.051 CHEMBL3091852

CHEMBL1203
0.0310.1070.13Alpha-mannosidase inhibitor

0.056 0.033 CHEMBL3544856

0.063 0.023 CHEMBL1203

0.071 0.016 CHEMBL3544636

0.13 0.004 CHEMBL3544637

0.064 0.022 CHEMBL3091859

0.101 0.006 CHEMBL1237174

0.071 0.016 CHEMBL3091852

CHEMBL3544637
0.0380.1150.075Histone deacetylase inhibitor

0.075 0.035 CHEMBL1442231

0.063 0.049 CHEMBL3091852

CHEMBL1442231
0.1020.180.249Melanin inhibitor

0.157 0.073 CHEMBL1203

0.249 0.029 CHEMBL3544637

0.13 0.113 CHEMBL3091859

0.16 0.069 CHEMBL1237174

0.162 0.067 CHEMBL3091852

CHEMBL3544637
0.0210.0990.052Glutamate (mGluR3) agonist

0.052 0.004 CHEMBL1203

0.031 0.027 CHEMBL3091859

0.042 0.008 CHEMBL1237174

0.038 0.011 CHEMBL3091852

CHEMBL1203
0.0660.1450.104CC chemokine 5 receptor agonist

0.104 0.018 CHEMBL1237174

0.089 0.038 CHEMBL3091852

CHEMBL1237174
0.0850.1660.18Antibacterial (Helicobacter pylori)

0.121 0.08 CHEMBL3544856

0.18 0.028 CHEMBL1203

0.126 0.073 CHEMBL1442231

0.136 0.06 CHEMBL3544636

0.126 0.072 CHEMBL3544637

0.138 0.058 CHEMBL3091852

CHEMBL1203
0.0630.1440.376Chelator

0.134 0.043 CHEMBL2111041

0.135 0.042 CHEMBL3544855

0.325 0.009 CHEMBL3544856

0.208 0.023 CHEMBL1203

0.107 0.068 CHEMBL1442231

0.376 0.007 CHEMBL3544636

0.105 0.07 CHEMBL3091852

CHEMBL3544636
0.0030.0840.011Thromboxane agonist

0.011 0.007 CHEMBL3091852

CHEMBL3091852
0.0080.090.019Integrin beta6 antagonist

0.014 0.009 CHEMBL3544855

0.019 0.005 CHEMBL3544636

CHEMBL3544636
0.0040.0860.114Egl nine homolog 1 inhibitor

0.042 0.004 CHEMBL1203

0.114 0.002 CHEMBL3544636

CHEMBL3544636
0.0030.0850.021Lysophosphatidic acid receptor 3 agonist

0.021 0.005 CHEMBL1237174

0.017 0.007 CHEMBL3091852

CHEMBL1237174
0.0250.1080.065Cathepsin L inhibitor

0.065 0.034 CHEMBL3091852

CHEMBL3091852
0.0150.0990.035 Hydroxytryptamine 6 agonist

0.03 0.017 CHEMBL1237174

CHEMBL1237174
0.0770.1610.18NADPH oxidase inhibitor

0.18 0.041 CHEMBL1203

0.105 0.104 CHEMBL1237174

0.137 0.065 CHEMBL3091852

CHEMBL1203
0.0130.0980.039Vanilloid 2 agonist

0.036 0.005 CHEMBL1203

0.039 0.004 CHEMBL3544637

0.036 0.005 CHEMBL1237174

0.028 0.012 CHEMBL3091852

CHEMBL3544637
0.0630.1480.232M18 aspartyl aminopeptidase inhibitor

0.1 0.092 CHEMBL1203

0.153 0.051 CHEMBL1442231

0.232 0.025 CHEMBL3091852

CHEMBL3091852
0.0050.090.031KiSS-1 receptor antagonist

0.031 0.005 CHEMBL3091852

CHEMBL3091852
0.0350.1210.205Catalase inhibitor

0.071 0.054 CHEMBL3544855

0.205 0.014 CHEMBL1203

0.15 0.026 CHEMBL3544636

0.13 0.031 CHEMBL3091859

0.161 0.024 CHEMBL1237174

0.199 0.015 CHEMBL3091852

CHEMBL1203
0.0050.0910.017Aminopeptidase A inhibitor

0.017 0.013 CHEMBL1203

CHEMBL1203
0.0160.1020.027Thrombin receptor antagonist

0.027 0.022 CHEMBL3091852

CHEMBL3091852
0.0190.1070.079Adenosine deaminase inhibitor

0.079 0.009 CHEMBL1203

0.055 0.025 CHEMBL3544636

0.069 0.014 CHEMBL3544637

0.061 0.02 CHEMBL1237174

0.047 0.033 CHEMBL3091852

CHEMBL1203
0.0450.1350.093CDK/cyclin complex inhibitor

0.092 0.058 CHEMBL3091859

0.093 0.057 CHEMBL3091852

CHEMBL3091852
0.0210.1110.152Mannosidase inhibitor

0.044 0.034 CHEMBL3544856

0.063 0.015 CHEMBL1203

0.059 0.017 CHEMBL3544636

0.152 0.004 CHEMBL3544637

0.048 0.028 CHEMBL3091859

0.09 0.007 CHEMBL1237174

0.056 0.019 CHEMBL3091852

CHEMBL3544637
0.030.1210.069Cytokine production stimulant

0.069 0.008 CHEMBL3544637

0.058 0.015 CHEMBL1237174

0.056 0.018 CHEMBL3091852

CHEMBL3544637
0.0180.110.089Dopamine D5 agonist

0.036 0.034 CHEMBL1203

0.089 0.005 CHEMBL1237174

0.049 0.018 CHEMBL3091852

CHEMBL1237174
0.0180.110.183Phosphorylase inhibitor

0.078 0.017 CHEMBL1203

0.135 0.009 CHEMBL3544636

0.183 0.005 CHEMBL3544637

CHEMBL3544637
0.0540.1470.129Glutathione S-transferase inhibitor

0.098 0.039 CHEMBL1203

0.076 0.069 CHEMBL1442231

0.121 0.022 CHEMBL3544636

0.088 0.05 CHEMBL3091859

0.085 0.054 CHEMBL1237174

0.129 0.019 CHEMBL3091852

CHEMBL3091852
0.0160.1090.026Baculoviral IAP repeat-containing protein 4 inhibitor

0.026 0.022 CHEMBL3091852

CHEMBL3091852
0.0840.1770.219Mcl-1 antagonist

0.13 0.111 CHEMBL2111041

0.219 0.047 CHEMBL1203

CHEMBL1203
0.0240.1170.075Protein kinase C epsilon inhibitor

0.075 0.022 CHEMBL1203

0.056 0.034 CHEMBL3544636

CHEMBL1203
0.0460.140.082I kappa B kinase inhibitor

0.082 0.058 CHEMBL1203

CHEMBL1203
0.010.1030.026Isoleucine-tRNA ligase inhibitor

0.021 0.019 CHEMBL1203

0.026 0.009 CHEMBL1237174

0.025 0.011 CHEMBL3091852

CHEMBL1237174
0.0060.10.019Alpha 2c adrenoreceptor agonist

0.019 0.013 CHEMBL1237174

CHEMBL1237174
0.0970.1910.196Adenylate cyclase stimulant

0.157 0.051 CHEMBL1203

0.156 0.054 CHEMBL3544636

0.148 0.066 CHEMBL3544637

0.143 0.075 CHEMBL3091859

0.196 0.015 CHEMBL1237174

0.171 0.034 CHEMBL3091852

CHEMBL1237174
0.1330.2270.296Lipoxygenase inhibitor

0.296 0.073 CHEMBL2111041

0.217 0.124 CHEMBL3544855

0.22 0.122 CHEMBL1203

0.22 0.121 CHEMBL3091859

0.204 0.137 CHEMBL3091852

CHEMBL2111041
0.0280.1220.065Aldosterone antagonist

0.065 0.017 CHEMBL1203

0.054 0.024 CHEMBL1237174

CHEMBL1203
0.0120.1060.048Potassium channel small-conductance Ca-activated activator

0.048 0.012 CHEMBL1237174

CHEMBL1237174
0.0890.1840.304Hexokinase inhibitor

0.138 0.093 CHEMBL3544856

0.302 0.011 CHEMBL1203

0.141 0.09 CHEMBL1442231

0.133 0.1 CHEMBL3544636

0.304 0.01 CHEMBL3544637

0.161 0.066 CHEMBL1237174

0.199 0.036 CHEMBL3091852

CHEMBL3544637
0.0280.1240.055Nicotinic receptor alpha7 subunit antagonist

0.055 0.035 CHEMBL1203

CHEMBL1203
0.0110.1070.031Neuraminidase (Influenza B) inhibitor

0.031 0.004 CHEMBL1203

0.023 0.01 CHEMBL3091859

0.025 0.008 CHEMBL1237174

0.03 0.004 CHEMBL3091852

CHEMBL1203
0.0060.1030.02Adenosine kinase inhibitor

0.02 0.017 CHEMBL1237174

CHEMBL1237174
0.0270.1240.048Purinergic P2X4 antagonist

0.048 0.029 CHEMBL1203

0.047 0.03 CHEMBL1237174

CHEMBL1203
0.040.1380.089Thrombin inhibitor

0.089 0.033 CHEMBL1237174

CHEMBL1237174
0.0520.150.109Vanilloid 4 agonist

0.081 0.038 CHEMBL3091859

0.109 0.011 CHEMBL1237174

0.101 0.016 CHEMBL3091852

CHEMBL1237174
0.0620.1610.139MAP kinase kinase 1 inhibitor

0.134 0.024 CHEMBL1203

0.118 0.037 CHEMBL1442231

0.104 0.052 CHEMBL1237174

0.139 0.021 CHEMBL3091852

CHEMBL3091852
0.0180.1170.068RNA-directed RNA polymerase inhibitor

0.068 0.008 CHEMBL1203

0.041 0.017 CHEMBL3544636

0.031 0.03 CHEMBL1237174

CHEMBL1203
0.1350.2340.26412-Lipoxygenase inhibitor

0.243 0.113 CHEMBL2111041

0.231 0.121 CHEMBL1203

0.221 0.13 CHEMBL1442231

0.264 0.101 CHEMBL3091852

CHEMBL3091852
0.0120.1120.085Plasmepsin I inhibitor

0.053 0.007 CHEMBL3544856

0.053 0.006 CHEMBL1442231

0.085 0.004 CHEMBL3091852

CHEMBL3091852
0.1010.2020.152Pregnane X receptor agonist

0.139 0.077 CHEMBL1203

0.152 0.049 CHEMBL1237174

0.139 0.075 CHEMBL3091852

CHEMBL1237174
0.0030.1050.012Imidazoline I2 receptor antagonist

0.012 0.006 CHEMBL1237174

CHEMBL1237174
0.0440.1460.154Histamine N-methyltransferase inhibitor

0.154 0.013 CHEMBL1203

0.131 0.023 CHEMBL1237174

0.075 0.073 CHEMBL3091852

CHEMBL1203
0.0830.1860.21Diuretic

0.21 0.041 CHEMBL1203

0.209 0.041 CHEMBL3544636

0.175 0.057 CHEMBL3544637

0.16 0.069 CHEMBL1237174

CHEMBL1203
0.0120.1160.034Lysophosphatidic acid receptor 1 agonist

0.025 0.017 CHEMBL1203

0.025 0.018 CHEMBL3091859

0.034 0.008 CHEMBL1237174

0.032 0.009 CHEMBL3091852

CHEMBL1237174
0.0020.1060.015Integrin alphaVbeta5 antagonist

0.015 0.005 CHEMBL3544636

CHEMBL3544636
0.0670.1720.132Glutamate (mGluR7) agonist

0.094 0.074 CHEMBL1203

0.098 0.065 CHEMBL3544636

0.097 0.067 CHEMBL3091859

0.132 0.02 CHEMBL1237174

0.126 0.025 CHEMBL3091852

CHEMBL1237174
0.0120.1160.059Phosphoglycerate kinase inhibitor

0.059 0.011 CHEMBL1203

0.046 0.016 CHEMBL1237174

CHEMBL1203
0.0180.1220.038Ceramide glucosyltransferase inhibitor

0.038 0.021 CHEMBL3544636

0.038 0.019 CHEMBL3544637

0.038 0.021 CHEMBL1237174

CHEMBL1237174
0.0270.1320.0843(or 17)beta-hydroxysteroid dehydrogenase inhibitor

0.084 0.014 CHEMBL1203

0.074 0.019 CHEMBL1237174

0.059 0.031 CHEMBL3091852

CHEMBL1203
0.1140.2190.163Death-associated protein kinase 2 inhibitor

0.152 0.102 CHEMBL1442231

0.163 0.079 CHEMBL3091852

CHEMBL3091852
0.0190.1240.057Integrin alpha2 antagonist

0.045 0.015 CHEMBL1203

0.057 0.008 CHEMBL3544636

0.039 0.022 CHEMBL1237174

CHEMBL3544636
0.030.1350.073Neuronal nicotinic receptor antagonist

0.073 0.042 CHEMBL1203

CHEMBL1203
0.0090.1140.02CXC chemokine 5 receptor antagonist

0.02 0.009 CHEMBL1203

CHEMBL1203
0.0420.1480.085HIV-1 integrase inhibitor

0.085 0.035 CHEMBL1203

0.072 0.046 CHEMBL3544636

CHEMBL1203
0.060.1660.162Interleukin 1 beta converting enzyme inhibitor

0.086 0.079 CHEMBL3544855

0.109 0.046 CHEMBL1203

0.104 0.053 CHEMBL1442231

0.162 0.013 CHEMBL3544636

0.088 0.076 CHEMBL1237174

0.107 0.049 CHEMBL3091852

CHEMBL3544636
0.0350.1410.0835 Hydroxytryptamine 3 agonist

0.083 0.025 CHEMBL1237174

CHEMBL1237174
0.0360.1430.099Cathepsin G inhibitor

0.064 0.062 CHEMBL1203

0.069 0.055 CHEMBL3091859

0.099 0.034 CHEMBL1237174

CHEMBL1237174
0.0330.1410.0565 Hydroxytryptamine 7 agonist

0.056 0.038 CHEMBL1237174

CHEMBL1237174
0.070.1780.192Folate antagonist

0.097 0.07 CHEMBL2111041

0.159 0.019 CHEMBL3544855

0.121 0.038 CHEMBL1203

0.192 0.011 CHEMBL3544636

CHEMBL3544636
0.0510.160.165Prolactin inhibitor

0.116 0.041 CHEMBL1203

0.088 0.069 CHEMBL3091859

0.165 0.017 CHEMBL1237174

0.132 0.031 CHEMBL3091852

CHEMBL1237174
0.0330.1430.115Na+ K+ transporting ATPase inhibitor

0.082 0.048 CHEMBL1203

0.115 0.02 CHEMBL3544637

0.105 0.027 CHEMBL1237174

0.088 0.043 CHEMBL3091852

CHEMBL3544637
0.1060.2150.175MAP kinase kinase 4 inhibitor

0.131 0.11 CHEMBL3544856

0.175 0.029 CHEMBL1203

CHEMBL1203
0.0520.1620.133GABA B receptor agonist

0.071 0.066 CHEMBL2111041

0.075 0.053 CHEMBL3544855

0.133 0.005 CHEMBL1203

0.095 0.021 CHEMBL3544636

0.07 0.068 CHEMBL3091859

0.102 0.015 CHEMBL1237174

0.091 0.025 CHEMBL3091852

CHEMBL1203
0.0170.1270.035Carboxypeptidase B inhibitor

0.034 0.021 CHEMBL1203

0.035 0.019 CHEMBL3544636

0.031 0.027 CHEMBL1237174

CHEMBL3544636
0.0110.1210.196Nicotinic acid receptor agonist

0.196 0.003 CHEMBL1203

0.032 0.031 CHEMBL1237174

0.035 0.026 CHEMBL3091852

CHEMBL1203
0.0570.1670.111mTOR complex 2 inhibitor

0.082 0.063 CHEMBL1203

0.111 0.023 CHEMBL1237174

0.085 0.056 CHEMBL3091852

CHEMBL1237174
0.0180.1290.057Retinoid X alpha receptor antagonist

0.057 0.004 CHEMBL1203

0.036 0.021 CHEMBL1237174

0.031 0.03 CHEMBL3091852

CHEMBL1203
0.050.1610.083MDM2 inhibitor

0.083 0.016 CHEMBL1203

0.073 0.032 CHEMBL3091859

0.083 0.016 CHEMBL1237174

0.068 0.044 CHEMBL3091852

CHEMBL1237174
0.040.1520.069Immunoglobulin Fc receptor antagonist

0.057 0.032 CHEMBL1203

0.053 0.047 CHEMBL3091859

0.069 0.012 CHEMBL1237174

0.064 0.018 CHEMBL3091852

CHEMBL1237174
0.0090.1210.044Lysophosphatidic acid 1 receptor antagonist

0.044 0.004 CHEMBL1203

CHEMBL1203
0.0290.1420.169Heparanase inhibitor

0.073 0.01 CHEMBL1203

0.062 0.02 CHEMBL3544636

0.169 0.003 CHEMBL3544637

0.055 0.033 CHEMBL1237174

0.05 0.045 CHEMBL3091852

CHEMBL3544637
0.0160.1290.054CDK2/cyclin E inhibitor

0.054 0.049 CHEMBL3091859

CHEMBL3091859
0.0130.1280.034Integrin alpha2beta1 antagonist

0.034 0.009 CHEMBL1203

0.029 0.013 CHEMBL3544636

0.028 0.015 CHEMBL1237174

CHEMBL1203
0.0410.1560.074Ryanodine receptor antagonist

0.074 0.013 CHEMBL1203

0.055 0.054 CHEMBL3544636

0.073 0.014 CHEMBL1237174

0.058 0.042 CHEMBL3091852

CHEMBL1203
0.0360.1520.076Corticotropin releasing factor 2 receptor antagonist

0.076 0.02 CHEMBL1237174

0.064 0.038 CHEMBL3091852

CHEMBL1237174
0.010.1260.04Retinoid X beta receptor antagonist

0.04 0.003 CHEMBL1203

0.022 0.011 CHEMBL1237174

CHEMBL1203
0.020.1370.104Dihydroorotase inhibitor

0.104 0.005 CHEMBL1203

0.049 0.026 CHEMBL1237174

0.04 0.039 CHEMBL3091852

CHEMBL1203
0.0090.1260.058HCV NS5B polymerase inhibitor

0.058 0.008 CHEMBL1203

0.032 0.021 CHEMBL3544636

CHEMBL1203
0.020.1380.066Retinoid X receptor antagonist

0.066 0.004 CHEMBL1203

0.04 0.023 CHEMBL1237174

0.035 0.033 CHEMBL3091852

CHEMBL1203
0.0110.1290.161Urate transporter 1 inhibitor

0.161 0.004 CHEMBL1203

CHEMBL1203
0.0870.2070.168Sphingosine 1-phosphate receptor 2 antagonist

0.158 0.031 CHEMBL1203

0.114 0.112 CHEMBL3544636

0.133 0.068 CHEMBL3091859

0.157 0.032 CHEMBL1237174

0.168 0.023 CHEMBL3091852

CHEMBL3091852
0.0220.1420.06Prolyl endopeptidase inhibitor

0.056 0.028 CHEMBL1203

0.06 0.024 CHEMBL3544636

0.049 0.038 CHEMBL1237174

CHEMBL3544636
0.0440.1640.125Glycine receptor agonist

0.125 0.011 CHEMBL1203

0.071 0.053 CHEMBL3544636

0.085 0.033 CHEMBL3544637

0.074 0.047 CHEMBL3091859

0.122 0.012 CHEMBL1237174

0.102 0.02 CHEMBL3091852

CHEMBL1203
0.0310.1520.064Nicotinic alpha3beta2 receptor antagonist

0.058 0.029 CHEMBL1203

0.064 0.022 CHEMBL1237174

0.049 0.047 CHEMBL3091852

CHEMBL1237174
0.1610.2840.203Ca(v)3.3 blocker

0.203 0.185 CHEMBL3544636

CHEMBL3544636
0.0080.1320.033Integrin alphaVbeta3 antagonist

0.024 0.013 CHEMBL3544855

0.022 0.015 CHEMBL1442231

0.033 0.007 CHEMBL3544636

CHEMBL3544636
0.0540.1780.266Cholesterol synthesis inhibitor

0.266 0.015 CHEMBL1203

0.152 0.043 CHEMBL3544636

0.171 0.035 CHEMBL3544637

0.129 0.057 CHEMBL1237174

CHEMBL1203
0.0170.1420.046Melatonin receptor 1A agonist

0.033 0.024 CHEMBL3091859

0.037 0.017 CHEMBL1237174

0.046 0.009 CHEMBL3091852

CHEMBL3091852
0.0160.1410.131Glutamate (mGluR3) antagonist

0.131 0.004 CHEMBL1203

0.047 0.014 CHEMBL1237174

0.034 0.03 CHEMBL3091852

CHEMBL1203
0.0290.1550.053Bombesin 2 receptor antagonist

0.047 0.039 CHEMBL1203

0.053 0.029 CHEMBL3544636

0.05 0.034 CHEMBL1237174

CHEMBL3544636
0.0070.1330.106Kynurenine 3 monooxygenase inhibitor

0.106 0.004 CHEMBL1203

CHEMBL1203
0.0260.1520.064HCV NS3/NS4A protease inhibitor

0.045 0.044 CHEMBL3544636

0.047 0.039 CHEMBL3091859

0.05 0.032 CHEMBL1237174

0.064 0.018 CHEMBL3091852

CHEMBL3091852
0.0110.140.025Myristoyl transferase inhibitor

0.025 0.024 CHEMBL1237174

CHEMBL1237174
0.0180.1470.067Neutrophil collagenase inhibitor

0.062 0.048 CHEMBL3544636

0.067 0.042 CHEMBL1237174

CHEMBL1237174
0.0420.1730.097Phosphodiesterase VI inhibitor

0.08 0.041 CHEMBL1203

0.097 0.022 CHEMBL3544637

CHEMBL3544637
0.0080.1390.028Protease (Human cytomegalovirus) inhibitor

0.023 0.014 CHEMBL1203

0.025 0.012 CHEMBL1237174

0.028 0.009 CHEMBL3091852

CHEMBL3091852
0.0330.1650.091Potassium channel intermediate-conductance Ca-activated blocker

0.091 0.012 CHEMBL1203

0.074 0.023 CHEMBL1237174

0.056 0.05 CHEMBL3091852

CHEMBL1203
0.0220.1550.05Benzodiazepine antagonist

0.05 0.027 CHEMBL3091852

CHEMBL3091852
0.0070.140.028Imidazoline I1 receptor antagonist

0.028 0.008 CHEMBL1237174

CHEMBL1237174
0.030.1640.127CD45 antagonist

0.081 0.012 CHEMBL1203

0.127 0.007 CHEMBL3544636

CHEMBL3544636
0.0050.1380.058Arginase inhibitor

0.056 0.012 CHEMBL1203

0.041 0.021 CHEMBL3544636

0.058 0.011 CHEMBL3544637

0.051 0.015 CHEMBL1237174

0.044 0.019 CHEMBL3091852

CHEMBL3544637
0.0530.1880.1Bromodomain-containing protein 2 inhibitor

0.089 0.058 CHEMBL1203

0.1 0.04 CHEMBL1237174

0.095 0.047 CHEMBL3091852

CHEMBL1237174
0.0290.1640.058Bombesin 3 receptor antagonist

0.058 0.035 CHEMBL1203

CHEMBL1203
0.0560.1910.151Proteasome inhibitor

0.096 0.093 CHEMBL1442231

0.118 0.067 CHEMBL3544636

0.1 0.088 CHEMBL1237174

0.151 0.046 CHEMBL3091852

CHEMBL3091852
0.0120.1470.031Acid ceramidase inhibitor

0.031 0.008 CHEMBL1237174

0.024 0.021 CHEMBL3091852

CHEMBL1237174
0.0150.1510.076Aromatase inhibitor

0.076 0.03 CHEMBL1203

CHEMBL1203
0.060.1970.247Microtubule formation inhibitor

0.149 0.038 CHEMBL1203

0.119 0.061 CHEMBL3544636

0.247 0.009 CHEMBL3544637

0.142 0.042 CHEMBL1237174

0.116 0.065 CHEMBL3091852

CHEMBL3544637
0.0270.1650.077Squalene epoxidase inhibitor

0.06 0.021 CHEMBL1203

0.077 0.01 CHEMBL3544637

0.061 0.019 CHEMBL1237174

0.047 0.039 CHEMBL3091852

CHEMBL3544637
0.0150.1530.031Dipeptidyl peptidase II inhibitor

0.031 0.026 CHEMBL1237174

CHEMBL1237174
0.0250.1640.082Sphingosine 1-phosphate receptor 3 antagonist

0.082 0.015 CHEMBL1203

0.07 0.026 CHEMBL3544636

0.059 0.04 CHEMBL1237174

CHEMBL1203
0.0270.1670.078Syk tyrosine kinase inhibitor

0.078 0.042 CHEMBL1203

CHEMBL1203
0.0550.1940.237Alkylator

0.108 0.08 CHEMBL1203

0.127 0.061 CHEMBL3544636

0.237 0.018 CHEMBL3544637

0.131 0.058 CHEMBL1237174

0.124 0.064 CHEMBL3091852

CHEMBL3544637
0.0030.1420.023Angiotensin AT1B receptor antagonist

0.023 0.005 CHEMBL1203

CHEMBL1203
0.0210.1610.083Diacylglycerol O-acyltransferase inhibitor

0.069 0.02 CHEMBL1203

0.083 0.013 CHEMBL3544636

CHEMBL3544636
0.0910.2320.334Interferon gamma antagonist

0.256 0.027 CHEMBL1203

0.334 0.016 CHEMBL3544637

0.179 0.051 CHEMBL1237174

0.155 0.071 CHEMBL3091852

CHEMBL3544637
0.0370.1770.068Metalloproteinase-9 inhibitor

0.068 0.059 CHEMBL1237174

CHEMBL1237174
0.0310.1720.123Phosphodiesterase IV inhibitor

0.123 0.032 CHEMBL1203

CHEMBL1203
0.0430.1870.101GABA A receptor agonist

0.101 0.037 CHEMBL1203

CHEMBL1203
0.0630.2070.207Photosensitizer

0.164 0.024 CHEMBL1203

0.117 0.061 CHEMBL3544636

0.207 0.011 CHEMBL3544637

0.099 0.091 CHEMBL3091859

0.152 0.03 CHEMBL1237174

0.134 0.043 CHEMBL3091852

CHEMBL3544637
0.0340.1790.059Phosphodiesterase 1A inhibitor

0.056 0.053 CHEMBL1203

0.059 0.044 CHEMBL1237174

CHEMBL1237174
0.0030.150.019G-protein-coupled receptor 120 agonist

0.019 0.01 CHEMBL1203

CHEMBL1203
0.020.1670.099Acetylcholine M5 receptor agonist

0.099 0.021 CHEMBL1237174

0.08 0.034 CHEMBL3091852

CHEMBL1237174
0.0090.1560.053Free fatty acid receptor 1 antagonist

0.053 0.008 CHEMBL1203

0.033 0.025 CHEMBL1237174

CHEMBL1203
0.0090.1580.474Protocollagen prolyl hydroxylase inhibitor

0.056 0.005 CHEMBL1203

0.474 0.002 CHEMBL3544636

CHEMBL3544636
0.0740.2230.124Transcription factor STAT6 inhibitor

0.117 0.065 CHEMBL1203

0.124 0.053 CHEMBL1237174

0.124 0.054 CHEMBL3091852

CHEMBL3091852
0.0210.1710.049Matrix metalloproteinase (membrane-type) inhibitor

0.049 0.048 CHEMBL1237174

CHEMBL1237174
0.030.1820.084Acetylcholine nicotinic antagonist

0.084 0.05 CHEMBL1203

CHEMBL1203
0.0030.1560.027Integrin beta2 antagonist

0.011 0.01 CHEMBL1203

0.027 0.004 CHEMBL3544636

CHEMBL3544636
0.020.1730.066Beta 1 adrenoreceptor antagonist

0.052 0.043 CHEMBL1203

0.06 0.036 CHEMBL3544636

0.066 0.03 CHEMBL1237174

CHEMBL1237174
0.0920.2470.455Spasmolytic

0.251 0.09 CHEMBL1203

0.455 0.03 CHEMBL3544637

0.185 0.133 CHEMBL3091859

0.241 0.095 CHEMBL1237174

CHEMBL3544637
0.0910.2470.249Ca2+/calmodulin-dependent protein kinase kinase B inhibitor

0.249 0.006 CHEMBL1203

0.132 0.112 CHEMBL3544636

CHEMBL1203
0.0080.1660.024Prostaglandin F2 alpha agonist

0.024 0.013 CHEMBL1237174

CHEMBL1237174
0.020.1780.056TRPA1 antagonist

0.056 0.05 CHEMBL1203

CHEMBL1203
0.0420.20.086Neuropeptide Y antagonist

0.086 0.051 CHEMBL1442231

0.083 0.055 CHEMBL3091852

CHEMBL1442231
0.0190.1770.0435 Hydroxytryptamine 2B agonist

0.043 0.02 CHEMBL1237174

CHEMBL1237174
0.0030.1630.012Melatonin 2 antagonist

0.012 0.009 CHEMBL3091852

CHEMBL3091852
0.0240.1840.061Alpha adrenoreceptor agonist

0.061 0.054 CHEMBL1237174

CHEMBL1237174
0.0320.1930.074Metalloproteinase-2 inhibitor

0.074 0.059 CHEMBL3544636

CHEMBL3544636
0.0140.1760.066Fructose-1,6-bisphosphatase inhibitor

0.048 0.027 CHEMBL1203

0.066 0.014 CHEMBL1237174

CHEMBL1237174
0.0370.1990.07Phosphodiesterase 1C inhibitor

0.07 0.029 CHEMBL1203

0.059 0.052 CHEMBL1237174

0.058 0.055 CHEMBL3091852

CHEMBL1203
0.0110.1750.034Lysophosphatidic acid 2 receptor antagonist

0.034 0.017 CHEMBL1237174

0.03 0.022 CHEMBL3091852

CHEMBL1237174
0.1190.2840.795Cholesterol antagonist

0.188 0.176 CHEMBL3544855

0.634 0.014 CHEMBL1203

0.355 0.062 CHEMBL3544636

0.795 0.004 CHEMBL3544637

0.319 0.079 CHEMBL1237174

0.252 0.124 CHEMBL3091852

CHEMBL3544637
0.0230.1880.043Leukotriene C4 antagonist

0.043 0.019 CHEMBL1203

0.037 0.034 CHEMBL1237174

CHEMBL1203
0.0160.1810.095Thromboxane antagonist

0.095 0.013 CHEMBL1203

0.055 0.037 CHEMBL3544636

CHEMBL1203
0.0210.1870.067Collagenase 3 inhibitor

0.067 0.034 CHEMBL1203

0.058 0.045 CHEMBL3544636

CHEMBL1203
0.0070.1730.083Sodium/glucose cotransporter 2 inhibitor

0.083 0.004 CHEMBL3544637

0.025 0.021 CHEMBL1237174

CHEMBL3544637
0.0110.1770.069Guanylate cyclase inhibitor

0.069 0.005 CHEMBL1203

0.058 0.014 CHEMBL3544637

0.066 0.007 CHEMBL1237174

0.042 0.03 CHEMBL3091852

CHEMBL1203
0.0590.2260.152Glutamate release inhibitor

0.119 0.023 CHEMBL1203

0.152 0.009 CHEMBL3544637

0.14 0.012 CHEMBL1237174

0.103 0.038 CHEMBL3091852

CHEMBL3544637
0.0210.1890.079Leukotriene antagonist

0.079 0.033 CHEMBL1203

CHEMBL1203
0.1030.2740.644Hypoglycemic

0.551 0.011 CHEMBL2111041

0.19 0.123 CHEMBL3544855

0.282 0.059 CHEMBL3544856

0.243 0.081 CHEMBL1203

0.204 0.109 CHEMBL3544636

0.644 0.006 CHEMBL3544637

CHEMBL3544637
0.0340.2050.067Secretase beta inhibitor

0.064 0.062 CHEMBL1203

0.067 0.054 CHEMBL1237174

CHEMBL1237174
0.0150.1870.125Dihydroorotate dehydrogenase inhibitor

0.125 0.007 CHEMBL1203

CHEMBL1203
0.0070.180.053AMPA 3 receptor antagonist

0.053 0.008 CHEMBL1203

0.041 0.013 CHEMBL3544636

CHEMBL1203
0.0040.1770.0155-Alpha-reductase 1 inhibitor

0.015 0.013 CHEMBL1203

CHEMBL1203
0.0160.1890.072AMPA 4 receptor antagonist

0.072 0.008 CHEMBL1203

0.039 0.028 CHEMBL1237174

0.036 0.035 CHEMBL3091852

CHEMBL1203
0.0070.180.025-Alpha-reductase 2 inhibitor

0.02 0.013 CHEMBL1203

CHEMBL1203
0.0020.1750.009Progesterone receptor A antagonist

0.009 0.008 CHEMBL1237174

CHEMBL1237174
0.0060.180.042Glutamate (mGluR2) antagonist

0.042 0.011 CHEMBL1203

CHEMBL1203
0.0750.2490.17Neuropeptide Y1 antagonist

0.146 0.072 CHEMBL3091859

0.164 0.046 CHEMBL1237174

0.17 0.039 CHEMBL3091852

CHEMBL3091852
0.0030.1780.055Kainate receptor 1 antagonist

0.055 0.005 CHEMBL1203

CHEMBL1203
0.0210.1970.061GABA B receptor antagonist

0.061 0.012 CHEMBL1203

0.043 0.03 CHEMBL1237174

CHEMBL1203
0.0490.2250.23Carbonic anhydrase III inhibitor

0.23 0.012 CHEMBL1203

0.089 0.076 CHEMBL3544636

0.101 0.061 CHEMBL3544637

0.133 0.036 CHEMBL1237174

0.125 0.041 CHEMBL3091852

CHEMBL1203
0.060.2370.168TRPA1 agonist

0.168 0.02 CHEMBL1203

0.109 0.073 CHEMBL3544636

0.125 0.053 CHEMBL1237174

0.098 0.091 CHEMBL3091852

CHEMBL1203
0.010.1880.063Oleamide hydrolase inhibitor

0.063 0.019 CHEMBL1203

CHEMBL1203
0.040.2170.131Gastric antisecretory

0.131 0.036 CHEMBL1203

0.094 0.073 CHEMBL3544636

0.093 0.075 CHEMBL1237174

CHEMBL1203
0.0170.1960.062Phosphodiesterase 4C inhibitor

0.062 0.033 CHEMBL1203

0.06 0.034 CHEMBL1442231

CHEMBL1203
0.0090.190.111Retinoid X alpha receptor agonist

0.111 0.004 CHEMBL1203

0.034 0.025 CHEMBL1237174

CHEMBL1203
0.0610.2430.149CDK3/cyclin E inhibitor

0.103 0.082 CHEMBL1442231

0.12 0.055 CHEMBL3544636

0.149 0.027 CHEMBL3091852

CHEMBL3091852
0.0940.2760.18Prostaglandin dehydrogenase inhibitor

0.18 0.172 CHEMBL1237174

CHEMBL1237174
0.0190.2020.0635 Hydroxytryptamine 2A agonist

0.063 0.044 CHEMBL1237174

CHEMBL1237174
0.0160.2010.039DNA topoisomerase IV inhibitor

0.039 0.009 CHEMBL1203

CHEMBL1203
0.0940.2790.209Phospholipase C inhibitor

0.209 0.038 CHEMBL1203

0.193 0.049 CHEMBL3544636

0.153 0.1 CHEMBL3544637

0.144 0.12 CHEMBL3091859

0.194 0.048 CHEMBL1237174

0.183 0.058 CHEMBL3091852

CHEMBL1203
0.0470.2320.462Amylase inhibitor

0.223 0.036 CHEMBL3544856

0.196 0.046 CHEMBL1203

0.462 0.007 CHEMBL3544637

0.185 0.05 CHEMBL1237174

0.139 0.07 CHEMBL3091852

CHEMBL3544637
0.0480.2340.187Mucolytic

0.168 0.024 CHEMBL1203

0.187 0.017 CHEMBL3544636

0.185 0.017 CHEMBL3544637

0.109 0.066 CHEMBL3091859

0.141 0.038 CHEMBL1237174

0.153 0.031 CHEMBL3091852

CHEMBL3544636
0.0390.2250.084Histamine H2 receptor antagonist

0.08 0.064 CHEMBL1203

0.084 0.057 CHEMBL1237174

CHEMBL1237174
0.0080.1950.056LFA antagonist

0.042 0.007 CHEMBL1203

0.056 0.005 CHEMBL3544636

CHEMBL3544636
0.0370.2240.405Mediator release inhibitor

0.178 0.019 CHEMBL1203

0.101 0.069 CHEMBL3544636

0.405 0.005 CHEMBL3544637

0.094 0.077 CHEMBL3091852

CHEMBL3544637
0.0280.2150.089Epoxide hydrolase inhibitor

0.065 0.061 CHEMBL1203

0.089 0.033 CHEMBL3544636

CHEMBL3544636
0.0330.2210.08Potassium channel large-conductance Ca-activated activator

0.08 0.035 CHEMBL1203

CHEMBL1203
0.0120.2010.086Thromboxane A2 antagonist

0.086 0.012 CHEMBL1203

0.052 0.034 CHEMBL3544636

CHEMBL1203
0.0090.1980.065Glutamate (mGluR group II) antagonist

0.065 0.009 CHEMBL1203

CHEMBL1203
0.0540.2440.18Cytokine production inhibitor

0.18 0.043 CHEMBL1203

CHEMBL1203
0.0060.1980.018O6-alkylguanine-DNA alkyltransferase inhibitor

0.018 0.009 CHEMBL3544637

CHEMBL3544637
0.0880.280.685Antioxidant

0.277 0.071 CHEMBL2111041

0.36 0.044 CHEMBL3544855

0.158 0.156 CHEMBL1203

0.685 0.006 CHEMBL3544637

CHEMBL3544637
0.020.2120.052VCAM-1 antagonist

0.04 0.025 CHEMBL1203

0.052 0.008 CHEMBL3544636

CHEMBL3544636
0.0310.2240.152Macrophage migration inhibitory factor inhibitor

0.152 0.015 CHEMBL1203

CHEMBL1203
0.0080.2010.073Sodium/glucose cotransporter inhibitor

0.073 0.004 CHEMBL3544637

0.024 0.023 CHEMBL1237174

CHEMBL3544637
0.020.2130.052VCAM antagonist

0.04 0.025 CHEMBL1203

0.052 0.008 CHEMBL3544636

CHEMBL3544636
0.0560.250.243Interleukin 1 antagonist

0.243 0.02 CHEMBL1203

0.128 0.078 CHEMBL3544637

CHEMBL1203
0.0670.2620.158Sphingosine 1-phosphate receptor 4 antagonist

0.158 0.027 CHEMBL1203

0.137 0.046 CHEMBL1237174

0.132 0.054 CHEMBL3091852

CHEMBL1203
0.1070.3030.329Gastrin inhibitor

0.311 0.026 CHEMBL1203

0.329 0.017 CHEMBL3544636

0.208 0.136 CHEMBL3544637

0.275 0.053 CHEMBL1237174

0.255 0.074 CHEMBL3091852

CHEMBL3544636
0.0610.2570.186Interleukin 8 antagonist

0.186 0.017 CHEMBL1203

0.122 0.059 CHEMBL3544636

0.11 0.076 CHEMBL1237174

CHEMBL1203
0.0050.2020.024Fructose-1,6-bisphosphatase 1 inhibitor

0.024 0.015 CHEMBL1237174

CHEMBL1237174
0.0850.2850.194Sphingosine 1-phosphate receptor 5 antagonist

0.194 0.014 CHEMBL1203

0.128 0.106 CHEMBL3091859

0.17 0.034 CHEMBL1237174

0.167 0.037 CHEMBL3091852

CHEMBL1203
0.0610.2610.267Protein kinase stimulant

0.176 0.052 CHEMBL1203

0.267 0.022 CHEMBL3544637

0.144 0.072 CHEMBL1237174

0.134 0.08 CHEMBL3091852

CHEMBL3544637
0.0030.2040.048Egl nine homolog 2 inhibitor

0.013 0.008 CHEMBL1203

0.048 0.004 CHEMBL3544636

CHEMBL3544636
0.0060.2070.095Retinoid X receptor agonist

0.095 0.005 CHEMBL1203

CHEMBL1203
0.010.2110.032ATP citrate lysase inhibitor

0.032 0.021 CHEMBL1203

0.031 0.023 CHEMBL1237174

CHEMBL1203
0.0250.2280.116NMDA receptor agonist

0.116 0.014 CHEMBL1203

0.084 0.026 CHEMBL3544636

0.087 0.025 CHEMBL1237174

0.088 0.024 CHEMBL3091852

CHEMBL1203
0.0030.2060.014NMDA receptor phencyclidine site antagonist

0.014 0.012 CHEMBL1237174

CHEMBL1237174
0.0070.210.119TRPM8 blocker

0.119 0.005 CHEMBL1203

CHEMBL1203
0.0150.220.097NMDA receptor glycine site agonist

0.097 0.018 CHEMBL1203

0.067 0.039 CHEMBL3544636

0.058 0.048 CHEMBL3091859

0.092 0.021 CHEMBL1237174

0.096 0.019 CHEMBL3091852

CHEMBL1203
0.0670.2730.207Anticonvulsant

0.149 0.131 CHEMBL1203

0.163 0.114 CHEMBL3544636

0.181 0.098 CHEMBL3091859

0.207 0.077 CHEMBL3091852

CHEMBL3091852
0.0750.2820.138Vanilloid 1 agonist

0.122 0.082 CHEMBL1203

0.138 0.052 CHEMBL3544636

0.124 0.078 CHEMBL3544637

0.136 0.056 CHEMBL1237174

0.128 0.07 CHEMBL3091852

CHEMBL3544636
0.0040.2110.045Prostaglandin EP2 agonist

0.045 0.007 CHEMBL1203

CHEMBL1203
0.0190.2280.21Glutamate receptor agonist

0.21 0.009 CHEMBL1203

CHEMBL1203
0.0770.2860.524Non-steroidal antiinflammatory agent

0.269 0.036 CHEMBL1203

0.139 0.131 CHEMBL1442231

0.172 0.093 CHEMBL3544636

0.524 0.006 CHEMBL3544637

0.153 0.112 CHEMBL1237174

0.228 0.053 CHEMBL3091852

CHEMBL3544637
0.040.2520.148GABA receptor agonist

0.148 0.037 CHEMBL1203

0.103 0.074 CHEMBL3544636

CHEMBL1203
0.0680.280.416Interleukin agonist

0.318 0.04 CHEMBL1203

0.251 0.078 CHEMBL3544636

0.416 0.017 CHEMBL3544637

0.238 0.088 CHEMBL3091859

0.287 0.055 CHEMBL1237174

0.32 0.039 CHEMBL3091852

CHEMBL3544637
0.020.2310.061Leukotriene B4 antagonist

0.061 0.027 CHEMBL1203

0.055 0.034 CHEMBL3544637

CHEMBL1203
0.0420.2540.124Bile acid receptor antagonist

0.124 0.016 CHEMBL1203

0.101 0.046 CHEMBL3544636

0.097 0.056 CHEMBL1237174

CHEMBL1203
0.0070.220.044Liver X receptor beta antagonist

0.044 0.01 CHEMBL1203

CHEMBL1203
0.0290.2410.0555 Hydroxytryptamine 5A antagonist

0.055 0.054 CHEMBL1237174

CHEMBL1237174
0.0910.3030.365DNA damaging

0.195 0.12 CHEMBL3544855

0.245 0.083 CHEMBL1203

0.25 0.08 CHEMBL3544636

0.365 0.037 CHEMBL3544637

CHEMBL3544637
0.0180.2310.067Amidase inhibitor

0.064 0.059 CHEMBL1203

0.067 0.053 CHEMBL3544636

CHEMBL3544636
0.0630.2760.203Amyloid beta precursor protein antagonist

0.179 0.073 CHEMBL2111041

0.139 0.115 CHEMBL1203

0.203 0.055 CHEMBL3091859

CHEMBL3091859
0.0350.2490.085Caspase 7 inhibitor

0.085 0.05 CHEMBL1203

0.085 0.05 CHEMBL3544636

0.084 0.053 CHEMBL1237174

0.076 0.072 CHEMBL3091852

CHEMBL3544636
0.0110.2260.071GABA uptake inhibitor

0.071 0.007 CHEMBL1203

0.052 0.014 CHEMBL1237174

CHEMBL1203
0.0440.2620.137Caspase 3 inhibitor

0.112 0.072 CHEMBL3544855

0.129 0.047 CHEMBL1203

0.137 0.039 CHEMBL3544636

0.101 0.09 CHEMBL1237174

0.132 0.044 CHEMBL3091852

CHEMBL3544636
0.0360.2540.133Protein kinase C mu inhibitor

0.089 0.068 CHEMBL3544636

0.133 0.034 CHEMBL3544637

CHEMBL3544637
0.0370.2570.092Aminoacyl-tRNA synthetase inhibitor

0.092 0.056 CHEMBL1203

0.091 0.057 CHEMBL3544636

CHEMBL1203
0.0240.2460.069Beta adrenoreceptor antagonist

0.067 0.043 CHEMBL3544636

0.069 0.04 CHEMBL1237174

CHEMBL1237174
0.0020.2280.018Ileal bile acid transport inhibitor

0.018 0.011 CHEMBL3544637

CHEMBL3544637
0.0230.2490.127NAD(P)H dehydrogenase (quinone) inhibitor

0.127 0.027 CHEMBL1203

0.082 0.049 CHEMBL1237174

CHEMBL1203
0.0240.250.064Potassium channel (ATP-sensitive) blocker

0.064 0.052 CHEMBL1237174

CHEMBL1237174
0.110.3360.552Vasodilator, coronary

0.354 0.053 CHEMBL1203

0.27 0.114 CHEMBL3544636

0.552 0.01 CHEMBL3544637

0.276 0.108 CHEMBL1237174

0.276 0.109 CHEMBL3091852

CHEMBL3544637
0.0170.2450.037Adenosine uptake inhibitor

0.037 0.019 CHEMBL1237174

0.033 0.031 CHEMBL3091852

CHEMBL1237174
0.0110.2390.042Leukocyte elastase inhibitor

0.042 0.031 CHEMBL1203

0.041 0.032 CHEMBL3091852

CHEMBL1203
0.0330.2620.086Peroxisome proliferator-activated receptor gamma antagonist

0.086 0.027 CHEMBL1203

0.078 0.037 CHEMBL3544636

CHEMBL1203
0.0170.2460.078Phosphodiesterase 4B inhibitor

0.078 0.038 CHEMBL1203

CHEMBL1203
0.0020.2350.017Integrin alpha4beta1 antagonist

0.017 0.01 CHEMBL3544636

CHEMBL3544636
0.0060.240.078Farnesoid X receptor agonist

0.078 0.005 CHEMBL1203

CHEMBL1203
0.0050.2420.0415-Alpha-reductase inhibitor

0.041 0.023 CHEMBL1203

CHEMBL1203
0.0280.2660.1Interferon inducer

0.064 0.045 CHEMBL1203

0.1 0.013 CHEMBL3544637

0.078 0.025 CHEMBL1237174

0.065 0.042 CHEMBL3091852

CHEMBL3544637
0.0020.2410.018Prostaglandin EP4 agonist

0.018 0.009 CHEMBL1203

CHEMBL1203
0.0140.2540.074Prostaglandin-E synthase inhibitor

0.074 0.044 CHEMBL1203

CHEMBL1203
0.0270.2670.137Glycine receptor antagonist

0.092 0.04 CHEMBL1203

0.137 0.011 CHEMBL3544637

0.096 0.037 CHEMBL3091859

0.126 0.015 CHEMBL1237174

0.128 0.014 CHEMBL3091852

CHEMBL3544637
0.0280.270.085DNA helicase inhibitor

0.054 0.038 CHEMBL2111041

0.062 0.025 CHEMBL1203

0.085 0.009 CHEMBL3544636

CHEMBL3544636
0.0030.2460.031Prostaglandin E2 agonist

0.031 0.01 CHEMBL1203

CHEMBL1203
0.0510.2960.108Nav1.2 sodium channel blocker

0.108 0.099 CHEMBL3544636

CHEMBL3544636
0.0180.2630.05CC chemokine 4 receptor antagonist

0.05 0.027 CHEMBL1237174

0.043 0.039 CHEMBL3091852

CHEMBL1237174
0.0210.2670.047Beta adrenoreceptor agonist

0.047 0.026 CHEMBL1203

CHEMBL1203
0.0170.2630.079Androgen agonist

0.064 0.036 CHEMBL1237174

0.079 0.024 CHEMBL3091852

CHEMBL3091852
0.0670.3140.451Hemostatic

0.219 0.027 CHEMBL1203

0.232 0.024 CHEMBL3544636

0.451 0.005 CHEMBL3544637

0.137 0.085 CHEMBL3091852

CHEMBL3544637
0.0170.2670.134Sphingosine 1-phosphate receptor 4 agonist

0.081 0.036 CHEMBL1203

0.134 0.012 CHEMBL3544636

0.087 0.032 CHEMBL1237174

CHEMBL3544636
0.0490.2990.291Cyclooxygenase 3 inhibitor

0.171 0.033 CHEMBL1203

0.291 0.006 CHEMBL3544637

0.12 0.078 CHEMBL3091859

0.154 0.045 CHEMBL1237174

0.166 0.036 CHEMBL3091852

CHEMBL3544637
0.0730.3240.393Ca2+/calmodulin-dependent kinase I alpha inhibitor

0.215 0.08 CHEMBL1442231

0.393 0.016 CHEMBL3091852

CHEMBL3091852
0.0770.3310.148Papain-like protease (SARS coronavirus) inhibitor

0.119 0.083 CHEMBL1442231

0.115 0.094 CHEMBL3544636

0.148 0.036 CHEMBL3091852

CHEMBL3091852
0.0420.2970.148Adenylate cyclase inhibitor

0.104 0.081 CHEMBL1203

0.148 0.047 CHEMBL3544636

0.124 0.064 CHEMBL1237174

0.102 0.082 CHEMBL3091852

CHEMBL3544636
0.0430.3020.127Dual specificity tyrosine-phosphorylation regulated kinase 1B inhibitor

0.127 0.098 CHEMBL1203

CHEMBL1203
0.0050.2650.041Prostaglandin agonist

0.041 0.013 CHEMBL1203

CHEMBL1203
0.0260.2890.365Expectorant

0.149 0.036 CHEMBL1203

0.15 0.035 CHEMBL3544636

0.365 0.005 CHEMBL3544637

0.112 0.056 CHEMBL1237174

0.119 0.051 CHEMBL3091852

CHEMBL3544637
0.0930.3560.157CC chemokine 6 receptor antagonist

0.148 0.025 CHEMBL1203

0.157 0.015 CHEMBL3544637

CHEMBL3544637
0.0160.2790.056Beta 2 adrenoreceptor antagonist

0.056 0.028 CHEMBL3544636

CHEMBL3544636
0.0040.2710.033Vitronectin receptor antagonist

0.033 0.01 CHEMBL3544636

CHEMBL3544636
0.0050.2740.069Glycine transporter inhibitor

0.069 0.021 CHEMBL3544636

CHEMBL3544636
0.0050.2740.023Beta 1 adrenoreceptor agonist

0.023 0.016 CHEMBL1203

CHEMBL1203
0.0340.3050.124Cyclooxygenase 1 inhibitor

0.124 0.076 CHEMBL2111041

CHEMBL2111041
0.0230.2950.124Pim-1 kinase inhibitor

0.124 0.04 CHEMBL1203

CHEMBL1203
0.0050.2820.038Prostaglandin EP4 antagonist

0.038 0.012 CHEMBL1203

CHEMBL1203
0.0090.2860.117Glycine transporter 2 inhibitor

0.117 0.01 CHEMBL3544636

CHEMBL3544636
0.0610.3380.12Interleukin 2 antagonist

0.12 0.045 CHEMBL1203

CHEMBL1203
0.0170.2950.093NMDA receptor antagonist

0.093 0.052 CHEMBL1203

CHEMBL1203
0.0880.3670.246MAP-kinase-activated kinase 5 inhibitor

0.169 0.151 CHEMBL1442231

0.246 0.062 CHEMBL3091852

CHEMBL3091852
0.0220.3010.071Glutamate (mGluR) antagonist

0.071 0.059 CHEMBL1203

CHEMBL1203
0.0160.2990.044Aggrecanase 1 inhibitor

0.037 0.033 CHEMBL1442231

0.044 0.019 CHEMBL3091852

CHEMBL3091852
0.0330.3160.535AMP-activated protein kinase stimulant

0.184 0.014 CHEMBL1203

0.115 0.053 CHEMBL3544636

0.535 0.003 CHEMBL3544637

CHEMBL3544637
0.0230.3070.097Adrenaline agonist

0.097 0.039 CHEMBL1203

0.074 0.066 CHEMBL3544636

CHEMBL1203
0.0080.2940.259Purinergic P2Y14 antagonist

0.259 0.003 CHEMBL1203

CHEMBL1203
0.0740.3590.2Thyroid hormone antagonist

0.2 0.162 CHEMBL3544636

0.196 0.165 CHEMBL3091852

CHEMBL3544636
0.0240.3130.119Interferon agonist

0.076 0.059 CHEMBL1203

0.119 0.018 CHEMBL3544637

0.093 0.035 CHEMBL1237174

0.078 0.056 CHEMBL3091852

CHEMBL3544637
0.0340.3260.081Phosphodiesterase I inhibitor

0.081 0.075 CHEMBL1203

CHEMBL1203
0.0040.30.05Aggrecanase 2 inhibitor

0.02 0.017 CHEMBL1442231

0.05 0.005 CHEMBL3091852

CHEMBL3091852
0.0060.3030.028Integrin alphaVbeta1 antagonist

0.028 0.007 CHEMBL3544636

CHEMBL3544636
0.0060.3060.05Purinergic P2Y antagonist

0.05 0.027 CHEMBL1203

CHEMBL1203
0.0250.3280.062Beta 3 adrenoreceptor antagonist

0.062 0.05 CHEMBL1237174

CHEMBL1237174
0.0080.3120.072NMDA 2C receptor antagonist

0.072 0.031 CHEMBL1203

0.056 0.051 CHEMBL1237174

CHEMBL1203
0.0360.3430.226Beta amyloid protein antagonist

0.12 0.067 CHEMBL1203

0.108 0.08 CHEMBL3544636

0.226 0.011 CHEMBL3544637

0.099 0.091 CHEMBL1237174

CHEMBL3544637
0.0370.3440.073Calcium channel P-type blocker

0.073 0.023 CHEMBL1237174

CHEMBL1237174
0.0190.3280.06Sphingosine 1-phosphate receptor 1 antagonist

0.055 0.039 CHEMBL1203

0.06 0.03 CHEMBL3544636

CHEMBL3544636
0.0570.3670.125Polo-like kinase-3 inhibitor

0.125 0.117 CHEMBL3091852

CHEMBL3091852
0.0590.370.536Vasodilator

0.19 0.113 CHEMBL1203

0.536 0.009 CHEMBL3544637

0.467 0.014 CHEMBL3091859

0.519 0.01 CHEMBL1237174

0.456 0.015 CHEMBL3091852

CHEMBL3544637
0.0040.3160.082GP IIb/IIIa receptor antagonist

0.082 0.021 CHEMBL3544636

CHEMBL3544636
0.0260.3390.085Sphingosine 1-phosphate receptor antagonist

0.08 0.045 CHEMBL1203

0.085 0.037 CHEMBL3544636

CHEMBL3544636
0.010.3280.039Liver X receptor alpha agonist

0.039 0.032 CHEMBL1203

CHEMBL1203
0.0320.3510.149Nav1.6 sodium channel blocker

0.118 0.099 CHEMBL1203

0.149 0.056 CHEMBL1237174

CHEMBL1237174
0.0050.3280.042Peroxisome proliferator-activated receptor alpha agonist

0.042 0.039 CHEMBL1203

CHEMBL1203
0.0430.3670.128MAP3K9 inhibitor

0.12 0.114 CHEMBL3544856

0.128 0.098 CHEMBL1203

CHEMBL1203
0.0050.3310.072NMDA 2 receptor antagonist

0.072 0.05 CHEMBL1203

CHEMBL1203
0.0130.3420.088Histamine H1 receptor antagonist

0.088 0.05 CHEMBL1203

CHEMBL1203
0.0060.3360.027Calcium-sensing receptor agonist

0.027 0.018 CHEMBL1203

0.026 0.019 CHEMBL3544636

CHEMBL1203
0.0080.3390.063Phosphodiesterase 4A inhibitor

0.063 0.028 CHEMBL1203

CHEMBL1203
0.0070.3410.047Neuropeptide Y5 antagonist

0.047 0.04 CHEMBL1442231

CHEMBL1442231
0.0350.3710.199Interleukin 1b antagonist

0.199 0.019 CHEMBL1203

0.151 0.04 CHEMBL3544637

CHEMBL1203
0.0070.3440.056NMDA receptor subunit 3B antagonist

0.056 0.021 CHEMBL1203

CHEMBL1203
0.0810.4190.21Catenin beta inhibitor

0.152 0.102 CHEMBL2111041

0.21 0.025 CHEMBL3544855

0.164 0.076 CHEMBL1203

CHEMBL3544855
0.0140.3550.076Androgen antagonist

0.076 0.071 CHEMBL1237174

CHEMBL1237174
0.0050.3490.046NMDA receptor subunit 3A antagonist

0.046 0.022 CHEMBL1203

CHEMBL1203
0.0590.4090.188Thyroid hormone beta antagonist

0.184 0.17 CHEMBL3544636

0.188 0.165 CHEMBL3091852

CHEMBL3091852
0.0130.3640.226Neuraminidase (influenza) inhibitor

0.088 0.02 CHEMBL3544856

0.128 0.01 CHEMBL1203

0.063 0.048 CHEMBL1442231

0.157 0.007 CHEMBL3544637

0.186 0.005 CHEMBL3091859

0.226 0.004 CHEMBL3091852

CHEMBL3091852
0.0350.390.143Acetylcholine M1 receptor antagonist

0.143 0.082 CHEMBL1237174

0.12 0.108 CHEMBL3091852

CHEMBL1237174
0.0040.3590.039Sphingosine 1-phosphate receptor 1 agonist

0.039 0.035 CHEMBL1203

CHEMBL1203
0.0170.3730.2135-Lipoxygenase inhibitor

0.213 0.022 CHEMBL2111041

0.12 0.05 CHEMBL3544855

CHEMBL2111041
0.0180.3740.098Autotaxin inhibitor

0.098 0.013 CHEMBL1203

CHEMBL1203
0.0530.4090.426NOS3 expression enhancer

0.285 0.02 CHEMBL1203

0.426 0.007 CHEMBL3544637

CHEMBL3544637
0.0220.3810.263Topoisomerase II inhibitor

0.152 0.048 CHEMBL1203

0.263 0.023 CHEMBL3544637

CHEMBL3544637
0.0140.3740.074Protein kinase C alpha inhibitor

0.064 0.053 CHEMBL1203

0.074 0.039 CHEMBL3544637

CHEMBL3544637
0.0070.3690.052Sphingosine 1-phosphate receptor agonist

0.052 0.023 CHEMBL1203

0.047 0.028 CHEMBL3544636

CHEMBL1203
0.0430.4120.166Histone deacetylase SIRT1 inhibitor

0.112 0.101 CHEMBL1203

0.119 0.093 CHEMBL1442231

0.166 0.049 CHEMBL3544636

0.127 0.084 CHEMBL3091852

CHEMBL3544636
0.020.3910.06Beta 2 adrenoreceptor agonist

0.06 0.051 CHEMBL1237174

CHEMBL1237174
0.0210.3970.07Factor III inhibitor

0.07 0.011 CHEMBL1203

0.058 0.019 CHEMBL3544636

0.052 0.03 CHEMBL3544637

CHEMBL1203
00.3780.117Mannitol 2-dehydrogenase inhibitor

0.117 0 CHEMBL3544856

0.017 0.003 CHEMBL1203

CHEMBL3544856
0.0160.3960.101Calcium antagonist

0.101 0.047 CHEMBL1237174

CHEMBL1237174
0.0140.4050.085Nitric oxide donor

0.085 0.018 CHEMBL3544637

CHEMBL3544637
0.0340.4270.226Insulin sensitizer

0.226 0.05 CHEMBL1203

0.216 0.058 CHEMBL3544636

0.151 0.132 CHEMBL3544637

0.168 0.11 CHEMBL1237174

0.158 0.122 CHEMBL3091852

CHEMBL1203
0.0040.40.024Bombesin agonist

0.024 0.013 CHEMBL1203

CHEMBL1203
0.0060.4080.125NMDA 2D receptor antagonist

0.125 0.003 CHEMBL1203

CHEMBL1203
0.0040.4070.02Bombesin 3 receptor agonist

0.02 0.012 CHEMBL1203

CHEMBL1203
0.010.420.175Protein kinase C eta inhibitor

0.12 0.012 CHEMBL1203

0.175 0.005 CHEMBL3544637

CHEMBL3544637
0.0230.4340.139Histone deacetylase class III inhibitor

0.096 0.094 CHEMBL1203

0.139 0.053 CHEMBL3544636

CHEMBL3544636
0.0170.4290.045Integrin alpha1beta1 antagonist

0.045 0.012 CHEMBL3544636

CHEMBL3544636
0.0150.430.083Guanylate cyclase stimulant

0.083 0.008 CHEMBL1203

CHEMBL1203
0.0550.4710.424Angiogenesis inhibitor

0.193 0.178 CHEMBL1203

0.424 0.047 CHEMBL3544637

CHEMBL3544637
0.0110.430.092Anesthetic local

0.092 0.091 CHEMBL1237174

CHEMBL1237174
0.0130.4350.066Carnitine palmitoyltransferase 1B inhibitor

0.066 0.013 CHEMBL1203

CHEMBL1203
0.0160.4370.062Transcription factor AP-1 inhibitor

0.056 0.053 CHEMBL1203

0.062 0.041 CHEMBL3544637

CHEMBL3544637
0.0060.430.027Cathepsin K inhibitor

0.027 0.018 CHEMBL3091852

CHEMBL3091852
0.0050.4310.186Nicotinic acid receptor 2 agonist

0.186 0.004 CHEMBL1203

CHEMBL1203
0.0890.520.409Peptidyltransferase inhibitor

0.173 0.141 CHEMBL3544856

0.196 0.105 CHEMBL1203

0.185 0.12 CHEMBL1442231

0.321 0.018 CHEMBL3544636

0.409 0.006 CHEMBL3544637

0.19 0.112 CHEMBL3091859

0.27 0.038 CHEMBL3091852

CHEMBL3544637
0.0150.4550.298Topoisomerase I inhibitor

0.298 0.011 CHEMBL3544637

CHEMBL3544637
0.0140.4570.049DNA gyrase subunit A inhibitor

0.049 0.018 CHEMBL1203

0.045 0.024 CHEMBL1237174

CHEMBL1203
0.0060.4530.035Protein kinase C beta II inhibitor

0.035 0.017 CHEMBL1203

0.032 0.025 CHEMBL3544637

CHEMBL1203
0.0090.4640.041Protein kinase C beta I inhibitor

0.039 0.01 CHEMBL1203

0.041 0.008 CHEMBL3544637

CHEMBL3544637
0.0070.4650.063Integrin alpha5beta1 antagonist

0.063 0.011 CHEMBL3544636

CHEMBL3544636
0.0320.4950.437Antiamyloidogenic

0.22 0.086 CHEMBL1203

0.159 0.135 CHEMBL3544636

0.437 0.023 CHEMBL3544637

CHEMBL3544637
0.0770.5430.796Cyclophilin D inhibitor

0.396 0.093 CHEMBL2111041

0.409 0.086 CHEMBL1203

0.362 0.114 CHEMBL3544636

0.796 0.007 CHEMBL3544637

CHEMBL3544637
0.0070.4830.02Tryptophan hydroxylase 1 inhibitor

0.02 0.006 CHEMBL3544636

CHEMBL3544636
0.0060.4850.114Glutamate (mGluR) agonist

0.114 0.02 CHEMBL1203

CHEMBL1203
0.0120.4970.078Nav1.8 sodium channel blocker

0.078 0.045 CHEMBL1203

CHEMBL1203
0.0060.4950.193Neuraminidase inhibitor

0.077 0.028 CHEMBL3544856

0.117 0.01 CHEMBL1203

0.117 0.01 CHEMBL3544637

0.144 0.006 CHEMBL3091859

0.193 0.004 CHEMBL3091852

CHEMBL3091852
0.010.5080.037Purinergic P2Y2 antagonist

0.037 0.019 CHEMBL1203

CHEMBL1203
0.0020.5070.088Retinoic acid beta receptor antagonist

0.088 0.003 CHEMBL1203

CHEMBL1203
0.0050.5140.125Phosphodiesterase 4D inhibitor

0.125 0.026 CHEMBL1203

CHEMBL1203
0.0190.530.373Thrombolytic

0.185 0.059 CHEMBL1203

0.244 0.035 CHEMBL3544636

0.373 0.014 CHEMBL3544637

CHEMBL3544637
0.0330.5520.211Interleukin 4 antagonist

0.211 0.019 CHEMBL1203

0.123 0.081 CHEMBL3544636

0.192 0.025 CHEMBL3544637

CHEMBL1203
0.010.530.201M17 leucyl aminopeptidase inhibitor

0.161 0.049 CHEMBL1203

0.201 0.032 CHEMBL3091852

CHEMBL3091852
0.0110.5320.055Acetyl-CoA transferase 2 inhibitor

0.055 0.042 CHEMBL1203

0.054 0.045 CHEMBL3544637

CHEMBL1203
0.0130.5340.113Glucose-6-phosphate translocase inhibitor

0.063 0.021 CHEMBL1203

0.113 0.005 CHEMBL3544637

CHEMBL3544637
0.0320.5540.174Antipruritic

0.174 0.07 CHEMBL1203

CHEMBL1203
0.0220.5640.066Caspase 9 inhibitor

0.058 0.053 CHEMBL3544855

0.066 0.037 CHEMBL3544636

CHEMBL3544636
0.0040.5610.066Glutamate (mGluR2) agonist

0.066 0.01 CHEMBL1203

CHEMBL1203
0.0020.560.076Retinoic acid receptor gamma antagonist

0.076 0.003 CHEMBL1203

CHEMBL1203
0.0040.5650.041Factor XI inhibitor

0.041 0.015 CHEMBL1203

CHEMBL1203
0.0050.5710.018Guanylate cyclase 1 stimulant

0.018 0.017 CHEMBL1203

CHEMBL1203
0.0040.5730.085Aldose reductase inhibitor

0.059 0.032 CHEMBL3544636

0.085 0.021 CHEMBL3544637

CHEMBL3544637
0.0050.5780.075Glutamate (mGluR group II) agonist

0.075 0.009 CHEMBL1203

CHEMBL1203
0.020.5990.26Platelet aggregation inhibitor

0.145 0.134 CHEMBL3544855

0.206 0.077 CHEMBL1203

0.26 0.047 CHEMBL3544636

CHEMBL3544636
0.0090.5890.188Glutamate receptor antagonist

0.188 0.03 CHEMBL1203

CHEMBL1203
0.0030.5840.046VLA-4 antagonist

0.046 0.014 CHEMBL3544636

CHEMBL3544636
0.0310.6150.114Hematopoietic

0.106 0.03 CHEMBL3544856

0.093 0.045 CHEMBL1203

0.114 0.025 CHEMBL3544636

CHEMBL3544636
0.0140.6120.045Glucagon-like peptide 1 receptor antagonist

0.045 0.018 CHEMBL3544636

CHEMBL3544636
0.0040.6020.024Kainate receptor 4 antagonist

0.024 0.018 CHEMBL1203

CHEMBL1203
0.0110.6130.179Topoisomerase II alpha inhibitor

0.179 0.018 CHEMBL3544637

CHEMBL3544637
0.0030.6080.02Kainate receptor 3 antagonist

0.02 0.009 CHEMBL1203

CHEMBL1203
0.0030.6090.026Integrin alpha4beta7 antagonist

0.026 0.01 CHEMBL3544636

CHEMBL3544636
0.0130.6260.106ATPase (Vacuolar H+) inhibitor

0.086 0.064 CHEMBL3544856

0.106 0.032 CHEMBL3544637

CHEMBL3544637
0.0040.6170.021Dopamine D1 agonist

0.021 0.02 CHEMBL3544637

CHEMBL3544637
0.0070.6220.083Leukotriene synthesis inhibitor

0.07 0.044 CHEMBL3544855

0.083 0.035 CHEMBL1203

CHEMBL1203
0.0040.620.026Diacylglycerol O-acyltransferase 1 inhibitor

0.026 0.023 CHEMBL3544636

CHEMBL3544636
0.0060.6230.091Lipase inhibitor

0.091 0.033 CHEMBL3544637

CHEMBL3544637
0.0270.6490.0893C-Like protease (SARS coronavirus) inhibitor

0.089 0.048 CHEMBL1203

CHEMBL1203
0.0040.630.115Integrin antagonist

0.115 0.014 CHEMBL3544636

CHEMBL3544636
0.0030.6360.078Retinoic acid receptor antagonist

0.078 0.003 CHEMBL1203

CHEMBL1203
0.0050.6430.065Factor XIa inhibitor

0.065 0.011 CHEMBL1203

CHEMBL1203
0.0130.6620.146Dual specificity tyrosine-phosphorylation regulated kinase 2 inhibitor

0.146 0.015 CHEMBL1203

CHEMBL1203
0.0040.6580.065Microtubule stabilization

0.065 0.009 CHEMBL3544637

CHEMBL3544637
0.020.6740.186P-glycoprotein inhibitor

0.186 0.074 CHEMBL3544637

CHEMBL3544637
0.0110.6670.306Anticoagulant

0.242 0.04 CHEMBL3544636

0.306 0.027 CHEMBL3544637

CHEMBL3544637
0.0430.7010.46Sodium/bile acid cotransporter inhibitor

0.253 0.125 CHEMBL2111041

0.305 0.074 CHEMBL3544855

0.352 0.038 CHEMBL1203

0.46 0.006 CHEMBL3544636

CHEMBL3544636
0.0040.6670.033Prostacyclin antagonist

0.033 0.023 CHEMBL3544855

0.029 0.026 CHEMBL3544636

CHEMBL3544855
0.0030.670.042Kainate receptor 5 antagonist

0.042 0.006 CHEMBL1203

CHEMBL1203
0.0220.6930.071Lipocortins synthesis agonist

0.071 0.02 CHEMBL3544637

CHEMBL3544637
0.0040.680.059Protein 30S ribosomal subunit inhibitor

0.059 0.006 CHEMBL3544637

CHEMBL3544637
0.0030.680.013Integrin alphaLbeta2 antagonist

0.013 0.009 CHEMBL3544636

CHEMBL3544636
0.0130.7050.851Angiogenesis stimulant

0.219 0.085 CHEMBL1203

0.261 0.065 CHEMBL3544636

0.851 0.003 CHEMBL3544637

CHEMBL3544637
0.0150.7090.106Thioredoxin inhibitor

0.106 0.042 CHEMBL3544637

CHEMBL3544637
0.0050.7160.115Retinoic acid alpha receptor agonist

0.115 0.004 CHEMBL1203

CHEMBL1203
0.0080.7210.062Nicotinic acid receptor 1 agonist

0.062 0.015 CHEMBL1203

CHEMBL1203
0.0160.7370.166Cardiotonic

0.166 0.156 CHEMBL3544636

CHEMBL3544636
0.0090.7340.421Platelet antagonist

0.156 0.138 CHEMBL2111041

0.323 0.045 CHEMBL3544855

0.252 0.071 CHEMBL1203

0.331 0.043 CHEMBL3544636

0.421 0.023 CHEMBL3544637

CHEMBL3544637
0.0030.730.033Integrin alpha4 antagonist

0.033 0.015 CHEMBL3544636

CHEMBL3544636
0.0080.7380.091Protease inhibitor

0.091 0.073 CHEMBL3091852

CHEMBL3091852
0.0070.7370.277Cell adhesion molecule inhibitor

0.138 0.018 CHEMBL1203

0.173 0.012 CHEMBL3544636

0.277 0.005 CHEMBL3544637

CHEMBL3544637
0.0120.7450.232Interleukin antagonist

0.232 0.069 CHEMBL1203

0.152 0.116 CHEMBL3544636

CHEMBL1203
0.0190.7550.541Immunosuppressant

0.273 0.133 CHEMBL1203

0.217 0.179 CHEMBL3544636

0.541 0.023 CHEMBL3544637

CHEMBL3544637
0.0070.7450.361Lipid peroxidase inhibitor

0.361 0.012 CHEMBL3544637

CHEMBL3544637
0.0140.7530.592Tumour necrosis factor alpha release inhibitor

0.185 0.122 CHEMBL1203

0.592 0.008 CHEMBL3544637

CHEMBL3544637
0.0220.7630.159ABCA1 expression enhancer

0.159 0.015 CHEMBL1203

CHEMBL1203
0.0180.7660.134Interleukin 5 antagonist

0.134 0.016 CHEMBL1203

CHEMBL1203
0.0120.7660.189Interleukin 6 antagonist

0.189 0.048 CHEMBL3544856

0.13 0.126 CHEMBL1203

0.166 0.068 CHEMBL3544636

0.182 0.053 CHEMBL3544637

CHEMBL3544856
0.0040.7590.034AMPA 2 receptor antagonist

0.034 0.018 CHEMBL1203

CHEMBL1203
0.020.7860.098T cell inhibitor

0.098 0.026 CHEMBL3544636

CHEMBL3544636
0.0670.8340.404Calcium channel L-type activator

0.404 0.079 CHEMBL1203

0.231 0.228 CHEMBL3544636

CHEMBL1203
0.0060.7760.184Erythropoietin receptor agonist

0.184 0.007 CHEMBL3544636

CHEMBL3544636
0.010.7840.079Thioredoxin reductase inhibitor

0.079 0.065 CHEMBL1203

CHEMBL1203
0.0310.8230.101Factor V inhibitor

0.101 0.068 CHEMBL1203

CHEMBL1203
0.0020.7940.021Angiotensin AT1A receptor antagonist

0.021 0.017 CHEMBL1203

CHEMBL1203
0.0210.8160.25Transcription factor NF kappa B stimulant

0.091 0.049 CHEMBL1203

0.25 0.006 CHEMBL3544637

CHEMBL3544637
0.0030.7990.203Antineoplastic antibiotic

0.203 0.021 CHEMBL3544637

CHEMBL3544637
0.0090.8070.15Multidrug resistance-associated protein 1 inhibitor

0.104 0.072 CHEMBL1203

0.093 0.092 CHEMBL3544636

0.15 0.025 CHEMBL3544637

CHEMBL3544637
0.0040.8040.144Prostaglandin EP2 antagonist

0.144 0.01 CHEMBL1203

0.065 0.037 CHEMBL3544636

CHEMBL1203
0.0290.8350.419Caspase 3 stimulant

0.419 0.039 CHEMBL3544637

0.208 0.158 CHEMBL3091852

CHEMBL3544637
0.0110.8210.107Factor IXa inhibitor

0.05 0.038 CHEMBL1203

0.107 0.008 CHEMBL3544637

CHEMBL3544637
0.0090.8230.038Calcium-independent phospholipase A2 inhibitor

0.038 0.014 CHEMBL1203

CHEMBL1203
0.0030.8210.054Somatostatin 5 antagonist

0.054 0.011 CHEMBL1203

CHEMBL1203
0.0040.8260.045Acetyl-CoA carboxylase inhibitor

0.045 0.024 CHEMBL3091852

CHEMBL3091852
0.0070.8310.094Prostaglandin F2 alpha antagonist

0.057 0.053 CHEMBL3544855

0.094 0.014 CHEMBL1203

CHEMBL1203
0.0020.8280.062Retinoic acid alpha receptor antagonist

0.062 0.004 CHEMBL1203

CHEMBL1203
0.0030.830.055Angiotensin-converting enzyme inhibitor

0.055 0.037 CHEMBL3544636

CHEMBL3544636
0.0290.8580.166Growth hormone agonist

0.166 0.075 CHEMBL3544855

CHEMBL3544855
0.0030.8360.048Retinoic acid gamma receptor agonist

0.048 0.004 CHEMBL1203

CHEMBL1203
0.0080.8420.397Cell adhesion inhibitor

0.195 0.026 CHEMBL1203

0.249 0.015 CHEMBL3544636

0.397 0.005 CHEMBL3544637

CHEMBL3544637
0.0310.8680.278Lipocortins synthesis antagonist

0.142 0.117 CHEMBL3544855

0.278 0.026 CHEMBL1203

0.15 0.105 CHEMBL3544637

CHEMBL1203
00.840.015Antibiotic Macrolide-like

0.015 0.009 CHEMBL3544637

CHEMBL3544637
0.0030.8460.028Melatonin antagonist

0.028 0.02 CHEMBL3091852

CHEMBL3091852
0.0020.8490.017Melatonin 1 antagonist

0.017 0.016 CHEMBL3091852

CHEMBL3091852
0.0030.8580.086Retinoic acid beta receptor agonist

0.086 0.003 CHEMBL1203

CHEMBL1203
0.0030.8610.042Melatonin agonist

0.042 0.014 CHEMBL3091852

CHEMBL3091852
0.0080.8670.28Toll-Like receptor 7 agonist

0.28 0.123 CHEMBL1203

0.228 0.169 CHEMBL3544636

CHEMBL1203
0.0020.8610.067Prostaglandin EP1 antagonist

0.067 0.005 CHEMBL1203

CHEMBL1203
0.0120.8720.696Apoptosis agonist

0.289 0.181 CHEMBL3544855

0.696 0.031 CHEMBL3544637

CHEMBL3544637
0.0030.8650.101Retinoic acid receptor agonist

0.101 0.004 CHEMBL1203

CHEMBL1203
0.0040.8660.213Prostaglandin E2 antagonist

0.213 0.005 CHEMBL1203

CHEMBL1203
0.0030.8670.069Peroxisome proliferator-activated receptor gamma agonist

0.069 0.049 CHEMBL1203

CHEMBL1203
0.0020.8670.032Leukotriene B4 receptor 1 antagonist

0.032 0.016 CHEMBL1203

CHEMBL1203
0.0030.8690.058Melatonin 2 agonist

0.058 0.008 CHEMBL3091852

CHEMBL3091852
0.0030.870.042Retinoid X gamma receptor antagonist

0.042 0.004 CHEMBL1203

CHEMBL1203
0.0070.8760.273Toll-Like receptor agonist

0.273 0.129 CHEMBL1203

0.236 0.162 CHEMBL3544636

CHEMBL1203
0.0050.8730.238Protein-tyrosine phosphatase inhibitor

0.238 0.034 CHEMBL1203

0.235 0.035 CHEMBL3544637

CHEMBL1203
0.0060.8750.54Nitric oxide antagonist

0.54 0.013 CHEMBL3544637

CHEMBL3544637
0.0130.8830.24DNA polymerase I inhibitor

0.137 0.057 CHEMBL1203

0.24 0.019 CHEMBL3544637

CHEMBL3544637
0.0020.8730.1Retinoid X gamma receptor agonist

0.1 0.004 CHEMBL1203

CHEMBL1203
0.0020.880.063Leukotriene A4 hydrolase inhibitor

0.063 0.014 CHEMBL1203

CHEMBL1203
0.0040.8820.079CDC25B inhibitor

0.079 0.029 CHEMBL1203

CHEMBL1203
0.0040.8880.071Neuraminidase (Influenza A) inhibitor

0.041 0.04 CHEMBL3544856

0.068 0.008 CHEMBL1203

0.071 0.007 CHEMBL3544637

0.043 0.036 CHEMBL3091859

0.069 0.008 CHEMBL3091852

CHEMBL3544637
0.0020.8870.096Retinoid X beta receptor agonist

0.096 0.004 CHEMBL1203

CHEMBL1203
0.0090.8940.144Farnesoid X receptor antagonist

0.144 0.06 CHEMBL1203

0.119 0.106 CHEMBL3544636

CHEMBL1203
0.0030.8930.05Melatonin 1 agonist

0.05 0.009 CHEMBL3091852

CHEMBL3091852
0.0070.8990.151Bone formation stimulant

0.151 0.058 CHEMBL3544636

CHEMBL3544636
0.0050.9070.119Protein 50S ribosomal subunit inhibitor

0.119 0.009 CHEMBL3544637

0.062 0.03 CHEMBL3091852

CHEMBL3544637
0.0030.9090.063Glucagon-like peptide 1 agonist

0.063 0.046 CHEMBL3544636

CHEMBL3544636
0.0090.9160.572Immunomodulator

0.572 0.014 CHEMBL3544637

CHEMBL3544637
0.0080.9170.857Antiinflammatory

0.39 0.145 CHEMBL1203

0.857 0.009 CHEMBL3544637

CHEMBL3544637
0.0070.9230.048Glutamate (mGluR8) antagonist

0.048 0.01 CHEMBL1203

CHEMBL1203
0.0030.9260.141Prostaglandin antagonist

0.141 0.011 CHEMBL1203

CHEMBL1203
0.0010.9250.023Corticosteroid-like

0.023 0.013 CHEMBL3544637

CHEMBL3544637
0.0050.9350.214Antiobesity

0.214 0.193 CHEMBL3544637

CHEMBL3544637
0.0050.9370.034Toll-Like receptor 4 agonist

0.034 0.008 CHEMBL3544637

CHEMBL3544637
0.0290.9670.508Interleukin 2 agonist

0.224 0.151 CHEMBL3544855

0.203 0.184 CHEMBL1203

0.22 0.157 CHEMBL3544636

0.508 0.007 CHEMBL3544637

0.206 0.178 CHEMBL3091859

0.307 0.069 CHEMBL3091852

CHEMBL3544637
0.0090.9540.1Adenine nucleotide translocase inhibitor

0.1 0.005 CHEMBL1203

0.089 0.006 CHEMBL3544637

CHEMBL1203
0.010.9570.602Hepatoprotectant

0.165 0.095 CHEMBL1203

0.164 0.096 CHEMBL3544636

0.602 0.005 CHEMBL3544637

CHEMBL3544637
0.0040.9540.079Antibiotic Aminoglycoside-like

0.079 0.004 CHEMBL3544637

CHEMBL3544637
0.0080.9680.615Apoptosis antagonist

0.245 0.132 CHEMBL1203

0.276 0.103 CHEMBL3544636

0.615 0.008 CHEMBL3544637

CHEMBL3544637
0.0010.9660.042Squalene synthetase inhibitor

0.042 0.017 CHEMBL3544637

CHEMBL3544637
0.0030.9740.06Sphingosine 1-phosphate receptor 5 agonist

0.06 0.025 CHEMBL3544636

CHEMBL3544636
0.0080.9820.185Toll-Like receptor 4 antagonist

0.185 0.009 CHEMBL3544637

CHEMBL3544637
0.0040.9790.326Hypolipemic

0.15 0.136 CHEMBL1203

0.326 0.042 CHEMBL3544637

CHEMBL3544637
0.0050.9820.431Insulin secretagoues

0.212 0.03 CHEMBL1203

0.177 0.05 CHEMBL3544636

0.431 0.005 CHEMBL3544637

CHEMBL3544637
0.0030.9850.216Protein-tyrosine phosphatase 1B inhibitor

0.152 0.045 CHEMBL1203

0.216 0.025 CHEMBL3544637

CHEMBL3544637
Ext Pa Pi Pmax Activity Other Results ID Pa_max