Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.7910.0030.791Protein kinase (Mos, Mil/Raf, MEKK, RIPK, TESK, LIMK, IRAK, ILK, Activin/TGF-beta) inhibitor

0.618 0.004 CHEMBL2059159

0.286 0.009 CHEMBL2030560

0.7770.0030.777Raf kinase inhibitor

0.615 0.004 CHEMBL2059159

0.264 0.008 CHEMBL2030560

0.7480.0010.748Raf kinase C inhibitor

0.733 0.002 CHEMBL2059159

0.545 0.003 CHEMBL2030560

0.7340.0030.734Raf kinase B inhibitor

0.56 0.004 CHEMBL2059159

0.216 0.008 CHEMBL2030560

0.5960.0060.596Calcium channel L-type activator

0.484 0.034 CHEMBL2059159

0.561 0.011 CHEMBL2030560

0.4360.0050.436TIE antagonist

0.208 0.014 CHEMBL2059159

0.185 0.017 CHEMBL2030560

0.440.0180.44Antimitotic

0.239 0.064 CHEMBL2059159

0.363 0.029 CHEMBL2030560

0.4230.0050.423TIE-2 antagonist

0.197 0.015 CHEMBL2059159

0.176 0.018 CHEMBL2030560

0.3880.0290.408Calcium channel activator

0.408 0.022 CHEMBL2030560

CHEMBL2030560
0.4060.0520.406Angiogenesis inhibitor

0.214 0.154 CHEMBL2059159

0.3 0.093 CHEMBL2030560

0.3740.020.374EphB2 antagonist

0.301 0.035 CHEMBL2059159

0.154 0.125 CHEMBL2030560

0.3440.0040.344Potassium channel (Ca-activated) blocker

0.139 0.005 CHEMBL2059159

0.332 0.004 CHEMBL2030560

0.3280.0160.328Tubulin antagonist

0.177 0.045 CHEMBL2059159

0.235 0.028 CHEMBL2030560

0.3420.0480.342Hypoxia-inducible factor 1 alpha inhibitor

0.229 0.119 CHEMBL2059159

0.226 0.123 CHEMBL2030560

0.2760.0050.276Hedgehog signaling inhibitor

0.122 0.038 CHEMBL2059159

0.134 0.031 CHEMBL2030560

0.2610.0080.261Catalase inhibitor

0.202 0.015 CHEMBL2059159

0.089 0.043 CHEMBL2030560

0.2490.0090.249Microtubule formation inhibitor

0.186 0.023 CHEMBL2059159

0.128 0.053 CHEMBL2030560

0.2770.0420.277Platelet aggregation inhibitor

0.173 0.104 CHEMBL2059159

0.2410.0070.241Gastric antisecretory

0.158 0.023 CHEMBL2059159

0.161 0.022 CHEMBL2030560

0.2290.0120.534Check point kinase 2 inhibitor

0.391 0.004 CHEMBL2059159

0.534 0.004 CHEMBL2030560

CHEMBL2030560
0.2780.0730.324Insulysin inhibitor

0.324 0.045 CHEMBL2030560

CHEMBL2030560
0.3470.1480.349Caspase 9 stimulant

0.283 0.213 CHEMBL2059159

0.349 0.146 CHEMBL2030560

CHEMBL2030560
0.2890.0970.291Vasodilator, coronary

0.269 0.116 CHEMBL2059159

0.291 0.095 CHEMBL2030560

CHEMBL2030560
0.2170.0260.217ATPase inhibitor

0.213 0.028 CHEMBL2059159

0.178 0.061 CHEMBL2030560

0.2140.0230.214Platelet activating factor antagonist

0.105 0.074 CHEMBL2030560

0.290.10.418Transcription factor NF kappa B inhibitor

0.418 0.06 CHEMBL2059159

0.244 0.132 CHEMBL2030560

CHEMBL2059159
0.20.0160.2Platelet activating factor alpha antagonist

0.094 0.064 CHEMBL2059159

0.1890.0140.497HIV-1 integrase (Overall Integration) inhibitor

0.104 0.051 CHEMBL2059159

0.497 0.002 CHEMBL2030560

CHEMBL2030560
0.2110.0370.286Dual specificity tyrosine-phosphorylation regulated kinase 1B inhibitor

0.286 0.018 CHEMBL2030560

CHEMBL2030560
0.1440.0060.199Granulocyte macrophage colony stimulating factor agonist

0.122 0.015 CHEMBL2059159

0.199 0.003 CHEMBL2030560

CHEMBL2030560
0.1330.0060.156Potassium channel (ATP-sensitive) blocker

0.072 0.038 CHEMBL2059159

0.156 0.005 CHEMBL2030560

CHEMBL2030560
0.1560.0360.179Interleukin 1b antagonist

0.179 0.025 CHEMBL2030560

CHEMBL2030560
0.1730.0540.173NOS3 expression enhancer

0.162 0.062 CHEMBL2059159

0.169 0.057 CHEMBL2030560

0.1860.0720.362Interleukin-1 receptor-associated protein kinase 1 inhibitor

0.137 0.107 CHEMBL2059159

0.362 0.017 CHEMBL2030560

CHEMBL2030560
0.1310.0190.131mTOR complex 1 inhibitor

0.113 0.038 CHEMBL2059159

0.118 0.032 CHEMBL2030560

0.120.0130.12DNA gyrase inhibitor

0.104 0.017 CHEMBL2059159

0.1660.0590.407Protein kinase (CK1) gamma inhibitor

0.407 0.007 CHEMBL2030560

CHEMBL2030560
0.1220.0190.125Prostaglandin-E synthase inhibitor

0.125 0.018 CHEMBL2030560

CHEMBL2030560
0.2370.1350.378Cholesterol antagonist

0.378 0.055 CHEMBL2059159

0.211 0.155 CHEMBL2030560

CHEMBL2059159
0.160.060.203Lck kinase inhibitor

0.203 0.039 CHEMBL2030560

CHEMBL2030560
0.1540.0540.236MAP kinase kinase 4 inhibitor

0.165 0.038 CHEMBL2059159

0.236 0.006 CHEMBL2030560

CHEMBL2030560
0.1020.0050.102Factor XIa inhibitor

0.086 0.007 CHEMBL2059159

0.1180.0230.18Glutamate release inhibitor

0.18 0.005 CHEMBL2030560

CHEMBL2030560
0.1490.0580.22Interleukin 1 antagonist

0.22 0.026 CHEMBL2030560

CHEMBL2030560
0.1480.0580.152Pregnane X receptor agonist

0.152 0.05 CHEMBL2030560

CHEMBL2030560
0.2040.1150.204Cardiotonic

0.203 0.116 CHEMBL2059159

0.183 0.136 CHEMBL2030560

0.1770.090.26Growth factor agonist

0.26 0.028 CHEMBL2030560

CHEMBL2030560
0.1410.0540.141Antibacterial (Helicobacter pylori)

0.138 0.058 CHEMBL2059159

0.133 0.063 CHEMBL2030560

0.1330.050.164DNA repair enzyme inhibitor

0.164 0.021 CHEMBL2030560

CHEMBL2030560
0.1290.0460.202Protein kinase C gamma inhibitor

0.202 0.014 CHEMBL2030560

CHEMBL2030560
0.1410.0580.367Protein kinase (CK1) delta inhibitor

0.367 0.008 CHEMBL2030560

CHEMBL2030560
0.1070.0280.112Histamine H2 receptor antagonist

0.079 0.068 CHEMBL2059159

0.112 0.025 CHEMBL2030560

CHEMBL2030560
0.090.0130.159Factor IXa inhibitor

0.131 0.005 CHEMBL2059159

0.159 0.004 CHEMBL2030560

CHEMBL2030560
0.1130.0370.149Potassium channel activator

0.149 0.021 CHEMBL2059159

0.093 0.057 CHEMBL2030560

CHEMBL2059159
0.1360.060.136Vascular endothelial growth factor antagonist

0.093 0.088 CHEMBL2030560

0.1850.1110.419Aryl hydrocarbon receptor agonist

0.419 0.034 CHEMBL2030560

CHEMBL2030560
0.0920.0180.092CDK4/cyclin D1 inhibitor

0.084 0.022 CHEMBL2030560

0.1590.0890.226LIM domain kinase 1 inhibitor

0.226 0.051 CHEMBL2030560

CHEMBL2030560
0.1230.0530.138Photosensitizer

0.138 0.039 CHEMBL2030560

CHEMBL2030560
0.1730.1030.173Insulin sensitizer

0.157 0.124 CHEMBL2030560

0.1250.0580.125Vascular endothelial growth factor 2 antagonist
0.1090.0460.175CDK/cyclin complex inhibitor

0.175 0.023 CHEMBL2030560

CHEMBL2030560
0.0670.0050.067Factor XI inhibitor

0.055 0.008 CHEMBL2059159

0.0770.0230.08CDK4/cyclin D inhibitor

0.08 0.022 CHEMBL2030560

CHEMBL2030560
0.0960.0440.164Platelet growth factor antagonist

0.164 0.015 CHEMBL2030560

CHEMBL2030560
0.1810.1310.303RNA-directed DNA polymerase inhibitor

0.303 0.031 CHEMBL2030560

CHEMBL2030560
0.0530.0040.053HCV NS5A inhibitor

0.045 0.004 CHEMBL2059159

0.1140.0660.141Protein kinase (CK2) alpha inhibitor

0.089 0.088 CHEMBL2059159

0.141 0.047 CHEMBL2030560

CHEMBL2030560
0.2830.2360.406Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.406 0.096 CHEMBL2030560

CHEMBL2030560
0.0730.0270.089Transcription factor AP-1 inhibitor

0.089 0.017 CHEMBL2059159

CHEMBL2059159
0.0690.0240.069Alpha tubulin antagonist

0.06 0.03 CHEMBL2059159

0.1470.1040.17Tumour necrosis factor antagonist

0.17 0.077 CHEMBL2030560

CHEMBL2030560
0.070.0280.08Cyclin D1 inhibitor

0.08 0.018 CHEMBL2030560

CHEMBL2030560
0.0980.0570.098Proto-oncogene tyrosine-protein kinase Kit inhibitor
0.10.0630.127Cyclin-dependent kinase 9 inhibitor

0.127 0.042 CHEMBL2030560

CHEMBL2030560
0.1240.0880.368Protein kinase (CK1) inhibitor

0.368 0.01 CHEMBL2030560

CHEMBL2030560
0.1090.0750.344Protein kinase (CK1) gamma 2 inhibitor

0.344 0.006 CHEMBL2030560

CHEMBL2030560
0.0360.0050.041Acid ceramidase inhibitor

0.041 0.004 CHEMBL2030560

CHEMBL2030560
0.1480.1170.287Pyruvate kinase inhibitor

0.287 0.051 CHEMBL2030560

CHEMBL2030560
0.1350.1070.249Protein kinase (CK1) gamma 3 inhibitor

0.249 0.027 CHEMBL2030560

CHEMBL2030560
0.1080.080.189Interleukin 8 antagonist

0.189 0.016 CHEMBL2030560

CHEMBL2030560
0.030.0030.048Granulocyte colony stimulating factor receptor agonist

0.027 0.004 CHEMBL2059159

0.048 0.002 CHEMBL2030560

CHEMBL2030560
0.120.0950.209CDC-like kinase 1 inhibitor

0.209 0.031 CHEMBL2030560

CHEMBL2030560
0.1570.1330.455Aldehyde oxidase inhibitor

0.455 0.039 CHEMBL2030560

CHEMBL2030560
0.0620.0390.062Beta tubulin antagonist
0.2270.2040.227Transcription factor inhibitor
0.0480.0260.074Potassium channel small-conductance Ca-activated blocker

0.074 0.012 CHEMBL2030560

CHEMBL2030560
0.1150.0930.246Interleukin 4 antagonist

0.126 0.077 CHEMBL2059159

0.246 0.014 CHEMBL2030560

CHEMBL2030560
0.0330.0150.035Elastase 2B inhibitor

0.035 0.013 CHEMBL2030560

CHEMBL2030560
0.0330.0150.035Elastase 3A inhibitor

0.035 0.013 CHEMBL2030560

CHEMBL2030560
0.0330.0150.035Elastase 3B inhibitor

0.035 0.013 CHEMBL2030560

CHEMBL2030560
0.060.0440.099Cyclin B1 inhibitor

0.099 0.011 CHEMBL2030560

CHEMBL2030560
0.0990.0830.104CDC-like kinase 3 inhibitor

0.104 0.07 CHEMBL2030560

CHEMBL2030560
0.1060.090.212MAP kinase 12 inhibitor

0.212 0.019 CHEMBL2030560

CHEMBL2030560
0.050.0350.069Potassium channel (Inward rectifier) activator

0.069 0.012 CHEMBL2059159

0.061 0.019 CHEMBL2030560

CHEMBL2059159
0.1430.1280.143P-glycoprotein inhibitor
0.0540.040.09Cyclin B2 inhibitor

0.09 0.011 CHEMBL2030560

CHEMBL2030560
0.0480.0340.065Potassium channel (ATP-sensitive) activator

0.065 0.012 CHEMBL2059159

0.058 0.018 CHEMBL2030560

CHEMBL2059159
0.1120.0980.189Cytokine production inhibitor

0.189 0.04 CHEMBL2059159

CHEMBL2059159
0.0830.0710.083ATPase (Vacuolar H+) inhibitor
0.1410.130.282I kappa B kinase epsilon inhibitor

0.282 0.022 CHEMBL2030560

CHEMBL2030560
0.0790.0670.088Stem cell growth factor agonist

0.088 0.056 CHEMBL2030560

CHEMBL2030560
0.0750.0640.104MAP kinase kinase 7 inhibitor

0.073 0.069 CHEMBL2059159

0.104 0.01 CHEMBL2030560

CHEMBL2030560
0.0320.0210.054Cholesterol ester transfer protein antagonist

0.054 0.005 CHEMBL2059159

CHEMBL2059159
0.0920.0830.222Folate antagonist

0.093 0.079 CHEMBL2059159

0.222 0.007 CHEMBL2030560

CHEMBL2030560
0.0620.0530.062Alpha adrenoreceptor agonist

0.06 0.055 CHEMBL2030560

0.0560.0480.056Alpha 2 adrenoreceptor agonist

0.055 0.05 CHEMBL2030560

0.0480.0410.06H+/K+-transporting ATPase inhibitor

0.06 0.025 CHEMBL2030560

CHEMBL2030560
0.0510.0440.052Heparanase inhibitor

0.052 0.04 CHEMBL2030560

CHEMBL2030560
0.0160.0090.024-Hydroxyphenylpyruvate dioxygenase inhibitor

0.02 0.004 CHEMBL2030560

CHEMBL2030560
0.0590.0530.079Fibroblast growth factor 2 antagonist

0.079 0.034 CHEMBL2030560

CHEMBL2030560
0.0290.0240.029Lysophosphatidic acid 2 receptor antagonist

0.028 0.026 CHEMBL2059159

0.0750.0720.076Dual specificity tyrosine-phosphorylation regulated kinase 2 inhibitor

0.076 0.072 CHEMBL2030560

CHEMBL2030560
0.0540.0530.17CDK1/cyclin B inhibitor

0.17 0.011 CHEMBL2030560

CHEMBL2030560
0.0860.0850.157Insulin receptor antagonist

0.157 0.025 CHEMBL2030560

CHEMBL2030560
0.0490.0490.085Cyclin B inhibitor

0.085 0.013 CHEMBL2030560

CHEMBL2030560
0.2130.2140.355Antibacterial

0.355 0.099 CHEMBL2059159

0.269 0.16 CHEMBL2030560

CHEMBL2059159
0.0470.0490.078Protein kinase C eta inhibitor

0.078 0.024 CHEMBL2030560

CHEMBL2030560
0.0790.0810.123CDK2/cyclin A inhibitor

0.123 0.04 CHEMBL2030560

CHEMBL2030560
0.0140.0190.02O6-alkylguanine-DNA alkyltransferase inhibitor

0.02 0.007 CHEMBL2030560

CHEMBL2030560
0.0790.0840.106Protein kinase (CK2) inhibitor

0.106 0.059 CHEMBL2030560

CHEMBL2030560
0.240.2470.259MAP kinase 1 inhibitor

0.259 0.223 CHEMBL2030560

CHEMBL2030560
0.1390.1470.444Dyrk kinase inhibitor

0.444 0.02 CHEMBL2030560

CHEMBL2030560
0.0410.0490.058Potassium channel (Inward rectifier) blocker

0.058 0.026 CHEMBL2030560

CHEMBL2030560
0.1760.1850.226Gastrin inhibitor

0.226 0.111 CHEMBL2030560

CHEMBL2030560
0.030.0390.037Protein kinase C beta I inhibitor

0.037 0.014 CHEMBL2030560

CHEMBL2030560
0.0440.0540.134Tyrosine-protein kinase EMT inhibitor

0.134 0.011 CHEMBL2030560

CHEMBL2030560
0.0320.0430.089CDK5/p25 inhibitor

0.089 0.008 CHEMBL2030560

CHEMBL2030560
0.0070.0220.011Imidazoline I2 receptor antagonist

0.011 0.008 CHEMBL2030560

CHEMBL2030560
0.0750.0910.113Hematopoietic

0.113 0.025 CHEMBL2030560

CHEMBL2030560
0.0270.0440.074Diamine oxidase inhibitor

0.074 0.006 CHEMBL2030560

CHEMBL2030560
0.070.0890.081MAP kinase 7 inhibitor

0.081 0.042 CHEMBL2030560

CHEMBL2030560
0.0730.0910.094mTOR complex 2 inhibitor

0.094 0.04 CHEMBL2030560

CHEMBL2030560
0.0860.1050.2MAP kinase 13 inhibitor

0.2 0.021 CHEMBL2030560

CHEMBL2030560
0.0270.0470.037Protein kinase (CK2) beta inhibitor

0.037 0.017 CHEMBL2030560

CHEMBL2030560
0.0590.0790.185Protein kinase (CaMK, MLCK, PhK, SNF, KIN, NIM1, MAPKAP, POLO, CHK, ULK, RSK-2nd domain) inhibitor

0.094 0.039 CHEMBL2059159

0.185 0.015 CHEMBL2030560

CHEMBL2030560
0.0860.110.133DOPA decarboxylase inhibitor

0.133 0.032 CHEMBL2030560

CHEMBL2030560
0.0710.0960.239Cyclin-dependent kinase 1 inhibitor

0.239 0.019 CHEMBL2030560

CHEMBL2030560
0.1490.1750.236DNA damaging

0.236 0.089 CHEMBL2030560

CHEMBL2030560
0.0620.0890.099Ornithine decarboxylase inhibitor

0.099 0.046 CHEMBL2059159

CHEMBL2059159
0.0410.070.076Adenosine A2a receptor antagonist

0.076 0.034 CHEMBL2030560

CHEMBL2030560
0.2290.2590.3255 Hydroxytryptamine release inhibitor

0.325 0.139 CHEMBL2030560

CHEMBL2030560
0.0360.0690.093CDK2/cyclin E inhibitor

0.093 0.025 CHEMBL2030560

CHEMBL2030560
0.0260.0580.042Urokinase inhibitor

0.042 0.037 CHEMBL2030560

CHEMBL2030560
0.0240.0570.034Protein kinase C beta II inhibitor

0.034 0.02 CHEMBL2030560

CHEMBL2030560
0.0290.0630.051Protein kinase (CK1) epsilon inhibitor

0.051 0.012 CHEMBL2030560

CHEMBL2030560
0.1120.1460.162GABA C receptor rho-2 antagonist

0.162 0.059 CHEMBL2030560

CHEMBL2030560
0.0480.0820.149Cyclin B3 inhibitor

0.149 0.014 CHEMBL2030560

CHEMBL2030560
0.0440.0790.085Cyclin-dependent kinase 4 inhibitor

0.085 0.032 CHEMBL2030560

CHEMBL2030560
0.0350.0690.145Adenosine A1 receptor antagonist

0.145 0.016 CHEMBL2030560

CHEMBL2030560
0.060.0960.083Carbonic anhydrase VI inhibitor

0.083 0.053 CHEMBL2030560

CHEMBL2030560
0.1250.1620.427Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor

0.427 0.021 CHEMBL2030560

CHEMBL2030560
0.0470.0840.0995 Hydroxytryptamine 5A antagonist

0.099 0.016 CHEMBL2030560

CHEMBL2030560
0.0550.0970.077Adenosine A3 receptor antagonist

0.077 0.047 CHEMBL2030560

CHEMBL2030560
0.0420.0850.0895 Hydroxytryptamine 5 antagonist

0.089 0.017 CHEMBL2030560

CHEMBL2030560
0.1850.2290.22715-Lipoxygenase inhibitor

0.227 0.185 CHEMBL2030560

CHEMBL2030560
0.0480.0950.106Interferon inducer

0.064 0.045 CHEMBL2059159

0.106 0.01 CHEMBL2030560

CHEMBL2030560
0.0390.0850.08Adenosine A2 receptor antagonist

0.08 0.035 CHEMBL2030560

CHEMBL2030560
0.0070.0580.022Sodium/hydrogen exchanger inhibitor

0.022 0.008 CHEMBL2030560

CHEMBL2030560
0.0670.1190.119DNA directed RNA polymerase inhibitor

0.119 0.038 CHEMBL2030560

CHEMBL2030560
0.0280.0810.053Adenosine A2b receptor antagonist

0.053 0.031 CHEMBL2030560

CHEMBL2030560
0.0490.1030.063Transforming growth factor antagonist

0.063 0.061 CHEMBL2030560

CHEMBL2030560
0.0240.0790.049MAP3K5 inhibitor

0.049 0.013 CHEMBL2030560

CHEMBL2030560
0.090.1450.156Src kinase inhibitor

0.156 0.079 CHEMBL2030560

CHEMBL2030560
0.0440.1020.087Protein kinase C beta inhibitor

0.087 0.021 CHEMBL2030560

CHEMBL2030560
0.1310.1910.178Cyclic AMP phosphodiesterase inhibitor

0.169 0.124 CHEMBL2059159

0.178 0.114 CHEMBL2030560

CHEMBL2030560
0.070.130.202Nav1.1 sodium channel blocker

0.202 0.018 CHEMBL2030560

CHEMBL2030560
0.080.1410.232Ribosomal protein S6 kinase inhibitor

0.232 0.026 CHEMBL2030560

CHEMBL2030560
0.0530.1140.115S-adenosyl-L-methionine decarboxylase inhibitor

0.115 0.007 CHEMBL2030560

CHEMBL2030560
0.0550.1170.09Insulin growth factor antagonist

0.09 0.054 CHEMBL2030560

CHEMBL2030560
0.110.1740.147Ca2+/calmodulin-dependent protein kinase kinase B inhibitor

0.147 0.078 CHEMBL2030560

CHEMBL2030560
0.0790.1450.134CDK3/cyclin E inhibitor

0.134 0.039 CHEMBL2030560

CHEMBL2030560
0.0720.1370.172Amylase inhibitor

0.172 0.054 CHEMBL2030560

CHEMBL2030560
0.0810.1470.107Toll-Like receptor 2 antagonist

0.107 0.093 CHEMBL2030560

CHEMBL2030560
0.0720.1390.165Nav1.4 sodium channel blocker

0.165 0.028 CHEMBL2030560

CHEMBL2030560
0.1380.2060.159MAP kinase kinase 5 inhibitor

0.159 0.119 CHEMBL2030560

CHEMBL2030560
0.0520.1210.124Fibroblast growth factor 1 antagonist

0.124 0.041 CHEMBL2030560

CHEMBL2030560
0.0050.0750.013Purine nucleoside phosphorylase inhibitor

0.013 0.006 CHEMBL2030560

CHEMBL2030560
0.0240.0930.064Nicotinic acid receptor 1 agonist

0.064 0.015 CHEMBL2030560

CHEMBL2030560
0.0860.1570.346Protein kinase (CK1) gamma 1 inhibitor

0.346 0.013 CHEMBL2030560

CHEMBL2030560
0.0480.1190.111Platelet activating factor beta antagonist

0.111 0.055 CHEMBL2030560

CHEMBL2030560
0.0690.140.172Cyclin-dependent kinase inhibitor

0.172 0.046 CHEMBL2030560

CHEMBL2030560
0.1440.2160.225DNA synthesis inhibitor

0.209 0.11 CHEMBL2059159

0.225 0.088 CHEMBL2030560

CHEMBL2030560
0.0960.1680.148Arachidonic acid antagonist

0.148 0.091 CHEMBL2030560

CHEMBL2030560
0.0390.1110.124CDK1/cyclin B1 inhibitor

0.124 0.021 CHEMBL2030560

CHEMBL2030560
0.0290.1030.078p38 MAP kinase inhibitor

0.078 0.041 CHEMBL2030560

CHEMBL2030560
0.0650.1410.184Adenylate cyclase inhibitor

0.184 0.029 CHEMBL2030560

CHEMBL2030560
0.0570.1330.081Antihistaminic

0.081 0.076 CHEMBL2030560

CHEMBL2030560
0.0250.1010.075Dihydrofolate reductase inhibitor

0.075 0.005 CHEMBL2030560

CHEMBL2030560
0.050.1270.126Interferon agonist

0.071 0.068 CHEMBL2059159

0.126 0.015 CHEMBL2030560

CHEMBL2030560
0.0820.1640.402Peroxidase inhibitor

0.402 0.02 CHEMBL2030560

CHEMBL2030560
0.0590.1410.134Glycogen synthase kinase-3 beta inhibitor

0.134 0.052 CHEMBL2030560

CHEMBL2030560
0.0590.1430.136Glycogen synthase kinase-3 inhibitor

0.136 0.052 CHEMBL2030560

CHEMBL2030560
0.0120.0980.025Toll-Like receptor 8 agonist

0.025 0.007 CHEMBL2030560

CHEMBL2030560
0.0330.1190.105MAP kinase 11 inhibitor

0.105 0.033 CHEMBL2030560

CHEMBL2030560
0.0380.1250.065Benzodiazepine agonist

0.065 0.059 CHEMBL2030560

CHEMBL2030560
0.070.1580.138Adenylate kinase inhibitor

0.138 0.031 CHEMBL2030560

CHEMBL2030560
0.1230.2120.182Histone acetyltransferase inhibitor

0.182 0.097 CHEMBL2030560

CHEMBL2030560
0.0190.1070.054Antimetabolite

0.054 0.029 CHEMBL2030560

CHEMBL2030560
0.1010.1920.186DNA methylase inhibitor

0.186 0.088 CHEMBL2030560

CHEMBL2030560
0.0080.1010.018CDK2/cyclin A3 inhibitor

0.018 0.008 CHEMBL2030560

CHEMBL2030560
0.0330.1270.065MAP kinase 14 inhibitor

0.065 0.06 CHEMBL2030560

CHEMBL2030560
0.1460.240.1855 Hydroxytryptamine 3E antagonist

0.185 0.092 CHEMBL2030560

CHEMBL2030560
0.0310.1260.097CDC7 inhibitor

0.097 0.025 CHEMBL2030560

CHEMBL2030560
0.0130.1080.037CDK4/cyclin D3 inhibitor

0.037 0.011 CHEMBL2030560

CHEMBL2030560
0.0370.1330.093Protein kinase C alpha inhibitor

0.093 0.025 CHEMBL2030560

CHEMBL2030560
0.0570.1550.118NADH dehydrogenase inhibitor

0.118 0.03 CHEMBL2030560

CHEMBL2030560
0.020.1180.059Histamine H2 receptor agonist

0.059 0.015 CHEMBL2030560

CHEMBL2030560
0.090.1890.272Dual specificity tyrosine-phosphorylation regulated kinase 3 inhibitor

0.272 0.036 CHEMBL2030560

CHEMBL2030560
0.0870.1880.242Clk dual-specificity kinase inhibitor

0.242 0.058 CHEMBL2030560

CHEMBL2030560
0.0660.1670.144Cyclin-dependent kinase 7 inhibitor

0.144 0.064 CHEMBL2030560

CHEMBL2030560
0.0560.1590.147Cyclin-dependent kinase 2 inhibitor

0.147 0.039 CHEMBL2030560

CHEMBL2030560
0.1410.2440.264Nitric-oxide synthase stimulant

0.264 0.024 CHEMBL2030560

CHEMBL2030560
0.0190.1250.086Thymidylate synthase inhibitor

0.086 0.005 CHEMBL2030560

CHEMBL2030560
0.0870.1940.189Heat shock protein 90 antagonist

0.189 0.043 CHEMBL2030560

CHEMBL2030560
0.0730.1820.113Activin receptor-like kinase 2 inhibitor

0.113 0.106 CHEMBL2030560

CHEMBL2030560
0.050.1590.116Protein kinase C delta inhibitor

0.116 0.039 CHEMBL2030560

CHEMBL2030560
0.1030.2140.1523C-like protease (Human coronavirus) inhibitor

0.152 0.098 CHEMBL2030560

CHEMBL2030560
0.10.2110.321Ca2+/calmodulin-dependent protein kinase inhibitor

0.321 0.037 CHEMBL2030560

CHEMBL2030560
0.1130.2260.217Streptokinase A inhibitor

0.217 0.122 CHEMBL2030560

CHEMBL2030560
0.0350.1490.055Heat shock protein 90 beta antagonist

0.055 0.048 CHEMBL2030560

CHEMBL2030560
0.0280.1420.053Androgen agonist

0.053 0.052 CHEMBL2059159

CHEMBL2059159
0.1570.2750.424GABA C receptor rho-3 antagonist

0.424 0.052 CHEMBL2030560

CHEMBL2030560
0.0260.1440.046Aldosterone antagonist

0.046 0.035 CHEMBL2030560

CHEMBL2030560
0.0590.1790.129MAP kinase kinase 1 inhibitor

0.129 0.028 CHEMBL2059159

0.118 0.037 CHEMBL2030560

CHEMBL2059159
0.0250.1510.103Mannitol-1-phosphate 5-dehydrogenase inhibitor

0.103 0.014 CHEMBL2030560

CHEMBL2030560
0.0680.1950.161Protein kinase C nu inhibitor

0.161 0.064 CHEMBL2030560

CHEMBL2030560
0.0580.1860.089D-Ala-D-Ala ligase inhibitor

0.089 0.047 CHEMBL2030560

CHEMBL2030560
0.1550.2850.284Interleukin 2 agonist

0.284 0.086 CHEMBL2030560

CHEMBL2030560
0.1190.250.238Superoxide dismutase inhibitor

0.238 0.083 CHEMBL2030560

CHEMBL2030560
0.0130.1430.06Dihydropteroate synthase inhibitor

0.06 0.011 CHEMBL2030560

CHEMBL2030560
0.0540.1880.11Thioredoxin inhibitor

0.11 0.039 CHEMBL2030560

CHEMBL2030560
0.0420.1770.067Glycine receptor agonist

0.067 0.06 CHEMBL2030560

CHEMBL2030560
0.0090.1460.036Phosphoglycerate kinase inhibitor

0.036 0.024 CHEMBL2030560

CHEMBL2030560
0.0370.1740.128Protein kinase A inhibitor

0.128 0.031 CHEMBL2030560

CHEMBL2030560
0.0830.220.191Heat shock protein 90 alpha antagonist

0.191 0.055 CHEMBL2030560

CHEMBL2030560
0.0380.1780.15Myeloperoxidase inhibitor

0.15 0.011 CHEMBL2030560

CHEMBL2030560
0.1350.2760.214Antithrombotic

0.214 0.16 CHEMBL2059159

CHEMBL2059159
0.0790.220.138Mannose-6-phosphate isomerase inhibitor

0.138 0.076 CHEMBL2030560

CHEMBL2030560
0.1630.3040.231Ca2+/calmodulin-dependent kinase IV inhibitor

0.231 0.094 CHEMBL2030560

CHEMBL2030560
0.0270.1690.071Check point kinase 1 inhibitor

0.071 0.045 CHEMBL2030560

CHEMBL2030560
0.0530.1960.108Xanthine oxidase inhibitor

0.108 0.054 CHEMBL2030560

CHEMBL2030560
0.0550.1990.172MAP kinase kinase inhibitor

0.138 0.059 CHEMBL2059159

0.172 0.04 CHEMBL2030560

CHEMBL2030560
0.0570.2010.119Tyrosine-protein kinase receptor antagonist

0.119 0.088 CHEMBL2030560

CHEMBL2030560
0.0920.2380.163MAP kinase 3 inhibitor

0.163 0.051 CHEMBL2030560

CHEMBL2030560
0.0520.1980.11GABA C receptor rho-1 antagonist

0.11 0.049 CHEMBL2030560

CHEMBL2030560
0.0510.20.085Bromodomain-containing protein 2 inhibitor

0.085 0.066 CHEMBL2059159

CHEMBL2059159
0.0240.1750.065Histamine H4 receptor antagonist

0.065 0.015 CHEMBL2030560

CHEMBL2030560
0.0460.1970.132Protein-tyrosine kinase Lyn inhibitor

0.132 0.076 CHEMBL2030560

CHEMBL2030560
0.0250.1760.064Carbonic anhydrase stimulant

0.064 0.037 CHEMBL2030560

CHEMBL2030560
0.1050.2570.142Death-associated protein kinase 2 inhibitor

0.142 0.125 CHEMBL2030560

CHEMBL2030560
0.0460.1990.145Ferrochelatase inhibitor

0.145 0.04 CHEMBL2030560

CHEMBL2030560
0.0570.2150.111Toll-Like receptor 9 antagonist

0.111 0.097 CHEMBL2030560

CHEMBL2030560
0.080.2380.199Interleukin antagonist

0.199 0.084 CHEMBL2030560

CHEMBL2030560
0.0350.1950.082Secretase beta inhibitor

0.082 0.034 CHEMBL2030560

CHEMBL2030560
0.0350.1990.113Histamine N-methyltransferase inhibitor

0.113 0.035 CHEMBL2030560

CHEMBL2030560
0.0560.2210.13Toll-Like receptor 3 antagonist

0.13 0.023 CHEMBL2030560

CHEMBL2030560
0.020.1850.076Biliverdin reductase inhibitor

0.076 0.028 CHEMBL2030560

CHEMBL2030560
0.0290.1940.08Phospholipase D inhibitor

0.08 0.035 CHEMBL2030560

CHEMBL2030560
0.0180.1840.045Histamine H1 receptor agonist

0.045 0.028 CHEMBL2030560

CHEMBL2030560
0.1020.2680.179Proto-oncogene tyrosine-protein kinase Fyn inhibitor

0.179 0.095 CHEMBL2030560

CHEMBL2030560
0.1360.3030.223Tyrosine 3 hydroxylase inhibitor

0.223 0.099 CHEMBL2030560

CHEMBL2030560
0.0480.2170.122Protein kinase C zeta inhibitor

0.122 0.031 CHEMBL2030560

CHEMBL2030560
0.0040.1730.032Hypoxanthine phosphoribosyltransferase inhibitor

0.032 0.016 CHEMBL2030560

CHEMBL2030560
0.020.1880.073Cyclin A2 inhibitor

0.073 0.036 CHEMBL2030560

CHEMBL2030560
0.1080.280.135Ca2+-transporting ATPase inhibitor

0.135 0.096 CHEMBL2030560

CHEMBL2030560
0.0430.2180.166GABA C receptor agonist

0.166 0.028 CHEMBL2030560

CHEMBL2030560
0.0140.1890.062Xanthine dehydrogenase inhibitor

0.062 0.037 CHEMBL2030560

CHEMBL2030560
0.0350.210.143Cyclin-dependent kinase 5 inhibitor

0.143 0.044 CHEMBL2030560

CHEMBL2030560
0.1670.3420.313MAP kinase kinase 6 inhibitor

0.313 0.123 CHEMBL2030560

CHEMBL2030560
0.1260.3040.251DNA directed DNA polymerase inhibitor

0.251 0.191 CHEMBL2030560

CHEMBL2030560
0.0180.2010.056AICAR transformylase inhibitor

0.056 0.017 CHEMBL2030560

CHEMBL2030560
0.0470.230.238Dual specificity tyrosine-phosphorylation-regulated kinase 4 inhibitor

0.238 0.039 CHEMBL2030560

CHEMBL2030560
0.0220.2070.055Dopamine beta hydroxylase inhibitor

0.055 0.022 CHEMBL2030560

CHEMBL2030560
0.0490.2340.116Electrolyte absorption antagonist

0.116 0.04 CHEMBL2030560

CHEMBL2030560
0.0560.2420.159CDC-like kinase 4 inhibitor

0.159 0.094 CHEMBL2030560

CHEMBL2030560
0.0430.230.086Phosphodiesterase I inhibitor

0.086 0.065 CHEMBL2030560

CHEMBL2030560
0.0170.2080.064Cyclin A inhibitor

0.064 0.041 CHEMBL2030560

CHEMBL2030560
0.0360.2270.052Immunoglobulin Fc receptor antagonist

0.052 0.048 CHEMBL2030560

CHEMBL2030560
0.0640.2560.169Diuretic

0.169 0.062 CHEMBL2030560

CHEMBL2030560
0.0420.2350.1175 Hydroxytryptamine 3A agonist

0.117 0.059 CHEMBL2030560

CHEMBL2030560
0.1210.3150.305Ca2+/calmodulin-dependent kinase II alpha inhibitor

0.305 0.06 CHEMBL2030560

CHEMBL2030560
0.0140.2160.042Adenosine deaminase inhibitor

0.042 0.038 CHEMBL2030560

CHEMBL2030560
0.0470.2490.187CDC-like kinase 2 inhibitor

0.187 0.074 CHEMBL2030560

CHEMBL2030560
0.0190.2240.0765 Hydroxytryptamine 3A antagonist

0.076 0.035 CHEMBL2030560

CHEMBL2030560
0.1290.3350.313Histamine release inhibitor

0.242 0.161 CHEMBL2059159

0.313 0.117 CHEMBL2030560

CHEMBL2030560
0.0390.2450.091Uric acid excretion stimulant

0.091 0.063 CHEMBL2030560

CHEMBL2030560
0.030.2380.094Adrenaline agonist

0.094 0.042 CHEMBL2059159

CHEMBL2059159
0.020.2310.172Phenylalanine 4-hydroxylase inhibitor

0.172 0.009 CHEMBL2030560

CHEMBL2030560
0.1370.3480.2045 Hydroxytryptamine uptake stimulant

0.204 0.143 CHEMBL2030560

CHEMBL2030560
0.1060.3180.131Heat shock protein 70 antagonist

0.131 0.114 CHEMBL2030560

CHEMBL2030560
0.0280.2420.097MAP kinase kinase kinase inhibitor

0.097 0.069 CHEMBL2030560

CHEMBL2030560
0.0170.2350.063Histamine agonist

0.063 0.024 CHEMBL2030560

CHEMBL2030560
0.0290.2480.082I kappa B kinase inhibitor

0.082 0.058 CHEMBL2030560

CHEMBL2030560
0.0520.270.098Nav1.5 sodium channel blocker

0.098 0.09 CHEMBL2030560

CHEMBL2030560
0.0460.2690.091Interleukin 5 antagonist

0.091 0.053 CHEMBL2030560

CHEMBL2030560
0.0040.2280.017Histamine H4 receptor agonist

0.017 0.015 CHEMBL2030560

CHEMBL2030560
0.0140.2410.083Argininosuccinate synthase inhibitor

0.083 0.024 CHEMBL2030560

CHEMBL2030560
0.0360.2670.115 Hydroxytryptamine 2B antagonist

0.11 0.072 CHEMBL2030560

CHEMBL2030560
0.0430.2750.116Beta amyloid protein antagonist

0.116 0.071 CHEMBL2030560

CHEMBL2030560
0.0330.2640.155Glycogen synthase kinase-3 alpha inhibitor

0.155 0.063 CHEMBL2030560

CHEMBL2030560
0.0310.2640.091Polo-like kinase-4 inhibitor

0.091 0.086 CHEMBL2030560

CHEMBL2030560
0.0190.2550.072Porphobilinogen synthase inhibitor

0.072 0.054 CHEMBL2030560

CHEMBL2030560
0.0270.2680.131Alcohol dehydrogenase inhibitor

0.131 0.028 CHEMBL2030560

CHEMBL2030560
0.0620.3030.22MAP kinase kinase 2 inhibitor

0.22 0.07 CHEMBL2030560

CHEMBL2030560
0.0380.2830.083GABA B receptor agonist

0.083 0.036 CHEMBL2030560

CHEMBL2030560
0.0520.2970.155TRKC antagonist

0.155 0.097 CHEMBL2030560

CHEMBL2030560
0.0450.2940.098Activin receptor-like kinase 4 inhibitor

0.098 0.09 CHEMBL2030560

CHEMBL2030560
0.0020.2630.009Phosphoribosylglycinamide formyltransferase inhibitor

0.009 0.004 CHEMBL2030560

CHEMBL2030560
0.0750.340.154Focal adhesion kinase 2 inhibitor

0.154 0.125 CHEMBL2030560

CHEMBL2030560
0.0230.2890.082Inducible nitric-oxide synthase inhibitor

0.082 0.059 CHEMBL2030560

CHEMBL2030560
0.0330.3020.105GABA C receptor antagonist

0.105 0.07 CHEMBL2030560

CHEMBL2030560
0.0380.3080.139Psychostimulant

0.139 0.126 CHEMBL2030560

CHEMBL2030560
0.0130.2940.038Tryptophan 5 hydroxylase inhibitor

0.038 0.019 CHEMBL2030560

CHEMBL2030560
0.0560.3390.294Interleukin agonist

0.294 0.051 CHEMBL2030560

CHEMBL2030560
0.0560.3390.158Hexokinase inhibitor

0.158 0.07 CHEMBL2030560

CHEMBL2030560
0.0590.3530.159Polo-like kinase-3 inhibitor

0.159 0.075 CHEMBL2030560

CHEMBL2030560
0.0340.3280.206Ca2+/calmodulin-dependent kinase II gamma inhibitor

0.206 0.061 CHEMBL2030560

CHEMBL2030560
0.0110.3060.063Phosphofructokinase-1 inhibitor

0.063 0.054 CHEMBL2030560

CHEMBL2030560
0.0140.3240.056Bromodomain-containing protein 4 inhibitor

0.056 0.036 CHEMBL2059159

CHEMBL2059159
0.0280.340.118Ca2+/calmodulin-dependent kinase II delta inhibitor

0.118 0.085 CHEMBL2030560

CHEMBL2030560
0.0360.3520.13DNA polymerase I inhibitor

0.13 0.061 CHEMBL2030560

CHEMBL2030560
0.0660.3860.166Neurotrophic factor enhancer

0.166 0.115 CHEMBL2030560

CHEMBL2030560
0.0250.3470.082Glutamate dehydrogenase inhibitor

0.082 0.043 CHEMBL2030560

CHEMBL2030560
0.0260.3490.123Nitric-oxide synthase inhibitor

0.123 0.036 CHEMBL2030560

CHEMBL2030560
0.0460.3710.14Cyclin-dependent kinase 8 inhibitor

0.14 0.09 CHEMBL2030560

CHEMBL2030560
0.0830.4140.1795 Hydroxytryptamine release stimulant

0.179 0.142 CHEMBL2030560

CHEMBL2030560
0.0440.3890.08T cell inhibitor

0.08 0.068 CHEMBL2030560

CHEMBL2030560
0.0750.4330.197MAP-kinase-activated kinase 5 inhibitor

0.197 0.107 CHEMBL2030560

CHEMBL2030560
0.0450.4180.195Ca2+/calmodulin-dependent kinase II beta inhibitor

0.195 0.08 CHEMBL2030560

CHEMBL2030560
0.0370.4180.11Nav1.2 sodium channel blocker

0.11 0.096 CHEMBL2030560

CHEMBL2030560
0.0470.4280.148Antipruritic

0.148 0.097 CHEMBL2030560

CHEMBL2030560
0.1130.5260.331MAP kinase kinase 3 inhibitor

0.331 0.004 CHEMBL2059159

0.194 0.142 CHEMBL2030560

CHEMBL2059159
0.0690.4860.232Immunomodulator

0.232 0.13 CHEMBL2030560

CHEMBL2030560
0.030.4540.16Death-associated protein kinase 3 inhibitor

0.16 0.108 CHEMBL2030560

CHEMBL2030560
0.030.4660.142Phosphodiesterase 7B inhibitor

0.142 0.025 CHEMBL2030560

CHEMBL2030560
0.0080.4560.077Dopamine transporter inhibitor

0.077 0.018 CHEMBL2059159

CHEMBL2059159
0.0520.5050.171Ca2+/calmodulin-dependent kinase I alpha inhibitor

0.171 0.117 CHEMBL2030560

CHEMBL2030560
0.010.4930.068Adrenaline uptake inhibitor

0.068 0.037 CHEMBL2059159

CHEMBL2059159
Ext Pa Pi Pmax Activity Other Results ID Pa_max