| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.582 | 0.008 | 0.636 | Anticonvulsant | 0.192 0.089 CHEMBL3544797 0.338 0.031 CHEMBL3544834 0.383 0.024 CHEMBL3544836 0.283 0.045 CHEMBL3544798 0.251 0.057 CHEMBL3544835 0.636 0.005 CHEMBL3544833 | CHEMBL3544833 | |
| 0.544 | 0.008 | 0.622 | Psychostimulant | 0.403 0.022 CHEMBL3544797 0.436 0.017 CHEMBL3544834 0.622 0.005 CHEMBL3544836 0.369 0.028 CHEMBL3544798 0.461 0.015 CHEMBL3544835 0.309 0.04 CHEMBL3544799 0.544 0.008 CHEMBL3544833 | CHEMBL3544836 | |
| 0.509 | 0.032 | 0.654 | Aldehyde oxidase inhibitor | 0.654 0.012 CHEMBL3544797 0.31 0.064 CHEMBL3544834 0.578 0.022 CHEMBL3544836 0.488 0.034 CHEMBL3544798 0.376 0.051 CHEMBL3544835 0.402 0.047 CHEMBL3544833 | CHEMBL3544797 | |
| 0.478 | 0.044 | 0.491 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.43 0.076 CHEMBL3544797 0.491 0.038 CHEMBL3544834 0.365 0.134 CHEMBL3544836 0.402 0.098 CHEMBL3544798 0.448 0.063 CHEMBL3544835 0.395 0.105 CHEMBL3544833 | CHEMBL3544834 | |
| 0.446 | 0.012 | 0.522 | Anesthetic general | 0.522 0.007 CHEMBL3544797 0.411 0.015 CHEMBL3544834 0.505 0.008 CHEMBL3544836 0.44 0.012 CHEMBL3544798 0.345 0.025 CHEMBL3544835 0.438 0.012 CHEMBL3544799 0.39 0.018 CHEMBL3544833 | CHEMBL3544797 | |
| 0.394 | 0.001 | 0.522 | p53 inhibitor | 0.05 0.014 CHEMBL3544797 0.066 0.006 CHEMBL3544836 0.282 0.001 CHEMBL3544798 0.11 0.003 CHEMBL3544799 0.522 0.001 CHEMBL3544833 | CHEMBL3544833 | |
| 0.409 | 0.025 | 0.568 | Interleukin 2 agonist | 0.398 0.028 CHEMBL3544797 0.382 0.033 CHEMBL3544834 0.474 0.011 CHEMBL3544836 0.413 0.024 CHEMBL3544798 0.46 0.014 CHEMBL3544835 0.568 0.004 CHEMBL3544799 0.479 0.011 CHEMBL3544833 | CHEMBL3544799 | |
| 0.428 | 0.05 | 0.458 | GABA C receptor rho-3 antagonist | 0.386 0.068 CHEMBL3544797 0.458 0.039 CHEMBL3544834 0.326 0.099 CHEMBL3544836 0.32 0.103 CHEMBL3544798 0.341 0.091 CHEMBL3544835 0.351 0.085 CHEMBL3544833 | CHEMBL3544834 | |
| 0.376 | 0.011 | 0.406 | Lipocortins synthesis antagonist | 0.357 0.013 CHEMBL3544797 0.406 0.008 CHEMBL3544834 0.356 0.013 CHEMBL3544836 0.33 0.016 CHEMBL3544798 0.335 0.015 CHEMBL3544835 0.266 0.029 CHEMBL3544799 0.364 0.012 CHEMBL3544833 | CHEMBL3544834 | |
| 0.424 | 0.066 | 0.6 | Calcium channel L-type activator | 0.328 0.134 CHEMBL3544797 0.426 0.065 CHEMBL3544834 0.533 0.017 CHEMBL3544836 0.453 0.049 CHEMBL3544798 0.6 0.005 CHEMBL3544835 0.275 0.18 CHEMBL3544799 0.446 0.053 CHEMBL3544833 | CHEMBL3544835 | |
| 0.367 | 0.03 | 0.414 | Sodium/bile acid cotransporter inhibitor | 0.414 0.013 CHEMBL3544797 0.375 0.026 CHEMBL3544836 0.237 0.143 CHEMBL3544798 0.293 0.086 CHEMBL3544835 0.362 0.033 CHEMBL3544833 | CHEMBL3544797 | |
| 0.43 | 0.094 | 0.545 | Caspase 9 stimulant | 0.545 0.046 CHEMBL3544797 0.45 0.083 CHEMBL3544834 0.443 0.087 CHEMBL3544836 0.48 0.068 CHEMBL3544798 0.494 0.062 CHEMBL3544835 0.462 0.077 CHEMBL3544799 0.45 0.083 CHEMBL3544833 | CHEMBL3544797 | |
| 0.402 | 0.077 | 0.52 | 5 Hydroxytryptamine release inhibitor | 0.426 0.063 CHEMBL3544797 0.52 0.027 CHEMBL3544834 0.35 0.115 CHEMBL3544836 0.45 0.051 CHEMBL3544798 0.496 0.034 CHEMBL3544835 0.396 0.081 CHEMBL3544799 0.439 0.057 CHEMBL3544833 | CHEMBL3544834 | |
| 0.326 | 0.003 | 0.326 | GABA aminotransferase inhibitor | 0.148 0.008 CHEMBL3544797 0.161 0.006 CHEMBL3544834 0.229 0.004 CHEMBL3544836 0.184 0.005 CHEMBL3544798 0.137 0.01 CHEMBL3544835 0.205 0.004 CHEMBL3544799 0.308 0.003 CHEMBL3544833 | ||
| 0.343 | 0.031 | 0.563 | Interleukin agonist | 0.359 0.027 CHEMBL3544797 0.325 0.037 CHEMBL3544834 0.405 0.018 CHEMBL3544836 0.35 0.029 CHEMBL3544798 0.427 0.015 CHEMBL3544835 0.563 0.006 CHEMBL3544799 0.429 0.015 CHEMBL3544833 | CHEMBL3544799 | |
| 0.348 | 0.037 | 0.383 | Ca2+/calmodulin-dependent kinase II alpha inhibitor | 0.345 0.038 CHEMBL3544797 0.383 0.025 CHEMBL3544834 0.338 0.041 CHEMBL3544836 0.29 0.071 CHEMBL3544798 0.267 0.091 CHEMBL3544835 0.26 0.097 CHEMBL3544833 | CHEMBL3544834 | |
| 0.345 | 0.04 | 0.465 | Cardiotonic | 0.223 0.1 CHEMBL3544797 0.465 0.019 CHEMBL3544834 0.338 0.043 CHEMBL3544836 0.189 0.13 CHEMBL3544798 0.32 0.048 CHEMBL3544835 0.19 0.129 CHEMBL3544833 | CHEMBL3544834 | |
| 0.31 | 0.007 | 0.47 | Ferrochelatase inhibitor | 0.303 0.007 CHEMBL3544797 0.267 0.011 CHEMBL3544834 0.288 0.009 CHEMBL3544836 0.254 0.013 CHEMBL3544798 0.47 0.003 CHEMBL3544835 0.405 0.004 CHEMBL3544833 | CHEMBL3544835 | |
| 0.354 | 0.056 | 0.385 | 5 Hydroxytryptamine release stimulant | 0.385 0.049 CHEMBL3544797 0.314 0.066 CHEMBL3544834 0.365 0.053 CHEMBL3544836 0.245 0.091 CHEMBL3544798 0.272 0.079 CHEMBL3544835 0.17 0.152 CHEMBL3544799 0.234 0.097 CHEMBL3544833 | CHEMBL3544797 | |
| 0.315 | 0.019 | 0.334 | Ca2+/calmodulin-dependent kinase IV inhibitor | 0.283 0.034 CHEMBL3544797 0.334 0.014 CHEMBL3544834 0.283 0.035 CHEMBL3544836 0.267 0.047 CHEMBL3544798 0.284 0.034 CHEMBL3544835 0.251 0.064 CHEMBL3544833 | CHEMBL3544834 | |
| 0.322 | 0.046 | 0.52 | Tumour necrosis factor alpha release inhibitor | 0.379 0.031 CHEMBL3544797 0.388 0.029 CHEMBL3544834 0.412 0.025 CHEMBL3544836 0.249 0.075 CHEMBL3544798 0.304 0.052 CHEMBL3544835 0.52 0.012 CHEMBL3544799 0.227 0.088 CHEMBL3544833 | CHEMBL3544799 | |
| 0.309 | 0.038 | 0.413 | Cyclic AMP phosphodiesterase inhibitor | 0.308 0.039 CHEMBL3544797 0.288 0.047 CHEMBL3544834 0.317 0.036 CHEMBL3544836 0.272 0.054 CHEMBL3544798 0.413 0.015 CHEMBL3544835 0.325 0.033 CHEMBL3544799 0.307 0.039 CHEMBL3544833 | CHEMBL3544835 | |
| 0.322 | 0.071 | 0.406 | Calcium channel activator | 0.336 0.059 CHEMBL3544797 0.332 0.063 CHEMBL3544834 0.309 0.083 CHEMBL3544836 0.296 0.096 CHEMBL3544798 0.406 0.023 CHEMBL3544835 0.404 0.023 CHEMBL3544833 | CHEMBL3544835 | |
| 0.295 | 0.045 | 0.417 | DNA synthesis inhibitor | 0.38 0.024 CHEMBL3544797 0.264 0.058 CHEMBL3544834 0.417 0.02 CHEMBL3544836 0.271 0.055 CHEMBL3544798 0.317 0.038 CHEMBL3544835 0.4 0.021 CHEMBL3544799 0.288 0.048 CHEMBL3544833 | CHEMBL3544836 | |
| 0.315 | 0.074 | 0.635 | Immunomodulator | 0.285 0.091 CHEMBL3544797 0.537 0.018 CHEMBL3544834 0.478 0.026 CHEMBL3544836 0.412 0.04 CHEMBL3544798 0.37 0.053 CHEMBL3544835 0.635 0.009 CHEMBL3544799 0.277 0.096 CHEMBL3544833 | CHEMBL3544799 | |
| 0.254 | 0.022 | 0.496 | Alpha-N-acetylglucosaminidase inhibitor | 0.474 0.006 CHEMBL3544797 0.254 0.022 CHEMBL3544834 0.496 0.005 CHEMBL3544836 0.375 0.01 CHEMBL3544798 0.361 0.011 CHEMBL3544835 0.48 0.006 CHEMBL3544799 0.41 0.008 CHEMBL3544833 | CHEMBL3544836 | |
| 0.313 | 0.083 | 0.647 | Cholesterol antagonist | 0.419 0.046 CHEMBL3544797 0.221 0.147 CHEMBL3544834 0.465 0.038 CHEMBL3544836 0.274 0.109 CHEMBL3544798 0.302 0.09 CHEMBL3544835 0.647 0.013 CHEMBL3544799 0.299 0.092 CHEMBL3544833 | CHEMBL3544799 | |
| 0.31 | 0.092 | 0.484 | Vasodilator, peripheral | 0.405 0.053 CHEMBL3544797 0.252 0.125 CHEMBL3544834 0.484 0.031 CHEMBL3544836 0.215 0.159 CHEMBL3544798 0.342 0.077 CHEMBL3544835 0.332 0.082 CHEMBL3544799 0.272 0.112 CHEMBL3544833 | CHEMBL3544836 | |
| 0.226 | 0.008 | 0.29 | Glutamate (mGluR) agonist | 0.29 0.005 CHEMBL3544797 0.204 0.009 CHEMBL3544834 0.11 0.021 CHEMBL3544836 0.15 0.014 CHEMBL3544798 0.13 0.017 CHEMBL3544835 0.18 0.011 CHEMBL3544833 | CHEMBL3544797 | |
| 0.263 | 0.056 | 0.315 | Tyrosine 3 hydroxylase inhibitor | 0.248 0.069 CHEMBL3544797 0.288 0.039 CHEMBL3544834 0.269 0.052 CHEMBL3544836 0.252 0.066 CHEMBL3544798 0.241 0.077 CHEMBL3544835 0.315 0.027 CHEMBL3544833 | CHEMBL3544833 | |
| 0.268 | 0.065 | 0.305 | 5 Hydroxytryptamine uptake stimulant | 0.283 0.055 CHEMBL3544797 0.305 0.042 CHEMBL3544834 0.299 0.045 CHEMBL3544836 0.202 0.147 CHEMBL3544798 0.238 0.093 CHEMBL3544835 0.26 0.072 CHEMBL3544833 | CHEMBL3544834 | |
| 0.244 | 0.053 | 0.346 | RNA-directed DNA polymerase inhibitor | 0.346 0.024 CHEMBL3544797 0.247 0.051 CHEMBL3544834 0.312 0.029 CHEMBL3544836 0.22 0.074 CHEMBL3544798 0.224 0.069 CHEMBL3544835 0.189 0.117 CHEMBL3544799 0.213 0.081 CHEMBL3544833 | CHEMBL3544797 | |
| 0.213 | 0.023 | 0.213 | GABA C receptor rho-2 antagonist | 0.18 0.042 CHEMBL3544797 0.18 0.042 CHEMBL3544834 0.195 0.032 CHEMBL3544836 0.159 0.062 CHEMBL3544798 0.151 0.072 CHEMBL3544835 0.164 0.056 CHEMBL3544833 | ||
| 0.207 | 0.019 | 0.516 | GABA C receptor agonist | 0.197 0.021 CHEMBL3544797 0.196 0.021 CHEMBL3544834 0.247 0.014 CHEMBL3544836 0.216 0.018 CHEMBL3544798 0.209 0.019 CHEMBL3544835 0.516 0.004 CHEMBL3544833 | CHEMBL3544833 | |
| 0.229 | 0.049 | 0.285 | Nitric-oxide synthase stimulant | 0.285 0.016 CHEMBL3544797 0.253 0.03 CHEMBL3544834 0.253 0.03 CHEMBL3544836 0.203 0.084 CHEMBL3544798 0.25 0.032 CHEMBL3544835 0.187 0.113 CHEMBL3544799 0.198 0.093 CHEMBL3544833 | CHEMBL3544797 | |
| 0.292 | 0.128 | 0.499 | Histamine release inhibitor | 0.329 0.109 CHEMBL3544797 0.418 0.066 CHEMBL3544834 0.335 0.107 CHEMBL3544836 0.35 0.1 CHEMBL3544798 0.407 0.072 CHEMBL3544835 0.499 0.029 CHEMBL3544799 0.424 0.063 CHEMBL3544833 | CHEMBL3544799 | |
| 0.179 | 0.018 | 0.204 | GABA C receptor antagonist | 0.165 0.023 CHEMBL3544797 0.15 0.03 CHEMBL3544834 0.18 0.018 CHEMBL3544836 0.14 0.036 CHEMBL3544798 0.149 0.03 CHEMBL3544835 0.204 0.012 CHEMBL3544833 | CHEMBL3544833 | |
| 0.177 | 0.028 | 0.224 | Adenylate cyclase stimulant | 0.224 0.006 CHEMBL3544797 0.18 0.026 CHEMBL3544834 0.192 0.017 CHEMBL3544836 0.186 0.022 CHEMBL3544798 0.215 0.008 CHEMBL3544835 0.146 0.07 CHEMBL3544799 0.194 0.016 CHEMBL3544833 | CHEMBL3544797 | |
| 0.236 | 0.096 | 0.29 | Gastrin inhibitor | 0.258 0.07 CHEMBL3544797 0.272 0.056 CHEMBL3544834 0.231 0.104 CHEMBL3544836 0.216 0.125 CHEMBL3544798 0.208 0.138 CHEMBL3544835 0.29 0.04 CHEMBL3544833 | CHEMBL3544833 | |
| 0.163 | 0.025 | 0.418 | UDP-glucose 4-epimerase inhibitor | 0.321 0.009 CHEMBL3544797 0.221 0.016 CHEMBL3544834 0.319 0.009 CHEMBL3544836 0.232 0.015 CHEMBL3544798 0.205 0.017 CHEMBL3544835 0.418 0.005 CHEMBL3544799 0.162 0.025 CHEMBL3544833 | CHEMBL3544799 | |
| 0.158 | 0.022 | 0.423 | DNA directed RNA polymerase inhibitor | 0.423 0.005 CHEMBL3544797 0.119 0.038 CHEMBL3544834 0.155 0.023 CHEMBL3544836 0.086 0.075 CHEMBL3544798 0.09 0.07 CHEMBL3544835 0.084 0.078 CHEMBL3544833 | CHEMBL3544797 | |
| 0.155 | 0.019 | 0.176 | GABA C receptor rho-1 antagonist | 0.129 0.033 CHEMBL3544797 0.124 0.036 CHEMBL3544834 0.152 0.02 CHEMBL3544836 0.115 0.045 CHEMBL3544798 0.121 0.039 CHEMBL3544835 0.176 0.013 CHEMBL3544833 | CHEMBL3544833 | |
| 0.183 | 0.051 | 0.218 | Arachidonic acid antagonist | 0.218 0.018 CHEMBL3544797 0.207 0.027 CHEMBL3544834 0.177 0.057 CHEMBL3544836 0.198 0.035 CHEMBL3544798 0.183 0.05 CHEMBL3544835 0.213 0.022 CHEMBL3544833 | CHEMBL3544797 | |
| 0.188 | 0.059 | 0.255 | Succinate dehydrogenase inhibitor | 0.196 0.052 CHEMBL3544797 0.224 0.033 CHEMBL3544834 0.2 0.048 CHEMBL3544836 0.238 0.027 CHEMBL3544798 0.214 0.039 CHEMBL3544835 0.255 0.02 CHEMBL3544833 | CHEMBL3544833 | |
| 0.157 | 0.032 | 0.172 | GABA receptor agonist | 0.166 0.028 CHEMBL3544834 0.139 0.042 CHEMBL3544836 0.151 0.035 CHEMBL3544798 0.172 0.026 CHEMBL3544833 | CHEMBL3544833 | |
| 0.25 | 0.127 | 0.571 | Transcription factor NF kappa B inhibitor | 0.324 0.085 CHEMBL3544797 0.268 0.115 CHEMBL3544834 0.335 0.081 CHEMBL3544836 0.218 0.153 CHEMBL3544798 0.253 0.125 CHEMBL3544835 0.571 0.035 CHEMBL3544799 0.3 0.094 CHEMBL3544833 | CHEMBL3544799 | |
| 0.138 | 0.016 | 0.138 | Cyclin B3 inhibitor | 0.118 0.022 CHEMBL3544834 0.12 0.021 CHEMBL3544836 0.084 0.036 CHEMBL3544798 0.063 0.052 CHEMBL3544835 | ||
| 0.131 | 0.013 | 0.152 | Glycine receptor antagonist | 0.152 0.007 CHEMBL3544797 0.137 0.011 CHEMBL3544834 0.127 0.015 CHEMBL3544836 0.1 0.032 CHEMBL3544798 0.116 0.02 CHEMBL3544835 0.141 0.01 CHEMBL3544799 0.12 0.018 CHEMBL3544833 | CHEMBL3544797 | |
| 0.212 | 0.095 | 0.44 | Vasodilator | 0.44 0.017 CHEMBL3544797 0.16 0.143 CHEMBL3544834 0.279 0.056 CHEMBL3544836 0.19 0.112 CHEMBL3544798 0.227 0.084 CHEMBL3544835 0.416 0.02 CHEMBL3544799 | CHEMBL3544797 | |
| 0.14 | 0.024 | 0.159 | Anabolic | 0.159 0.014 CHEMBL3544797 0.135 0.027 CHEMBL3544834 0.141 0.023 CHEMBL3544836 0.124 0.036 CHEMBL3544798 0.158 0.014 CHEMBL3544835 0.136 0.027 CHEMBL3544833 | CHEMBL3544797 | |
| 0.149 | 0.038 | 0.209 | Microtubule formation inhibitor | 0.192 0.022 CHEMBL3544797 0.155 0.035 CHEMBL3544834 0.137 0.046 CHEMBL3544836 0.15 0.037 CHEMBL3544798 0.177 0.026 CHEMBL3544835 0.209 0.018 CHEMBL3544799 0.143 0.041 CHEMBL3544833 | CHEMBL3544799 | |
| 0.207 | 0.096 | 0.456 | Platelet antagonist | 0.197 0.103 CHEMBL3544797 0.182 0.115 CHEMBL3544834 0.31 0.05 CHEMBL3544836 0.2 0.101 CHEMBL3544798 0.269 0.064 CHEMBL3544835 0.393 0.029 CHEMBL3544799 0.456 0.019 CHEMBL3544833 | CHEMBL3544833 | |
| 0.193 | 0.084 | 0.242 | Neurotrophic factor enhancer | 0.242 0.043 CHEMBL3544797 0.227 0.054 CHEMBL3544834 0.225 0.055 CHEMBL3544836 0.178 0.1 CHEMBL3544798 0.193 0.083 CHEMBL3544835 0.175 0.104 CHEMBL3544833 | CHEMBL3544797 | |
| 0.12 | 0.012 | 0.142 | Protein kinase C eta inhibitor | 0.13 0.01 CHEMBL3544797 0.133 0.009 CHEMBL3544834 0.134 0.009 CHEMBL3544836 0.114 0.014 CHEMBL3544798 0.142 0.008 CHEMBL3544835 0.128 0.01 CHEMBL3544799 0.093 0.019 CHEMBL3544833 | CHEMBL3544835 | |
| 0.175 | 0.069 | 0.193 | Antipruritic | 0.17 0.074 CHEMBL3544797 0.13 0.123 CHEMBL3544834 0.19 0.056 CHEMBL3544836 0.193 0.054 CHEMBL3544798 0.148 0.097 CHEMBL3544835 | CHEMBL3544798 | |
| 0.216 | 0.111 | 0.551 | Immunostimulant | 0.302 0.078 CHEMBL3544797 0.215 0.111 CHEMBL3544834 0.361 0.061 CHEMBL3544836 0.235 0.102 CHEMBL3544798 0.282 0.084 CHEMBL3544835 0.551 0.022 CHEMBL3544799 0.273 0.087 CHEMBL3544833 | CHEMBL3544799 | |
| 0.136 | 0.031 | 0.233 | UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor | 0.213 0.014 CHEMBL3544797 0.17 0.021 CHEMBL3544834 0.228 0.012 CHEMBL3544836 0.156 0.025 CHEMBL3544798 0.152 0.026 CHEMBL3544835 0.173 0.021 CHEMBL3544799 0.233 0.011 CHEMBL3544833 | CHEMBL3544833 | |
| 0.213 | 0.109 | 0.33 | Spasmolytic | 0.24 0.096 CHEMBL3544797 0.189 0.129 CHEMBL3544834 0.33 0.059 CHEMBL3544836 0.215 0.108 CHEMBL3544798 0.314 0.065 CHEMBL3544835 0.256 0.089 CHEMBL3544799 0.168 0.147 CHEMBL3544833 | CHEMBL3544836 | |
| 0.188 | 0.085 | 0.189 | 5 Hydroxytryptamine 3E antagonist | 0.189 0.083 CHEMBL3544834 0.163 0.16 CHEMBL3544798 | CHEMBL3544834 | |
| 0.14 | 0.038 | 0.175 | Photosensitizer | 0.175 0.019 CHEMBL3544797 0.123 0.054 CHEMBL3544834 0.161 0.025 CHEMBL3544836 0.1 0.088 CHEMBL3544798 0.139 0.038 CHEMBL3544835 0.15 0.031 CHEMBL3544799 0.116 0.062 CHEMBL3544833 | CHEMBL3544797 | |
| 0.148 | 0.048 | 0.165 | Ca2+-transporting ATPase inhibitor | 0.165 0.017 CHEMBL3544797 0.165 0.018 CHEMBL3544834 0.151 0.04 CHEMBL3544836 0.153 0.036 CHEMBL3544798 0.163 0.02 CHEMBL3544835 0.158 0.027 CHEMBL3544799 0.152 0.038 CHEMBL3544833 | CHEMBL3544834 | |
| 0.162 | 0.064 | 0.346 | Interferon gamma antagonist | 0.201 0.04 CHEMBL3544797 0.196 0.042 CHEMBL3544834 0.172 0.056 CHEMBL3544836 0.165 0.061 CHEMBL3544798 0.201 0.04 CHEMBL3544835 0.346 0.014 CHEMBL3544799 0.186 0.047 CHEMBL3544833 | CHEMBL3544799 | |
| 0.111 | 0.018 | 0.159 | Protein kinase C alpha inhibitor | 0.101 0.022 CHEMBL3544797 0.114 0.018 CHEMBL3544834 0.159 0.009 CHEMBL3544836 0.115 0.017 CHEMBL3544798 0.104 0.02 CHEMBL3544835 0.064 0.053 CHEMBL3544799 0.072 0.041 CHEMBL3544833 | CHEMBL3544836 | |
| 0.263 | 0.174 | 0.321 | MAP kinase kinase 6 inhibitor | 0.287 0.149 CHEMBL3544797 0.321 0.117 CHEMBL3544834 | CHEMBL3544834 | |
| 0.101 | 0.022 | 0.101 | Phosphodiesterase III inhibitor | 0.069 0.045 CHEMBL3544797 0.075 0.04 CHEMBL3544834 0.084 0.032 CHEMBL3544836 | ||
| 0.198 | 0.119 | 0.234 | Superoxide dismutase inhibitor | 0.234 0.086 CHEMBL3544797 0.221 0.097 CHEMBL3544834 0.189 0.13 CHEMBL3544836 0.202 0.115 CHEMBL3544798 0.167 0.16 CHEMBL3544835 0.211 0.106 CHEMBL3544833 | CHEMBL3544797 | |
| 0.154 | 0.074 | 0.182 | Diuretic | 0.133 0.092 CHEMBL3544797 0.128 0.096 CHEMBL3544834 0.178 0.055 CHEMBL3544836 0.118 0.107 CHEMBL3544798 0.142 0.084 CHEMBL3544835 0.182 0.052 CHEMBL3544799 0.146 0.081 CHEMBL3544833 | CHEMBL3544799 | |
| 0.089 | 0.012 | 0.131 | MDM2 inhibitor | 0.071 0.036 CHEMBL3544797 0.078 0.023 CHEMBL3544834 0.088 0.013 CHEMBL3544836 0.103 0.006 CHEMBL3544798 0.069 0.041 CHEMBL3544835 0.131 0.004 CHEMBL3544833 | CHEMBL3544833 | |
| 0.117 | 0.039 | 0.152 | Electrolyte absorption antagonist | 0.119 0.037 CHEMBL3544797 0.111 0.044 CHEMBL3544834 0.099 0.058 CHEMBL3544836 0.095 0.066 CHEMBL3544798 0.105 0.051 CHEMBL3544835 0.152 0.019 CHEMBL3544833 | CHEMBL3544833 | |
| 0.147 | 0.072 | 0.321 | Hemostatic | 0.143 0.077 CHEMBL3544797 0.13 0.096 CHEMBL3544834 0.19 0.037 CHEMBL3544836 0.131 0.094 CHEMBL3544798 0.14 0.081 CHEMBL3544835 0.321 0.014 CHEMBL3544799 0.148 0.07 CHEMBL3544833 | CHEMBL3544799 | |
| 0.081 | 0.009 | 0.123 | Guanylate cyclase stimulant | 0.069 0.011 CHEMBL3544797 0.077 0.009 CHEMBL3544834 0.068 0.011 CHEMBL3544836 0.069 0.011 CHEMBL3544798 0.068 0.011 CHEMBL3544835 0.123 0.005 CHEMBL3544833 | CHEMBL3544833 | |
| 0.099 | 0.028 | 0.118 | Lipase inhibitor | 0.118 0.019 CHEMBL3544834 0.103 0.025 CHEMBL3544836 0.078 0.045 CHEMBL3544798 0.085 0.038 CHEMBL3544835 0.069 0.055 CHEMBL3544799 0.083 0.04 CHEMBL3544833 | CHEMBL3544834 | |
| 0.211 | 0.141 | 0.284 | Insulysin inhibitor | 0.235 0.111 CHEMBL3544834 0.214 0.136 CHEMBL3544836 0.193 0.169 CHEMBL3544798 0.284 0.069 CHEMBL3544833 | CHEMBL3544833 | |
| 0.104 | 0.035 | 0.44 | Phosphodiesterase 4D inhibitor | 0.126 0.026 CHEMBL3544834 0.079 0.048 CHEMBL3544836 0.44 0.004 CHEMBL3544835 0.085 0.044 CHEMBL3544833 | CHEMBL3544835 | |
| 0.107 | 0.042 | 0.192 | Androgen antagonist | 0.192 0.014 CHEMBL3544797 0.156 0.021 CHEMBL3544834 0.083 0.062 CHEMBL3544836 0.112 0.038 CHEMBL3544835 | CHEMBL3544797 | |
| 0.075 | 0.01 | 0.103 | Adenylate cyclase 1 inhibitor | 0.103 0.004 CHEMBL3544797 0.059 0.018 CHEMBL3544834 0.05 0.026 CHEMBL3544798 0.048 0.029 CHEMBL3544835 0.043 0.036 CHEMBL3544833 | CHEMBL3544797 | |
| 0.084 | 0.021 | 0.084 | Calcium channel T-type blocker | |||
| 0.068 | 0.008 | 0.092 | Membrane dipeptidase inhibitor | 0.063 0.009 CHEMBL3544797 0.048 0.017 CHEMBL3544834 0.063 0.009 CHEMBL3544836 0.063 0.009 CHEMBL3544798 0.092 0.004 CHEMBL3544835 0.075 0.006 CHEMBL3544833 | CHEMBL3544835 | |
| 0.072 | 0.012 | 0.077 | Pregnane X receptor antagonist | 0.077 0.008 CHEMBL3544797 0.062 0.027 CHEMBL3544834 0.056 0.04 CHEMBL3544836 0.061 0.028 CHEMBL3544798 0.074 0.01 CHEMBL3544835 0.061 0.027 CHEMBL3544833 | CHEMBL3544797 | |
| 0.128 | 0.07 | 0.156 | Vanilloid 1 agonist | 0.13 0.066 CHEMBL3544797 0.124 0.079 CHEMBL3544834 0.156 0.033 CHEMBL3544836 0.126 0.075 CHEMBL3544798 0.128 0.07 CHEMBL3544799 0.136 0.057 CHEMBL3544833 | CHEMBL3544836 | |
| 0.081 | 0.025 | 0.149 | Biliverdin reductase inhibitor | 0.147 0.01 CHEMBL3544797 0.071 0.032 CHEMBL3544834 0.112 0.015 CHEMBL3544836 0.092 0.021 CHEMBL3544798 0.097 0.019 CHEMBL3544835 0.053 0.049 CHEMBL3544799 0.149 0.009 CHEMBL3544833 | CHEMBL3544833 | |
| 0.1 | 0.045 | 0.116 | Ornithine decarboxylase inhibitor | 0.116 0.029 CHEMBL3544797 0.096 0.049 CHEMBL3544834 0.101 0.043 CHEMBL3544836 0.081 0.066 CHEMBL3544798 0.105 0.039 CHEMBL3544835 0.096 0.049 CHEMBL3544833 | CHEMBL3544797 | |
| 0.114 | 0.059 | 0.14 | Acetylcholine release stimulant | 0.128 0.037 CHEMBL3544834 0.101 0.086 CHEMBL3544836 0.115 0.057 CHEMBL3544798 0.14 0.024 CHEMBL3544799 0.101 0.086 CHEMBL3544833 | CHEMBL3544799 | |
| 0.075 | 0.022 | 0.075 | Corticotropin releasing factor 2 receptor antagonist | 0.067 0.032 CHEMBL3544834 | ||
| 0.109 | 0.055 | 0.187 | Adenylate kinase inhibitor | 0.187 0.017 CHEMBL3544797 0.112 0.051 CHEMBL3544834 0.148 0.027 CHEMBL3544836 0.117 0.046 CHEMBL3544798 0.17 0.02 CHEMBL3544835 0.094 0.079 CHEMBL3544799 0.184 0.017 CHEMBL3544833 | CHEMBL3544797 | |
| 0.078 | 0.025 | 0.12 | Androgen agonist | 0.12 0.01 CHEMBL3544797 0.056 0.047 CHEMBL3544834 0.096 0.016 CHEMBL3544836 0.076 0.026 CHEMBL3544835 | CHEMBL3544797 | |
| 0.143 | 0.089 | 0.18 | CF transmembrane conductance regulator agonist | 0.18 0.036 CHEMBL3544797 0.133 0.111 CHEMBL3544834 0.171 0.046 CHEMBL3544836 | CHEMBL3544797 | |
| 0.102 | 0.051 | 0.114 | Protein kinase C delta inhibitor | 0.098 0.054 CHEMBL3544797 0.108 0.046 CHEMBL3544834 0.114 0.041 CHEMBL3544836 0.089 0.063 CHEMBL3544798 0.088 0.065 CHEMBL3544835 | CHEMBL3544836 | |
| 0.091 | 0.04 | 0.186 | Porphobilinogen synthase inhibitor | 0.091 0.04 CHEMBL3544797 0.096 0.038 CHEMBL3544834 0.17 0.017 CHEMBL3544836 0.08 0.047 CHEMBL3544798 0.089 0.041 CHEMBL3544835 0.186 0.014 CHEMBL3544833 | CHEMBL3544833 | |
| 0.143 | 0.092 | 0.191 | Melanin inhibitor | 0.177 0.053 CHEMBL3544797 0.16 0.07 CHEMBL3544834 0.155 0.074 CHEMBL3544836 0.143 0.092 CHEMBL3544798 0.191 0.045 CHEMBL3544835 0.175 0.055 CHEMBL3544799 0.144 0.09 CHEMBL3544833 | CHEMBL3544835 | |
| 0.1 | 0.053 | 0.152 | Interleukin 12 antagonist | 0.099 0.055 CHEMBL3544834 0.112 0.038 CHEMBL3544836 0.117 0.032 CHEMBL3544798 0.091 0.07 CHEMBL3544835 0.152 0.012 CHEMBL3544799 0.12 0.029 CHEMBL3544833 | CHEMBL3544799 | |
| 0.061 | 0.014 | 0.072 | AICAR transformylase inhibitor | 0.072 0.009 CHEMBL3544797 0.055 0.018 CHEMBL3544836 0.043 0.033 CHEMBL3544798 0.068 0.01 CHEMBL3544833 | CHEMBL3544797 | |
| 0.052 | 0.005 | 0.057 | Protein kinase C beta II inhibitor | 0.05 0.006 CHEMBL3544797 0.051 0.006 CHEMBL3544834 0.057 0.005 CHEMBL3544836 0.052 0.005 CHEMBL3544798 0.045 0.008 CHEMBL3544835 0.041 0.01 CHEMBL3544799 0.042 0.009 CHEMBL3544833 | CHEMBL3544836 | |
| 0.149 | 0.104 | 0.191 | Neurotensin receptor agonist | 0.15 0.102 CHEMBL3544834 0.151 0.099 CHEMBL3544836 0.191 0.04 CHEMBL3544833 | CHEMBL3544833 | |
| 0.066 | 0.021 | 0.077 | Dihydroorotate oxidase inhibitor | 0.077 0.012 CHEMBL3544834 0.066 0.021 CHEMBL3544836 0.059 0.031 CHEMBL3544798 0.073 0.014 CHEMBL3544835 0.059 0.03 CHEMBL3544833 | CHEMBL3544834 | |
| 0.09 | 0.046 | 0.09 | Acetylcholine nicotinic antagonist | 0.081 0.053 CHEMBL3544834 0.086 0.048 CHEMBL3544836 | ||
| 0.046 | 0.004 | 0.051 | Retinoic acid gamma receptor agonist | 0.046 0.004 CHEMBL3544834 0.031 0.006 CHEMBL3544836 0.043 0.004 CHEMBL3544798 0.051 0.003 CHEMBL3544835 0.024 0.012 CHEMBL3544799 0.049 0.004 CHEMBL3544833 | CHEMBL3544835 | |
| 0.046 | 0.004 | 0.046 | Nicotinic acid receptor 2 antagonist | 0.038 0.006 CHEMBL3544797 0.028 0.015 CHEMBL3544834 0.046 0.004 CHEMBL3544836 0.028 0.016 CHEMBL3544798 0.038 0.005 CHEMBL3544835 0.032 0.01 CHEMBL3544833 | ||
| 0.093 | 0.052 | 0.246 | NADH dehydrogenase inhibitor | 0.153 0.017 CHEMBL3544797 0.097 0.047 CHEMBL3544834 0.146 0.019 CHEMBL3544836 0.114 0.032 CHEMBL3544798 0.114 0.032 CHEMBL3544835 0.246 0.008 CHEMBL3544799 0.122 0.028 CHEMBL3544833 | CHEMBL3544799 | |
| 0.162 | 0.122 | 0.263 | Glyceraldehyde-3-phosphate dehydrogenase inhibitor | 0.263 0.037 CHEMBL3544797 0.171 0.106 CHEMBL3544834 0.216 0.06 CHEMBL3544836 0.164 0.118 CHEMBL3544798 0.218 0.059 CHEMBL3544835 0.193 0.078 CHEMBL3544833 | CHEMBL3544797 | |
| 0.044 | 0.004 | 0.058 | Retinoic acid beta receptor agonist | 0.039 0.004 CHEMBL3544834 0.027 0.007 CHEMBL3544836 0.058 0.004 CHEMBL3544798 0.046 0.004 CHEMBL3544835 0.019 0.016 CHEMBL3544799 0.05 0.004 CHEMBL3544833 | CHEMBL3544798 | |
| 0.085 | 0.045 | 0.117 | Na+ K+ transporting ATPase inhibitor | 0.107 0.026 CHEMBL3544797 0.098 0.033 CHEMBL3544834 0.091 0.04 CHEMBL3544836 0.103 0.029 CHEMBL3544798 0.112 0.021 CHEMBL3544835 0.117 0.018 CHEMBL3544799 0.089 0.042 CHEMBL3544833 | CHEMBL3544799 | |
| 0.059 | 0.02 | 0.061 | Aldosterone antagonist | 0.061 0.019 CHEMBL3544797 0.059 0.02 CHEMBL3544834 | CHEMBL3544797 | |
| 0.067 | 0.028 | 0.128 | Acyl-CoA dehydrogenase inhibitor | 0.128 0.011 CHEMBL3544797 0.066 0.029 CHEMBL3544834 0.105 0.015 CHEMBL3544836 0.074 0.025 CHEMBL3544798 0.082 0.021 CHEMBL3544835 0.091 0.019 CHEMBL3544833 | CHEMBL3544797 | |
| 0.045 | 0.006 | 0.047 | Retinoic acid receptor agonist | 0.035 0.008 CHEMBL3544834 0.024 0.015 CHEMBL3544836 0.043 0.006 CHEMBL3544798 0.047 0.005 CHEMBL3544835 0.022 0.017 CHEMBL3544799 0.043 0.006 CHEMBL3544833 | CHEMBL3544835 | |
| 0.096 | 0.057 | 0.096 | Alpha 2d adrenoreceptor antagonist | |||
| 0.093 | 0.055 | 0.21 | Triose-phosphate isomerase inhibitor | 0.151 0.019 CHEMBL3544797 0.099 0.049 CHEMBL3544834 0.161 0.017 CHEMBL3544836 0.142 0.022 CHEMBL3544798 0.158 0.018 CHEMBL3544835 0.21 0.01 CHEMBL3544799 0.149 0.02 CHEMBL3544833 | CHEMBL3544799 | |
| 0.106 | 0.069 | 0.106 | 5 Hydroxytryptamine 3A agonist | |||
| 0.101 | 0.065 | 0.104 | Alpha 2c adrenoreceptor antagonist | 0.104 0.062 CHEMBL3544836 0.101 0.065 CHEMBL3544835 | CHEMBL3544836 | |
| 0.053 | 0.017 | 0.078 | Thymidine kinase inhibitor | 0.078 0.009 CHEMBL3544797 0.043 0.025 CHEMBL3544834 0.067 0.011 CHEMBL3544836 0.064 0.012 CHEMBL3544798 0.052 0.018 CHEMBL3544835 0.037 0.036 CHEMBL3544799 0.044 0.024 CHEMBL3544833 | CHEMBL3544797 | |
| 0.136 | 0.1 | 0.227 | Growth hormone agonist | 0.227 0.05 CHEMBL3544797 0.159 0.08 CHEMBL3544798 0.13 0.107 CHEMBL3544835 0.218 0.052 CHEMBL3544833 | CHEMBL3544797 | |
| 0.209 | 0.174 | 0.428 | Vasodilator, coronary | 0.267 0.118 CHEMBL3544797 0.222 0.161 CHEMBL3544834 0.263 0.122 CHEMBL3544836 0.214 0.169 CHEMBL3544798 0.249 0.135 CHEMBL3544835 0.428 0.028 CHEMBL3544799 | CHEMBL3544799 | |
| 0.042 | 0.007 | 0.045 | Protein kinase C beta I inhibitor | 0.043 0.006 CHEMBL3544797 0.042 0.007 CHEMBL3544834 0.045 0.005 CHEMBL3544836 0.041 0.008 CHEMBL3544798 0.04 0.009 CHEMBL3544835 0.045 0.005 CHEMBL3544799 0.039 0.01 CHEMBL3544833 | CHEMBL3544799 | |
| 0.094 | 0.059 | 0.162 | ABCA1 expression enhancer | 0.089 0.067 CHEMBL3544834 0.124 0.028 CHEMBL3544798 0.11 0.039 CHEMBL3544835 0.162 0.015 CHEMBL3544833 | CHEMBL3544833 | |
| 0.061 | 0.026 | 0.069 | Nicotinic alpha3beta2 receptor antagonist | 0.069 0.018 CHEMBL3544834 0.053 0.038 CHEMBL3544836 0.061 0.026 CHEMBL3544798 | CHEMBL3544834 | |
| 0.155 | 0.121 | 0.155 | Ca2+/calmodulin-dependent kinase II beta inhibitor | 0.154 0.123 CHEMBL3544834 0.147 0.132 CHEMBL3544836 0.145 0.135 CHEMBL3544798 | ||
| 0.049 | 0.015 | 0.083 | Kainate receptor agonist | 0.061 0.007 CHEMBL3544797 0.047 0.018 CHEMBL3544834 0.052 0.012 CHEMBL3544836 0.046 0.019 CHEMBL3544798 0.051 0.013 CHEMBL3544835 0.083 0.004 CHEMBL3544833 | CHEMBL3544833 | |
| 0.08 | 0.046 | 0.08 | Acetylcholine M4 receptor antagonist | 0.077 0.05 CHEMBL3544834 | ||
| 0.069 | 0.035 | 0.128 | Carbamoyl phosphate synthetase inhibitor | 0.128 0.014 CHEMBL3544797 0.075 0.031 CHEMBL3544834 0.112 0.017 CHEMBL3544836 0.111 0.018 CHEMBL3544798 0.096 0.022 CHEMBL3544835 0.121 0.015 CHEMBL3544833 | CHEMBL3544797 | |
| 0.057 | 0.024 | 0.058 | HCV NS3/NS4A protease inhibitor | 0.058 0.023 CHEMBL3544834 0.046 0.04 CHEMBL3544836 0.049 0.035 CHEMBL3544835 0.055 0.026 CHEMBL3544833 | CHEMBL3544834 | |
| 0.069 | 0.037 | 0.151 | NMDA receptor agonist | 0.062 0.044 CHEMBL3544797 0.056 0.053 CHEMBL3544834 0.077 0.031 CHEMBL3544836 0.056 0.053 CHEMBL3544798 0.059 0.049 CHEMBL3544835 0.151 0.008 CHEMBL3544833 | CHEMBL3544833 | |
| 0.084 | 0.054 | 0.101 | Estrogen-related receptor beta agonist | 0.101 0.023 CHEMBL3544797 0.085 0.053 CHEMBL3544834 0.087 0.046 CHEMBL3544836 0.096 0.031 CHEMBL3544798 0.082 0.062 CHEMBL3544835 0.087 0.048 CHEMBL3544833 | CHEMBL3544797 | |
| 0.081 | 0.052 | 0.118 | Glutamate receptor agonist | 0.067 0.066 CHEMBL3544834 0.118 0.027 CHEMBL3544833 | CHEMBL3544833 | |
| 0.073 | 0.046 | 0.19 | Phosphofructokinase-1 inhibitor | 0.151 0.018 CHEMBL3544797 0.061 0.055 CHEMBL3544834 0.148 0.018 CHEMBL3544836 0.109 0.028 CHEMBL3544798 0.086 0.038 CHEMBL3544835 0.19 0.012 CHEMBL3544799 0.123 0.024 CHEMBL3544833 | CHEMBL3544799 | |
| 0.093 | 0.066 | 0.141 | Phosphodiesterase 6D inhibitor | 0.097 0.059 CHEMBL3544797 0.097 0.058 CHEMBL3544834 0.106 0.042 CHEMBL3544836 0.106 0.041 CHEMBL3544798 0.109 0.038 CHEMBL3544835 0.141 0.012 CHEMBL3544799 | CHEMBL3544799 | |
| 0.095 | 0.069 | 0.152 | Aminopeptidase B inhibitor | 0.087 0.075 CHEMBL3544797 0.084 0.078 CHEMBL3544834 0.126 0.049 CHEMBL3544836 0.12 0.053 CHEMBL3544798 0.1 0.065 CHEMBL3544835 0.152 0.037 CHEMBL3544833 | CHEMBL3544833 | |
| 0.05 | 0.025 | 0.057 | Phosphodiesterase 3B inhibitor | 0.041 0.035 CHEMBL3544797 0.057 0.02 CHEMBL3544834 0.051 0.024 CHEMBL3544836 0.048 0.027 CHEMBL3544798 0.041 0.034 CHEMBL3544835 0.04 0.036 CHEMBL3544833 | CHEMBL3544834 | |
| 0.073 | 0.047 | 0.075 | Phospholipase D inhibitor | 0.071 0.05 CHEMBL3544797 0.075 0.043 CHEMBL3544834 0.068 0.057 CHEMBL3544836 0.069 0.055 CHEMBL3544798 0.074 0.045 CHEMBL3544835 0.071 0.051 CHEMBL3544833 | CHEMBL3544834 | |
| 0.061 | 0.036 | 0.118 | Argininosuccinate synthase inhibitor | 0.118 0.015 CHEMBL3544797 0.082 0.024 CHEMBL3544834 0.099 0.019 CHEMBL3544836 0.057 0.04 CHEMBL3544798 0.075 0.027 CHEMBL3544835 0.112 0.017 CHEMBL3544833 | CHEMBL3544797 | |
| 0.058 | 0.033 | 0.07 | Protein kinase C epsilon inhibitor | 0.07 0.024 CHEMBL3544834 0.048 0.043 CHEMBL3544798 0.058 0.033 CHEMBL3544835 | CHEMBL3544834 | |
| 0.1 | 0.075 | 0.149 | DOPA decarboxylase inhibitor | 0.099 0.078 CHEMBL3544797 0.108 0.061 CHEMBL3544834 0.112 0.056 CHEMBL3544836 0.109 0.06 CHEMBL3544798 0.093 0.092 CHEMBL3544835 0.149 0.022 CHEMBL3544833 | CHEMBL3544833 | |
| 0.109 | 0.085 | 0.125 | Cholinergic antagonist | 0.123 0.071 CHEMBL3544836 0.125 0.069 CHEMBL3544835 | CHEMBL3544835 | |
| 0.045 | 0.02 | 0.079 | Progesterone antagonist | 0.048 0.019 CHEMBL3544797 0.079 0.011 CHEMBL3544834 0.03 0.029 CHEMBL3544835 | CHEMBL3544834 | |
| 0.048 | 0.025 | 0.048 | Oxytocin agonist | 0.038 0.034 CHEMBL3544797 0.042 0.03 CHEMBL3544834 0.043 0.029 CHEMBL3544836 0.038 0.034 CHEMBL3544798 | ||
| 0.031 | 0.009 | 0.044 | Thymidine kinase (Herpes simplex virus 1) inhibitor | 0.044 0.004 CHEMBL3544797 0.027 0.018 CHEMBL3544834 0.035 0.007 CHEMBL3544836 0.035 0.007 CHEMBL3544798 0.028 0.015 CHEMBL3544835 0.025 0.023 CHEMBL3544833 | CHEMBL3544797 | |
| 0.082 | 0.06 | 0.092 | GABA A receptor agonist | 0.092 0.046 CHEMBL3544834 0.083 0.059 CHEMBL3544798 | CHEMBL3544834 | |
| 0.036 | 0.014 | 0.066 | Uridine phosphorylase inhibitor | 0.062 0.005 CHEMBL3544797 0.028 0.02 CHEMBL3544834 0.066 0.005 CHEMBL3544836 0.049 0.009 CHEMBL3544798 0.034 0.015 CHEMBL3544835 0.039 0.012 CHEMBL3544799 0.03 0.018 CHEMBL3544833 | CHEMBL3544836 | |
| 0.089 | 0.068 | 0.107 | Prolactin inhibitor | 0.085 0.073 CHEMBL3544797 0.085 0.074 CHEMBL3544834 0.107 0.048 CHEMBL3544836 0.094 0.061 CHEMBL3544833 | CHEMBL3544836 | |
| 0.072 | 0.051 | 0.107 | Glycine receptor agonist | 0.107 0.017 CHEMBL3544797 0.103 0.019 CHEMBL3544834 0.076 0.045 CHEMBL3544836 0.083 0.035 CHEMBL3544798 0.081 0.037 CHEMBL3544835 0.075 0.045 CHEMBL3544799 0.089 0.029 CHEMBL3544833 | CHEMBL3544797 | |
| 0.026 | 0.006 | 0.038 | Thymidine kinase (Herpes simplex virus 2) inhibitor | 0.038 0.003 CHEMBL3544797 0.021 0.014 CHEMBL3544834 0.027 0.005 CHEMBL3544836 0.027 0.005 CHEMBL3544798 0.021 0.013 CHEMBL3544835 0.02 0.017 CHEMBL3544833 | CHEMBL3544797 | |
| 0.034 | 0.014 | 0.034 | Calcitonin gene-related peptide antagonist | 0.024 0.018 CHEMBL3544834 | ||
| 0.077 | 0.057 | 0.122 | Interferon agonist | 0.09 0.038 CHEMBL3544797 0.075 0.06 CHEMBL3544834 0.119 0.018 CHEMBL3544836 0.086 0.043 CHEMBL3544798 0.087 0.042 CHEMBL3544835 0.122 0.017 CHEMBL3544799 0.085 0.045 CHEMBL3544833 | CHEMBL3544799 | |
| 0.057 | 0.038 | 0.137 | Alcohol oxidase inhibitor | 0.137 0.012 CHEMBL3544797 0.069 0.029 CHEMBL3544834 0.09 0.021 CHEMBL3544836 0.107 0.016 CHEMBL3544798 0.095 0.019 CHEMBL3544835 0.119 0.014 CHEMBL3544833 | CHEMBL3544797 | |
| 0.102 | 0.083 | 0.154 | Adenylate cyclase inhibitor | 0.152 0.044 CHEMBL3544797 0.094 0.09 CHEMBL3544834 0.127 0.062 CHEMBL3544836 0.106 0.079 CHEMBL3544798 0.154 0.043 CHEMBL3544835 0.137 0.054 CHEMBL3544833 | CHEMBL3544835 | |
| 0.038 | 0.02 | 0.052 | Tryptophan 5 hydroxylase inhibitor | 0.033 0.032 CHEMBL3544834 0.036 0.025 CHEMBL3544836 0.036 0.023 CHEMBL3544798 0.047 0.007 CHEMBL3544835 0.052 0.005 CHEMBL3544833 | CHEMBL3544833 | |
| 0.058 | 0.041 | 0.058 | CDK4/cyclin D1 inhibitor | |||
| 0.024 | 0.009 | 0.031 | Guanylate cyclase 1 stimulant | 0.018 0.015 CHEMBL3544797 0.022 0.011 CHEMBL3544834 0.02 0.013 CHEMBL3544836 0.02 0.012 CHEMBL3544798 0.02 0.013 CHEMBL3544835 0.031 0.006 CHEMBL3544833 | CHEMBL3544833 | |
| 0.054 | 0.041 | 0.059 | Cyclin B2 inhibitor | 0.059 0.033 CHEMBL3544834 0.055 0.04 CHEMBL3544836 | CHEMBL3544834 | |
| 0.1 | 0.087 | 0.116 | Proteasome inhibitor | 0.116 0.068 CHEMBL3544834 0.104 0.082 CHEMBL3544835 0.109 0.076 CHEMBL3544833 | CHEMBL3544834 | |
| 0.065 | 0.052 | 0.086 | Glutamate (mGluR6) antagonist | 0.076 0.029 CHEMBL3544797 0.064 0.053 CHEMBL3544834 0.074 0.032 CHEMBL3544836 0.07 0.039 CHEMBL3544798 0.077 0.028 CHEMBL3544835 0.086 0.019 CHEMBL3544833 | CHEMBL3544833 | |
| 0.072 | 0.06 | 0.087 | Nicotinic alpha4beta2 receptor antagonist | 0.087 0.043 CHEMBL3544834 | CHEMBL3544834 | |
| 0.072 | 0.06 | 0.107 | Keratolytic | 0.097 0.033 CHEMBL3544797 0.078 0.052 CHEMBL3544834 0.077 0.053 CHEMBL3544836 0.103 0.028 CHEMBL3544798 0.107 0.027 CHEMBL3544835 0.099 0.031 CHEMBL3544833 | CHEMBL3544835 | |
| 0.068 | 0.056 | 0.099 | Aminopeptidase I inhibitor | 0.083 0.039 CHEMBL3544797 0.079 0.044 CHEMBL3544836 0.085 0.038 CHEMBL3544798 0.075 0.047 CHEMBL3544835 0.099 0.029 CHEMBL3544833 | CHEMBL3544833 | |
| 0.058 | 0.047 | 0.064 | Cyclin B1 inhibitor | 0.064 0.039 CHEMBL3544834 0.057 0.048 CHEMBL3544836 | CHEMBL3544834 | |
| 0.101 | 0.091 | 0.116 | Acetylcholine antagonist | 0.113 0.077 CHEMBL3544836 0.116 0.074 CHEMBL3544835 | CHEMBL3544835 | |
| 0.121 | 0.112 | 0.147 | CC chemokine 6 receptor antagonist | 0.13 0.07 CHEMBL3544797 0.132 0.064 CHEMBL3544836 0.147 0.027 CHEMBL3544799 | CHEMBL3544799 | |
| 0.058 | 0.049 | 0.07 | NMDA 2C receptor antagonist | 0.067 0.036 CHEMBL3544835 0.07 0.033 CHEMBL3544833 | CHEMBL3544833 | |
| 0.02 | 0.012 | 0.021 | Progesterone receptor B antagonist | 0.019 0.015 CHEMBL3544797 0.021 0.01 CHEMBL3544834 | CHEMBL3544834 | |
| 0.037 | 0.029 | 0.037 | Cyclin D3 inhibitor | |||
| 0.1 | 0.092 | 0.102 | Interleukin 2 antagonist | 0.102 0.086 CHEMBL3544834 | CHEMBL3544834 | |
| 0.068 | 0.06 | 0.115 | Glutamate dehydrogenase inhibitor | 0.114 0.025 CHEMBL3544797 0.071 0.055 CHEMBL3544834 0.094 0.034 CHEMBL3544836 0.072 0.054 CHEMBL3544798 0.086 0.039 CHEMBL3544835 0.115 0.024 CHEMBL3544833 | CHEMBL3544833 | |
| 0.07 | 0.063 | 0.078 | Vanilloid 4 agonist | 0.078 0.044 CHEMBL3544797 0.07 0.065 CHEMBL3544834 | CHEMBL3544797 | |
| 0.038 | 0.031 | 0.115 | AMPA 4 receptor antagonist | 0.036 0.035 CHEMBL3544836 0.038 0.029 CHEMBL3544798 0.115 0.004 CHEMBL3544833 | CHEMBL3544833 | |
| 0.05 | 0.043 | 0.138 | Alpha-mannosidase inhibitor | 0.084 0.01 CHEMBL3544797 0.079 0.012 CHEMBL3544836 0.078 0.012 CHEMBL3544798 0.07 0.017 CHEMBL3544835 0.138 0.004 CHEMBL3544799 0.06 0.027 CHEMBL3544833 | CHEMBL3544799 | |
| 0.036 | 0.03 | 0.036 | Glutamate (mGluR group II) antagonist | 0.035 0.032 CHEMBL3544833 | ||
| 0.059 | 0.054 | 0.059 | Cyclin-dependent kinase 4 inhibitor | |||
| 0.029 | 0.024 | 0.048 | Cyclophilin A inhibitor | 0.048 0.008 CHEMBL3544797 0.035 0.017 CHEMBL3544836 0.041 0.011 CHEMBL3544835 | CHEMBL3544797 | |
| 0.073 | 0.069 | 0.09 | MAP kinase kinase 7 inhibitor | 0.086 0.032 CHEMBL3544797 0.079 0.049 CHEMBL3544834 0.085 0.033 CHEMBL3544836 0.09 0.025 CHEMBL3544798 | CHEMBL3544798 | |
| 0.037 | 0.032 | 0.053 | Retinoic acid alpha receptor agonist | 0.036 0.033 CHEMBL3544834 0.053 0.012 CHEMBL3544798 0.044 0.02 CHEMBL3544835 0.049 0.015 CHEMBL3544833 | CHEMBL3544798 | |
| 0.082 | 0.078 | 0.087 | Polo-like kinase-1 inhibitor | 0.087 0.067 CHEMBL3544835 | CHEMBL3544835 | |
| 0.017 | 0.013 | 0.023 | Telomerase stimulant | 0.023 0.005 CHEMBL3544797 0.017 0.011 CHEMBL3544834 0.018 0.01 CHEMBL3544836 0.02 0.008 CHEMBL3544835 0.022 0.006 CHEMBL3544799 0.018 0.011 CHEMBL3544833 | CHEMBL3544797 | |
| 0.097 | 0.094 | 0.098 | TRPA1 agonist | 0.098 0.091 CHEMBL3544834 | CHEMBL3544834 | |
| 0.024 | 0.022 | 0.093 | Sodium/glucose cotransporter inhibitor | 0.029 0.012 CHEMBL3544797 0.045 0.006 CHEMBL3544836 0.026 0.017 CHEMBL3544798 0.029 0.012 CHEMBL3544835 0.093 0.003 CHEMBL3544799 | CHEMBL3544799 | |
| 0.027 | 0.025 | 0.027 | Acetylcholine M4 receptor agonist | |||
| 0.027 | 0.025 | 0.027 | Glutamate (mGluR2) antagonist | |||
| 0.032 | 0.03 | 0.04 | Nicotinic acid receptor agonist | 0.04 0.021 CHEMBL3544836 | CHEMBL3544836 | |
| 0.063 | 0.062 | 0.077 | Protein kinase C beta inhibitor | 0.069 0.05 CHEMBL3544797 0.064 0.061 CHEMBL3544834 0.077 0.035 CHEMBL3544836 0.071 0.045 CHEMBL3544798 0.068 0.051 CHEMBL3544835 | CHEMBL3544836 | |
| 0.007 | 0.006 | 0.007 | DNA topoisomerase III inhibitor | |||
| 0.071 | 0.07 | 0.071 | Acetylcholine M3 receptor agonist | |||
| 0.079 | 0.079 | 0.112 | Granulocyte macrophage colony stimulating factor agonist | 0.112 0.022 CHEMBL3544834 0.102 0.032 CHEMBL3544836 | CHEMBL3544834 | |
| 0.116 | 0.116 | 0.303 | Thrombolytic | 0.167 0.07 CHEMBL3544797 0.125 0.104 CHEMBL3544834 0.217 0.044 CHEMBL3544836 0.142 0.088 CHEMBL3544798 0.156 0.077 CHEMBL3544835 0.303 0.023 CHEMBL3544799 0.224 0.041 CHEMBL3544833 | CHEMBL3544799 | |
| 0.102 | 0.103 | 0.122 | Cathepsin H inhibitor | 0.122 0.073 CHEMBL3544834 | CHEMBL3544834 | |
| 0.029 | 0.03 | 0.072 | Retinoid X receptor agonist | 0.043 0.021 CHEMBL3544835 0.072 0.01 CHEMBL3544833 | CHEMBL3544833 | |
| 0.059 | 0.061 | 0.062 | Calcium channel P-type blocker | 0.062 0.049 CHEMBL3544797 | CHEMBL3544797 | |
| 0.031 | 0.033 | 0.051 | 5-Alpha-reductase inhibitor | 0.051 0.018 CHEMBL3544834 0.051 0.018 CHEMBL3544835 0.051 0.018 CHEMBL3544833 | CHEMBL3544833 | |
| 0.057 | 0.059 | 0.059 | Histone deacetylase SIRT3 inhibitor | 0.059 0.053 CHEMBL3544836 | CHEMBL3544836 | |
| 0.057 | 0.059 | 0.07 | Protease 3C (Human rhinovirus) inhibitor | 0.07 0.037 CHEMBL3544834 | CHEMBL3544834 | |
| 0.022 | 0.025 | 0.03 | Lysophosphatidic acid receptor 1 agonist | 0.026 0.017 CHEMBL3544836 0.025 0.018 CHEMBL3544798 0.03 0.011 CHEMBL3544835 0.028 0.014 CHEMBL3544833 | CHEMBL3544835 | |
| 0.136 | 0.139 | 0.189 | Phospholipase C inhibitor | 0.189 0.052 CHEMBL3544797 0.15 0.107 CHEMBL3544834 0.159 0.089 CHEMBL3544836 0.147 0.113 CHEMBL3544798 0.164 0.081 CHEMBL3544833 | CHEMBL3544797 | |
| 0.04 | 0.043 | 0.045 | Glutamate (mGluR5) agonist | 0.045 0.034 CHEMBL3544834 | CHEMBL3544834 | |
| 0.039 | 0.042 | 0.042 | Alpha 1L adrenoreceptor agonist | 0.042 0.034 CHEMBL3544834 | CHEMBL3544834 | |
| 0.141 | 0.145 | 0.161 | Focal adhesion kinase 2 inhibitor | 0.161 0.114 CHEMBL3544834 | CHEMBL3544834 | |
| 0.106 | 0.11 | 0.204 | Protein kinase stimulant | 0.18 0.05 CHEMBL3544797 0.12 0.092 CHEMBL3544834 0.147 0.07 CHEMBL3544836 0.151 0.068 CHEMBL3544798 0.204 0.04 CHEMBL3544835 0.151 0.068 CHEMBL3544799 0.131 0.083 CHEMBL3544833 | CHEMBL3544835 | |
| 0.042 | 0.046 | 0.076 | Glucose-6-phosphate isomerase inhibitor | 0.065 0.015 CHEMBL3544797 0.045 0.038 CHEMBL3544834 0.064 0.015 CHEMBL3544836 0.061 0.018 CHEMBL3544798 0.052 0.026 CHEMBL3544835 0.076 0.01 CHEMBL3544799 0.061 0.018 CHEMBL3544833 | CHEMBL3544799 | |
| 0.052 | 0.056 | 0.072 | Sphingosine kinase inhibitor | 0.072 0.023 CHEMBL3544797 0.071 0.024 CHEMBL3544836 0.064 0.032 CHEMBL3544798 0.055 0.049 CHEMBL3544835 | CHEMBL3544797 | |
| 0.016 | 0.021 | 0.021 | Methylmalonyl-CoA mutase inhibitor | 0.021 0.008 CHEMBL3544797 0.019 0.011 CHEMBL3544836 0.017 0.016 CHEMBL3544835 0.018 0.013 CHEMBL3544833 | CHEMBL3544797 | |
| 0.121 | 0.126 | 0.136 | Pregnane X receptor agonist | 0.136 0.082 CHEMBL3544797 0.134 0.088 CHEMBL3544835 | CHEMBL3544797 | |
| 0.023 | 0.028 | 0.03 | Thymidine phosphorylase inhibitor | 0.028 0.014 CHEMBL3544797 0.03 0.012 CHEMBL3544836 0.027 0.017 CHEMBL3544798 | CHEMBL3544836 | |
| 0.018 | 0.024 | 0.021 | Retinoid X beta receptor antagonist | 0.021 0.012 CHEMBL3544833 | CHEMBL3544833 | |
| 0.056 | 0.062 | 0.103 | Phosphodiesterase 4B inhibitor | 0.103 0.024 CHEMBL3544835 | CHEMBL3544835 | |
| 0.048 | 0.053 | 0.09 | Mannitol-1-phosphate 5-dehydrogenase inhibitor | 0.09 0.017 CHEMBL3544797 0.05 0.049 CHEMBL3544834 0.088 0.017 CHEMBL3544836 0.068 0.027 CHEMBL3544798 0.062 0.033 CHEMBL3544835 0.067 0.028 CHEMBL3544799 0.058 0.037 CHEMBL3544833 | CHEMBL3544797 | |
| 0.011 | 0.017 | 0.014 | Cyclin D2 inhibitor | 0.014 0.007 CHEMBL3544834 | CHEMBL3544834 | |
| 0.033 | 0.039 | 0.041 | Potassium channel Kv1.1 blocker | 0.041 0.021 CHEMBL3544834 | CHEMBL3544834 | |
| 0.093 | 0.099 | 0.124 | Acetylcholine muscarinic antagonist | 0.106 0.083 CHEMBL3544836 0.124 0.063 CHEMBL3544835 | CHEMBL3544835 | |
| 0.039 | 0.045 | 0.044 | Glutamate (mGluR group I) agonist | 0.044 0.037 CHEMBL3544834 | CHEMBL3544834 | |
| 0.083 | 0.091 | 0.107 | Bile acid receptor antagonist | 0.107 0.035 CHEMBL3544797 0.093 0.067 CHEMBL3544834 0.107 0.036 CHEMBL3544836 0.091 0.07 CHEMBL3544835 0.102 0.045 CHEMBL3544833 | CHEMBL3544836 | |
| 0.068 | 0.076 | 0.077 | Phosphodiesterase 3A inhibitor | 0.077 0.061 CHEMBL3544834 | CHEMBL3544834 | |
| 0.06 | 0.068 | 0.108 | Cathepsin G inhibitor | 0.069 0.055 CHEMBL3544834 0.07 0.054 CHEMBL3544836 0.108 0.03 CHEMBL3544835 0.094 0.035 CHEMBL3544833 | CHEMBL3544835 | |
| 0.029 | 0.039 | 0.041 | Tubulin agonist | 0.041 0.014 CHEMBL3544797 0.032 0.03 CHEMBL3544834 0.032 0.028 CHEMBL3544835 | CHEMBL3544797 | |
| 0.021 | 0.031 | 0.024 | Vanilloid 2 agonist | 0.024 0.02 CHEMBL3544797 0.023 0.022 CHEMBL3544836 0.024 0.02 CHEMBL3544799 | CHEMBL3544799 | |
| 0.009 | 0.019 | 0.014 | Lysophosphatidic acid receptor 3 agonist | 0.012 0.011 CHEMBL3544836 0.014 0.009 CHEMBL3544835 | CHEMBL3544835 | |
| 0.103 | 0.113 | 0.139 | Sphingosine 1-phosphate receptor 4 antagonist | 0.107 0.101 CHEMBL3544836 0.139 0.044 CHEMBL3544833 | CHEMBL3544833 | |
| 0.097 | 0.107 | 0.193 | Cyclooxygenase 3 inhibitor | 0.136 0.061 CHEMBL3544797 0.145 0.052 CHEMBL3544835 0.193 0.021 CHEMBL3544799 0.136 0.061 CHEMBL3544833 | CHEMBL3544799 | |
| 0.07 | 0.081 | 0.157 | Antineoplastic alkaloid | 0.157 0.025 CHEMBL3544797 0.09 0.054 CHEMBL3544836 | CHEMBL3544797 | |
| 0.106 | 0.117 | 0.29 | Peroxidase inhibitor | 0.148 0.079 CHEMBL3544797 0.123 0.097 CHEMBL3544834 0.122 0.098 CHEMBL3544836 0.142 0.082 CHEMBL3544798 0.29 0.039 CHEMBL3544835 0.16 0.073 CHEMBL3544833 | CHEMBL3544835 | |
| 0.011 | 0.022 | 0.107 | Progesterone agonist | 0.107 0.003 CHEMBL3544834 | CHEMBL3544834 | |
| 0.024 | 0.035 | 0.037 | Purinergic P2Y15 antagonist | 0.037 0.009 CHEMBL3544797 0.031 0.015 CHEMBL3544835 | CHEMBL3544797 | |
| 0.09 | 0.102 | 0.149 | Cholesterol synthesis inhibitor | 0.132 0.056 CHEMBL3544797 0.104 0.083 CHEMBL3544834 0.107 0.079 CHEMBL3544798 0.137 0.052 CHEMBL3544835 0.149 0.045 CHEMBL3544833 | CHEMBL3544833 | |
| 0.078 | 0.09 | 0.125 | Creatine kinase inhibitor | 0.125 0.037 CHEMBL3544797 0.089 0.073 CHEMBL3544834 0.091 0.07 CHEMBL3544836 0.105 0.054 CHEMBL3544798 0.09 0.071 CHEMBL3544835 0.099 0.061 CHEMBL3544833 | CHEMBL3544797 | |
| 0.016 | 0.029 | 0.044 | Retinoid X gamma receptor agonist | 0.044 0.006 CHEMBL3544833 | CHEMBL3544833 | |
| 0.025 | 0.038 | 0.05 | Fumarate hydratase inhibitor | 0.05 0.013 CHEMBL3544797 0.039 0.019 CHEMBL3544836 0.034 0.024 CHEMBL3544835 0.048 0.014 CHEMBL3544833 | CHEMBL3544797 | |
| 0.032 | 0.045 | 0.044 | Glutamate (mGluR8) agonist | 0.038 0.025 CHEMBL3544836 0.044 0.017 CHEMBL3544833 | CHEMBL3544833 | |
| 0.03 | 0.044 | 0.036 | Delayed rectifier potassium channel blocker | 0.036 0.028 CHEMBL3544797 | CHEMBL3544797 | |
| 0.042 | 0.056 | 0.053 | Potassium channel (Inward rectifier) activator | 0.053 0.03 CHEMBL3544797 | CHEMBL3544797 | |
| 0.047 | 0.06 | 0.065 | Acetylcholine M3 receptor antagonist | 0.057 0.045 CHEMBL3544836 0.065 0.036 CHEMBL3544835 | CHEMBL3544835 | |
| 0.044 | 0.058 | 0.049 | Cyclin B inhibitor | 0.049 0.048 CHEMBL3544834 | CHEMBL3544834 | |
| 0.154 | 0.169 | 0.165 | ErbB-1 antagonist | 0.165 0.142 CHEMBL3544834 | CHEMBL3544834 | |
| 0.039 | 0.054 | 0.049 | Parathyroid hormone antagonist | 0.049 0.023 CHEMBL3544797 | CHEMBL3544797 | |
| 0.11 | 0.125 | 0.138 | Acetylcholine M1 receptor antagonist | 0.138 0.087 CHEMBL3544835 | CHEMBL3544835 | |
| 0.022 | 0.038 | 0.028 | CXC chemokine 3 receptor antagonist | 0.028 0.027 CHEMBL3544833 | CHEMBL3544833 | |
| 0.013 | 0.029 | 0.021 | 5-Alpha-reductase 2 inhibitor | 0.019 0.014 CHEMBL3544834 0.021 0.012 CHEMBL3544835 0.019 0.014 CHEMBL3544833 | CHEMBL3544835 | |
| 0.051 | 0.066 | 0.095 | Transcription factor AP-1 inhibitor | 0.056 0.054 CHEMBL3544797 0.058 0.049 CHEMBL3544834 0.095 0.014 CHEMBL3544798 0.072 0.028 CHEMBL3544799 | CHEMBL3544798 | |
| 0.034 | 0.05 | 0.047 | Sphingosine kinase 1 inhibitor | 0.047 0.02 CHEMBL3544797 0.046 0.02 CHEMBL3544836 0.044 0.024 CHEMBL3544798 0.038 0.037 CHEMBL3544835 | CHEMBL3544797 | |
| 0.041 | 0.057 | 0.068 | GABA A receptor antagonist | 0.068 0.026 CHEMBL3544834 | CHEMBL3544834 | |
| 0.04 | 0.056 | 0.05 | Potassium channel (ATP-sensitive) activator | 0.05 0.03 CHEMBL3544797 | CHEMBL3544797 | |
| 0.039 | 0.057 | 0.057 | Lysophosphatidic acid 3 receptor antagonist | 0.053 0.031 CHEMBL3544836 0.057 0.026 CHEMBL3544835 0.054 0.03 CHEMBL3544833 | CHEMBL3544835 | |
| 0.027 | 0.044 | 0.034 | Glutamate (mGluR3) agonist | 0.031 0.027 CHEMBL3544797 0.033 0.021 CHEMBL3544836 0.034 0.017 CHEMBL3544833 | CHEMBL3544833 | |
| 0.067 | 0.085 | 0.133 | NMDA receptor antagonist | 0.089 0.055 CHEMBL3544797 0.082 0.063 CHEMBL3544836 0.133 0.03 CHEMBL3544833 | CHEMBL3544833 | |
| 0.042 | 0.061 | 0.056 | 3(or 17)beta-hydroxysteroid dehydrogenase inhibitor | 0.056 0.034 CHEMBL3544797 0.053 0.038 CHEMBL3544834 | CHEMBL3544797 | |
| 0.027 | 0.045 | 0.039 | Retinoid X alpha receptor antagonist | 0.039 0.016 CHEMBL3544833 | CHEMBL3544833 | |
| 0.041 | 0.06 | 0.068 | GABA receptor antagonist | 0.068 0.027 CHEMBL3544834 | CHEMBL3544834 | |
| 0.034 | 0.053 | 0.138 | Mannosidase inhibitor | 0.069 0.012 CHEMBL3544797 0.066 0.014 CHEMBL3544836 0.064 0.014 CHEMBL3544798 0.058 0.018 CHEMBL3544835 0.138 0.004 CHEMBL3544799 0.045 0.032 CHEMBL3544833 | CHEMBL3544799 | |
| 0.007 | 0.026 | 0.013 | Immunosuppressant Cyclosporine-like | 0.013 0.006 CHEMBL3544835 | CHEMBL3544835 | |
| 0.021 | 0.041 | 0.03 | Retinoid X gamma receptor antagonist | 0.03 0.013 CHEMBL3544833 | CHEMBL3544833 | |
| 0.029 | 0.05 | 0.044 | Retinoid X receptor antagonist | 0.044 0.019 CHEMBL3544833 | CHEMBL3544833 | |
| 0.111 | 0.133 | 0.172 | MAP3K9 inhibitor | 0.152 0.057 CHEMBL3544836 0.145 0.067 CHEMBL3544798 0.172 0.033 CHEMBL3544835 | CHEMBL3544835 | |
| 0.026 | 0.048 | 0.033 | Angiotensin II receptor antagonist | 0.033 0.027 CHEMBL3544836 | CHEMBL3544836 | |
| 0.014 | 0.036 | 0.03 | Antibiotic Anthracycline-like | 0.02 0.011 CHEMBL3544797 0.018 0.017 CHEMBL3544835 0.03 0.004 CHEMBL3544799 | CHEMBL3544799 | |
| 0.016 | 0.038 | 0.021 | Neuraminidase (Influenza B) inhibitor | 0.02 0.018 CHEMBL3544836 0.021 0.015 CHEMBL3544835 | CHEMBL3544835 | |
| 0.032 | 0.054 | 0.041 | Angiotensin AT1 receptor antagonist | 0.041 0.031 CHEMBL3544836 | CHEMBL3544836 | |
| 0.062 | 0.084 | 0.071 | S-adenosyl-L-methionine decarboxylase inhibitor | 0.071 0.057 CHEMBL3544797 | CHEMBL3544797 | |
| 0.026 | 0.048 | 0.032 | Carboxypeptidase B inhibitor | 0.032 0.025 CHEMBL3544833 | CHEMBL3544833 | |
| 0.023 | 0.046 | 0.051 | Retinoid X alpha receptor agonist | 0.051 0.014 CHEMBL3544833 | CHEMBL3544833 | |
| 0.014 | 0.038 | 0.028 | Hypoxanthine phosphoribosyltransferase inhibitor | 0.028 0.019 CHEMBL3544797 0.025 0.022 CHEMBL3544836 | CHEMBL3544797 | |
| 0.013 | 0.037 | 0.036 | Retinoid X beta receptor agonist | 0.036 0.007 CHEMBL3544833 | CHEMBL3544833 | |
| 0.022 | 0.046 | 0.029 | Hedgehog signaling activator | 0.029 0.015 CHEMBL3544797 | CHEMBL3544797 | |
| 0.125 | 0.15 | 0.14 | Heat shock protein 70 antagonist | 0.14 0.076 CHEMBL3544797 | CHEMBL3544797 | |
| 0.06 | 0.086 | 0.131 | Phosphodiesterase IV inhibitor | 0.131 0.029 CHEMBL3544834 0.114 0.036 CHEMBL3544835 | CHEMBL3544834 | |
| 0.018 | 0.045 | 0.03 | Thyroid hormone agonist | 0.03 0.012 CHEMBL3544833 | CHEMBL3544833 | |
| 0.045 | 0.071 | 0.059 | Acetylcholine M5 receptor antagonist | 0.059 0.043 CHEMBL3544835 | CHEMBL3544835 | |
| 0.126 | 0.152 | 0.158 | 3C-like protease (Human coronavirus) inhibitor | 0.158 0.088 CHEMBL3544834 | CHEMBL3544834 | |
| 0.042 | 0.07 | 0.116 | NMDA receptor glycine site agonist | 0.116 0.01 CHEMBL3544833 | CHEMBL3544833 | |
| 0.052 | 0.08 | 0.063 | Heme oxygenase stimulant | 0.063 0.039 CHEMBL3544834 | CHEMBL3544834 | |
| 0.013 | 0.042 | 0.037 | NMDA receptor glycine site antagonist | 0.037 0.009 CHEMBL3544833 | CHEMBL3544833 | |
| 0.033 | 0.063 | 0.061 | Ornithine carbamoyltransferase inhibitor | 0.061 0.031 CHEMBL3544797 0.054 0.036 CHEMBL3544836 0.052 0.037 CHEMBL3544798 0.061 0.031 CHEMBL3544833 | CHEMBL3544833 | |
| 0.083 | 0.113 | 0.112 | Protein kinase C gamma inhibitor | 0.096 0.085 CHEMBL3544834 0.111 0.061 CHEMBL3544836 0.101 0.074 CHEMBL3544798 0.112 0.059 CHEMBL3544835 | CHEMBL3544835 | |
| 0.051 | 0.082 | 0.078 | Interferon inducer | 0.068 0.037 CHEMBL3544797 0.076 0.027 CHEMBL3544836 0.078 0.026 CHEMBL3544799 | CHEMBL3544799 | |
| 0.02 | 0.052 | 0.037 | Lysophosphatidic acid 2 receptor antagonist | 0.037 0.014 CHEMBL3544835 | CHEMBL3544835 | |
| 0.154 | 0.186 | 0.175 | 5 Hydroxytryptamine 1E antagonist | 0.175 0.16 CHEMBL3544834 | CHEMBL3544834 | |
| 0.018 | 0.05 | 0.026 | Glutamate (mGluR1) agonist | 0.026 0.014 CHEMBL3544833 | CHEMBL3544833 | |
| 0.052 | 0.085 | 0.115 | Glutamate decarboxylase inhibitor | 0.065 0.061 CHEMBL3544834 0.065 0.061 CHEMBL3544836 0.069 0.057 CHEMBL3544798 0.09 0.036 CHEMBL3544835 0.115 0.023 CHEMBL3544833 | CHEMBL3544833 | |
| 0.007 | 0.041 | 0.02 | Ileal bile acid transport inhibitor | 0.02 0.009 CHEMBL3544797 | CHEMBL3544797 | |
| 0.025 | 0.059 | 0.043 | Glutamate (mGluR3) antagonist | 0.038 0.024 CHEMBL3544836 0.043 0.018 CHEMBL3544833 | CHEMBL3544833 | |
| 0.113 | 0.147 | 0.146 | Sphingosine 1-phosphate receptor 5 antagonist | 0.125 0.112 CHEMBL3544798 0.146 0.067 CHEMBL3544833 | CHEMBL3544833 | |
| 0.118 | 0.155 | 0.175 | MAP kinase kinase 2 inhibitor | 0.162 0.111 CHEMBL3544834 0.175 0.1 CHEMBL3544798 | CHEMBL3544798 | |
| 0.048 | 0.085 | 0.143 | Histidine decarboxylase inhibitor | 0.09 0.037 CHEMBL3544797 0.113 0.028 CHEMBL3544836 0.143 0.02 CHEMBL3544833 | CHEMBL3544833 | |
| 0.046 | 0.084 | 0.103 | Phenylalanine 4-hydroxylase inhibitor | 0.077 0.039 CHEMBL3544797 0.062 0.056 CHEMBL3544836 0.082 0.036 CHEMBL3544798 0.103 0.024 CHEMBL3544835 0.091 0.03 CHEMBL3544833 | CHEMBL3544835 | |
| 0.127 | 0.167 | 0.144 | Cyclin-dependent kinase 3 inhibitor | 0.144 0.111 CHEMBL3544836 0.136 0.135 CHEMBL3544798 | CHEMBL3544836 | |
| 0.066 | 0.106 | 0.094 | Protein kinase C mu inhibitor | 0.086 0.073 CHEMBL3544797 0.094 0.063 CHEMBL3544834 | CHEMBL3544834 | |
| 0.085 | 0.129 | 0.114 | Aldehyde dehydrogenase inhibitor | 0.114 0.077 CHEMBL3544834 0.11 0.082 CHEMBL3544836 0.102 0.094 CHEMBL3544798 | CHEMBL3544834 | |
| 0.027 | 0.071 | 0.033 | Adenosine uptake inhibitor | 0.033 0.032 CHEMBL3544834 | CHEMBL3544834 | |
| 0.035 | 0.08 | 0.063 | Aconitate hydratase inhibitor | 0.063 0.023 CHEMBL3544833 | CHEMBL3544833 | |
| 0.014 | 0.058 | 0.024 | Lysine carboxypeptidase inhibitor | 0.024 0.023 CHEMBL3544833 | CHEMBL3544833 | |
| 0.077 | 0.122 | 0.12 | Mucolytic | 0.12 0.055 CHEMBL3544797 0.114 0.06 CHEMBL3544836 0.113 0.062 CHEMBL3544798 0.11 0.064 CHEMBL3544835 0.12 0.054 CHEMBL3544833 | CHEMBL3544833 | |
| 0.015 | 0.063 | 0.032 | Sirtuin 2 inhibitor | 0.032 0.023 CHEMBL3544834 | CHEMBL3544834 | |
| 0.012 | 0.062 | 0.052 | AMPA 3 receptor antagonist | 0.052 0.008 CHEMBL3544833 | CHEMBL3544833 | |
| 0.048 | 0.099 | 0.077 | NAD(P)H dehydrogenase (quinone) inhibitor | 0.077 0.053 CHEMBL3544797 0.074 0.057 CHEMBL3544836 | CHEMBL3544797 | |
| 0.021 | 0.073 | 0.035 | Toll-Like receptor 2 agonist | 0.035 0.034 CHEMBL3544799 | CHEMBL3544799 | |
| 0.025 | 0.076 | 0.038 | Guanylate cyclase inhibitor | 0.038 0.037 CHEMBL3544836 | CHEMBL3544836 | |
| 0.015 | 0.067 | 0.052 | Kainate receptor 2 antagonist | 0.052 0.015 CHEMBL3544833 | CHEMBL3544833 | |
| 0.012 | 0.064 | 0.053 | Arginase inhibitor | 0.053 0.013 CHEMBL3544799 0.036 0.026 CHEMBL3544833 | CHEMBL3544799 | |
| 0.072 | 0.125 | 0.099 | Anesthetic local | 0.099 0.084 CHEMBL3544835 | CHEMBL3544835 | |
| 0.018 | 0.072 | 0.061 | Kainate receptor antagonist | 0.061 0.016 CHEMBL3544833 | CHEMBL3544833 | |
| 0.063 | 0.117 | 0.093 | Alcohol dehydrogenase inhibitor | 0.085 0.072 CHEMBL3544836 0.088 0.067 CHEMBL3544798 0.093 0.06 CHEMBL3544833 | CHEMBL3544833 | |
| 0.168 | 0.224 | 0.605 | Antithrombotic | 0.226 0.147 CHEMBL3544797 0.262 0.117 CHEMBL3544836 0.259 0.119 CHEMBL3544835 0.605 0.016 CHEMBL3544799 0.285 0.099 CHEMBL3544833 | CHEMBL3544799 | |
| 0.037 | 0.093 | 0.058 | Sphingosine kinase 2 inhibitor | 0.058 0.035 CHEMBL3544797 0.056 0.037 CHEMBL3544836 | CHEMBL3544797 | |
| 0.04 | 0.099 | 0.069 | Purinergic P2X1 antagonist | 0.069 0.033 CHEMBL3544797 0.055 0.051 CHEMBL3544834 | CHEMBL3544797 | |
| 0.031 | 0.09 | 0.068 | Diacylglycerol O-acyltransferase inhibitor | 0.068 0.02 CHEMBL3544833 | CHEMBL3544833 | |
| 0.007 | 0.066 | 0.051 | AMPA 1 receptor antagonist | 0.051 0.011 CHEMBL3544833 | CHEMBL3544833 | |
| 0.068 | 0.128 | 0.089 | Alpha 2b adrenoreceptor antagonist | 0.089 0.087 CHEMBL3544835 | CHEMBL3544835 | |
| 0.071 | 0.132 | 0.096 | Glutamate release inhibitor | 0.096 0.049 CHEMBL3544835 | CHEMBL3544835 | |
| 0.031 | 0.091 | 0.046 | Glutamate (mGluR group III) antagonist | 0.046 0.026 CHEMBL3544833 | CHEMBL3544833 | |
| 0.009 | 0.071 | 0.03 | RNA-directed RNA polymerase stimulant | 0.03 0.021 CHEMBL3544797 | CHEMBL3544797 | |
| 0.03 | 0.091 | 0.048 | Glutamate (mGluR4) antagonist | 0.048 0.023 CHEMBL3544833 | CHEMBL3544833 | |
| 0.066 | 0.128 | 0.119 | Lanosterol 14 alpha demethylase inhibitor | 0.104 0.05 CHEMBL3544797 0.119 0.032 CHEMBL3544835 | CHEMBL3544835 | |
| 0.04 | 0.103 | 0.121 | Catalase inhibitor | 0.072 0.053 CHEMBL3544836 0.069 0.056 CHEMBL3544798 0.087 0.044 CHEMBL3544835 0.121 0.033 CHEMBL3544833 | CHEMBL3544833 | |
| 0.028 | 0.09 | 0.057 | Microtubule stabilization | 0.044 0.036 CHEMBL3544797 0.057 0.019 CHEMBL3544799 | CHEMBL3544799 | |
| 0.067 | 0.131 | 0.088 | Hematopoietic | 0.083 0.065 CHEMBL3544834 0.079 0.076 CHEMBL3544835 0.088 0.053 CHEMBL3544833 | CHEMBL3544833 | |
| 0.022 | 0.087 | 0.056 | Adenosine deaminase inhibitor | 0.056 0.025 CHEMBL3544797 0.051 0.029 CHEMBL3544836 | CHEMBL3544797 | |
| 0.14 | 0.205 | 0.18 | MAP-kinase-activated kinase 5 inhibitor | 0.18 0.132 CHEMBL3544834 | CHEMBL3544834 | |
| 0.114 | 0.183 | 0.191 | Insulin sensitizer | 0.171 0.106 CHEMBL3544797 0.175 0.101 CHEMBL3544835 0.191 0.083 CHEMBL3544833 | CHEMBL3544833 | |
| 0.036 | 0.106 | 0.071 | Sphingosine 1-phosphate receptor 4 agonist | 0.071 0.043 CHEMBL3544833 | CHEMBL3544833 | |
| 0.182 | 0.253 | 0.607 | Antibacterial | 0.38 0.086 CHEMBL3544797 0.231 0.195 CHEMBL3544834 0.297 0.138 CHEMBL3544836 0.436 0.062 CHEMBL3544835 0.607 0.018 CHEMBL3544799 | CHEMBL3544799 | |
| 0.004 | 0.076 | 0.02 | Kainate receptor 1 antagonist | 0.02 0.015 CHEMBL3544833 | CHEMBL3544833 | |
| 0.113 | 0.185 | 0.302 | Hypolipemic | 0.302 0.048 CHEMBL3544797 0.202 0.093 CHEMBL3544836 0.295 0.05 CHEMBL3544799 0.168 0.12 CHEMBL3544833 | CHEMBL3544797 | |
| 0.017 | 0.09 | 0.062 | NMDA receptor subunit 3A antagonist | 0.062 0.016 CHEMBL3544833 | CHEMBL3544833 | |
| 0.057 | 0.131 | 0.089 | GABA B receptor agonist | 0.075 0.052 CHEMBL3544834 0.089 0.027 CHEMBL3544833 | CHEMBL3544833 | |
| 0.069 | 0.144 | 0.203 | Alkylator | 0.13 0.059 CHEMBL3544836 0.121 0.067 CHEMBL3544835 0.203 0.025 CHEMBL3544799 | CHEMBL3544799 | |
| 0.022 | 0.099 | 0.053 | NMDA receptor subunit 3B antagonist | 0.053 0.023 CHEMBL3544833 | CHEMBL3544833 | |
| 0.043 | 0.12 | 0.06 | Leukotriene C antagonist | 0.06 0.028 CHEMBL3544833 | CHEMBL3544833 | |
| 0.105 | 0.183 | 0.174 | Tumour necrosis factor antagonist | 0.129 0.128 CHEMBL3544797 0.174 0.072 CHEMBL3544834 | CHEMBL3544834 | |
| 0.011 | 0.092 | 0.033 | Prostaglandin agonist | 0.033 0.019 CHEMBL3544797 | CHEMBL3544797 | |
| 0.027 | 0.111 | 0.039 | Leukotriene C4 antagonist | 0.039 0.026 CHEMBL3544833 | CHEMBL3544833 | |
| 0.033 | 0.117 | 0.18 | Antineoplastic antibiotic | 0.123 0.037 CHEMBL3544797 0.068 0.067 CHEMBL3544835 0.18 0.025 CHEMBL3544799 | CHEMBL3544799 | |
| 0.018 | 0.102 | 0.039 | Toll-Like receptor 4 agonist | 0.039 0.005 CHEMBL3544799 | CHEMBL3544799 | |
| 0.057 | 0.143 | 0.158 | Expectorant | 0.1 0.068 CHEMBL3544797 0.11 0.058 CHEMBL3544836 0.088 0.084 CHEMBL3544798 0.089 0.083 CHEMBL3544835 0.158 0.032 CHEMBL3544799 0.093 0.078 CHEMBL3544833 | CHEMBL3544799 | |
| 0.009 | 0.099 | 0.051 | Sodium/glucose cotransporter 2 inhibitor | 0.051 0.006 CHEMBL3544799 | CHEMBL3544799 | |
| 0.023 | 0.115 | 0.059 | Mineralocorticoid receptor antagonist | 0.059 0.02 CHEMBL3544834 | CHEMBL3544834 | |
| 0.025 | 0.118 | 0.039 | Glucose-6-phosphate dehydrogenase inhibitor | 0.039 0.023 CHEMBL3544834 | CHEMBL3544834 | |
| 0.044 | 0.138 | 0.153 | Somatostatin 1 agonist | 0.088 0.043 CHEMBL3544836 0.153 0.013 CHEMBL3544835 | CHEMBL3544835 | |
| 0.024 | 0.118 | 0.057 | Neutrophil collagenase inhibitor | 0.057 0.054 CHEMBL3544833 | CHEMBL3544833 | |
| 0.059 | 0.155 | 0.105 | Cystathionine beta-synthase inhibitor | 0.093 0.085 CHEMBL3544797 0.105 0.071 CHEMBL3544833 | CHEMBL3544833 | |
| 0.084 | 0.18 | 0.208 | Cell wall synthesis inhibitor | 0.143 0.072 CHEMBL3544797 0.208 0.027 CHEMBL3544835 0.187 0.036 CHEMBL3544799 0.113 0.11 CHEMBL3544833 | CHEMBL3544835 | |
| 0.051 | 0.154 | 0.082 | HIV-1 integrase (Overall Integration) inhibitor | 0.082 0.074 CHEMBL3544836 | CHEMBL3544836 | |
| 0.035 | 0.138 | 0.069 | Beta adrenoreceptor antagonist | 0.069 0.04 CHEMBL3544835 | CHEMBL3544835 | |
| 0.065 | 0.17 | 0.098 | Caspase 3 inhibitor | 0.098 0.095 CHEMBL3544833 | CHEMBL3544833 | |
| 0.121 | 0.226 | 0.17 | DNA damaging | 0.17 0.146 CHEMBL3544836 | CHEMBL3544836 | |
| 0.045 | 0.151 | 0.061 | Beta 2 adrenoreceptor agonist | 0.061 0.047 CHEMBL3544836 0.061 0.043 CHEMBL3544835 | CHEMBL3544835 | |
| 0.011 | 0.118 | 0.033 | Free fatty acid receptor 1 antagonist | 0.033 0.025 CHEMBL3544833 | CHEMBL3544833 | |
| 0.102 | 0.21 | 0.191 | Non-steroidal antiinflammatory agent | 0.145 0.121 CHEMBL3544836 0.19 0.079 CHEMBL3544799 0.191 0.079 CHEMBL3544833 | CHEMBL3544833 | |
| 0.012 | 0.125 | 0.037 | 1,3-Beta-glucan synthase inhibitor | 0.037 0.005 CHEMBL3544835 0.029 0.018 CHEMBL3544799 | CHEMBL3544835 | |
| 0.041 | 0.157 | 0.067 | Lipocortins synthesis agonist | 0.064 0.029 CHEMBL3544797 0.06 0.035 CHEMBL3544834 0.067 0.024 CHEMBL3544799 | CHEMBL3544799 | |
| 0.021 | 0.143 | 0.094 | Protein 50S ribosomal subunit inhibitor | 0.052 0.037 CHEMBL3544797 0.094 0.015 CHEMBL3544799 | CHEMBL3544799 | |
| 0.057 | 0.179 | 0.151 | Glutamate receptor antagonist | 0.151 0.05 CHEMBL3544833 | CHEMBL3544833 | |
| 0.007 | 0.13 | 0.016 | Thyroid hormone alpha agonist | 0.016 0.013 CHEMBL3544833 | CHEMBL3544833 | |
| 0.028 | 0.154 | 0.093 | Heparanase inhibitor | 0.093 0.004 CHEMBL3544799 | CHEMBL3544799 | |
| 0.041 | 0.167 | 0.11 | Adrenaline agonist | 0.079 0.059 CHEMBL3544836 0.11 0.031 CHEMBL3544835 | CHEMBL3544835 | |
| 0.087 | 0.214 | 0.428 | Nitric oxide antagonist | 0.157 0.089 CHEMBL3544797 0.128 0.123 CHEMBL3544834 0.168 0.083 CHEMBL3544836 0.138 0.108 CHEMBL3544798 0.222 0.06 CHEMBL3544835 0.428 0.022 CHEMBL3544799 0.133 0.114 CHEMBL3544833 | CHEMBL3544799 | |
| 0.103 | 0.233 | 0.153 | ATPase inhibitor | 0.153 0.096 CHEMBL3544797 0.136 0.128 CHEMBL3544799 | CHEMBL3544797 | |
| 0.031 | 0.168 | 0.052 | Glucosylceramidase inhibitor | 0.052 0.044 CHEMBL3544797 | CHEMBL3544797 | |
| 0.055 | 0.192 | 0.283 | Amylase inhibitor | 0.147 0.065 CHEMBL3544797 0.122 0.08 CHEMBL3544836 0.105 0.092 CHEMBL3544835 0.283 0.021 CHEMBL3544799 | CHEMBL3544799 | |
| 0.039 | 0.179 | 0.19 | Topoisomerase I inhibitor | 0.108 0.063 CHEMBL3544797 0.088 0.081 CHEMBL3544836 0.19 0.029 CHEMBL3544799 | CHEMBL3544799 | |
| 0.021 | 0.162 | 0.049 | Beta 1 adrenoreceptor antagonist | 0.049 0.048 CHEMBL3544835 | CHEMBL3544835 | |
| 0.036 | 0.178 | 0.152 | Monophenol monooxygenase inhibitor | 0.152 0.046 CHEMBL3544799 | CHEMBL3544799 | |
| 0.007 | 0.151 | 0.022 | Corticosteroid-like | 0.022 0.014 CHEMBL3544799 | CHEMBL3544799 | |
| 0.082 | 0.226 | 0.159 | DNA repair enzyme inhibitor | 0.159 0.024 CHEMBL3544799 | CHEMBL3544799 | |
| 0.046 | 0.197 | 0.071 | Estrogen receptor alpha antagonist | 0.071 0.066 CHEMBL3544797 | CHEMBL3544797 | |
| 0.015 | 0.171 | 0.16 | Aldose reductase inhibitor | 0.053 0.036 CHEMBL3544799 0.16 0.01 CHEMBL3544833 | CHEMBL3544833 | |
| 0.065 | 0.221 | 0.765 | Angiogenesis stimulant | 0.234 0.078 CHEMBL3544797 0.256 0.067 CHEMBL3544836 0.183 0.103 CHEMBL3544798 0.765 0.004 CHEMBL3544799 0.208 0.09 CHEMBL3544833 | CHEMBL3544799 | |
| 0.015 | 0.172 | 0.042 | Growth hormone release inhibitor | 0.042 0.029 CHEMBL3544835 | CHEMBL3544835 | |
| 0.085 | 0.244 | 0.145 | Interleukin 6 antagonist | 0.136 0.113 CHEMBL3544797 0.139 0.106 CHEMBL3544798 0.145 0.097 CHEMBL3544799 | CHEMBL3544799 | |
| 0.026 | 0.189 | 0.05 | Thromboxane synthase inhibitor | 0.05 0.048 CHEMBL3544833 | CHEMBL3544833 | |
| 0.022 | 0.186 | 0.119 | HIV-1 reverse transcriptase inhibitor | 0.119 0.023 CHEMBL3544797 | CHEMBL3544797 | |
| 0.054 | 0.221 | 0.409 | Phosphodiesterase inhibitor | 0.129 0.074 CHEMBL3544834 0.409 0.006 CHEMBL3544835 | CHEMBL3544835 | |
| 0.014 | 0.184 | 0.104 | Phosphodiesterase 4A inhibitor | 0.104 0.014 CHEMBL3544834 | CHEMBL3544834 | |
| 0.05 | 0.227 | 0.158 | Transcription factor NF kappa B stimulant | 0.085 0.06 CHEMBL3544836 0.158 0.014 CHEMBL3544799 | CHEMBL3544799 | |
| 0.047 | 0.227 | 0.158 | Beta glucuronidase inhibitor | 0.094 0.08 CHEMBL3544797 0.158 0.021 CHEMBL3544799 | CHEMBL3544799 | |
| 0.047 | 0.229 | 0.193 | DNA polymerase I inhibitor | 0.142 0.054 CHEMBL3544797 0.187 0.032 CHEMBL3544836 0.193 0.03 CHEMBL3544799 | CHEMBL3544799 | |
| 0.12 | 0.306 | 0.364 | Peptidyltransferase inhibitor | 0.254 0.048 CHEMBL3544797 0.164 0.16 CHEMBL3544836 0.209 0.088 CHEMBL3544798 0.265 0.041 CHEMBL3544835 0.364 0.01 CHEMBL3544799 0.171 0.145 CHEMBL3544833 | CHEMBL3544799 | |
| 0.076 | 0.262 | 0.186 | DNA methylase inhibitor | 0.186 0.089 CHEMBL3544799 | CHEMBL3544799 | |
| 0.066 | 0.253 | 0.119 | Phospholipase A2 inhibitor | 0.119 0.118 CHEMBL3544833 | CHEMBL3544833 | |
| 0.019 | 0.208 | 0.038 | Glutamate (mGluR8) antagonist | 0.038 0.02 CHEMBL3544833 | CHEMBL3544833 | |
| 0.046 | 0.236 | 0.189 | AMP-activated protein kinase stimulant | 0.126 0.044 CHEMBL3544797 0.189 0.013 CHEMBL3544799 | CHEMBL3544799 | |
| 0.111 | 0.316 | 0.508 | Immunosuppressant | 0.393 0.066 CHEMBL3544797 0.292 0.12 CHEMBL3544836 0.236 0.16 CHEMBL3544798 0.424 0.055 CHEMBL3544835 0.508 0.031 CHEMBL3544799 | CHEMBL3544799 | |
| 0.006 | 0.213 | 0.141 | Diacylglycerol O-acyltransferase 1 inhibitor | 0.141 0.004 CHEMBL3544833 | CHEMBL3544833 | |
| 0.056 | 0.265 | 0.158 | EphB2 antagonist | 0.158 0.122 CHEMBL3544835 | CHEMBL3544835 | |
| 0.071 | 0.279 | 0.441 | Hepatoprotectant | 0.164 0.095 CHEMBL3544797 0.201 0.064 CHEMBL3544834 0.187 0.074 CHEMBL3544836 0.441 0.01 CHEMBL3544799 0.143 0.118 CHEMBL3544833 | CHEMBL3544799 | |
| 0.027 | 0.239 | 0.089 | Adrenaline antagonist | 0.089 0.061 CHEMBL3544835 | CHEMBL3544835 | |
| 0.028 | 0.24 | 0.09 | Antiadrenergic | 0.09 0.062 CHEMBL3544835 | CHEMBL3544835 | |
| 0.01 | 0.227 | 0.057 | Somatostatin 1 antagonist | 0.057 0.017 CHEMBL3544835 | CHEMBL3544835 | |
| 0.083 | 0.34 | 0.143 | MAP kinase kinase 4 inhibitor | 0.143 0.078 CHEMBL3544798 | CHEMBL3544798 | |
| 0.037 | 0.301 | 0.086 | Xanthine oxidase inhibitor | 0.086 0.079 CHEMBL3544799 | CHEMBL3544799 | |
| 0.009 | 0.275 | 0.038 | Integrin alpha5beta1 antagonist | 0.038 0.033 CHEMBL3544833 | CHEMBL3544833 | |
| 0.006 | 0.274 | 0.079 | AMPA 2 receptor antagonist | 0.079 0.007 CHEMBL3544833 | CHEMBL3544833 | |
| 0.004 | 0.291 | 0.038 | Somatostatin 5 antagonist | 0.038 0.019 CHEMBL3544835 | CHEMBL3544835 | |
| 0.016 | 0.312 | 0.056 | Sphingosine 1-phosphate receptor 5 agonist | 0.056 0.033 CHEMBL3544833 | CHEMBL3544833 | |
| 0.007 | 0.309 | 0.021 | Somatostatin 4 antagonist | 0.021 0.02 CHEMBL3544835 | CHEMBL3544835 | |
| 0.048 | 0.352 | 0.119 | Farnesoid X receptor antagonist | 0.118 0.109 CHEMBL3544797 0.119 0.105 CHEMBL3544836 | CHEMBL3544836 | |
| 0.015 | 0.329 | 0.068 | Antibiotic Aminoglycoside-like | 0.068 0.006 CHEMBL3544799 | CHEMBL3544799 | |
| 0.005 | 0.321 | 0.02 | Integrin beta5 antagonist | 0.02 0.015 CHEMBL3544833 | CHEMBL3544833 | |
| 0.053 | 0.369 | 0.145 | Platelet aggregation inhibitor | 0.145 0.134 CHEMBL3544833 | CHEMBL3544833 | |
| 0.014 | 0.361 | 0.129 | CDC25A inhibitor | 0.129 0.017 CHEMBL3544798 0.068 0.06 CHEMBL3544799 | CHEMBL3544798 | |
| 0.034 | 0.4 | 0.126 | Electron transport complex I inhibitor | 0.126 0.04 CHEMBL3544835 | CHEMBL3544835 | |
| 0.011 | 0.38 | 0.047 | Neuraminidase (Influenza A) inhibitor | 0.047 0.029 CHEMBL3544799 | CHEMBL3544799 | |
| 0.043 | 0.42 | 0.361 | Platelet adhesion inhibitor | 0.361 0.017 CHEMBL3544799 | CHEMBL3544799 | |
| 0.007 | 0.406 | 0.056 | Cathepsin L2 inhibitor | 0.056 0.019 CHEMBL3544797 | CHEMBL3544797 | |
| 0.105 | 0.515 | 0.728 | Antiinflammatory | 0.718 0.028 CHEMBL3544797 0.383 0.15 CHEMBL3544836 0.728 0.026 CHEMBL3544835 0.725 0.026 CHEMBL3544799 0.308 0.208 CHEMBL3544833 | CHEMBL3544835 | |
| 0.024 | 0.453 | 0.073 | Adenine nucleotide translocase inhibitor | 0.073 0.013 CHEMBL3544799 | CHEMBL3544799 | |
| 0.004 | 0.44 | 0.034 | Leukotriene D4 antagonist | 0.034 0.013 CHEMBL3544833 | CHEMBL3544833 | |
| 0.003 | 0.453 | 0.019 | Free fatty acid receptor 1 agonist | 0.019 0.011 CHEMBL3544833 | CHEMBL3544833 | |
| 0.008 | 0.474 | 0.097 | Protein-tyrosine phosphatase 1B inhibitor | 0.097 0.081 CHEMBL3544799 | CHEMBL3544799 | |
| 0.017 | 0.507 | 0.084 | ATPase (Vacuolar H+) inhibitor | 0.081 0.075 CHEMBL3544797 0.084 0.068 CHEMBL3544799 | CHEMBL3544799 | |
| 0.006 | 0.509 | 0.057 | Neuraminidase inhibitor | 0.057 0.047 CHEMBL3544799 | CHEMBL3544799 | |
| 0.008 | 0.517 | 0.084 | CDC25B inhibitor | 0.084 0.025 CHEMBL3544798 | CHEMBL3544798 | |
| 0.004 | 0.528 | 0.016 | O6-alkylguanine-DNA alkyltransferase inhibitor | 0.016 0.014 CHEMBL3544799 | CHEMBL3544799 | |
| 0.015 | 0.569 | 0.197 | Lipid peroxidase inhibitor | 0.197 0.043 CHEMBL3544799 | CHEMBL3544799 | |
| 0.003 | 0.56 | 0.045 | GP IIb/IIIa receptor antagonist | 0.045 0.037 CHEMBL3544833 | CHEMBL3544833 | |
| 0.053 | 0.627 | 0.754 | Cyclophilin D inhibitor | 0.401 0.091 CHEMBL3544836 0.316 0.149 CHEMBL3544835 0.754 0.009 CHEMBL3544799 0.435 0.073 CHEMBL3544833 | CHEMBL3544799 | |
| 0.019 | 0.595 | 0.105 | Estrogen antagonist | 0.104 0.088 CHEMBL3544797 0.105 0.086 CHEMBL3544834 | CHEMBL3544834 | |
| 0.007 | 0.591 | 0.072 | Neuraminidase (influenza) inhibitor | 0.059 0.057 CHEMBL3544835 0.072 0.032 CHEMBL3544799 | CHEMBL3544799 | |
| 0.004 | 0.603 | 0.033 | Protein 30S ribosomal subunit inhibitor | 0.033 0.011 CHEMBL3544799 | CHEMBL3544799 | |
| 0.021 | 0.619 | 0.529 | Antioxidant | 0.529 0.017 CHEMBL3544799 | CHEMBL3544799 | |
| 0.014 | 0.62 | 0.239 | Anticoagulant | 0.239 0.041 CHEMBL3544799 | CHEMBL3544799 | |
| 0.035 | 0.646 | 0.236 | NOS3 expression enhancer | 0.236 0.029 CHEMBL3544799 | CHEMBL3544799 | |
| 0.01 | 0.623 | 0.091 | Estrogen receptor beta antagonist | 0.091 0.082 CHEMBL3544797 | CHEMBL3544797 | |
| 0.003 | 0.621 | 0.054 | Prostaglandin D2 antagonist | 0.054 0.006 CHEMBL3544833 | CHEMBL3544833 | |
| 0.046 | 0.685 | 0.419 | Apoptosis antagonist | 0.23 0.147 CHEMBL3544836 0.419 0.033 CHEMBL3544799 | CHEMBL3544799 | |
| 0.009 | 0.65 | 0.119 | Topoisomerase II inhibitor | 0.119 0.068 CHEMBL3544799 | CHEMBL3544799 | |
| 0.015 | 0.685 | 0.2 | Interleukin antagonist | 0.2 0.084 CHEMBL3544835 | CHEMBL3544835 | |
| 0.004 | 0.679 | 0.099 | Prostaglandin antagonist | 0.099 0.018 CHEMBL3544833 | CHEMBL3544833 | |
| 0.016 | 0.695 | 0.064 | DNA helicase inhibitor | 0.064 0.023 CHEMBL3544833 | CHEMBL3544833 | |
| 0.004 | 0.689 | 0.353 | Selectin antagonist | 0.353 0.004 CHEMBL3544799 | CHEMBL3544799 | |
| 0.034 | 0.721 | 0.546 | Apoptosis agonist | 0.546 0.061 CHEMBL3544799 | CHEMBL3544799 | |
| 0.008 | 0.713 | 0.049 | Phosphodiesterase 7A inhibitor | 0.049 0.043 CHEMBL3544834 | CHEMBL3544834 | |
| 0.006 | 0.73 | 0.116 | Bronchodilator | 0.116 0.047 CHEMBL3544835 | CHEMBL3544835 | |
| 0.022 | 0.754 | 0.079 | T cell inhibitor | 0.079 0.072 CHEMBL3544798 | CHEMBL3544798 | |
| 0.023 | 0.771 | 0.557 | Hypoglycemic | 0.557 0.011 CHEMBL3544799 | CHEMBL3544799 | |
| 0.015 | 0.765 | 0.13 | Nav1.4 sodium channel blocker | 0.13 0.044 CHEMBL3544835 | CHEMBL3544835 | |
| 0.009 | 0.761 | 0.047 | Carnitine palmitoyltransferase 1B inhibitor | 0.047 0.034 CHEMBL3544833 | CHEMBL3544833 | |
| 0.017 | 0.769 | 0.171 | Toll-Like receptor 4 antagonist | 0.171 0.012 CHEMBL3544799 | CHEMBL3544799 | |
| 0.011 | 0.79 | 0.071 | Factor IXa inhibitor | 0.071 0.02 CHEMBL3544799 | CHEMBL3544799 | |
| 0.01 | 0.818 | 0.18 | Insulin secretagoues | 0.18 0.048 CHEMBL3544799 | CHEMBL3544799 | |
| 0.006 | 0.82 | 0.437 | Free radical scavenger | 0.437 0.023 CHEMBL3544799 | CHEMBL3544799 | |
| 0.008 | 0.827 | 0.054 | Glucose-6-phosphate translocase inhibitor | 0.054 0.032 CHEMBL3544799 | CHEMBL3544799 | |
| 0.016 | 0.861 | 0.108 | Interleukin 4 antagonist | 0.108 0.104 CHEMBL3544799 | CHEMBL3544799 | |
| 0.005 | 0.89 | 0.091 | Topoisomerase II alpha inhibitor | 0.075 0.056 CHEMBL3544834 0.091 0.045 CHEMBL3544799 | CHEMBL3544799 | |
| 0.006 | 0.892 | 0.776 | Toll-Like receptor 7 agonist | 0.776 0.005 CHEMBL3544835 | CHEMBL3544835 | |
| 0.006 | 0.895 | 0.771 | Toll-Like receptor agonist | 0.771 0.005 CHEMBL3544835 | CHEMBL3544835 | |
| 0.005 | 0.896 | 0.193 | Cell adhesion inhibitor | 0.193 0.027 CHEMBL3544799 | CHEMBL3544799 | |
| 0.004 | 0.919 | 0.101 | Cell adhesion molecule inhibitor | 0.101 0.034 CHEMBL3544799 | CHEMBL3544799 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |