| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.912 | 0 | 0.912 | 5-Alpha-reductase 2 inhibitor | 0.71 0.001 CHEMBL4525755 0.835 0.001 CHEMBL3542374 | ||
| 0.909 | 0 | 0.909 | 5-Alpha-reductase 1 inhibitor | 0.714 0.001 CHEMBL4525755 0.795 0.001 CHEMBL3542374 | ||
| 0.898 | 0.001 | 0.976 | 5-Alpha-reductase inhibitor | 0.876 0.001 CHEMBL4525755 0.976 0 CHEMBL3542374 | CHEMBL3542374 | |
| 0.869 | 0.002 | 0.901 | Androgen antagonist | 0.901 0.002 CHEMBL4525755 0.677 0.003 CHEMBL3542374 | CHEMBL4525755 | |
| 0.475 | 0.002 | 0.488 | Androgen agonist | 0.488 0.002 CHEMBL4525755 0.377 0.003 CHEMBL3542374 | CHEMBL4525755 | |
| 0.436 | 0.009 | 0.441 | Sodium/bile acid cotransporter inhibitor | 0.43 0.01 CHEMBL4525755 0.441 0.009 CHEMBL3542374 | CHEMBL3542374 | |
| 0.334 | 0.015 | 0.338 | Lipocortins synthesis antagonist | 0.319 0.018 CHEMBL4525755 0.338 0.015 CHEMBL3542374 | CHEMBL3542374 | |
| 0.421 | 0.127 | 0.485 | Antiinflammatory | 0.444 0.113 CHEMBL4525755 0.485 0.094 CHEMBL3542374 | CHEMBL3542374 | |
| 0.288 | 0.016 | 0.407 | Antipruritic | 0.225 0.034 CHEMBL4525755 0.407 0.006 CHEMBL3542374 | CHEMBL3542374 | |
| 0.272 | 0.022 | 0.272 | NOS3 expression enhancer | 0.181 0.05 CHEMBL4525755 0.197 0.042 CHEMBL3542374 | ||
| 0.288 | 0.046 | 0.288 | Psychostimulant | 0.167 0.102 CHEMBL4525755 0.193 0.084 CHEMBL3542374 | ||
| 0.302 | 0.072 | 0.339 | Interleukin 2 agonist | 0.32 0.061 CHEMBL4525755 0.339 0.05 CHEMBL3542374 | CHEMBL3542374 | |
| 0.327 | 0.099 | 0.488 | Immunosuppressant | 0.488 0.036 CHEMBL4525755 0.377 0.073 CHEMBL3542374 | CHEMBL4525755 | |
| 0.246 | 0.031 | 0.345 | Diuretic | 0.345 0.017 CHEMBL4525755 0.184 0.051 CHEMBL3542374 | CHEMBL4525755 | |
| 0.183 | 0.017 | 0.183 | Pregnane X receptor agonist | 0.144 0.064 CHEMBL4525755 0.142 0.069 CHEMBL3542374 | ||
| 0.188 | 0.023 | 0.188 | Microtubule formation inhibitor | 0.155 0.035 CHEMBL4525755 0.161 0.032 CHEMBL3542374 | ||
| 0.243 | 0.084 | 0.353 | Interleukin agonist | 0.353 0.028 CHEMBL4525755 0.267 0.067 CHEMBL3542374 | CHEMBL4525755 | |
| 0.158 | 0.005 | 0.158 | Aldosterone antagonist | 0.11 0.008 CHEMBL4525755 0.088 0.009 CHEMBL3542374 | ||
| 0.156 | 0.015 | 0.156 | Anabolic | 0.134 0.028 CHEMBL4525755 0.145 0.021 CHEMBL3542374 | ||
| 0.162 | 0.024 | 0.162 | Antineoplastic alkaloid | 0.142 0.03 CHEMBL4525755 0.153 0.027 CHEMBL3542374 | ||
| 0.185 | 0.048 | 0.2 | Arachidonic acid antagonist | 0.199 0.034 CHEMBL4525755 0.2 0.033 CHEMBL3542374 | CHEMBL3542374 | |
| 0.161 | 0.04 | 0.161 | Proteasome inhibitor | 0.106 0.08 CHEMBL4525755 0.132 0.057 CHEMBL3542374 | ||
| 0.16 | 0.042 | 0.161 | Farnesoid X receptor antagonist | 0.16 0.042 CHEMBL4525755 0.161 0.041 CHEMBL3542374 | CHEMBL3542374 | |
| 0.236 | 0.123 | 0.236 | Ca(v)3.3 blocker | |||
| 0.107 | 0.004 | 0.107 | Lipocortins synthesis agonist | 0.103 0.005 CHEMBL4525755 0.102 0.005 CHEMBL3542374 | ||
| 0.107 | 0.008 | 0.107 | Gonadotropin-releasing hormone receptor agonist | 0.101 0.01 CHEMBL4525755 0.064 0.033 CHEMBL3542374 | ||
| 0.232 | 0.138 | 0.34 | Cholesterol antagonist | 0.34 0.069 CHEMBL4525755 0.303 0.089 CHEMBL3542374 | CHEMBL4525755 | |
| 0.159 | 0.067 | 0.17 | Interferon gamma antagonist | 0.16 0.066 CHEMBL4525755 0.17 0.057 CHEMBL3542374 | CHEMBL3542374 | |
| 0.096 | 0.008 | 0.096 | Mineralocorticoid receptor antagonist | 0.078 0.012 CHEMBL4525755 0.075 0.013 CHEMBL3542374 | ||
| 0.083 | 0.007 | 0.083 | Chemokine receptor agonist | 0.056 0.03 CHEMBL4525755 | ||
| 0.104 | 0.029 | 0.104 | Glycine receptor antagonist | 0.077 0.061 CHEMBL3542374 | ||
| 0.082 | 0.008 | 0.082 | RNA-directed RNA polymerase stimulant | 0.066 0.01 CHEMBL4525755 0.067 0.01 CHEMBL3542374 | ||
| 0.072 | 0.002 | 0.072 | Corticosteroid-like | 0.06 0.003 CHEMBL4525755 0.058 0.003 CHEMBL3542374 | ||
| 0.076 | 0.007 | 0.076 | Glucocorticoid antagonist | 0.063 0.01 CHEMBL4525755 0.063 0.01 CHEMBL3542374 | ||
| 0.109 | 0.047 | 0.109 | Prolactin inhibitor | 0.084 0.075 CHEMBL4525755 0.105 0.051 CHEMBL3542374 | ||
| 0.067 | 0.005 | 0.067 | Glucose-6-phosphate dehydrogenase inhibitor | 0.062 0.006 CHEMBL4525755 0.059 0.007 CHEMBL3542374 | ||
| 0.099 | 0.04 | 0.099 | Acetylcholine nicotinic antagonist | |||
| 0.059 | 0.001 | 0.059 | 3 Beta-hydroxy-delta 5-steroid dehydrogenase inhibitor | 0.046 0.001 CHEMBL4525755 0.046 0.001 CHEMBL3542374 | ||
| 0.078 | 0.02 | 0.078 | Bombesin 3 receptor antagonist | |||
| 0.203 | 0.146 | 0.203 | 5 Hydroxytryptamine uptake stimulant | 0.188 0.178 CHEMBL3542374 | ||
| 0.149 | 0.095 | 0.15 | Nitric oxide antagonist | 0.146 0.099 CHEMBL4525755 0.15 0.094 CHEMBL3542374 | CHEMBL3542374 | |
| 0.098 | 0.046 | 0.098 | Acetylcholine M3 receptor agonist | 0.076 0.064 CHEMBL4525755 | ||
| 0.12 | 0.07 | 0.12 | Acetylcholine antagonist | |||
| 0.122 | 0.072 | 0.122 | Cholinergic antagonist | |||
| 0.256 | 0.208 | 0.296 | Apoptosis agonist | 0.24 0.225 CHEMBL4525755 0.296 0.175 CHEMBL3542374 | CHEMBL3542374 | |
| 0.063 | 0.015 | 0.063 | Nicotinic acid receptor 1 agonist | 0.05 0.02 CHEMBL4525755 0.045 0.023 CHEMBL3542374 | ||
| 0.08 | 0.034 | 0.08 | Phospholipase D inhibitor | 0.069 0.055 CHEMBL4525755 0.071 0.051 CHEMBL3542374 | ||
| 0.048 | 0.005 | 0.048 | CXC chemokine receptor agonist | 0.036 0.023 CHEMBL4525755 | ||
| 0.056 | 0.013 | 0.056 | Nicotinic receptor beta4 subunit antagonist | 0.033 0.032 CHEMBL4525755 | ||
| 0.21 | 0.167 | 0.28 | Apoptosis antagonist | 0.28 0.1 CHEMBL3542374 | CHEMBL3542374 | |
| 0.08 | 0.038 | 0.093 | Glycine receptor agonist | 0.086 0.032 CHEMBL4525755 0.093 0.026 CHEMBL3542374 | CHEMBL3542374 | |
| 0.057 | 0.015 | 0.057 | Progesterone antagonist | 0.031 0.028 CHEMBL4525755 | ||
| 0.088 | 0.048 | 0.088 | Opioid kappa receptor antagonist | 0.086 0.05 CHEMBL3542374 | ||
| 0.15 | 0.11 | 0.196 | Hepatoprotectant | 0.188 0.073 CHEMBL4525755 0.196 0.067 CHEMBL3542374 | CHEMBL3542374 | |
| 0.042 | 0.005 | 0.042 | Glucocorticoid agonist | 0.03 0.006 CHEMBL4525755 0.025 0.007 CHEMBL3542374 | ||
| 0.066 | 0.031 | 0.066 | Heme oxygenase stimulant | 0.062 0.04 CHEMBL4525755 0.064 0.036 CHEMBL3542374 | ||
| 0.052 | 0.018 | 0.052 | Parathyroid hormone antagonist | 0.05 0.022 CHEMBL4525755 0.047 0.026 CHEMBL3542374 | ||
| 0.042 | 0.009 | 0.042 | Estrone sulfatase inhibitor | 0.024 0.013 CHEMBL4525755 0.024 0.013 CHEMBL3542374 | ||
| 0.181 | 0.152 | 0.236 | DNA synthesis inhibitor | 0.236 0.077 CHEMBL4525755 0.201 0.121 CHEMBL3542374 | CHEMBL4525755 | |
| 0.05 | 0.024 | 0.05 | Opioid kappa receptor agonist | 0.041 0.032 CHEMBL3542374 | ||
| 0.145 | 0.119 | 0.171 | Anesthetic general | 0.171 0.093 CHEMBL4525755 0.155 0.109 CHEMBL3542374 | CHEMBL4525755 | |
| 0.096 | 0.072 | 0.096 | Hedgehog signaling inhibitor | |||
| 0.032 | 0.009 | 0.032 | Steroid 17-alpha-hydroxylase/17,20 lyase inhibitor | |||
| 0.027 | 0.008 | 0.027 | Progesterone agonist | 0.02 0.011 CHEMBL4525755 0.021 0.01 CHEMBL3542374 | ||
| 0.102 | 0.084 | 0.124 | DNA polymerase I inhibitor | 0.114 0.073 CHEMBL4525755 0.124 0.065 CHEMBL3542374 | CHEMBL3542374 | |
| 0.033 | 0.015 | 0.033 | 11-Beta-hydroxysteroid dehydrogenase 2 inhibitor | |||
| 0.028 | 0.017 | 0.028 | Hedgehog signaling activator | |||
| 0.046 | 0.039 | 0.046 | HCV NS3/NS4A protease inhibitor | |||
| 0.022 | 0.015 | 0.022 | Vitamin D receptor antagonist | 0.022 0.015 CHEMBL4525755 0.021 0.017 CHEMBL3542374 | ||
| 0.164 | 0.16 | 0.299 | Peptidyltransferase inhibitor | 0.299 0.025 CHEMBL4525755 0.2 0.099 CHEMBL3542374 | CHEMBL4525755 | |
| 0.181 | 0.178 | 0.204 | Gastrin inhibitor | 0.204 0.143 CHEMBL3542374 | CHEMBL3542374 | |
| 0.054 | 0.053 | 0.054 | Ca(v)3.2 blocker | |||
| 0.018 | 0.017 | 0.018 | Progesterone receptor B antagonist | |||
| 0.063 | 0.067 | 0.067 | Na+ K+ transporting ATPase inhibitor | 0.067 0.063 CHEMBL4525755 | CHEMBL4525755 | |
| 0.116 | 0.128 | 0.149 | Growth hormone agonist | 0.125 0.113 CHEMBL4525755 0.149 0.088 CHEMBL3542374 | CHEMBL3542374 | |
| 0.012 | 0.031 | 0.017 | Vitamin D receptor agonist | 0.017 0.01 CHEMBL3542374 | CHEMBL3542374 | |
| 0.059 | 0.081 | 0.067 | CDC25A inhibitor | 0.067 0.062 CHEMBL3542374 | CHEMBL3542374 | |
| 0.129 | 0.176 | 0.275 | Immunostimulant | 0.185 0.129 CHEMBL4525755 0.275 0.087 CHEMBL3542374 | CHEMBL3542374 | |
| 0.107 | 0.228 | 0.144 | Phospholipase C inhibitor | 0.144 0.119 CHEMBL4525755 | CHEMBL4525755 | |
| 0.007 | 0.138 | 0.043 | Diacylglycerol O-acyltransferase 1 inhibitor | 0.043 0.012 CHEMBL3542374 | CHEMBL3542374 | |
| 0.02 | 0.173 | 0.053 | Diacylglycerol O-acyltransferase inhibitor | 0.053 0.032 CHEMBL3542374 | CHEMBL3542374 | |
| 0.105 | 0.374 | 0.445 | Toll-Like receptor 7 agonist | 0.445 0.045 CHEMBL3542374 | CHEMBL3542374 | |
| 0.102 | 0.382 | 0.441 | Toll-Like receptor agonist | 0.441 0.046 CHEMBL3542374 | CHEMBL3542374 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |