| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.687 | 0.003 | 0.687 | Dopamine D5 antagonist | 0.156 0.006 CHEMBL3544613 0.542 0.003 CHEMBL100454 0.63 0.003 CHEMBL440512 0.644 0.003 CHEMBL1125 0.501 0.003 CHEMBL3544641 0.399 0.003 CHEMBL3544615 | ||
| 0.534 | 0.003 | 0.708 | Acetylcholine M4 receptor antagonist | 0.082 0.044 CHEMBL3544613 0.394 0.004 CHEMBL100454 0.708 0.002 CHEMBL440512 0.4 0.003 CHEMBL1125 0.18 0.007 CHEMBL3544641 0.134 0.013 CHEMBL3544615 | CHEMBL440512 | |
| 0.512 | 0.003 | 0.609 | Dopamine D1 antagonist | 0.43 0.004 CHEMBL100454 0.609 0.003 CHEMBL440512 0.338 0.005 CHEMBL1125 0.202 0.01 CHEMBL3544641 0.101 0.025 CHEMBL3544615 | CHEMBL440512 | |
| 0.509 | 0.007 | 0.509 | 5 Hydroxytryptamine antagonist | 0.277 0.021 CHEMBL100454 0.444 0.009 CHEMBL440512 0.389 0.012 CHEMBL1125 0.13 0.059 CHEMBL3544641 | ||
| 0.504 | 0.006 | 0.547 | 5 Hydroxytryptamine 2 antagonist | 0.369 0.011 CHEMBL100454 0.547 0.005 CHEMBL440512 0.423 0.009 CHEMBL1125 0.175 0.037 CHEMBL3544641 0.133 0.052 CHEMBL3544615 | CHEMBL440512 | |
| 0.5 | 0.004 | 0.5 | 5 Hydroxytryptamine 1F antagonist | 0.404 0.005 CHEMBL100454 0.171 0.013 CHEMBL440512 0.462 0.004 CHEMBL1125 0.267 0.007 CHEMBL3544641 0.224 0.009 CHEMBL3544615 | ||
| 0.497 | 0.003 | 0.497 | 5 Hydroxytryptamine 3 antagonist | 0.151 0.009 CHEMBL100454 0.301 0.004 CHEMBL440512 0.362 0.004 CHEMBL1125 0.164 0.008 CHEMBL3544641 0.098 0.018 CHEMBL3544615 | ||
| 0.49 | 0.021 | 0.499 | MAP kinase kinase 6 inhibitor | 0.226 0.225 CHEMBL3544613 0.382 0.07 CHEMBL100454 0.409 0.053 CHEMBL440512 0.23 0.219 CHEMBL3544614 0.499 0.019 CHEMBL1125 0.406 0.055 CHEMBL3544641 0.41 0.053 CHEMBL3544615 | CHEMBL1125 | |
| 0.465 | 0.006 | 0.489 | Dopamine antagonist | 0.189 0.02 CHEMBL100454 0.489 0.005 CHEMBL440512 0.295 0.012 CHEMBL1125 0.083 0.046 CHEMBL3544641 | CHEMBL440512 | |
| 0.459 | 0.004 | 0.459 | Alpha 2a adrenoreceptor antagonist | 0.316 0.006 CHEMBL100454 0.308 0.006 CHEMBL440512 0.413 0.005 CHEMBL1125 0.106 0.034 CHEMBL3544641 0.092 0.041 CHEMBL3544615 | ||
| 0.455 | 0.004 | 0.455 | Dopamine D4 antagonist | 0.145 0.018 CHEMBL100454 0.16 0.016 CHEMBL440512 0.229 0.01 CHEMBL1125 0.092 0.029 CHEMBL3544641 | ||
| 0.456 | 0.006 | 0.521 | 5 Hydroxytryptamine 2B antagonist | 0.418 0.008 CHEMBL100454 0.521 0.005 CHEMBL440512 0.386 0.009 CHEMBL1125 0.16 0.037 CHEMBL3544641 0.13 0.051 CHEMBL3544615 | CHEMBL440512 | |
| 0.45 | 0.005 | 0.457 | 5 Hydroxytryptamine 2A antagonist | 0.183 0.022 CHEMBL100454 0.457 0.005 CHEMBL440512 0.364 0.008 CHEMBL1125 0.121 0.037 CHEMBL3544641 0.089 0.053 CHEMBL3544615 | CHEMBL440512 | |
| 0.445 | 0.002 | 0.445 | 5 Hydroxytryptamine 3A antagonist | 0.183 0.004 CHEMBL100454 0.144 0.005 CHEMBL440512 0.383 0.002 CHEMBL1125 0.196 0.004 CHEMBL3544641 0.156 0.005 CHEMBL3544615 | ||
| 0.445 | 0.004 | 0.445 | Alpha 1 adrenoreceptor agonist | 0.156 0.009 CHEMBL100454 0.08 0.023 CHEMBL440512 0.382 0.004 CHEMBL1125 0.106 0.015 CHEMBL3544641 0.087 0.02 CHEMBL3544615 | ||
| 0.398 | 0.005 | 0.398 | Alpha 2 adrenoreceptor antagonist | 0.265 0.01 CHEMBL100454 0.237 0.013 CHEMBL440512 0.359 0.006 CHEMBL1125 0.093 0.053 CHEMBL3544641 0.083 0.062 CHEMBL3544615 | ||
| 0.447 | 0.055 | 0.447 | 15-Lipoxygenase inhibitor | 0.219 0.193 CHEMBL100454 0.394 0.077 CHEMBL1125 0.418 0.067 CHEMBL3544641 0.362 0.092 CHEMBL3544615 | ||
| 0.373 | 0.005 | 0.373 | Alpha 2b adrenoreceptor antagonist | 0.139 0.044 CHEMBL100454 0.325 0.008 CHEMBL440512 0.333 0.007 CHEMBL1125 0.124 0.055 CHEMBL3544641 0.106 0.07 CHEMBL3544615 | ||
| 0.369 | 0.007 | 0.418 | Acetylcholine M1 receptor antagonist | 0.181 0.051 CHEMBL3544613 0.313 0.012 CHEMBL100454 0.418 0.005 CHEMBL440512 0.291 0.016 CHEMBL1125 0.298 0.015 CHEMBL3544641 0.228 0.031 CHEMBL3544615 | CHEMBL440512 | |
| 0.367 | 0.008 | 0.422 | Dopamine D2 antagonist | 0.156 0.022 CHEMBL100454 0.422 0.006 CHEMBL440512 0.233 0.014 CHEMBL1125 0.059 0.05 CHEMBL3544641 | CHEMBL440512 | |
| 0.345 | 0.006 | 0.466 | Alpha 1b adrenoreceptor antagonist | 0.26 0.009 CHEMBL100454 0.466 0.004 CHEMBL440512 0.284 0.008 CHEMBL1125 0.13 0.026 CHEMBL3544641 0.101 0.035 CHEMBL3544615 | CHEMBL440512 | |
| 0.339 | 0.004 | 0.343 | Alpha adrenoreceptor agonist | 0.129 0.02 CHEMBL100454 0.07 0.045 CHEMBL440512 0.343 0.004 CHEMBL1125 0.074 0.043 CHEMBL3544641 0.075 0.042 CHEMBL3544615 | CHEMBL1125 | |
| 0.423 | 0.092 | 0.423 | MAP kinase 1 inhibitor | 0.247 0.237 CHEMBL100454 0.33 0.151 CHEMBL1125 0.264 0.218 CHEMBL3544641 | ||
| 0.317 | 0.005 | 0.602 | GABA receptor agonist | 0.094 0.084 CHEMBL3544613 0.162 0.03 CHEMBL100454 0.602 0.003 CHEMBL440512 0.287 0.007 CHEMBL1125 0.237 0.012 CHEMBL3544641 0.209 0.016 CHEMBL3544615 | CHEMBL440512 | |
| 0.329 | 0.033 | 0.329 | Anticonvulsant | 0.143 0.138 CHEMBL100454 0.243 0.06 CHEMBL1125 0.203 0.08 CHEMBL3544641 0.15 0.13 CHEMBL3544615 | ||
| 0.288 | 0.003 | 0.288 | 5 Hydroxytryptamine 6 antagonist | 0.149 0.006 CHEMBL100454 0.099 0.015 CHEMBL440512 0.253 0.003 CHEMBL1125 0.087 0.02 CHEMBL3544641 0.075 0.026 CHEMBL3544615 | ||
| 0.29 | 0.005 | 0.29 | 5 Hydroxytryptamine 1B antagonist | 0.148 0.013 CHEMBL100454 0.188 0.009 CHEMBL1125 0.064 0.047 CHEMBL3544641 | ||
| 0.315 | 0.034 | 0.426 | Death-associated protein kinase 3 inhibitor | 0.226 0.062 CHEMBL100454 0.183 0.085 CHEMBL440512 0.361 0.024 CHEMBL1125 0.385 0.019 CHEMBL3544641 0.426 0.013 CHEMBL3544615 | CHEMBL3544615 | |
| 0.296 | 0.016 | 0.372 | Alpha adrenoreceptor antagonist | 0.214 0.025 CHEMBL100454 0.372 0.011 CHEMBL440512 0.254 0.02 CHEMBL1125 0.077 0.074 CHEMBL3544641 | CHEMBL440512 | |
| 0.298 | 0.026 | 0.346 | Dual specificity tyrosine-phosphorylation-regulated kinase 4 inhibitor | 0.22 0.044 CHEMBL100454 0.221 0.044 CHEMBL440512 0.346 0.016 CHEMBL1125 0.249 0.037 CHEMBL3544641 0.308 0.024 CHEMBL3544615 | CHEMBL1125 | |
| 0.287 | 0.019 | 0.314 | Protein kinase (CK1) inhibitor | 0.156 0.063 CHEMBL100454 0.143 0.073 CHEMBL440512 0.314 0.016 CHEMBL1125 0.225 0.033 CHEMBL3544641 0.242 0.028 CHEMBL3544615 | CHEMBL1125 | |
| 0.377 | 0.122 | 0.39 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.273 0.252 CHEMBL100454 0.39 0.109 CHEMBL1125 0.36 0.14 CHEMBL3544641 0.373 0.126 CHEMBL3544615 | CHEMBL1125 | |
| 0.259 | 0.004 | 0.31 | Acetylcholine M5 receptor antagonist | 0.14 0.009 CHEMBL100454 0.31 0.003 CHEMBL440512 0.18 0.005 CHEMBL1125 0.135 0.01 CHEMBL3544641 0.086 0.022 CHEMBL3544615 | CHEMBL440512 | |
| 0.285 | 0.04 | 0.285 | Ca2+/calmodulin-dependent kinase II beta inhibitor | 0.213 0.067 CHEMBL100454 0.239 0.055 CHEMBL1125 0.216 0.066 CHEMBL3544641 0.184 0.09 CHEMBL3544615 | ||
| 0.268 | 0.028 | 0.331 | I kappa B kinase epsilon inhibitor | 0.237 0.045 CHEMBL100454 0.261 0.032 CHEMBL1125 0.331 0.007 CHEMBL3544641 0.326 0.008 CHEMBL3544615 | CHEMBL3544641 | |
| 0.241 | 0.011 | 0.241 | Alpha 2c adrenoreceptor antagonist | 0.122 0.048 CHEMBL100454 0.2 0.018 CHEMBL440512 0.206 0.017 CHEMBL1125 0.085 0.081 CHEMBL3544641 | ||
| 0.238 | 0.009 | 0.238 | 5 Hydroxytryptamine 7 antagonist | 0.087 0.028 CHEMBL100454 0.231 0.009 CHEMBL1125 0.07 0.037 CHEMBL3544641 0.063 0.043 CHEMBL3544615 | ||
| 0.231 | 0.004 | 0.231 | Histamine agonist | 0.07 0.019 CHEMBL100454 0.054 0.034 CHEMBL440512 0.161 0.005 CHEMBL1125 0.062 0.026 CHEMBL3544641 0.047 0.045 CHEMBL3544615 | ||
| 0.271 | 0.047 | 0.274 | MAP-kinase-activated kinase 5 inhibitor | 0.211 0.09 CHEMBL100454 0.274 0.045 CHEMBL1125 0.22 0.082 CHEMBL3544641 0.219 0.083 CHEMBL3544615 | CHEMBL1125 | |
| 0.232 | 0.011 | 0.325 | Histamine H1 receptor antagonist | 0.225 0.012 CHEMBL100454 0.325 0.005 CHEMBL440512 0.141 0.027 CHEMBL1125 0.165 0.02 CHEMBL3544641 0.095 0.044 CHEMBL3544615 | CHEMBL440512 | |
| 0.227 | 0.01 | 0.317 | Acetylcholine agonist | 0.171 0.02 CHEMBL100454 0.317 0.005 CHEMBL440512 0.204 0.013 CHEMBL1125 0.109 0.041 CHEMBL3544641 0.093 0.052 CHEMBL3544615 | CHEMBL440512 | |
| 0.301 | 0.085 | 0.402 | Apoptosis antagonist | 0.361 0.051 CHEMBL3544613 0.258 0.12 CHEMBL100454 0.402 0.038 CHEMBL3544614 0.304 0.083 CHEMBL1125 0.263 0.115 CHEMBL3544641 0.263 0.115 CHEMBL3544615 | CHEMBL3544614 | |
| 0.287 | 0.074 | 0.287 | Ca2+/calmodulin-dependent kinase II alpha inhibitor | 0.261 0.096 CHEMBL1125 | ||
| 0.223 | 0.015 | 0.223 | 5 Hydroxytryptamine 2C antagonist | 0.12 0.036 CHEMBL100454 0.102 0.044 CHEMBL440512 0.183 0.02 CHEMBL1125 | ||
| 0.21 | 0.004 | 0.232 | Alpha 2 adrenoreceptor agonist | 0.083 0.022 CHEMBL100454 0.065 0.037 CHEMBL440512 0.232 0.004 CHEMBL1125 0.059 0.044 CHEMBL3544615 | CHEMBL1125 | |
| 0.255 | 0.049 | 0.268 | Platelet aggregation inhibitor | 0.18 0.098 CHEMBL100454 0.268 0.045 CHEMBL440512 0.26 0.048 CHEMBL1125 0.193 0.087 CHEMBL3544641 0.192 0.087 CHEMBL3544615 | CHEMBL440512 | |
| 0.243 | 0.042 | 0.243 | LIM domain kinase 1 inhibitor | 0.145 0.103 CHEMBL100454 0.239 0.044 CHEMBL1125 0.178 0.075 CHEMBL3544641 0.173 0.078 CHEMBL3544615 | ||
| 0.21 | 0.01 | 0.21 | Dopamine D3 antagonist | 0.065 0.04 CHEMBL100454 0.104 0.024 CHEMBL440512 0.118 0.02 CHEMBL1125 | ||
| 0.241 | 0.049 | 0.283 | CDC-like kinase 4 inhibitor | 0.144 0.106 CHEMBL100454 0.283 0.036 CHEMBL1125 0.166 0.088 CHEMBL3544641 0.192 0.071 CHEMBL3544615 | CHEMBL1125 | |
| 0.21 | 0.019 | 0.311 | Alpha 1 adrenoreceptor antagonist | 0.139 0.032 CHEMBL100454 0.311 0.01 CHEMBL440512 0.189 0.022 CHEMBL1125 | CHEMBL440512 | |
| 0.199 | 0.01 | 0.199 | Alpha 1d adrenoreceptor antagonist | 0.12 0.019 CHEMBL100454 0.141 0.016 CHEMBL440512 0.178 0.011 CHEMBL1125 0.056 0.044 CHEMBL3544641 | ||
| 0.247 | 0.069 | 0.255 | Ca2+/calmodulin-dependent kinase IV inhibitor | 0.235 0.086 CHEMBL100454 0.255 0.059 CHEMBL1125 0.219 0.118 CHEMBL3544641 0.223 0.108 CHEMBL3544615 | CHEMBL1125 | |
| 0.199 | 0.025 | 0.27 | Acetylcholine muscarinic antagonist | 0.098 0.094 CHEMBL3544613 0.201 0.024 CHEMBL100454 0.27 0.012 CHEMBL440512 0.155 0.041 CHEMBL1125 0.16 0.038 CHEMBL3544641 0.126 0.061 CHEMBL3544615 | CHEMBL440512 | |
| 0.205 | 0.033 | 0.205 | Toll-Like receptor 9 antagonist | 0.116 0.09 CHEMBL100454 0.146 0.066 CHEMBL1125 | ||
| 0.205 | 0.035 | 0.226 | Ribosomal protein S6 kinase inhibitor | 0.114 0.097 CHEMBL100454 0.226 0.028 CHEMBL1125 0.156 0.06 CHEMBL3544641 0.172 0.051 CHEMBL3544615 | CHEMBL1125 | |
| 0.229 | 0.065 | 0.229 | MAP kinase kinase 2 inhibitor | 0.205 0.079 CHEMBL1125 | ||
| 0.193 | 0.031 | 0.193 | Protein kinase (CK1) delta inhibitor | 0.106 0.085 CHEMBL100454 0.191 0.032 CHEMBL1125 0.16 0.047 CHEMBL3544641 0.156 0.05 CHEMBL3544615 | ||
| 0.23 | 0.071 | 0.23 | Ca2+/calmodulin-dependent kinase I alpha inhibitor | 0.162 0.128 CHEMBL100454 0.206 0.086 CHEMBL1125 | ||
| 0.313 | 0.155 | 0.313 | DNA directed DNA polymerase inhibitor | 0.228 0.206 CHEMBL3544614 0.255 0.188 CHEMBL1125 0.277 0.174 CHEMBL3544641 0.222 0.21 CHEMBL3544615 | ||
| 0.192 | 0.034 | 0.283 | Cholinergic antagonist | 0.209 0.03 CHEMBL100454 0.283 0.016 CHEMBL440512 0.157 0.049 CHEMBL1125 0.149 0.053 CHEMBL3544641 0.12 0.074 CHEMBL3544615 | CHEMBL440512 | |
| 0.19 | 0.033 | 0.266 | Acetylcholine antagonist | 0.207 0.029 CHEMBL100454 0.266 0.018 CHEMBL440512 0.154 0.048 CHEMBL1125 0.146 0.052 CHEMBL3544641 0.117 0.073 CHEMBL3544615 | CHEMBL440512 | |
| 0.27 | 0.117 | 0.277 | Prostaglandin dehydrogenase inhibitor | 0.277 0.113 CHEMBL1125 0.18 0.172 CHEMBL3544615 | CHEMBL1125 | |
| 0.22 | 0.068 | 0.234 | Clk dual-specificity kinase inhibitor | 0.234 0.062 CHEMBL1125 0.147 0.117 CHEMBL3544641 0.152 0.112 CHEMBL3544615 | CHEMBL1125 | |
| 0.234 | 0.088 | 0.358 | Aldehyde oxidase inhibitor | 0.235 0.088 CHEMBL100454 0.148 0.141 CHEMBL1125 0.358 0.054 CHEMBL3544641 0.228 0.091 CHEMBL3544615 | CHEMBL3544641 | |
| 0.236 | 0.09 | 0.236 | 5 Hydroxytryptamine 1E antagonist | |||
| 0.145 | 0.005 | 0.145 | 5 Hydroxytryptamine 3 agonist | 0.118 0.009 CHEMBL100454 0.122 0.008 CHEMBL1125 0.101 0.015 CHEMBL3544641 0.082 0.025 CHEMBL3544615 | ||
| 0.208 | 0.071 | 0.211 | Ca2+/calmodulin-dependent protein kinase inhibitor | 0.211 0.07 CHEMBL1125 | CHEMBL1125 | |
| 0.214 | 0.079 | 0.214 | EphB2 antagonist | 0.168 0.113 CHEMBL1125 | ||
| 0.187 | 0.053 | 0.38 | Polo-like kinase-3 inhibitor | 0.122 0.121 CHEMBL3544613 0.154 0.079 CHEMBL100454 0.38 0.004 CHEMBL440512 0.151 0.083 CHEMBL1125 0.242 0.027 CHEMBL3544641 0.213 0.038 CHEMBL3544615 | CHEMBL440512 | |
| 0.145 | 0.012 | 0.182 | Acetylcholine M2 receptor antagonist | 0.059 0.046 CHEMBL100454 0.182 0.008 CHEMBL440512 0.095 0.023 CHEMBL1125 0.078 0.03 CHEMBL3544641 | CHEMBL440512 | |
| 0.148 | 0.018 | 0.148 | Phosphodiesterase I inhibitor | 0.095 0.051 CHEMBL100454 0.1 0.045 CHEMBL1125 0.114 0.031 CHEMBL3544641 0.081 0.075 CHEMBL3544615 | ||
| 0.138 | 0.008 | 0.138 | Phosphodiesterase 1B inhibitor | 0.074 0.027 CHEMBL100454 0.091 0.017 CHEMBL1125 0.076 0.025 CHEMBL3544641 | ||
| 0.154 | 0.031 | 0.154 | Antihistaminic | 0.139 0.035 CHEMBL100454 0.152 0.031 CHEMBL440512 0.095 0.059 CHEMBL1125 | ||
| 0.149 | 0.027 | 0.149 | Gastric antisecretory | 0.134 0.034 CHEMBL1125 | ||
| 0.133 | 0.012 | 0.133 | Benzodiazepine agonist | 0.072 0.048 CHEMBL100454 0.067 0.056 CHEMBL440512 0.102 0.024 CHEMBL1125 | ||
| 0.228 | 0.107 | 0.25 | Gastrin inhibitor | 0.223 0.114 CHEMBL100454 0.25 0.079 CHEMBL3544641 | CHEMBL3544641 | |
| 0.135 | 0.014 | 0.15 | Alpha 2d adrenoreceptor antagonist | 0.118 0.026 CHEMBL440512 0.15 0.009 CHEMBL1125 0.087 0.08 CHEMBL3544615 | CHEMBL1125 | |
| 0.153 | 0.034 | 0.164 | 5 Hydroxytryptamine 3A agonist | 0.164 0.028 CHEMBL1125 | CHEMBL1125 | |
| 0.141 | 0.025 | 0.141 | 5 Hydroxytryptamine 1 antagonist | 0.091 0.04 CHEMBL1125 | ||
| 0.287 | 0.172 | 0.287 | DNA polymerase beta inhibitor | 0.231 0.204 CHEMBL1125 0.24 0.199 CHEMBL3544641 | ||
| 0.15 | 0.036 | 0.202 | Antiadrenergic | 0.138 0.039 CHEMBL100454 0.202 0.024 CHEMBL440512 0.174 0.03 CHEMBL1125 0.076 0.075 CHEMBL3544641 0.085 0.067 CHEMBL3544615 | CHEMBL440512 | |
| 0.148 | 0.035 | 0.201 | Adrenaline antagonist | 0.136 0.039 CHEMBL100454 0.201 0.023 CHEMBL440512 0.172 0.029 CHEMBL1125 0.075 0.073 CHEMBL3544641 0.083 0.065 CHEMBL3544615 | CHEMBL440512 | |
| 0.143 | 0.031 | 0.143 | Histamine antagonist | 0.125 0.037 CHEMBL100454 0.143 0.031 CHEMBL440512 0.084 0.059 CHEMBL1125 | ||
| 0.119 | 0.007 | 0.18 | 5 Hydroxytryptamine 2 agonist | 0.068 0.02 CHEMBL100454 0.18 0.004 CHEMBL1125 | CHEMBL1125 | |
| 0.281 | 0.17 | 0.491 | Alpha-glucosidase inhibitor | 0.491 0.083 CHEMBL3544613 0.306 0.157 CHEMBL3544614 0.274 0.174 CHEMBL1125 | CHEMBL3544613 | |
| 0.116 | 0.004 | 0.116 | Histamine H4 receptor antagonist | 0.079 0.009 CHEMBL100454 0.084 0.007 CHEMBL1125 0.059 0.02 CHEMBL3544641 0.046 0.039 CHEMBL3544615 | ||
| 0.113 | 0.004 | 0.113 | 5 Hydroxytryptamine 3B antagonist | 0.044 0.018 CHEMBL100454 0.074 0.008 CHEMBL1125 0.048 0.015 CHEMBL3544641 | ||
| 0.155 | 0.053 | 0.168 | MAP3K9 inhibitor | 0.168 0.037 CHEMBL100454 0.158 0.049 CHEMBL1125 0.157 0.05 CHEMBL3544641 0.16 0.047 CHEMBL3544615 | CHEMBL100454 | |
| 0.197 | 0.095 | 0.197 | Potassium channel blocker | 0.18 0.107 CHEMBL1125 | ||
| 0.122 | 0.025 | 0.122 | 5 Hydroxytryptamine 1A antagonist | 0.095 0.034 CHEMBL1125 | ||
| 0.105 | 0.01 | 0.105 | Phosphodiesterase VII inhibitor | 0.091 0.017 CHEMBL100454 0.071 0.035 CHEMBL440512 0.105 0.01 CHEMBL1125 0.095 0.015 CHEMBL3544641 0.094 0.015 CHEMBL3544615 | ||
| 0.099 | 0.004 | 0.099 | Protein kinase (CK1) epsilon inhibitor | 0.042 0.022 CHEMBL100454 0.038 0.029 CHEMBL440512 0.09 0.004 CHEMBL1125 0.036 0.035 CHEMBL3544641 | ||
| 0.134 | 0.039 | 0.2 | Check point kinase 2 inhibitor | 0.106 0.06 CHEMBL100454 0.186 0.02 CHEMBL1125 0.155 0.03 CHEMBL3544641 0.2 0.017 CHEMBL3544615 | CHEMBL3544615 | |
| 0.123 | 0.03 | 0.123 | Protein kinase C zeta inhibitor | 0.121 0.032 CHEMBL100454 0.105 0.045 CHEMBL1125 0.11 0.04 CHEMBL3544641 0.094 0.059 CHEMBL3544615 | ||
| 0.117 | 0.029 | 0.219 | 5 Hydroxytryptamine agonist | 0.106 0.032 CHEMBL100454 0.219 0.013 CHEMBL1125 | CHEMBL1125 | |
| 0.109 | 0.024 | 0.109 | Dopamine agonist | 0.064 0.049 CHEMBL100454 0.084 0.035 CHEMBL1125 | ||
| 0.188 | 0.105 | 0.229 | Dyrk kinase inhibitor | 0.186 0.106 CHEMBL1125 0.228 0.083 CHEMBL3544641 0.229 0.082 CHEMBL3544615 | CHEMBL3544615 | |
| 0.09 | 0.009 | 0.09 | Potassium channel (Inward rectifier) blocker | 0.082 0.012 CHEMBL100454 0.082 0.012 CHEMBL1125 | ||
| 0.148 | 0.068 | 0.148 | Activin receptor-like kinase 2 inhibitor | 0.147 0.069 CHEMBL1125 | ||
| 0.112 | 0.032 | 0.112 | Alpha 1a adrenoreceptor antagonist | 0.069 0.051 CHEMBL100454 0.072 0.05 CHEMBL440512 0.104 0.034 CHEMBL1125 | ||
| 0.085 | 0.005 | 0.095 | Purinergic P2T antagonist | 0.024 0.014 CHEMBL3544613 0.083 0.006 CHEMBL100454 0.029 0.013 CHEMBL440512 0.037 0.011 CHEMBL3544614 0.095 0.005 CHEMBL1125 0.081 0.006 CHEMBL3544641 0.09 0.005 CHEMBL3544615 | CHEMBL1125 | |
| 0.215 | 0.14 | 0.215 | Nootropic | 0.204 0.152 CHEMBL1125 | ||
| 0.094 | 0.02 | 0.141 | Protein kinase C iota inhibitor | 0.054 0.047 CHEMBL440512 0.141 0.01 CHEMBL1125 0.07 0.032 CHEMBL3544615 | CHEMBL1125 | |
| 0.133 | 0.061 | 0.182 | Tyrosine-protein kinase receptor FLT3 inhibitor | 0.182 0.042 CHEMBL440512 0.111 0.073 CHEMBL1125 | CHEMBL440512 | |
| 0.08 | 0.01 | 0.093 | Gonadotropin-releasing hormone receptor antagonist | 0.058 0.014 CHEMBL100454 0.033 0.025 CHEMBL440512 0.093 0.008 CHEMBL1125 0.057 0.015 CHEMBL3544641 0.064 0.013 CHEMBL3544615 | CHEMBL1125 | |
| 0.076 | 0.008 | 0.076 | Phosphodiesterase 7A inhibitor | 0.069 0.012 CHEMBL100454 0.06 0.022 CHEMBL440512 0.076 0.008 CHEMBL1125 0.069 0.012 CHEMBL3544641 0.068 0.013 CHEMBL3544615 | ||
| 0.128 | 0.061 | 0.151 | MAP kinase 12 inhibitor | 0.151 0.041 CHEMBL1125 | CHEMBL1125 | |
| 0.11 | 0.043 | 0.11 | mTOR complex 1 inhibitor | 0.102 0.058 CHEMBL100454 0.106 0.051 CHEMBL1125 0.094 0.077 CHEMBL3544641 | ||
| 0.145 | 0.079 | 0.15 | Dual specificity tyrosine-phosphorylation regulated kinase 1B inhibitor | 0.15 0.074 CHEMBL1125 | CHEMBL1125 | |
| 0.178 | 0.112 | 0.181 | 5 Hydroxytryptamine 3E antagonist | 0.181 0.104 CHEMBL1125 | CHEMBL1125 | |
| 0.124 | 0.06 | 0.239 | Protein kinase (CK2) alpha inhibitor | 0.138 0.049 CHEMBL1125 0.212 0.022 CHEMBL3544641 0.239 0.018 CHEMBL3544615 | CHEMBL3544615 | |
| 0.178 | 0.116 | 0.178 | Aryl hydrocarbon receptor agonist | 0.153 0.133 CHEMBL1125 | ||
| 0.08 | 0.021 | 0.08 | Cyclin-dependent kinase 6 inhibitor | 0.062 0.039 CHEMBL100454 0.08 0.022 CHEMBL1125 | ||
| 0.195 | 0.137 | 0.195 | MAP kinase kinase 3 inhibitor | 0.194 0.139 CHEMBL1125 | ||
| 0.148 | 0.09 | 0.148 | Ca2+/calmodulin-dependent kinase II gamma inhibitor | |||
| 0.119 | 0.064 | 0.119 | Platelet activating factor antagonist | 0.115 0.067 CHEMBL440512 | ||
| 0.085 | 0.029 | 0.096 | Purinergic P2 antagonist | 0.096 0.023 CHEMBL1125 | CHEMBL1125 | |
| 0.11 | 0.055 | 0.234 | Protein kinase (CK2) inhibitor | 0.125 0.045 CHEMBL1125 0.208 0.017 CHEMBL3544641 0.234 0.013 CHEMBL3544615 | CHEMBL3544615 | |
| 0.056 | 0.006 | 0.056 | Purinergic P2Y12 antagonist | 0.024 0.015 CHEMBL3544613 0.053 0.006 CHEMBL100454 0.022 0.017 CHEMBL440512 0.037 0.01 CHEMBL3544614 0.055 0.006 CHEMBL1125 0.053 0.006 CHEMBL3544641 0.051 0.007 CHEMBL3544615 | ||
| 0.227 | 0.176 | 0.227 | GABA C receptor rho-3 antagonist | |||
| 0.166 | 0.117 | 0.224 | Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor | 0.164 0.119 CHEMBL1125 0.222 0.08 CHEMBL3544641 0.224 0.079 CHEMBL3544615 | CHEMBL3544615 | |
| 0.097 | 0.049 | 0.128 | Pim-3 kinase inhibitor | 0.128 0.026 CHEMBL1125 0.092 0.055 CHEMBL3544615 | CHEMBL1125 | |
| 0.111 | 0.065 | 0.127 | Polo-like kinase-4 inhibitor | 0.092 0.085 CHEMBL100454 0.127 0.051 CHEMBL3544641 0.09 0.088 CHEMBL3544615 | CHEMBL3544641 | |
| 0.074 | 0.029 | 0.106 | Acetylcholine M3 receptor antagonist | 0.059 0.042 CHEMBL100454 0.106 0.017 CHEMBL440512 0.065 0.035 CHEMBL1125 0.059 0.042 CHEMBL3544641 0.052 0.051 CHEMBL3544615 | CHEMBL440512 | |
| 0.111 | 0.065 | 0.136 | Activin receptor-like kinase 4 inhibitor | 0.136 0.037 CHEMBL1125 0.104 0.078 CHEMBL3544615 | CHEMBL1125 | |
| 0.102 | 0.058 | 0.102 | Insulin receptor antagonist | |||
| 0.079 | 0.035 | 0.079 | Adenosine A2 receptor antagonist | |||
| 0.099 | 0.057 | 0.138 | Protein kinase C mu inhibitor | 0.084 0.075 CHEMBL100454 0.138 0.032 CHEMBL1125 0.107 0.051 CHEMBL3544615 | CHEMBL1125 | |
| 0.086 | 0.046 | 0.088 | Transforming growth factor beta 3 antagonist | 0.088 0.041 CHEMBL440512 0.085 0.049 CHEMBL1125 | CHEMBL440512 | |
| 0.122 | 0.083 | 0.197 | Glycogen synthase kinase-3 alpha inhibitor | 0.15 0.067 CHEMBL1125 0.168 0.054 CHEMBL3544641 0.197 0.042 CHEMBL3544615 | CHEMBL3544615 | |
| 0.05 | 0.011 | 0.05 | Potassium channel small-conductance Ca-activated activator | 0.037 0.017 CHEMBL1125 | ||
| 0.111 | 0.072 | 0.111 | Aurora-B kinase inhibitor | 0.105 0.076 CHEMBL1125 | ||
| 0.046 | 0.008 | 0.046 | CDK4/cyclin D3 inhibitor | 0.045 0.008 CHEMBL1125 | ||
| 0.072 | 0.035 | 0.072 | Adenosine A2a receptor antagonist | |||
| 0.217 | 0.184 | 0.457 | Histamine release inhibitor | 0.27 0.141 CHEMBL3544613 0.25 0.155 CHEMBL100454 0.211 0.189 CHEMBL3544614 0.457 0.046 CHEMBL3544641 0.401 0.075 CHEMBL3544615 | CHEMBL3544641 | |
| 0.231 | 0.2 | 0.231 | Transcription factor inhibitor | |||
| 0.114 | 0.085 | 0.168 | DNA repair enzyme inhibitor | 0.16 0.023 CHEMBL3544613 0.163 0.022 CHEMBL100454 0.168 0.019 CHEMBL3544614 0.157 0.026 CHEMBL3544641 0.145 0.036 CHEMBL3544615 | CHEMBL3544614 | |
| 0.043 | 0.014 | 0.043 | Acetylcholine M4 receptor agonist | 0.032 0.02 CHEMBL1125 | ||
| 0.065 | 0.036 | 0.065 | Corticotropin releasing factor 2 receptor antagonist | 0.06 0.047 CHEMBL1125 | ||
| 0.083 | 0.056 | 0.097 | I kappa B kinase inhibitor | 0.093 0.045 CHEMBL100454 0.097 0.041 CHEMBL1125 0.074 0.07 CHEMBL3544641 0.087 0.052 CHEMBL3544615 | CHEMBL1125 | |
| 0.063 | 0.036 | 0.096 | Glutamate (mGluR1) antagonist | 0.069 0.031 CHEMBL1125 0.086 0.021 CHEMBL3544641 0.096 0.017 CHEMBL3544615 | CHEMBL3544615 | |
| 0.038 | 0.013 | 0.052 | Poly(ADP-ribose) polymerase 2 inhibitor | 0.052 0.009 CHEMBL1125 0.031 0.018 CHEMBL3544615 | CHEMBL1125 | |
| 0.035 | 0.01 | 0.036 | Potassium channel (Inward rectifier) 1 blocker | 0.036 0.01 CHEMBL100454 0.034 0.012 CHEMBL1125 0.031 0.02 CHEMBL3544641 0.029 0.024 CHEMBL3544615 | CHEMBL100454 | |
| 0.067 | 0.044 | 0.096 | Cyclin-dependent kinase 4 inhibitor | 0.096 0.027 CHEMBL1125 | CHEMBL1125 | |
| 0.189 | 0.166 | 0.276 | Hypoxia-inducible factor 1 alpha inhibitor | 0.276 0.079 CHEMBL100454 0.231 0.118 CHEMBL3544614 0.197 0.156 CHEMBL1125 | CHEMBL100454 | |
| 0.059 | 0.038 | 0.064 | Protein kinase C theta inhibitor | 0.064 0.03 CHEMBL440512 0.062 0.033 CHEMBL1125 | CHEMBL440512 | |
| 0.149 | 0.132 | 0.149 | HERG channel blocker | |||
| 0.061 | 0.045 | 0.073 | I kappa B kinase 2 inhibitor | 0.067 0.036 CHEMBL100454 0.073 0.029 CHEMBL1125 | CHEMBL1125 | |
| 0.065 | 0.049 | 0.089 | CDC7 inhibitor | 0.089 0.03 CHEMBL1125 0.066 0.049 CHEMBL3544641 0.089 0.03 CHEMBL3544615 | CHEMBL3544615 | |
| 0.085 | 0.07 | 0.17 | Fibroblast growth factor 1 antagonist | 0.17 0.025 CHEMBL440512 | CHEMBL440512 | |
| 0.09 | 0.075 | 0.09 | Aurora-A kinase inhibitor | |||
| 0.023 | 0.009 | 0.023 | Histamine H4 receptor agonist | |||
| 0.156 | 0.142 | 0.296 | Cyclic AMP phosphodiesterase inhibitor | 0.167 0.126 CHEMBL100454 0.296 0.044 CHEMBL3544641 0.276 0.052 CHEMBL3544615 | CHEMBL3544641 | |
| 0.141 | 0.128 | 0.194 | Dual specificity tyrosine-phosphorylation regulated kinase 3 inhibitor | 0.194 0.081 CHEMBL1125 0.163 0.108 CHEMBL3544615 | CHEMBL1125 | |
| 0.044 | 0.033 | 0.044 | Potassium channel small-conductance Ca-activated blocker | |||
| 0.13 | 0.12 | 0.13 | TRKC antagonist | |||
| 0.057 | 0.047 | 0.057 | Cyclin A inhibitor | 0.054 0.049 CHEMBL1125 | ||
| 0.042 | 0.034 | 0.131 | 5 Hydroxytryptamine 2C agonist | 0.131 0.005 CHEMBL1125 0.071 0.014 CHEMBL3544615 | CHEMBL1125 | |
| 0.046 | 0.039 | 0.046 | Dopamine beta hydroxylase inhibitor | |||
| 0.068 | 0.062 | 0.116 | Protein kinase (CaMK, MLCK, PhK, SNF, KIN, NIM1, MAPKAP, POLO, CHK, ULK, RSK-2nd domain) inhibitor | 0.116 0.029 CHEMBL1125 0.084 0.047 CHEMBL3544615 | CHEMBL1125 | |
| 0.076 | 0.07 | 0.077 | Bcr-Abl kinase inhibitor | 0.077 0.068 CHEMBL100454 | CHEMBL100454 | |
| 0.021 | 0.015 | 0.03 | Glutaminyl-peptide cyclotransferase inhibitor | 0.03 0.006 CHEMBL1125 | CHEMBL1125 | |
| 0.055 | 0.05 | 0.061 | Cyclin A1 inhibitor | 0.061 0.036 CHEMBL1125 | CHEMBL1125 | |
| 0.076 | 0.071 | 0.076 | GABA A receptor agonist | 0.076 0.071 CHEMBL1125 | ||
| 0.05 | 0.045 | 0.05 | Lysine-specific demethylase 1A inhibitor | |||
| 0.01 | 0.006 | 0.01 | CXC chemokine 3 receptor agonist | 0.009 0.008 CHEMBL1125 | ||
| 0.016 | 0.012 | 0.016 | CDK2/cyclin A3 inhibitor | 0.016 0.013 CHEMBL1125 | ||
| 0.08 | 0.077 | 0.145 | Protein kinase C delta inhibitor | 0.145 0.023 CHEMBL440512 0.103 0.05 CHEMBL1125 0.087 0.066 CHEMBL3544615 | CHEMBL440512 | |
| 0.081 | 0.078 | 0.104 | Platelet activating factor beta antagonist | 0.104 0.06 CHEMBL440512 | CHEMBL440512 | |
| 0.094 | 0.091 | 0.114 | MAP kinase 13 inhibitor | 0.114 0.062 CHEMBL1125 | CHEMBL1125 | |
| 0.033 | 0.03 | 0.033 | Adenosine uptake inhibitor | |||
| 0.159 | 0.158 | 0.159 | ErbB-1 antagonist | |||
| 0.079 | 0.086 | 0.11 | Polo-like kinase-1 inhibitor | 0.11 0.036 CHEMBL440512 0.106 0.039 CHEMBL3544641 | CHEMBL440512 | |
| 0.017 | 0.025 | 0.024 | Alpha 2d adrenoreceptor agonist | 0.024 0.012 CHEMBL1125 | CHEMBL1125 | |
| 0.058 | 0.067 | 0.073 | Protein kinase B alpha inhibitor | 0.073 0.045 CHEMBL1125 | CHEMBL1125 | |
| 0.043 | 0.053 | 0.087 | Acetylcholine muscarinic agonist | 0.087 0.02 CHEMBL440512 | CHEMBL440512 | |
| 0.07 | 0.084 | 0.088 | MAP kinase kinase 7 inhibitor | 0.078 0.052 CHEMBL100454 0.086 0.031 CHEMBL1125 0.088 0.028 CHEMBL3544615 | CHEMBL3544615 | |
| 0.117 | 0.132 | 0.124 | Interleukin-1 receptor-associated protein kinase 1 inhibitor | 0.124 0.122 CHEMBL1125 | CHEMBL1125 | |
| 0.1 | 0.116 | 0.175 | Lipid peroxidase inhibitor | 0.175 0.053 CHEMBL3544613 0.137 0.077 CHEMBL3544614 | CHEMBL3544613 | |
| 0.115 | 0.133 | 0.135 | Death-associated protein kinase 1 inhibitor | 0.135 0.069 CHEMBL1125 | CHEMBL1125 | |
| 0.095 | 0.116 | 0.167 | Phosphodiesterase inhibitor | 0.167 0.048 CHEMBL440512 | CHEMBL440512 | |
| 0.041 | 0.065 | 0.069 | Myc inhibitor | 0.063 0.026 CHEMBL1125 0.052 0.042 CHEMBL3544641 0.069 0.02 CHEMBL3544615 | CHEMBL3544615 | |
| 0.055 | 0.081 | 0.08 | Rho-associated kinase I inhibitor | 0.08 0.046 CHEMBL1125 | CHEMBL1125 | |
| 0.034 | 0.062 | 0.066 | Poly(ADP-ribose) polymerase inhibitor | 0.066 0.014 CHEMBL440512 | CHEMBL440512 | |
| 0.028 | 0.057 | 0.049 | Glutamate (mGluR1a) antagonist | 0.049 0.021 CHEMBL3544641 | CHEMBL3544641 | |
| 0.027 | 0.058 | 0.069 | Purinergic P2Y antagonist | 0.066 0.017 CHEMBL3544641 0.069 0.015 CHEMBL3544615 | CHEMBL3544615 | |
| 0.075 | 0.108 | 0.109 | Granulocyte macrophage colony stimulating factor antagonist | 0.109 0.062 CHEMBL440512 | CHEMBL440512 | |
| 0.05 | 0.084 | 0.074 | Phosphodiesterase 5A inhibitor | 0.074 0.046 CHEMBL440512 | CHEMBL440512 | |
| 0.024 | 0.06 | 0.062 | Poly(ADP-ribose) polymerase 1 inhibitor | 0.062 0.012 CHEMBL440512 | CHEMBL440512 | |
| 0.048 | 0.086 | 0.072 | Phosphodiesterase V inhibitor | 0.072 0.049 CHEMBL440512 | CHEMBL440512 | |
| 0.047 | 0.089 | 0.073 | Check point kinase 1 inhibitor | 0.073 0.043 CHEMBL1125 | CHEMBL1125 | |
| 0.025 | 0.068 | 0.05 | Acetylcholine M1 receptor agonist | 0.05 0.026 CHEMBL440512 | CHEMBL440512 | |
| 0.024 | 0.071 | 0.046 | Protein kinase (CK2) beta inhibitor | 0.046 0.009 CHEMBL3544641 0.045 0.009 CHEMBL3544615 | CHEMBL3544641 | |
| 0.123 | 0.169 | 0.136 | Heat shock protein 70 antagonist | 0.136 0.09 CHEMBL3544641 | CHEMBL3544641 | |
| 0.055 | 0.106 | 0.081 | Adrenaline agonist | 0.081 0.057 CHEMBL1125 0.081 0.056 CHEMBL3544615 | CHEMBL3544615 | |
| 0.045 | 0.101 | 0.087 | Protein kinase C beta inhibitor | 0.087 0.021 CHEMBL100454 | CHEMBL100454 | |
| 0.014 | 0.071 | 0.055 | HCV NS5B polymerase inhibitor | 0.055 0.009 CHEMBL3544641 0.048 0.01 CHEMBL3544615 | CHEMBL3544641 | |
| 0.06 | 0.118 | 0.094 | Pim-1 kinase inhibitor | 0.091 0.067 CHEMBL1125 0.094 0.064 CHEMBL3544615 | CHEMBL3544615 | |
| 0.037 | 0.106 | 0.062 | Glucosylceramidase inhibitor | 0.062 0.028 CHEMBL1125 | CHEMBL1125 | |
| 0.108 | 0.179 | 0.139 | Ca2+/calmodulin-dependent protein kinase kinase B inhibitor | 0.139 0.095 CHEMBL3544641 | CHEMBL3544641 | |
| 0.018 | 0.091 | 0.034 | DNA gyrase subunit B inhibitor | 0.034 0.033 CHEMBL3544615 | CHEMBL3544615 | |
| 0.019 | 0.095 | 0.058 | RNA-directed RNA polymerase inhibitor | 0.055 0.011 CHEMBL3544641 0.058 0.01 CHEMBL3544615 | CHEMBL3544615 | |
| 0.028 | 0.109 | 0.041 | DNA gyrase subunit A inhibitor | 0.041 0.033 CHEMBL3544615 | CHEMBL3544615 | |
| 0.173 | 0.259 | 0.261 | Calcium channel activator | 0.261 0.134 CHEMBL1125 0.249 0.149 CHEMBL3544615 | CHEMBL1125 | |
| 0.066 | 0.161 | 0.112 | Multidrug resistance-associated protein 1 inhibitor | 0.112 0.058 CHEMBL3544614 | CHEMBL3544614 | |
| 0.035 | 0.138 | 0.095 | DNA gyrase inhibitor | 0.087 0.023 CHEMBL3544641 0.095 0.019 CHEMBL3544615 | CHEMBL3544615 | |
| 0.091 | 0.196 | 0.302 | Platelet adhesion inhibitor | 0.262 0.046 CHEMBL3544613 0.302 0.033 CHEMBL3544614 0.146 0.111 CHEMBL1125 0.182 0.081 CHEMBL3544615 | CHEMBL3544614 | |
| 0.003 | 0.116 | 0.011 | Egl nine homolog 3 inhibitor | 0.011 0.01 CHEMBL3544615 | CHEMBL3544615 | |
| 0.182 | 0.303 | 0.441 | Cyclophilin D inhibitor | 0.441 0.071 CHEMBL3544613 0.324 0.142 CHEMBL100454 0.408 0.087 CHEMBL3544614 0.253 0.209 CHEMBL1125 0.343 0.127 CHEMBL3544641 0.41 0.085 CHEMBL3544615 | CHEMBL3544613 | |
| 0.046 | 0.167 | 0.091 | Vascular endothelial growth factor 1 antagonist | 0.091 0.072 CHEMBL440512 | CHEMBL440512 | |
| 0.08 | 0.212 | 0.102 | Sphingosine 1-phosphate receptor 2 agonist | 0.102 0.096 CHEMBL1125 | CHEMBL1125 | |
| 0.128 | 0.263 | 0.169 | RNA-directed DNA polymerase inhibitor | 0.169 0.154 CHEMBL100454 | CHEMBL100454 | |
| 0.018 | 0.167 | 0.028 | DNA topoisomerase IV inhibitor | 0.028 0.025 CHEMBL3544615 | CHEMBL3544615 | |
| 0.072 | 0.226 | 0.128 | Dual specificity phosphatase 3 inhibitor | 0.128 0.119 CHEMBL3544641 | CHEMBL3544641 | |
| 0.041 | 0.198 | 0.114 | Protein-tyrosine kinase (PTK, not ETK, WZC) inhibitor | 0.114 0.074 CHEMBL440512 | CHEMBL440512 | |
| 0.041 | 0.197 | 0.114 | Abl kinase inhibitor | 0.114 0.074 CHEMBL440512 | CHEMBL440512 | |
| 0.101 | 0.273 | 0.132 | CC chemokine 6 receptor antagonist | 0.13 0.069 CHEMBL3544613 0.132 0.064 CHEMBL3544614 | CHEMBL3544614 | |
| 0.024 | 0.203 | 0.045 | Alpha 1L adrenoreceptor agonist | 0.045 0.024 CHEMBL1125 | CHEMBL1125 | |
| 0.024 | 0.206 | 0.062 | Factor IXa inhibitor | 0.062 0.025 CHEMBL3544613 0.055 0.032 CHEMBL3544614 | CHEMBL3544613 | |
| 0.097 | 0.291 | 0.374 | Hypoglycemic | 0.374 0.032 CHEMBL3544613 0.338 0.041 CHEMBL3544614 0.185 0.127 CHEMBL3544615 | CHEMBL3544613 | |
| 0.108 | 0.307 | 0.233 | DNA synthesis inhibitor | 0.221 0.093 CHEMBL3544613 0.173 0.164 CHEMBL100454 0.233 0.08 CHEMBL3544614 0.184 0.147 CHEMBL3544615 | CHEMBL3544614 | |
| 0.071 | 0.274 | 0.167 | NOS3 expression enhancer | 0.167 0.058 CHEMBL3544613 0.148 0.075 CHEMBL3544614 | CHEMBL3544613 | |
| 0.017 | 0.221 | 0.233 | Selectin antagonist | 0.208 0.01 CHEMBL3544613 0.063 0.047 CHEMBL100454 0.233 0.009 CHEMBL3544614 | CHEMBL3544614 | |
| 0.058 | 0.261 | 0.167 | Cholinergic | 0.167 0.064 CHEMBL440512 | CHEMBL440512 | |
| 0.079 | 0.291 | 0.144 | Interferon gamma antagonist | 0.127 0.117 CHEMBL3544613 0.144 0.087 CHEMBL3544614 | CHEMBL3544614 | |
| 0.041 | 0.266 | 0.095 | Beta glucuronidase inhibitor | 0.094 0.079 CHEMBL3544613 0.095 0.078 CHEMBL3544615 | CHEMBL3544615 | |
| 0.07 | 0.296 | 0.202 | Platelet antagonist | 0.2 0.101 CHEMBL3544613 0.202 0.099 CHEMBL3544614 0.148 0.147 CHEMBL3544641 0.197 0.103 CHEMBL3544615 | CHEMBL3544614 | |
| 0.109 | 0.342 | 0.247 | Vasodilator, coronary | 0.247 0.138 CHEMBL3544614 | CHEMBL3544614 | |
| 0.033 | 0.268 | 0.13 | Ephrin antagonist | 0.13 0.044 CHEMBL440512 | CHEMBL440512 | |
| 0.03 | 0.292 | 0.081 | ATPase (Vacuolar H+) inhibitor | 0.081 0.075 CHEMBL3544613 | CHEMBL3544613 | |
| 0.141 | 0.422 | 0.292 | Calcium channel L-type activator | 0.292 0.164 CHEMBL100454 0.253 0.202 CHEMBL3544615 | CHEMBL100454 | |
| 0.006 | 0.324 | 0.018 | Retinoic acid beta receptor agonist | 0.018 0.017 CHEMBL3544615 | CHEMBL3544615 | |
| 0.027 | 0.357 | 0.123 | GABA C receptor agonist | 0.123 0.047 CHEMBL3544615 | CHEMBL3544615 | |
| 0.025 | 0.41 | 0.149 | Uric acid excretion stimulant | 0.141 0.027 CHEMBL3544641 0.149 0.024 CHEMBL3544615 | CHEMBL3544615 | |
| 0.037 | 0.427 | 0.207 | Interleukin 1 antagonist | 0.207 0.03 CHEMBL100454 | CHEMBL100454 | |
| 0.014 | 0.486 | 0.575 | Topoisomerase I inhibitor | 0.363 0.007 CHEMBL3544613 0.575 0.003 CHEMBL3544614 | CHEMBL3544614 | |
| 0.05 | 0.553 | 0.564 | Antibacterial | 0.471 0.049 CHEMBL3544613 0.564 0.025 CHEMBL3544614 | CHEMBL3544614 | |
| 0.028 | 0.555 | 0.159 | Vasodilator | 0.159 0.145 CHEMBL3544614 | CHEMBL3544614 | |
| 0.078 | 0.606 | 0.328 | Interleukin 2 agonist | 0.328 0.056 CHEMBL3544613 0.325 0.058 CHEMBL3544614 | CHEMBL3544613 | |
| 0.024 | 0.551 | 0.116 | Cell wall synthesis inhibitor | 0.116 0.105 CHEMBL3544614 | CHEMBL3544614 | |
| 0.026 | 0.577 | 0.129 | Insulin secretagoues | 0.129 0.098 CHEMBL3544614 | CHEMBL3544614 | |
| 0.017 | 0.631 | 0.109 | Thioredoxin inhibitor | 0.109 0.039 CHEMBL100454 | CHEMBL100454 | |
| 0.013 | 0.642 | 0.208 | Immunostimulant | 0.208 0.115 CHEMBL3544613 | CHEMBL3544613 | |
| 0.051 | 0.681 | 0.33 | Antiinflammatory | 0.282 0.232 CHEMBL3544613 0.33 0.188 CHEMBL3544614 | CHEMBL3544614 | |
| 0.023 | 0.656 | 0.158 | Tumour necrosis factor alpha release inhibitor | 0.158 0.147 CHEMBL100454 | CHEMBL100454 | |
| 0.025 | 0.661 | 0.2 | Antithrombotic | 0.2 0.177 CHEMBL3544614 | CHEMBL3544614 | |
| 0.033 | 0.692 | 0.201 | Immunomodulator | 0.201 0.164 CHEMBL3544613 | CHEMBL3544613 | |
| 0.065 | 0.766 | 0.291 | Peptidyltransferase inhibitor | 0.291 0.028 CHEMBL3544613 0.29 0.028 CHEMBL3544614 | CHEMBL3544613 | |
| 0.007 | 0.73 | 0.055 | Protein 50S ribosomal subunit inhibitor | 0.051 0.038 CHEMBL3544613 0.055 0.035 CHEMBL3544614 | CHEMBL3544614 | |
| 0.023 | 0.797 | 0.235 | Hepatoprotectant | 0.224 0.052 CHEMBL3544613 0.235 0.048 CHEMBL3544614 | CHEMBL3544614 | |
| 0.007 | 0.809 | 0.244 | Free radical scavenger | 0.185 0.11 CHEMBL3544613 0.244 0.071 CHEMBL3544614 | CHEMBL3544614 | |
| 0.01 | 0.819 | 0.366 | Angiogenesis stimulant | 0.359 0.03 CHEMBL3544613 0.366 0.028 CHEMBL3544614 | CHEMBL3544614 | |
| 0.008 | 0.84 | 0.162 | Nitric oxide antagonist | 0.162 0.086 CHEMBL3544613 0.162 0.086 CHEMBL3544614 | CHEMBL3544614 | |
| 0.012 | 0.875 | 0.224 | Immunosuppressant | 0.224 0.172 CHEMBL3544614 | CHEMBL3544614 | |
| 0.005 | 0.887 | 0.259 | Antioxidant | 0.203 0.111 CHEMBL3544613 0.259 0.079 CHEMBL3544614 | CHEMBL3544614 | |
| 0.006 | 0.889 | 0.046 | Antibiotic Aminoglycoside-like | 0.046 0.016 CHEMBL3544613 0.046 0.016 CHEMBL3544614 | CHEMBL3544614 | |
| 0.008 | 0.913 | 0.378 | Apoptosis agonist | 0.378 0.124 CHEMBL3544614 | CHEMBL3544614 | |
| 0.001 | 0.976 | 0.044 | Prostaglandin D2 agonist | 0.037 0.015 CHEMBL3544641 0.044 0.01 CHEMBL3544615 | CHEMBL3544615 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |