Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.7210.0050.721Immunomodulator

0.668 0.007 CHEMBL3527332

0.7140.0010.714Glutamate release inhibitor

0.24 0.004 CHEMBL3527332

0.6990.0040.699Proto-oncogene tyrosine-protein kinase Yes inhibitor
0.5870.0190.587Toll-Like receptor agonist
0.570.0210.57Toll-Like receptor 7 agonist
0.4410.0220.441HERG channel blocker
0.4240.0070.424Protein kinase (CK1) gamma 1 inhibitor
0.4190.0060.419c-Src kinase inhibitor
0.4420.0440.442GABA C receptor rho-3 antagonist
0.3890.0080.389Nav1.2 sodium channel blocker
0.3840.030.384Potassium channel (Voltage-sensitive) blocker
0.3650.0160.365Src kinase inhibitor
0.3560.0110.356LIM domain kinase 1 inhibitor
0.3420.0120.342Protein kinase (CK1) gamma inhibitor
0.3370.0190.337Dual specificity tyrosine-phosphorylation regulated kinase 3 inhibitor

0.183 0.09 CHEMBL3527332

0.3180.0090.318Sodium channel blocker
0.3110.0090.311Heat shock protein 90 antagonist
0.3240.030.324Ca2+/calmodulin-dependent kinase II gamma inhibitor
0.310.0340.31Ca2+/calmodulin-dependent kinase II beta inhibitor
0.3690.10.3695 Hydroxytryptamine release inhibitor
0.3020.040.302Anticonvulsant
0.2580.0050.258Folate antagonist

0.162 0.018 CHEMBL3527332

0.2890.0410.289Death-associated protein kinase 3 inhibitor
0.2590.0240.259Heat shock protein 90 alpha antagonist
0.2370.0050.237Electrolyte absorption antagonist
0.2340.0080.234Adenosine A2 receptor antagonist

0.2 0.01 CHEMBL3527332

0.2640.0430.264Interleukin-1 receptor-associated protein kinase 1 inhibitor
0.2290.0080.229Adenosine A2a receptor antagonist

0.201 0.01 CHEMBL3527332

0.2230.0090.333Adenosine A1 receptor antagonist

0.333 0.005 CHEMBL3527332

CHEMBL3527332
0.2450.0360.245Nitric-oxide synthase stimulant
0.2520.0480.315RNA-directed DNA polymerase inhibitor

0.315 0.029 CHEMBL3527332

CHEMBL3527332
0.2250.0210.225Sodium channel (voltage-gated) blocker
0.2560.0580.256Ca2+/calmodulin-dependent kinase I alpha inhibitor

0.149 0.147 CHEMBL3527332

0.2430.0480.243CDC-like kinase 2 inhibitor
0.2220.0430.222Dual specificity tyrosine-phosphorylation-regulated kinase 4 inhibitor
0.20.0240.2Ephrin antagonist
0.2260.060.226Tyrosine kinase inhibitor
0.2220.0570.222CDC-like kinase 4 inhibitor
0.3340.1690.334Ca2+/calmodulin-dependent protein kinase kinase A inhibitor
0.2070.0430.207Protein kinase (CK1) gamma 3 inhibitor
0.1870.0270.187Interleukin 4 antagonist

0.146 0.054 CHEMBL3527332

0.2250.0660.225Clk dual-specificity kinase inhibitor
0.2140.0550.214Peroxidase inhibitor
0.2360.0780.236Antiamyloidogenic
0.190.0320.19Protein kinase (CK1) delta inhibitor
0.2330.080.233Dyrk kinase inhibitor
0.1880.0350.188Cell wall synthesis inhibitor

0.167 0.05 CHEMBL3527332

0.1610.0090.161Purinergic P2X2 antagonist

0.141 0.014 CHEMBL3527332

0.1930.0420.193Protein kinase (CK1) inhibitor
0.220.0810.22Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor
0.1450.0060.145Adenosine A2b receptor antagonist

0.054 0.03 CHEMBL3527332

0.2070.0720.207Ca2+/calmodulin-dependent protein kinase inhibitor
0.1440.0130.144Interleukin 5 antagonist

0.086 0.062 CHEMBL3527332

0.1770.0490.177Glycogen synthase kinase-3 alpha inhibitor
0.1610.0360.161Protein kinase (CK2) alpha inhibitor
0.1930.0710.193TRKC antagonist
0.2520.1330.433Vasodilator, coronary

0.433 0.026 CHEMBL3527332

CHEMBL3527332
0.1390.0250.139Interleukin 2 antagonist
0.1190.0070.119Heat shock protein 90 beta antagonist
0.1370.0270.137Phosphodiesterase 7B inhibitor
0.1460.0380.146MAP kinase 13 inhibitor
0.1230.0150.123Phosphatidylinositol 3-kinase delta inhibitor
0.1230.0170.39Adenosine A3 receptor antagonist

0.39 0.004 CHEMBL3527332

CHEMBL3527332
0.1480.0430.148MAP kinase 12 inhibitor
0.2040.10.204Aryl hydrocarbon receptor agonist
0.1650.0650.178Diuretic

0.178 0.055 CHEMBL3527332

CHEMBL3527332
0.1590.0610.159Ca2+/calmodulin-dependent kinase II delta inhibitor
0.1070.010.108S-adenosyl-L-methionine decarboxylase inhibitor

0.108 0.009 CHEMBL3527332

CHEMBL3527332
0.1610.0640.161Protein kinase C nu inhibitor
0.1190.0270.119AXL receptor tyrosine kinase inhibitor
0.1150.0260.115Factor XII inhibitor
0.0930.0040.093Dihydrofolate reductase inhibitor
0.1510.0640.151Ribosomal protein S6 kinase inhibitor
0.1080.0250.108mTOR complex 2 inhibitor
0.0980.0150.098Phosphodiesterase VIII inhibitor

0.07 0.053 CHEMBL3527332

0.1990.1160.199DNA damaging
0.1160.0330.116Histamine N-methyltransferase inhibitor
0.1140.0320.222NADH dehydrogenase inhibitor

0.222 0.009 CHEMBL3527332

CHEMBL3527332
0.2010.1210.428DNA synthesis inhibitor

0.428 0.019 CHEMBL3527332

CHEMBL3527332
0.1440.0690.144Protein-tyrosine kinase Lyn inhibitor
0.1130.0440.113HIV-1 integrase (Overall Integration) inhibitor
0.1720.1040.244Glyceraldehyde-3-phosphate dehydrogenase inhibitor

0.244 0.045 CHEMBL3527332

CHEMBL3527332
0.130.0630.13M18 aspartyl aminopeptidase inhibitor
0.1710.1050.171Proto-oncogene tyrosine-protein kinase Fyn inhibitor
0.1260.0610.126Protein kinase (CK1) gamma 2 inhibitor
0.120.0570.12Polo-like kinase-4 inhibitor
0.0840.0220.084EphB4 antagonist
0.1140.0520.114Protein kinase (CK2) inhibitor
0.0910.030.091Phenylalanine 4-hydroxylase inhibitor
0.1660.1070.166MAP kinase kinase 2 inhibitor
0.1410.0830.141MAP kinase 3 inhibitor
0.1710.1150.171Potassium channel blocker
0.0850.0320.085CDC7 inhibitor
0.1160.0670.116Aurora-B kinase inhibitor
0.140.0960.14Polo-like kinase-3 inhibitor
0.0540.0110.054Phenylethanolamine N methyltransferase inhibitor
0.1090.0660.109EphA2 antagonist
0.1360.0950.136GABA C receptor rho-2 antagonist
0.0670.0280.101Mannitol-1-phosphate 5-dehydrogenase inhibitor

0.101 0.014 CHEMBL3527332

CHEMBL3527332
0.1260.0860.126Nav1.6 sodium channel blocker
0.0590.020.059Histamine H4 receptor antagonist
0.1310.0930.131Dual specificity tyrosine-phosphorylation regulated kinase 1B inhibitor
0.1570.120.157Focal adhesion kinase 2 inhibitor
0.0950.0590.095Toll-Like receptor 3 antagonist
0.1110.0770.111Protein-tyrosine kinase (PTK, not ETK, WZC) inhibitor
0.0580.0240.058Purinergic P2X antagonist
0.110.0770.11Abl kinase inhibitor
0.180.1460.18Streptokinase A inhibitor
0.0750.0420.075Secretase beta inhibitor
0.1320.10.132Cyclin-dependent kinase 8 inhibitor
0.0990.0680.099Carbonic anhydrase XV inhibitor
0.0480.0180.0483-Hydroxyanthranilate 3,4-dioxygenase inhibitor
0.0770.0480.077GABA B receptor agonist
0.1040.0770.104Nav1.5 sodium channel blocker
0.0430.0170.088Phosphoglycerate kinase inhibitor

0.088 0.008 CHEMBL3527332

CHEMBL3527332
0.030.0050.03Toll-Like receptor 8 agonist
0.0750.0490.075Nav1.8 sodium channel blocker
0.0590.0330.059Cyclin B inhibitor
0.0510.0260.051Cytokine production stimulant

0.048 0.036 CHEMBL3527332

0.1290.1050.174Hexokinase inhibitor

0.174 0.055 CHEMBL3527332

CHEMBL3527332
0.0470.0240.047Guanylate cyclase stimulant
0.0830.0610.083D-Ala-D-Ala ligase inhibitor
0.0960.0750.096Ferrochelatase inhibitor
0.0840.0650.084Granulocyte macrophage colony stimulating factor agonist
0.040.0220.04Growth hormone secretagogue receptor antagonist
0.0390.0240.039Integrin alpha1beta1 antagonist
0.090.0770.09Insulin receptor antagonist
0.0960.0820.096Cystathionine beta-synthase inhibitor
0.0620.0490.062Interferon inducer
0.0590.0490.059Purinergic P2 antagonist
0.0320.0210.032Potassium channel small-conductance Ca-activated activator
0.0450.0350.045Thymidylate synthase inhibitor
0.0270.0170.031Thymidine phosphorylase inhibitor

0.031 0.011 CHEMBL3527332

CHEMBL3527332
0.1290.120.129CF transmembrane conductance regulator agonist
0.0640.0550.064ZAP-70 protein tyrosine kinase inhibitor
0.0820.0730.082Pim-3 kinase inhibitor
0.0730.0650.073Interferon agonist
0.1230.1170.123Neuropeptide Y1 antagonist
0.0180.0130.018Cyclin T1 inhibitor
0.0910.0850.144Adenylate kinase inhibitor

0.144 0.029 CHEMBL3527332

CHEMBL3527332
0.0270.0230.035Purinergic P2Y15 antagonist

0.035 0.01 CHEMBL3527332

CHEMBL3527332
0.0970.0930.097Beta amyloid protein antagonist
0.0310.0290.031Purinergic P2X7 antagonist
0.0070.0050.007DNA topoisomerase III inhibitor
0.0190.0170.034Adenosine kinase inhibitor

0.034 0.009 CHEMBL3527332

CHEMBL3527332
0.080.0780.202Aminoacyl-tRNA synthetase inhibitor

0.202 0.01 CHEMBL3527332

CHEMBL3527332
0.0540.0530.089Purinergic P2X1 antagonist

0.089 0.021 CHEMBL3527332

CHEMBL3527332
0.0390.040.049AICAR transformylase inhibitor

0.049 0.024 CHEMBL3527332

CHEMBL3527332
0.0130.0140.027S-adenosyl-L-homocysteine hydrolase inhibitor

0.027 0.005 CHEMBL3527332

CHEMBL3527332
0.0220.0240.041Purinergic P2X agonist

0.041 0.012 CHEMBL3527332

CHEMBL3527332
0.0120.0160.021Adenosine A2b receptor agonist

0.021 0.005 CHEMBL3527332

CHEMBL3527332
0.050.0550.085Carbamoyl phosphate synthetase inhibitor

0.085 0.026 CHEMBL3527332

CHEMBL3527332
0.0140.020.021O6-alkylguanine-DNA alkyltransferase inhibitor

0.021 0.006 CHEMBL3527332

CHEMBL3527332
0.1040.1150.18DNA repair enzyme inhibitor

0.18 0.013 CHEMBL3527332

CHEMBL3527332
0.0610.0720.096Glutamate dehydrogenase inhibitor

0.096 0.033 CHEMBL3527332

CHEMBL3527332
0.0080.020.011Purine nucleoside phosphorylase inhibitor

0.011 0.01 CHEMBL3527332

CHEMBL3527332
0.0090.0230.021Adenosine A2a receptor agonist

0.021 0.008 CHEMBL3527332

CHEMBL3527332
0.0120.0290.024Adenosine A3 receptor agonist

0.024 0.006 CHEMBL3527332

CHEMBL3527332
0.0330.0490.04Thymidine kinase inhibitor

0.04 0.03 CHEMBL3527332

CHEMBL3527332
0.1260.1440.401DNA methylase inhibitor

0.401 0.011 CHEMBL3527332

CHEMBL3527332
0.010.030.022Adenosine A2 receptor agonist

0.022 0.007 CHEMBL3527332

CHEMBL3527332
0.0750.0960.085DNA directed RNA polymerase inhibitor

0.085 0.077 CHEMBL3527332

CHEMBL3527332
0.0390.0650.077Argininosuccinate synthase inhibitor

0.077 0.027 CHEMBL3527332

CHEMBL3527332
0.0210.050.039Fumarate hydratase inhibitor

0.039 0.02 CHEMBL3527332

CHEMBL3527332
0.0290.060.071Adenosine deaminase inhibitor

0.071 0.013 CHEMBL3527332

CHEMBL3527332
0.0150.0480.023Isoleucine-tRNA ligase inhibitor

0.023 0.015 CHEMBL3527332

CHEMBL3527332
0.1390.1730.183Cyclic AMP phosphodiesterase inhibitor

0.183 0.108 CHEMBL3527332

CHEMBL3527332
0.1150.1530.356DNA methyltransferase I inhibitor

0.356 0.013 CHEMBL3527332

CHEMBL3527332
0.0410.0850.126Phosphofructokinase-1 inhibitor

0.126 0.024 CHEMBL3527332

CHEMBL3527332
0.0370.0820.063Biliverdin reductase inhibitor

0.063 0.038 CHEMBL3527332

CHEMBL3527332
0.1230.1680.141Heat shock protein 70 antagonist

0.141 0.071 CHEMBL3527332

CHEMBL3527332
0.0680.1150.159UDP-glucose 4-epimerase inhibitor

0.159 0.026 CHEMBL3527332

CHEMBL3527332
0.0030.0550.016Purinergic P2 agonist

0.016 0.01 CHEMBL3527332

CHEMBL3527332
0.0030.0550.016Purinergic receptor agonist

0.016 0.01 CHEMBL3527332

CHEMBL3527332
0.0030.0560.012Purinergic P2Y agonist

0.012 0.009 CHEMBL3527332

CHEMBL3527332
0.010.0630.042Adenosine A1 receptor agonist

0.042 0.007 CHEMBL3527332

CHEMBL3527332
0.2290.2920.344Antiinflammatory

0.344 0.177 CHEMBL3527332

CHEMBL3527332
0.0230.0860.059Antimetabolite

0.059 0.026 CHEMBL3527332

CHEMBL3527332
0.150.2220.237Cholesterol antagonist

0.237 0.135 CHEMBL3527332

CHEMBL3527332
0.1090.2030.424Immunostimulant

0.424 0.043 CHEMBL3527332

CHEMBL3527332
0.0610.1560.125Adenylate cyclase inhibitor

0.125 0.063 CHEMBL3527332

CHEMBL3527332
0.0070.1130.021Inosine monophosphate dehydrogenase 1 inhibitor

0.021 0.013 CHEMBL3527332

CHEMBL3527332
0.0510.1840.085UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor

0.085 0.073 CHEMBL3527332

CHEMBL3527332
0.0260.1730.07Factor IXa inhibitor

0.07 0.02 CHEMBL3527332

CHEMBL3527332
0.0710.2770.12NOS3 expression enhancer

0.12 0.116 CHEMBL3527332

CHEMBL3527332
0.1220.350.381Antibacterial

0.381 0.086 CHEMBL3527332

CHEMBL3527332
0.0320.4180.192DNA polymerase I inhibitor

0.192 0.031 CHEMBL3527332

CHEMBL3527332
0.0750.6580.285Peptidyltransferase inhibitor

0.285 0.03 CHEMBL3527332

CHEMBL3527332
0.0660.6950.213Interleukin 2 agonist

0.213 0.168 CHEMBL3527332

CHEMBL3527332
0.0170.670.231Vasodilator

0.231 0.081 CHEMBL3527332

CHEMBL3527332
0.0090.7060.034Antibiotic Aminoglycoside-like

0.034 0.029 CHEMBL3527332

CHEMBL3527332
0.0270.7380.168Hepatoprotectant

0.168 0.091 CHEMBL3527332

CHEMBL3527332
0.0120.7560.463Angiogenesis stimulant

0.463 0.014 CHEMBL3527332

CHEMBL3527332
0.0050.8130.123Topoisomerase I inhibitor

0.123 0.054 CHEMBL3527332

CHEMBL3527332
0.0060.8150.049Protein 50S ribosomal subunit inhibitor

0.049 0.041 CHEMBL3527332

CHEMBL3527332
0.0060.9030.123Thrombolytic

0.123 0.107 CHEMBL3527332

CHEMBL3527332
0.0070.9210.302Apoptosis agonist

0.302 0.17 CHEMBL3527332

CHEMBL3527332
0.0080.9310.155Platelet adhesion inhibitor

0.155 0.1 CHEMBL3527332

CHEMBL3527332
Ext Pa Pi Pmax Activity Other Results ID Pa_max