Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.8560.0020.956Estrogen antagonist

0.787 0.003 CHEMBL4525767

0.871 0.002 CHEMBL2137046

0.956 0.001 CHEMBL50995

0.822 0.003 CHEMBL1093458

0.813 0.003 CHEMBL1743350

0.832 0.002 CHEMBL4525766

CHEMBL50995
0.830.0070.865Caspase 9 stimulant

0.767 0.016 CHEMBL4525767

0.849 0.005 CHEMBL2137046

0.865 0.004 CHEMBL50995

0.8 0.011 CHEMBL1093458

0.779 0.014 CHEMBL1743350

0.857 0.005 CHEMBL4525766

CHEMBL50995
0.8030.0040.923Aldehyde oxidase inhibitor

0.539 0.027 CHEMBL4525767

0.918 0.003 CHEMBL2137046

0.867 0.004 CHEMBL50995

0.672 0.01 CHEMBL1093458

0.618 0.017 CHEMBL1743350

0.923 0.003 CHEMBL4525766

CHEMBL4525766
0.6920.0050.758Vasodilator, coronary

0.648 0.005 CHEMBL4525767

0.697 0.005 CHEMBL2137046

0.485 0.018 CHEMBL50995

0.651 0.005 CHEMBL1093458

0.625 0.007 CHEMBL1743350

0.758 0.004 CHEMBL4525766

CHEMBL4525766
0.6630.0040.736Growth factor agonist

0.652 0.004 CHEMBL4525767

0.554 0.004 CHEMBL2137046

0.736 0.003 CHEMBL50995

0.55 0.004 CHEMBL1093458

0.587 0.004 CHEMBL1743350

0.546 0.004 CHEMBL4525766

CHEMBL50995
0.6050.0120.674Spasmolytic

0.525 0.02 CHEMBL4525767

0.646 0.009 CHEMBL2137046

0.318 0.063 CHEMBL50995

0.578 0.015 CHEMBL1093458

0.383 0.044 CHEMBL1743350

0.674 0.007 CHEMBL4525766

CHEMBL4525766
0.5780.0070.578Vasodilator

0.551 0.009 CHEMBL4525767

0.559 0.008 CHEMBL2137046

0.535 0.009 CHEMBL50995

0.535 0.009 CHEMBL1093458

0.569 0.007 CHEMBL1743350

0.569 0.007 CHEMBL4525766

0.5720.0040.572Anesthetic local

0.474 0.005 CHEMBL4525767

0.517 0.004 CHEMBL2137046

0.21 0.03 CHEMBL50995

0.431 0.005 CHEMBL1093458

0.302 0.012 CHEMBL1743350

0.549 0.004 CHEMBL4525766

0.5340.0010.841Estrogen-related receptor gamma agonist

0.468 0.001 CHEMBL4525767

0.841 0.001 CHEMBL2137046

0.27 0.001 CHEMBL50995

0.735 0.001 CHEMBL1093458

0.086 0.002 CHEMBL1743350

0.788 0.001 CHEMBL4525766

CHEMBL2137046
0.5210.0010.657Estrogen-related receptor beta agonist

0.308 0.001 CHEMBL4525767

0.657 0 CHEMBL2137046

0.349 0.001 CHEMBL50995

0.432 0.001 CHEMBL1093458

0.258 0.002 CHEMBL1743350

0.592 0.001 CHEMBL4525766

CHEMBL2137046
0.50600.913Estrogen-related receptor beta antagonist

0.41 0.001 CHEMBL4525767

0.474 0.001 CHEMBL2137046

0.913 0 CHEMBL50995

0.383 0.001 CHEMBL1093458

0.469 0.001 CHEMBL1743350

0.425 0.001 CHEMBL4525766

CHEMBL50995
0.5030.0040.83Estrogen agonist

0.415 0.004 CHEMBL4525767

0.565 0.003 CHEMBL2137046

0.83 0.002 CHEMBL50995

0.499 0.004 CHEMBL1093458

0.455 0.004 CHEMBL1743350

0.504 0.004 CHEMBL4525766

CHEMBL50995
0.460.0040.815Estrogen receptor beta antagonist

0.36 0.004 CHEMBL4525767

0.568 0.003 CHEMBL2137046

0.815 0.002 CHEMBL50995

0.485 0.004 CHEMBL1093458

0.399 0.004 CHEMBL1743350

0.49 0.004 CHEMBL4525766

CHEMBL50995
0.4570.0280.701Caspase 3 stimulant

0.428 0.036 CHEMBL4525767

0.472 0.025 CHEMBL2137046

0.701 0.005 CHEMBL50995

0.445 0.031 CHEMBL1093458

0.44 0.032 CHEMBL1743350

0.487 0.022 CHEMBL4525766

CHEMBL50995
0.440.0210.49DNA damaging

0.435 0.021 CHEMBL4525767

0.455 0.019 CHEMBL2137046

0.42 0.024 CHEMBL50995

0.45 0.019 CHEMBL1093458

0.49 0.015 CHEMBL1743350

0.462 0.018 CHEMBL4525766

CHEMBL1743350
0.4110.0050.414Alpha 2b adrenoreceptor antagonist

0.414 0.005 CHEMBL4525767

0.351 0.006 CHEMBL2137046

0.236 0.017 CHEMBL50995

0.354 0.006 CHEMBL1093458

0.304 0.009 CHEMBL1743350

0.36 0.006 CHEMBL4525766

CHEMBL4525767
0.3910.0040.663Estrogen receptor alpha antagonist

0.174 0.009 CHEMBL4525767

0.663 0.003 CHEMBL2137046

0.5 0.003 CHEMBL50995

0.374 0.004 CHEMBL1093458

0.153 0.011 CHEMBL1743350

0.63 0.003 CHEMBL4525766

CHEMBL2137046
0.3930.0230.394Psychostimulant

0.363 0.029 CHEMBL4525767

0.392 0.024 CHEMBL2137046

0.239 0.063 CHEMBL50995

0.361 0.029 CHEMBL1093458

0.236 0.064 CHEMBL1743350

0.394 0.023 CHEMBL4525766

CHEMBL4525766
0.4060.0530.457Vasodilator, peripheral

0.292 0.101 CHEMBL4525767

0.412 0.051 CHEMBL2137046

0.215 0.159 CHEMBL50995

0.298 0.098 CHEMBL1093458

0.457 0.039 CHEMBL4525766

CHEMBL4525766
0.3480.0090.356Acetylcholine M1 receptor antagonist

0.278 0.019 CHEMBL4525767

0.356 0.008 CHEMBL2137046

0.26 0.023 CHEMBL50995

0.283 0.018 CHEMBL1093458

0.239 0.028 CHEMBL1743350

0.335 0.01 CHEMBL4525766

CHEMBL2137046
0.3340.0040.3375 Hydroxytryptamine 3E antagonist

0.337 0.004 CHEMBL4525767

0.263 0.011 CHEMBL2137046

0.183 0.097 CHEMBL50995

0.266 0.01 CHEMBL1093458

0.317 0.004 CHEMBL1743350

0.25 0.016 CHEMBL4525766

CHEMBL4525767
0.3510.0210.375P-glycoprotein inhibitor

0.303 0.028 CHEMBL4525767

0.319 0.026 CHEMBL2137046

0.375 0.019 CHEMBL50995

0.281 0.033 CHEMBL1093458

0.295 0.03 CHEMBL1743350

0.346 0.022 CHEMBL4525766

CHEMBL50995
0.3260.0030.326Phosphodiesterase 1B inhibitor

0.132 0.009 CHEMBL4525767

0.278 0.004 CHEMBL2137046

0.191 0.005 CHEMBL50995

0.104 0.013 CHEMBL1093458

0.156 0.006 CHEMBL1743350

0.246 0.004 CHEMBL4525766

0.3240.0030.324Phosphodiesterase 1C inhibitor

0.14 0.005 CHEMBL4525767

0.288 0.003 CHEMBL2137046

0.184 0.004 CHEMBL50995

0.121 0.006 CHEMBL1093458

0.16 0.004 CHEMBL1743350

0.271 0.003 CHEMBL4525766

0.3090.0050.422Phosphodiesterase 4A inhibitor

0.235 0.005 CHEMBL4525767

0.221 0.006 CHEMBL2137046

0.422 0.004 CHEMBL50995

0.166 0.009 CHEMBL1093458

0.284 0.005 CHEMBL1743350

0.234 0.005 CHEMBL4525766

CHEMBL50995
0.3020.0050.302Phosphodiesterase I inhibitor

0.153 0.017 CHEMBL4525767

0.275 0.005 CHEMBL2137046

0.248 0.007 CHEMBL50995

0.13 0.023 CHEMBL1093458

0.219 0.009 CHEMBL1743350

0.255 0.006 CHEMBL4525766

0.2950.0040.323Histamine H2 receptor antagonist

0.323 0.003 CHEMBL4525767

0.202 0.005 CHEMBL2137046

0.111 0.026 CHEMBL50995

0.226 0.005 CHEMBL1093458

0.218 0.005 CHEMBL1743350

0.219 0.005 CHEMBL4525766

CHEMBL4525767
0.3460.0570.6115 Hydroxytryptamine release stimulant

0.492 0.029 CHEMBL4525767

0.364 0.053 CHEMBL2137046

0.611 0.013 CHEMBL50995

0.506 0.026 CHEMBL1093458

0.572 0.017 CHEMBL1743350

0.231 0.099 CHEMBL4525766

CHEMBL50995
0.2890.0040.367CYP2A6 inhibitor

0.275 0.004 CHEMBL4525767

0.219 0.005 CHEMBL2137046

0.239 0.005 CHEMBL50995

0.21 0.006 CHEMBL1093458

0.367 0.003 CHEMBL1743350

0.188 0.009 CHEMBL4525766

CHEMBL1743350
0.370.090.429Histamine release inhibitor

0.211 0.189 CHEMBL4525767

0.424 0.063 CHEMBL2137046

0.429 0.061 CHEMBL50995

0.269 0.142 CHEMBL1093458

0.235 0.167 CHEMBL1743350

0.425 0.063 CHEMBL4525766

CHEMBL50995
0.2980.0330.342Anesthetic general

0.192 0.079 CHEMBL4525767

0.342 0.025 CHEMBL2137046

0.277 0.039 CHEMBL50995

0.226 0.061 CHEMBL1093458

0.212 0.068 CHEMBL1743350

0.324 0.028 CHEMBL4525766

CHEMBL2137046
0.2630.0010.506Estrogen-related receptor gamma antagonist

0.137 0.001 CHEMBL4525767

0.506 0 CHEMBL2137046

0.107 0.001 CHEMBL50995

0.253 0.001 CHEMBL1093458

0.088 0.001 CHEMBL1743350

0.35 0 CHEMBL4525766

CHEMBL2137046
0.3470.0870.578GABA C receptor rho-3 antagonist

0.365 0.078 CHEMBL4525767

0.384 0.069 CHEMBL2137046

0.578 0.01 CHEMBL50995

0.402 0.06 CHEMBL1093458

0.399 0.062 CHEMBL1743350

0.28 0.13 CHEMBL4525766

CHEMBL50995
0.3780.1240.512Apoptosis agonist

0.382 0.123 CHEMBL4525767

0.432 0.099 CHEMBL2137046

0.512 0.071 CHEMBL50995

0.432 0.099 CHEMBL1093458

0.359 0.134 CHEMBL1743350

0.472 0.083 CHEMBL4525766

CHEMBL50995
0.2560.0030.366Beta 3 adrenoreceptor antagonist

0.289 0.003 CHEMBL4525767

0.332 0.002 CHEMBL2137046

0.195 0.004 CHEMBL50995

0.366 0.002 CHEMBL1093458

0.165 0.005 CHEMBL1743350

0.339 0.002 CHEMBL4525766

CHEMBL1093458
0.2560.0040.256Sphingomyelinase inhibitor

0.219 0.007 CHEMBL4525767

0.227 0.005 CHEMBL2137046

0.135 0.032 CHEMBL50995

0.192 0.011 CHEMBL1093458

0.218 0.007 CHEMBL1743350

0.238 0.005 CHEMBL4525766

0.2610.020.261Nav1.2 sodium channel blocker

0.216 0.029 CHEMBL4525767

0.208 0.032 CHEMBL2137046

0.173 0.045 CHEMBL1093458

0.177 0.044 CHEMBL1743350

0.17 0.047 CHEMBL4525766

0.2370.0030.237Phosphodiesterase 1A inhibitor

0.13 0.006 CHEMBL4525767

0.173 0.004 CHEMBL2137046

0.139 0.005 CHEMBL50995

0.088 0.013 CHEMBL1093458

0.126 0.006 CHEMBL1743350

0.158 0.004 CHEMBL4525766

0.2630.0390.298Proto-oncogene tyrosine-protein kinase Fyn inhibitor

0.244 0.045 CHEMBL4525767

0.232 0.051 CHEMBL2137046

0.298 0.03 CHEMBL50995

0.221 0.057 CHEMBL1093458

0.22 0.057 CHEMBL1743350

0.237 0.048 CHEMBL4525766

CHEMBL50995
0.2230.0130.223Nav1.6 sodium channel blocker

0.18 0.028 CHEMBL4525767

0.18 0.028 CHEMBL2137046

0.123 0.091 CHEMBL50995

0.149 0.055 CHEMBL1093458

0.147 0.057 CHEMBL1743350

0.174 0.032 CHEMBL4525766

0.2160.0210.224Acetylcholine muscarinic antagonist

0.146 0.046 CHEMBL4525767

0.224 0.019 CHEMBL2137046

0.142 0.049 CHEMBL50995

0.152 0.043 CHEMBL1093458

0.117 0.07 CHEMBL1743350

0.205 0.023 CHEMBL4525766

CHEMBL2137046
0.2180.0230.2185 Hydroxytryptamine 2B antagonist

0.135 0.048 CHEMBL4525767

0.151 0.04 CHEMBL2137046

0.106 0.076 CHEMBL50995

0.102 0.081 CHEMBL1093458

0.121 0.06 CHEMBL1743350

0.146 0.043 CHEMBL4525766

0.2010.0130.201Calcium antagonist

0.105 0.044 CHEMBL4525767

0.113 0.039 CHEMBL2137046

0.123 0.033 CHEMBL1743350

0.122 0.034 CHEMBL4525766

0.2010.0140.201Alpha 2a adrenoreceptor antagonist

0.196 0.014 CHEMBL4525767

0.18 0.017 CHEMBL2137046

0.121 0.029 CHEMBL50995

0.176 0.018 CHEMBL1093458

0.166 0.019 CHEMBL1743350

0.2 0.014 CHEMBL4525766

0.1920.0060.192Acetylcholine M4 receptor antagonist

0.107 0.023 CHEMBL4525767

0.119 0.018 CHEMBL2137046

0.088 0.039 CHEMBL50995

0.072 0.054 CHEMBL1093458

0.088 0.039 CHEMBL1743350

0.105 0.024 CHEMBL4525766

0.2310.0460.256Insulin sensitizer

0.244 0.038 CHEMBL4525767

0.242 0.039 CHEMBL2137046

0.223 0.052 CHEMBL50995

0.255 0.032 CHEMBL1093458

0.246 0.037 CHEMBL1743350

0.256 0.031 CHEMBL4525766

CHEMBL4525766
0.2070.0220.207Nav1.3 sodium channel blocker

0.183 0.031 CHEMBL4525767

0.155 0.044 CHEMBL2137046

0.135 0.06 CHEMBL1093458

0.101 0.096 CHEMBL1743350

0.137 0.057 CHEMBL4525766

0.2830.1020.37Cholesterol antagonist

0.299 0.092 CHEMBL4525767

0.329 0.074 CHEMBL2137046

0.37 0.057 CHEMBL50995

0.346 0.066 CHEMBL1093458

0.275 0.108 CHEMBL1743350

0.336 0.071 CHEMBL4525766

CHEMBL50995
0.1830.0050.183Acetylcholine M5 receptor antagonist

0.123 0.012 CHEMBL4525767

0.158 0.007 CHEMBL2137046

0.1 0.017 CHEMBL50995

0.107 0.016 CHEMBL1093458

0.086 0.022 CHEMBL1743350

0.14 0.009 CHEMBL4525766

0.2070.030.207Cholinergic antagonist

0.154 0.05 CHEMBL4525767

0.203 0.031 CHEMBL2137046

0.111 0.082 CHEMBL50995

0.151 0.052 CHEMBL1093458

0.123 0.071 CHEMBL1743350

0.184 0.036 CHEMBL4525766

0.210.0330.305Bone formation stimulant

0.177 0.043 CHEMBL4525767

0.244 0.026 CHEMBL2137046

0.305 0.016 CHEMBL50995

0.21 0.033 CHEMBL1093458

0.232 0.028 CHEMBL1743350

0.217 0.031 CHEMBL4525766

CHEMBL50995
0.20.0310.2Acetylcholine antagonist

0.147 0.051 CHEMBL4525767

0.195 0.032 CHEMBL2137046

0.108 0.082 CHEMBL50995

0.144 0.053 CHEMBL1093458

0.115 0.075 CHEMBL1743350

0.177 0.037 CHEMBL4525766

0.1880.0190.189Alpha 2 adrenoreceptor antagonist

0.189 0.019 CHEMBL4525767

0.151 0.027 CHEMBL2137046

0.09 0.055 CHEMBL50995

0.151 0.027 CHEMBL1093458

0.13 0.033 CHEMBL1743350

0.171 0.023 CHEMBL4525766

CHEMBL4525767
0.1760.0080.198Anabolic

0.157 0.015 CHEMBL4525767

0.184 0.006 CHEMBL2137046

0.198 0.004 CHEMBL50995

0.166 0.011 CHEMBL1093458

0.166 0.011 CHEMBL1743350

0.178 0.008 CHEMBL4525766

CHEMBL50995
0.1770.0110.274Thioredoxin inhibitor

0.185 0.01 CHEMBL4525767

0.175 0.011 CHEMBL2137046

0.274 0.004 CHEMBL50995

0.182 0.01 CHEMBL1093458

0.203 0.008 CHEMBL1743350

0.175 0.011 CHEMBL4525766

CHEMBL50995
0.1690.0040.299Estrogen-related receptor alpha antagonist

0.142 0.004 CHEMBL4525767

0.163 0.004 CHEMBL2137046

0.299 0.002 CHEMBL50995

0.141 0.004 CHEMBL1093458

0.154 0.004 CHEMBL1743350

0.153 0.004 CHEMBL4525766

CHEMBL50995
0.190.0290.247Cholesterol synthesis inhibitor

0.098 0.091 CHEMBL4525767

0.236 0.02 CHEMBL2137046

0.227 0.021 CHEMBL50995

0.12 0.065 CHEMBL1093458

0.108 0.077 CHEMBL1743350

0.247 0.018 CHEMBL4525766

CHEMBL4525766
0.2010.0420.404Cyclooxygenase inhibitor

0.197 0.043 CHEMBL4525767

0.2 0.042 CHEMBL2137046

0.404 0.007 CHEMBL50995

0.197 0.043 CHEMBL1093458

0.224 0.033 CHEMBL1743350

0.202 0.041 CHEMBL4525766

CHEMBL50995
0.2380.0810.479Tyrosine 3 hydroxylase inhibitor

0.245 0.073 CHEMBL4525767

0.286 0.04 CHEMBL2137046

0.479 0.004 CHEMBL50995

0.295 0.035 CHEMBL1093458

0.303 0.032 CHEMBL1743350

0.293 0.037 CHEMBL4525766

CHEMBL50995
0.2740.1190.363Calcium channel activator

0.363 0.042 CHEMBL4525767

0.252 0.144 CHEMBL2137046

0.304 0.088 CHEMBL50995

0.344 0.054 CHEMBL1093458

0.36 0.044 CHEMBL1743350

0.233 0.167 CHEMBL4525766

CHEMBL4525767
0.1890.0390.427Cyclooxygenase 1 inhibitor

0.197 0.035 CHEMBL4525767

0.203 0.033 CHEMBL2137046

0.427 0.006 CHEMBL50995

0.21 0.03 CHEMBL1093458

0.206 0.032 CHEMBL1743350

0.206 0.032 CHEMBL4525766

CHEMBL50995
0.2120.0630.276Glyceraldehyde-3-phosphate dehydrogenase inhibitor

0.261 0.038 CHEMBL2137046

0.239 0.048 CHEMBL50995

0.155 0.137 CHEMBL1093458

0.168 0.11 CHEMBL1743350

0.276 0.032 CHEMBL4525766

CHEMBL4525766
0.160.0120.16Acetylcholine release stimulant

0.136 0.028 CHEMBL4525767

0.129 0.035 CHEMBL2137046

0.144 0.021 CHEMBL50995

0.108 0.069 CHEMBL1093458

0.117 0.053 CHEMBL1743350

0.125 0.041 CHEMBL4525766

0.1860.0470.214Arachidonic acid antagonist

0.124 0.121 CHEMBL4525767

0.19 0.043 CHEMBL2137046

0.214 0.021 CHEMBL50995

0.131 0.112 CHEMBL1093458

0.145 0.094 CHEMBL1743350

0.195 0.038 CHEMBL4525766

CHEMBL50995
0.1430.0040.153Phospholipase D inhibitor

0.153 0.003 CHEMBL4525767

0.135 0.004 CHEMBL2137046

0.142 0.004 CHEMBL50995

0.146 0.004 CHEMBL1093458

0.12 0.006 CHEMBL1743350

0.125 0.005 CHEMBL4525766

CHEMBL4525767
0.2990.1630.386Cyclophilin D inhibitor

0.318 0.147 CHEMBL4525767

0.326 0.141 CHEMBL2137046

0.386 0.099 CHEMBL50995

0.34 0.129 CHEMBL1093458

0.377 0.104 CHEMBL1743350

0.354 0.119 CHEMBL4525766

CHEMBL50995
0.1590.0280.168Alpha 2c adrenoreceptor antagonist

0.168 0.025 CHEMBL4525767

0.137 0.039 CHEMBL2137046

0.095 0.071 CHEMBL50995

0.144 0.035 CHEMBL1093458

0.129 0.043 CHEMBL1743350

0.138 0.038 CHEMBL4525766

CHEMBL4525767
0.1670.0370.219Proteasome inhibitor

0.177 0.033 CHEMBL4525767

0.165 0.038 CHEMBL2137046

0.219 0.02 CHEMBL50995

0.174 0.034 CHEMBL1093458

0.183 0.031 CHEMBL1743350

0.167 0.037 CHEMBL4525766

CHEMBL50995
0.1440.0160.144Histamine N-methyltransferase inhibitor

0.083 0.064 CHEMBL4525767

0.141 0.018 CHEMBL2137046

0.092 0.053 CHEMBL50995

0.078 0.069 CHEMBL1093458

0.116 0.033 CHEMBL1743350

0.112 0.035 CHEMBL4525766

0.1420.0160.229Dopamine D1 antagonist

0.098 0.025 CHEMBL4525767

0.225 0.009 CHEMBL2137046

0.176 0.012 CHEMBL50995

0.15 0.015 CHEMBL1093458

0.067 0.042 CHEMBL1743350

0.229 0.009 CHEMBL4525766

CHEMBL4525766
0.2520.1260.345Sodium/bile acid cotransporter inhibitor

0.306 0.074 CHEMBL4525767

0.319 0.063 CHEMBL2137046

0.324 0.058 CHEMBL50995

0.345 0.043 CHEMBL1093458

0.234 0.146 CHEMBL1743350

0.308 0.072 CHEMBL4525766

CHEMBL1093458
0.2060.0830.21ErbB-1 antagonist

0.21 0.079 CHEMBL2137046

0.179 0.117 CHEMBL4525766

CHEMBL2137046
0.150.0270.155 Hydroxytryptamine 2C antagonist

0.104 0.043 CHEMBL4525767

0.091 0.052 CHEMBL2137046

0.08 0.061 CHEMBL1743350

0.087 0.055 CHEMBL4525766

0.1270.0060.23Beta 1 adrenoreceptor antagonist

0.189 0.004 CHEMBL4525767

0.154 0.005 CHEMBL2137046

0.116 0.008 CHEMBL50995

0.23 0.003 CHEMBL1093458

0.124 0.007 CHEMBL1743350

0.163 0.004 CHEMBL4525766

CHEMBL1093458
0.1240.0040.151Squalene epoxidase inhibitor

0.085 0.008 CHEMBL4525767

0.122 0.004 CHEMBL2137046

0.063 0.018 CHEMBL50995

0.083 0.009 CHEMBL1093458

0.072 0.013 CHEMBL1743350

0.151 0.003 CHEMBL4525766

CHEMBL4525766
0.1280.0090.216Beta adrenoreceptor antagonist

0.172 0.005 CHEMBL4525767

0.16 0.005 CHEMBL2137046

0.116 0.011 CHEMBL50995

0.216 0.004 CHEMBL1093458

0.137 0.007 CHEMBL1743350

0.171 0.005 CHEMBL4525766

CHEMBL1093458
0.2250.110.4345 Hydroxytryptamine uptake stimulant

0.229 0.105 CHEMBL4525767

0.215 0.125 CHEMBL2137046

0.434 0.009 CHEMBL50995

0.218 0.12 CHEMBL1093458

0.302 0.044 CHEMBL1743350

0.25 0.081 CHEMBL4525766

CHEMBL50995
0.1290.0140.129Acetylcholine M2 receptor antagonist

0.075 0.033 CHEMBL4525767

0.122 0.016 CHEMBL2137046

0.069 0.037 CHEMBL50995

0.071 0.036 CHEMBL1093458

0.054 0.05 CHEMBL1743350

0.084 0.027 CHEMBL4525766

0.1240.0140.124Dopamine uptake inhibitor

0.121 0.014 CHEMBL4525767

0.095 0.02 CHEMBL2137046

0.076 0.027 CHEMBL50995

0.092 0.021 CHEMBL1093458

0.071 0.03 CHEMBL1743350

0.08 0.025 CHEMBL4525766

0.1120.0050.145 Hydroxytryptamine 1B agonist

0.14 0.004 CHEMBL4525767

0.084 0.011 CHEMBL2137046

0.102 0.006 CHEMBL1093458

0.12 0.005 CHEMBL1743350

0.075 0.015 CHEMBL4525766

CHEMBL4525767
0.1550.050.339Cyclooxygenase 2 inhibitor

0.142 0.06 CHEMBL4525767

0.149 0.054 CHEMBL2137046

0.339 0.009 CHEMBL50995

0.138 0.063 CHEMBL1093458

0.177 0.039 CHEMBL1743350

0.151 0.053 CHEMBL4525766

CHEMBL50995
0.1770.0730.177Lipocortins synthesis antagonist

0.176 0.074 CHEMBL2137046

0.167 0.084 CHEMBL4525766

0.1950.0980.222Cyclic AMP phosphodiesterase inhibitor

0.198 0.095 CHEMBL2137046

0.222 0.079 CHEMBL4525766

CHEMBL4525766
0.170.0730.181Sigma receptor agonist

0.181 0.068 CHEMBL2137046

0.142 0.091 CHEMBL4525766

CHEMBL2137046
0.1520.0570.152Calcium channel blocker

0.11 0.099 CHEMBL4525767

0.1110.0160.154Acetylcholine M3 receptor antagonist

0.076 0.028 CHEMBL4525767

0.154 0.011 CHEMBL2137046

0.095 0.02 CHEMBL50995

0.094 0.02 CHEMBL1093458

0.06 0.041 CHEMBL1743350

0.114 0.015 CHEMBL4525766

CHEMBL2137046
0.1040.0110.104Glycine transporter inhibitor

0.074 0.019 CHEMBL4525767

0.058 0.026 CHEMBL2137046

0.044 0.037 CHEMBL1743350

0.048 0.033 CHEMBL4525766

0.2790.1890.4935 Hydroxytryptamine release inhibitor

0.284 0.184 CHEMBL4525767

0.292 0.174 CHEMBL2137046

0.493 0.035 CHEMBL50995

0.297 0.168 CHEMBL1093458

0.398 0.079 CHEMBL1743350

CHEMBL50995
0.1240.0350.194Prolactin inhibitor

0.159 0.019 CHEMBL2137046

0.194 0.01 CHEMBL50995

0.108 0.048 CHEMBL1093458

0.087 0.071 CHEMBL1743350

0.157 0.019 CHEMBL4525766

CHEMBL50995
0.1260.040.126Antihistaminic

0.084 0.072 CHEMBL4525767

0.2070.1230.2075 Hydroxytryptamine 1E antagonist

0.194 0.138 CHEMBL4525767

0.188 0.144 CHEMBL2137046

0.201 0.13 CHEMBL50995

0.174 0.161 CHEMBL1093458

0.0840.0050.084GABA uptake inhibitor

0.04 0.025 CHEMBL4525767

0.078 0.005 CHEMBL2137046

0.062 0.009 CHEMBL50995

0.037 0.03 CHEMBL1093458

0.065 0.008 CHEMBL1743350

0.069 0.007 CHEMBL4525766

0.1180.0390.118Histamine antagonist

0.075 0.07 CHEMBL4525767

0.1010.0230.131Alpha 1d adrenoreceptor antagonist

0.131 0.017 CHEMBL4525767

0.066 0.037 CHEMBL2137046

0.086 0.028 CHEMBL1093458

0.085 0.028 CHEMBL1743350

0.051 0.048 CHEMBL4525766

CHEMBL4525767
0.1040.0260.104Interferon agonist

0.099 0.029 CHEMBL2137046

0.072 0.065 CHEMBL50995

0.082 0.049 CHEMBL1743350

0.089 0.039 CHEMBL4525766

0.0880.010.356Estrogen receptor alpha agonist

0.056 0.016 CHEMBL4525767

0.168 0.005 CHEMBL2137046

0.356 0.003 CHEMBL50995

0.119 0.007 CHEMBL1093458

0.062 0.015 CHEMBL1743350

0.114 0.007 CHEMBL4525766

CHEMBL50995
0.2230.1470.223Ca(v)3.3 blocker
0.1090.0390.168Phosphodiesterase IV inhibitor

0.074 0.068 CHEMBL4525767

0.168 0.018 CHEMBL50995

0.1 0.045 CHEMBL1743350

0.079 0.063 CHEMBL4525766

CHEMBL50995
0.1230.0570.1235 Hydroxytryptamine 2 antagonist

0.093 0.077 CHEMBL4525767

0.1070.0430.1075 Hydroxytryptamine 2A antagonist

0.071 0.066 CHEMBL4525767

0.0680.0050.0682,3-Oxidosqualene-lanosterol cyclase inhibitor

0.05 0.011 CHEMBL2137046

0.049 0.012 CHEMBL4525766

0.190.1280.19Cardiotonic

0.176 0.144 CHEMBL4525766

0.1410.0790.19Adenylate cyclase stimulant

0.172 0.033 CHEMBL4525767

0.158 0.05 CHEMBL2137046

0.183 0.023 CHEMBL50995

0.19 0.019 CHEMBL1093458

0.153 0.058 CHEMBL1743350

0.17 0.035 CHEMBL4525766

CHEMBL1093458
0.1310.0690.164MAO inhibitor

0.101 0.089 CHEMBL4525767

0.162 0.055 CHEMBL2137046

0.125 0.072 CHEMBL1093458

0.158 0.057 CHEMBL1743350

0.164 0.054 CHEMBL4525766

CHEMBL4525766
0.1640.1040.167MAP kinase kinase 5 inhibitor

0.167 0.095 CHEMBL4525767

0.151 0.147 CHEMBL1093458

0.154 0.135 CHEMBL1743350

CHEMBL4525767
0.0690.010.069Glycine transporter 1 inhibitor

0.042 0.019 CHEMBL4525767

0.034 0.024 CHEMBL2137046

0.03 0.027 CHEMBL4525766

0.1860.1290.247Immunostimulant

0.157 0.149 CHEMBL4525767

0.238 0.101 CHEMBL2137046

0.242 0.099 CHEMBL50995

0.207 0.116 CHEMBL1093458

0.247 0.097 CHEMBL1743350

0.227 0.106 CHEMBL4525766

CHEMBL1743350
0.1380.0820.182Ca2+-transporting ATPase inhibitor

0.129 0.126 CHEMBL4525767

0.141 0.071 CHEMBL2137046

0.182 0.006 CHEMBL50995

0.132 0.111 CHEMBL1093458

0.139 0.075 CHEMBL1743350

0.136 0.088 CHEMBL4525766

CHEMBL50995
0.1070.0520.142Antiadrenergic

0.142 0.038 CHEMBL4525767

0.093 0.06 CHEMBL2137046

0.119 0.046 CHEMBL1093458

0.08 0.071 CHEMBL1743350

0.1 0.056 CHEMBL4525766

CHEMBL4525767
0.0810.0260.179Adrenaline uptake inhibitor

0.179 0.007 CHEMBL4525767

0.063 0.042 CHEMBL2137046

0.139 0.011 CHEMBL1093458

0.056 0.049 CHEMBL4525766

CHEMBL4525767
0.110.0550.131MAO B inhibitor

0.131 0.045 CHEMBL2137046

0.082 0.074 CHEMBL1093458

0.128 0.047 CHEMBL1743350

0.13 0.045 CHEMBL4525766

CHEMBL2137046
0.1070.0530.109Alpha adrenoreceptor antagonist

0.109 0.052 CHEMBL4525767

0.079 0.073 CHEMBL2137046

0.08 0.071 CHEMBL1093458

0.084 0.069 CHEMBL4525766

CHEMBL4525767
0.1020.0480.319Toll-Like receptor 3 antagonist

0.239 0.004 CHEMBL4525767

0.18 0.008 CHEMBL1093458

0.319 0.003 CHEMBL1743350

CHEMBL1743350
0.0870.0330.087Calcium channel L-type blocker

0.066 0.057 CHEMBL4525767

0.1250.0720.16Cyclooxygenase 3 inhibitor

0.118 0.08 CHEMBL4525767

0.136 0.061 CHEMBL2137046

0.16 0.04 CHEMBL50995

0.129 0.068 CHEMBL1093458

0.15 0.048 CHEMBL1743350

0.137 0.06 CHEMBL4525766

CHEMBL50995
0.1010.0490.131ABCA1 expression enhancer

0.099 0.051 CHEMBL4525767

0.101 0.049 CHEMBL2137046

0.131 0.024 CHEMBL50995

0.099 0.051 CHEMBL1093458

0.09 0.065 CHEMBL1743350

0.1 0.051 CHEMBL4525766

CHEMBL50995
0.0760.0240.083Acyl-CoA dehydrogenase inhibitor

0.066 0.029 CHEMBL2137046

0.083 0.021 CHEMBL50995

0.059 0.034 CHEMBL1743350

0.057 0.035 CHEMBL4525766

CHEMBL50995
0.1030.0520.137Adrenaline antagonist

0.137 0.038 CHEMBL4525767

0.09 0.06 CHEMBL2137046

0.115 0.046 CHEMBL1093458

0.077 0.071 CHEMBL1743350

0.097 0.056 CHEMBL4525766

CHEMBL4525767
0.1250.0750.177Vanilloid 1 agonist

0.162 0.028 CHEMBL4525767

0.137 0.055 CHEMBL2137046

0.152 0.036 CHEMBL50995

0.177 0.02 CHEMBL1093458

0.155 0.033 CHEMBL1743350

0.155 0.034 CHEMBL4525766

CHEMBL1093458
0.1040.0550.305Creatine kinase inhibitor

0.16 0.02 CHEMBL2137046

0.305 0.004 CHEMBL50995

0.112 0.047 CHEMBL1093458

0.116 0.044 CHEMBL1743350

0.143 0.027 CHEMBL4525766

CHEMBL50995
0.0680.0190.097Thromboxane synthase inhibitor

0.073 0.016 CHEMBL4525767

0.068 0.019 CHEMBL2137046

0.097 0.007 CHEMBL50995

0.073 0.015 CHEMBL1093458

0.077 0.013 CHEMBL1743350

0.066 0.02 CHEMBL4525766

CHEMBL50995
0.0560.0080.056Delayed rectifier potassium channel blocker

0.045 0.015 CHEMBL4525767

0.045 0.016 CHEMBL2137046

0.034 0.032 CHEMBL50995

0.036 0.028 CHEMBL1093458

0.041 0.02 CHEMBL1743350

0.036 0.029 CHEMBL4525766

0.0770.0290.077Exportin-1 inhibitor

0.076 0.031 CHEMBL50995

0.076 0.031 CHEMBL1743350

0.0930.0460.094Alpha 1 adrenoreceptor antagonist

0.094 0.045 CHEMBL4525767

CHEMBL4525767
0.0760.030.289Aromatase inhibitor

0.065 0.038 CHEMBL4525767

0.087 0.025 CHEMBL2137046

0.289 0.005 CHEMBL50995

0.074 0.031 CHEMBL1093458

0.175 0.01 CHEMBL1743350

0.079 0.028 CHEMBL4525766

CHEMBL50995
0.1120.0690.141Photosensitizer

0.119 0.059 CHEMBL2137046

0.141 0.037 CHEMBL50995

0.104 0.081 CHEMBL1743350

0.102 0.084 CHEMBL4525766

CHEMBL50995
0.0620.020.062Alpha 1L adrenoreceptor antagonist

0.053 0.034 CHEMBL2137046

0.054 0.033 CHEMBL4525766

0.070.030.075 Hydroxytryptamine 6 antagonist

0.053 0.044 CHEMBL4525767

0.0760.0360.1745 Hydroxytryptamine uptake inhibitor

0.174 0.013 CHEMBL4525767

0.103 0.025 CHEMBL1093458

CHEMBL4525767
0.0870.0480.087Acetylcholine nicotinic antagonist

0.077 0.058 CHEMBL4525767

0.0510.0140.059Diamine oxidase inhibitor

0.053 0.013 CHEMBL4525767

0.034 0.032 CHEMBL1093458

0.059 0.01 CHEMBL1743350

CHEMBL1743350
0.1020.0640.104Nav1.1 sodium channel blocker

0.104 0.062 CHEMBL2137046

0.087 0.085 CHEMBL4525766

CHEMBL2137046
0.1350.0980.146Heat shock protein 70 antagonist

0.145 0.06 CHEMBL2137046

0.145 0.058 CHEMBL50995

0.146 0.056 CHEMBL4525766

CHEMBL4525766
0.1120.0760.128Alkylator

0.109 0.079 CHEMBL4525767

0.128 0.06 CHEMBL2137046

0.125 0.063 CHEMBL1093458

0.122 0.067 CHEMBL4525766

CHEMBL2137046
0.0780.0420.079Peroxisome proliferator-activated receptor gamma agonist

0.068 0.051 CHEMBL4525767

0.072 0.048 CHEMBL2137046

0.068 0.051 CHEMBL50995

0.063 0.055 CHEMBL1093458

0.061 0.057 CHEMBL1743350

0.079 0.041 CHEMBL4525766

CHEMBL4525766
0.1470.1120.219Phospholipase C inhibitor

0.175 0.066 CHEMBL2137046

0.219 0.034 CHEMBL50995

0.145 0.116 CHEMBL1093458

0.172 0.07 CHEMBL1743350

0.18 0.061 CHEMBL4525766

CHEMBL50995
0.0820.0480.092Na+ K+ transporting ATPase inhibitor

0.092 0.039 CHEMBL2137046

0.085 0.045 CHEMBL50995

0.085 0.046 CHEMBL1743350

0.089 0.041 CHEMBL4525766

CHEMBL2137046
0.080.0470.085 Hydroxytryptamine 1 antagonist

0.066 0.057 CHEMBL4525767

0.0760.0430.0765 Hydroxytryptamine 1A antagonist

0.062 0.051 CHEMBL4525767

0.0770.0460.091Alpha 1a adrenoreceptor antagonist

0.091 0.04 CHEMBL4525767

CHEMBL4525767
0.0570.0260.117Plasminogen activator inhibitor antagonist

0.062 0.023 CHEMBL2137046

0.117 0.008 CHEMBL50995

0.047 0.036 CHEMBL1093458

0.052 0.031 CHEMBL1743350

0.08 0.015 CHEMBL4525766

CHEMBL50995
0.2030.1730.266Antithrombotic

0.223 0.15 CHEMBL2137046

0.245 0.13 CHEMBL50995

0.206 0.17 CHEMBL1093458

0.266 0.114 CHEMBL1743350

0.237 0.137 CHEMBL4525766

CHEMBL1743350
0.0770.0470.105Adenosine A3 receptor antagonist

0.099 0.027 CHEMBL4525767

0.072 0.055 CHEMBL2137046

0.105 0.024 CHEMBL50995

0.091 0.031 CHEMBL1093458

0.085 0.037 CHEMBL1743350

CHEMBL50995
0.0680.0380.068Interferon inducer

0.065 0.042 CHEMBL2137046

0.06 0.053 CHEMBL50995

0.061 0.051 CHEMBL1743350

0.059 0.055 CHEMBL4525766

0.2760.2470.335Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.331 0.173 CHEMBL4525767

0.335 0.168 CHEMBL50995

0.275 0.248 CHEMBL1743350

CHEMBL50995
0.0980.070.141Adenylate kinase inhibitor

0.094 0.077 CHEMBL2137046

0.141 0.03 CHEMBL50995

0.103 0.063 CHEMBL1743350

CHEMBL50995
0.0380.010.065Dopamine autoreceptor agonist

0.059 0.006 CHEMBL4525767

0.042 0.009 CHEMBL2137046

0.065 0.005 CHEMBL1093458

0.038 0.01 CHEMBL1743350

CHEMBL1093458
0.090.0620.101Glutamate release inhibitor

0.09 0.061 CHEMBL4525767

0.101 0.042 CHEMBL50995

0.097 0.048 CHEMBL1743350

CHEMBL50995
0.0830.0570.083ErbB-3 antagonist
0.1460.120.292Succinate dehydrogenase inhibitor

0.14 0.132 CHEMBL4525767

0.153 0.106 CHEMBL2137046

0.292 0.012 CHEMBL50995

0.147 0.118 CHEMBL1093458

0.19 0.058 CHEMBL1743350

0.168 0.082 CHEMBL4525766

CHEMBL50995
0.1010.0760.193GABA C receptor antagonist

0.102 0.075 CHEMBL4525767

0.111 0.062 CHEMBL2137046

0.193 0.014 CHEMBL50995

0.112 0.062 CHEMBL1093458

0.191 0.015 CHEMBL1743350

CHEMBL50995
0.0650.040.065Dopamine D3 antagonist

0.06 0.045 CHEMBL4525767

0.0450.0220.057Leukotriene A4 hydrolase inhibitor

0.057 0.017 CHEMBL1743350

CHEMBL1743350
0.0380.0160.046Melatonin receptor 1A agonist

0.046 0.009 CHEMBL4525767

0.035 0.021 CHEMBL1743350

CHEMBL4525767
0.0560.0350.066Epithelial sodium channel blocker

0.056 0.035 CHEMBL4525767

0.051 0.047 CHEMBL2137046

0.051 0.046 CHEMBL1093458

0.066 0.021 CHEMBL1743350

CHEMBL1743350
0.0250.0050.037Antibiotic Anthracycline-like

0.023 0.006 CHEMBL4525767

0.028 0.004 CHEMBL2137046

0.037 0.003 CHEMBL50995

0.027 0.004 CHEMBL1093458

0.026 0.005 CHEMBL1743350

0.026 0.005 CHEMBL4525766

CHEMBL50995
0.0630.0430.074Nitric oxide donor

0.066 0.039 CHEMBL4525767

0.057 0.054 CHEMBL2137046

0.06 0.048 CHEMBL1093458

0.074 0.028 CHEMBL1743350

0.061 0.046 CHEMBL4525766

CHEMBL1743350
0.1280.1090.217GABA C receptor rho-2 antagonist

0.17 0.05 CHEMBL4525767

0.132 0.102 CHEMBL2137046

0.217 0.021 CHEMBL50995

0.175 0.046 CHEMBL1093458

0.134 0.098 CHEMBL1743350

CHEMBL50995
0.1350.1150.152Interleukin 6 antagonist

0.151 0.088 CHEMBL2137046

0.152 0.085 CHEMBL4525766

CHEMBL4525766
0.0630.0450.063Calcium channel P-type blocker
0.0540.0360.058Nicotinic alpha3beta2 receptor antagonist

0.058 0.028 CHEMBL4525767

0.053 0.038 CHEMBL50995

CHEMBL4525767
0.0320.0150.032Thiazolidinedione

0.029 0.021 CHEMBL2137046

0.03 0.02 CHEMBL4525766

0.0540.0370.067Leukotriene B4 antagonist

0.061 0.026 CHEMBL2137046

0.067 0.021 CHEMBL50995

0.05 0.044 CHEMBL1093458

0.051 0.042 CHEMBL1743350

0.066 0.022 CHEMBL4525766

CHEMBL50995
0.1010.0850.155Topoisomerase II inhibitor

0.155 0.047 CHEMBL2137046

0.146 0.052 CHEMBL50995

0.106 0.08 CHEMBL1093458

0.15 0.049 CHEMBL4525766

CHEMBL2137046
0.0450.0290.048Geranyltranstransferase inhibitor

0.042 0.033 CHEMBL2137046

0.048 0.025 CHEMBL50995

0.039 0.038 CHEMBL1743350

CHEMBL50995
0.150.1370.186Hypolipemic

0.165 0.122 CHEMBL2137046

0.186 0.105 CHEMBL50995

0.162 0.125 CHEMBL4525766

CHEMBL50995
0.0360.0240.074Retinoid X receptor agonist

0.074 0.009 CHEMBL50995

0.04 0.022 CHEMBL1743350

CHEMBL50995
0.0890.0790.089Gastric antisecretory

0.089 0.079 CHEMBL4525767

0.0910.0820.143Carbonic anhydrase XV inhibitor

0.11 0.055 CHEMBL2137046

0.143 0.033 CHEMBL50995

0.118 0.048 CHEMBL1743350

0.112 0.054 CHEMBL4525766

CHEMBL50995
0.0610.0530.061Neuronal nicotinic receptor antagonist

0.059 0.056 CHEMBL4525767

0.060.0510.089Leukotriene antagonist

0.069 0.041 CHEMBL2137046

0.089 0.027 CHEMBL50995

0.076 0.035 CHEMBL4525766

CHEMBL50995
0.0540.0460.054Dopamine D4 antagonist
0.0170.0110.017Vitamin D receptor agonist

0.017 0.011 CHEMBL2137046

0.017 0.01 CHEMBL50995

0.015 0.014 CHEMBL4525766

0.0570.0510.064Bcl-xL inhibitor

0.056 0.053 CHEMBL2137046

0.064 0.03 CHEMBL4525766

CHEMBL4525766
0.0570.0530.0575 Hydroxytryptamine 1D antagonist
0.0440.0410.044Benzodiazepine antagonist
0.020.0180.024Leukotriene B4 receptor 2 antagonist

0.022 0.015 CHEMBL2137046

0.024 0.013 CHEMBL50995

0.023 0.014 CHEMBL4525766

CHEMBL50995
0.0250.0230.0255 Hydroxytryptamine 1D agonist
0.1650.1630.393Superoxide dismutase inhibitor

0.168 0.158 CHEMBL4525767

0.197 0.12 CHEMBL2137046

0.393 0.028 CHEMBL50995

0.202 0.116 CHEMBL1093458

0.354 0.036 CHEMBL1743350

0.227 0.092 CHEMBL4525766

CHEMBL50995
0.1060.1050.106Cytokine production inhibitor
0.1480.1470.426Free radical scavenger

0.274 0.059 CHEMBL2137046

0.426 0.025 CHEMBL50995

0.251 0.068 CHEMBL1093458

0.362 0.036 CHEMBL4525766

CHEMBL50995
0.0890.0880.095DNA intercalator

0.095 0.08 CHEMBL2137046

CHEMBL2137046
0.0990.0990.201Aldehyde dehydrogenase inhibitor

0.138 0.055 CHEMBL2137046

0.201 0.027 CHEMBL50995

0.125 0.066 CHEMBL1093458

0.12 0.071 CHEMBL1743350

CHEMBL50995
0.070.0690.07Histamine H1 receptor antagonist
0.0860.0860.095Falcipain 3 inhibitor

0.095 0.075 CHEMBL50995

CHEMBL50995
0.0180.0190.043Retinoid X beta receptor agonist

0.043 0.005 CHEMBL50995

CHEMBL50995
0.1840.1850.338Transcription factor NF kappa B inhibitor

0.215 0.155 CHEMBL4525767

0.265 0.117 CHEMBL2137046

0.338 0.081 CHEMBL50995

0.292 0.099 CHEMBL1093458

0.216 0.154 CHEMBL1743350

0.291 0.099 CHEMBL4525766

CHEMBL50995
0.0520.0540.084Pregnane X receptor antagonist

0.084 0.005 CHEMBL50995

CHEMBL50995
0.0290.0320.053Retinoid X alpha receptor agonist

0.053 0.013 CHEMBL50995

0.031 0.03 CHEMBL1743350

CHEMBL50995
0.0940.0970.106Electron transport complex I inhibitor

0.106 0.069 CHEMBL50995

0.106 0.069 CHEMBL4525766

CHEMBL4525766
0.1130.1160.161Sphingosine 1-phosphate receptor 2 antagonist

0.118 0.101 CHEMBL4525767

0.161 0.028 CHEMBL50995

0.114 0.113 CHEMBL1093458

0.135 0.065 CHEMBL1743350

0.118 0.101 CHEMBL4525766

CHEMBL50995
0.0530.0570.056Gonadotropin-releasing hormone receptor agonist

0.056 0.05 CHEMBL2137046

CHEMBL2137046
0.0720.0760.141Ornithine decarboxylase inhibitor

0.105 0.039 CHEMBL4525767

0.082 0.065 CHEMBL2137046

0.141 0.014 CHEMBL50995

0.112 0.032 CHEMBL1093458

0.127 0.021 CHEMBL1743350

0.088 0.059 CHEMBL4525766

CHEMBL50995
0.1550.1590.398Antioxidant

0.273 0.073 CHEMBL2137046

0.398 0.035 CHEMBL50995

0.255 0.081 CHEMBL1093458

0.164 0.148 CHEMBL1743350

0.337 0.05 CHEMBL4525766

CHEMBL50995
0.0340.0390.052Retinoic acid alpha receptor agonist

0.052 0.013 CHEMBL50995

CHEMBL50995
0.0770.0830.116MAO A inhibitor

0.089 0.072 CHEMBL4525767

0.102 0.063 CHEMBL2137046

0.116 0.054 CHEMBL1093458

0.099 0.065 CHEMBL1743350

0.1 0.064 CHEMBL4525766

CHEMBL1093458
0.0440.050.058Cytokine production stimulant

0.058 0.014 CHEMBL1743350

CHEMBL1743350
0.0850.0910.092Phosphodiesterase 6D inhibitor

0.088 0.082 CHEMBL50995

0.092 0.071 CHEMBL4525766

CHEMBL4525766
0.020.0280.304Estrogen receptor beta agonist

0.119 0.009 CHEMBL2137046

0.304 0.004 CHEMBL50995

0.074 0.015 CHEMBL1093458

0.081 0.014 CHEMBL4525766

CHEMBL50995
0.1160.1230.183Phospholipase A2 inhibitor

0.13 0.101 CHEMBL2137046

0.154 0.071 CHEMBL50995

0.183 0.052 CHEMBL1743350

0.128 0.103 CHEMBL4525766

CHEMBL1743350
0.0120.020.018Ileal bile acid transport inhibitor

0.017 0.012 CHEMBL2137046

0.018 0.011 CHEMBL50995

CHEMBL50995
0.0210.030.034Vanilloid 2 agonist

0.034 0.006 CHEMBL50995

CHEMBL50995
0.0330.0420.059Oxytocin agonist

0.044 0.028 CHEMBL2137046

0.059 0.018 CHEMBL50995

0.047 0.026 CHEMBL1093458

CHEMBL50995
0.0180.030.022Vitamin D receptor antagonist

0.022 0.015 CHEMBL50995

CHEMBL50995
0.080.0920.158Carbonic anhydrase III inhibitor

0.117 0.046 CHEMBL2137046

0.158 0.026 CHEMBL50995

0.09 0.075 CHEMBL1743350

0.121 0.043 CHEMBL4525766

CHEMBL50995
0.0210.0330.024Acid ceramidase inhibitor

0.024 0.022 CHEMBL4525767

CHEMBL4525767
0.0330.0470.049Glycine transporter 2 inhibitor

0.046 0.033 CHEMBL2137046

0.049 0.031 CHEMBL50995

0.041 0.038 CHEMBL1093458

0.04 0.039 CHEMBL1743350

CHEMBL50995
0.1580.1720.268Peptidyltransferase inhibitor

0.246 0.053 CHEMBL4525767

0.203 0.096 CHEMBL2137046

0.191 0.111 CHEMBL50995

0.268 0.039 CHEMBL1093458

0.232 0.065 CHEMBL1743350

0.211 0.086 CHEMBL4525766

CHEMBL1093458
0.1090.1230.23Thrombolytic

0.128 0.101 CHEMBL2137046

0.147 0.084 CHEMBL50995

0.23 0.039 CHEMBL1743350

0.145 0.086 CHEMBL4525766

CHEMBL1743350
0.0220.0360.03Retinoid X gamma receptor antagonist

0.03 0.012 CHEMBL50995

0.028 0.017 CHEMBL1743350

CHEMBL50995
0.0630.080.076S-adenosyl-L-methionine decarboxylase inhibitor

0.073 0.051 CHEMBL50995

0.076 0.046 CHEMBL1743350

CHEMBL1743350
0.0170.0340.029Leukotriene B4 receptor 1 antagonist

0.029 0.019 CHEMBL50995

CHEMBL50995
0.0750.0920.125Granulocyte macrophage colony stimulating factor agonist

0.08 0.075 CHEMBL4525767

0.125 0.013 CHEMBL50995

0.098 0.037 CHEMBL1743350

CHEMBL50995
0.0170.0340.029Retinoic acid receptor agonist

0.029 0.01 CHEMBL50995

CHEMBL50995
0.0160.0350.024Retinoid X beta receptor antagonist

0.024 0.008 CHEMBL50995

0.02 0.016 CHEMBL1743350

CHEMBL50995
0.0270.0460.042Retinoid X alpha receptor antagonist

0.042 0.013 CHEMBL50995

0.032 0.028 CHEMBL1743350

CHEMBL50995
0.0370.0570.09Beta 2 adrenoreceptor antagonist

0.07 0.017 CHEMBL4525767

0.055 0.029 CHEMBL2137046

0.048 0.039 CHEMBL50995

0.09 0.009 CHEMBL1093458

0.058 0.026 CHEMBL1743350

0.058 0.026 CHEMBL4525766

CHEMBL1093458
0.0290.050.05Retinoid X receptor antagonist

0.05 0.012 CHEMBL50995

0.036 0.03 CHEMBL1743350

CHEMBL50995
0.0150.0360.024Retinoic acid beta receptor agonist

0.024 0.008 CHEMBL50995

CHEMBL50995
0.0650.0860.188Androgen antagonist

0.086 0.059 CHEMBL2137046

0.188 0.015 CHEMBL50995

0.077 0.069 CHEMBL1093458

0.082 0.063 CHEMBL4525766

CHEMBL50995
0.0730.0950.12CC chemokine 5 receptor agonist

0.081 0.061 CHEMBL2137046

0.12 0.009 CHEMBL50995

CHEMBL50995
0.0890.1110.173TRPA1 agonist

0.1 0.087 CHEMBL2137046

0.173 0.018 CHEMBL50995

0.105 0.079 CHEMBL1093458

0.097 0.093 CHEMBL4525766

CHEMBL50995
0.0220.0450.028Hedgehog signaling activator

0.028 0.016 CHEMBL50995

CHEMBL50995
0.0170.040.028Retinoic acid gamma receptor agonist

0.028 0.008 CHEMBL50995

CHEMBL50995
0.0670.0910.098Glutathione S-transferase inhibitor

0.098 0.039 CHEMBL50995

0.095 0.042 CHEMBL1743350

0.075 0.069 CHEMBL4525766

CHEMBL50995
0.020.0470.053Kainate receptor 2 antagonist

0.034 0.027 CHEMBL4525767

0.053 0.015 CHEMBL50995

0.039 0.023 CHEMBL1743350

CHEMBL50995
0.0370.0640.056Lysophosphatidic acid 3 receptor antagonist

0.056 0.027 CHEMBL50995

0.049 0.037 CHEMBL1743350

CHEMBL50995
0.0070.0360.0131-Deoxy-D-xylulose-5-phosphate reductoisomerase inhibitor

0.013 0.01 CHEMBL50995

CHEMBL50995
0.0480.0770.064Leukotriene C antagonist

0.064 0.022 CHEMBL50995

CHEMBL50995
0.040.070.059Alpha-mannosidase inhibitor

0.059 0.028 CHEMBL50995

CHEMBL50995
0.0460.0760.062Sphingosine 1-phosphate receptor 4 agonist

0.058 0.057 CHEMBL50995

0.062 0.052 CHEMBL1743350

CHEMBL1743350
0.0340.0660.041Histamine H1 receptor agonist

0.041 0.037 CHEMBL4525767

CHEMBL4525767
0.0530.0850.106Aminopeptidase I inhibitor

0.106 0.025 CHEMBL50995

0.07 0.054 CHEMBL1743350

CHEMBL50995
0.0130.0460.025Retinoid X gamma receptor agonist

0.025 0.014 CHEMBL50995

CHEMBL50995
0.1560.1910.236Nitric-oxide synthase stimulant

0.178 0.133 CHEMBL4525767

0.169 0.154 CHEMBL2137046

0.236 0.043 CHEMBL50995

0.192 0.104 CHEMBL1093458

0.195 0.098 CHEMBL1743350

0.177 0.135 CHEMBL4525766

CHEMBL50995
0.0870.1230.291Alpha-N-acetylglucosaminidase inhibitor

0.291 0.017 CHEMBL50995

0.105 0.095 CHEMBL1743350

CHEMBL50995
0.0650.1010.154Aminopeptidase B inhibitor

0.154 0.036 CHEMBL50995

0.116 0.055 CHEMBL1743350

CHEMBL50995
0.0410.0770.105Androgen agonist

0.053 0.052 CHEMBL2137046

0.105 0.013 CHEMBL50995

CHEMBL50995
0.0180.0540.088Progesterone antagonist

0.088 0.01 CHEMBL50995

CHEMBL50995
0.0410.0790.053Sphingosine 1-phosphate receptor 3 antagonist

0.053 0.05 CHEMBL50995

CHEMBL50995
0.0160.0540.023Lysophosphatidic acid receptor 1 agonist

0.023 0.022 CHEMBL50995

CHEMBL50995
0.1620.2010.19Neuropeptide Y2 antagonist

0.19 0.139 CHEMBL50995

CHEMBL50995
0.0270.0660.042Sphingosine 1-phosphate receptor 1 agonist

0.042 0.03 CHEMBL1743350

CHEMBL1743350
0.0310.0710.042Leukotriene C4 antagonist

0.042 0.021 CHEMBL50995

CHEMBL50995
0.0480.0880.067Protease 3C (Human rhinovirus) inhibitor

0.067 0.041 CHEMBL50995

0.061 0.05 CHEMBL1743350

CHEMBL50995
0.1130.1540.167Pregnane X receptor agonist

0.167 0.029 CHEMBL50995

CHEMBL50995
0.050.0930.096NAD(P)H dehydrogenase (quinone) inhibitor

0.081 0.05 CHEMBL2137046

0.096 0.04 CHEMBL50995

0.079 0.052 CHEMBL4525766

CHEMBL50995
0.0240.0670.134Dopamine D5 agonist

0.038 0.03 CHEMBL2137046

0.134 0.003 CHEMBL50995

0.039 0.029 CHEMBL1093458

0.056 0.014 CHEMBL1743350

0.043 0.024 CHEMBL4525766

CHEMBL50995
0.0130.0560.024Prostaglandin F2 alpha agonist

0.024 0.013 CHEMBL50995

CHEMBL50995
0.0130.0560.032Uridine phosphorylase inhibitor

0.032 0.016 CHEMBL50995

0.03 0.018 CHEMBL1743350

CHEMBL50995
0.0280.0720.046Mannosidase inhibitor

0.046 0.03 CHEMBL50995

CHEMBL50995
0.0520.0970.068Beta 2 adrenoreceptor agonist

0.059 0.054 CHEMBL4525767

0.061 0.044 CHEMBL2137046

0.063 0.039 CHEMBL50995

0.068 0.023 CHEMBL1093458

0.059 0.056 CHEMBL1743350

0.062 0.04 CHEMBL4525766

CHEMBL1093458
0.110.1560.158Sphingosine 1-phosphate receptor 5 antagonist

0.158 0.049 CHEMBL50995

0.135 0.09 CHEMBL1743350

CHEMBL50995
0.070.1170.128Lanosterol 14 alpha demethylase inhibitor

0.128 0.023 CHEMBL50995

0.1 0.055 CHEMBL1743350

CHEMBL50995
0.0330.0820.066Glucose-6-phosphate isomerase inhibitor

0.066 0.014 CHEMBL50995

CHEMBL50995
0.0770.1280.115Glutamate (mGluR7) agonist

0.115 0.036 CHEMBL4525767

0.091 0.082 CHEMBL1743350

CHEMBL4525767
0.0660.120.169UDP-glucose 4-epimerase inhibitor

0.169 0.023 CHEMBL50995

CHEMBL50995
0.0210.0760.042Vascular adhesion protein 1 inhibitor

0.042 0.023 CHEMBL1743350

CHEMBL1743350
0.0350.0930.051Beta adrenoreceptor agonist

0.043 0.04 CHEMBL4525767

0.043 0.041 CHEMBL2137046

0.051 0.015 CHEMBL1093458

0.043 0.04 CHEMBL4525766

CHEMBL1093458
0.0290.0860.047Adenylate cyclase 1 inhibitor

0.047 0.031 CHEMBL50995

CHEMBL50995
0.0630.1230.149Triose-phosphate isomerase inhibitor

0.149 0.02 CHEMBL50995

0.085 0.067 CHEMBL1743350

CHEMBL50995
0.0540.1150.168Keratolytic

0.072 0.062 CHEMBL2137046

0.168 0.012 CHEMBL50995

0.092 0.036 CHEMBL1743350

0.072 0.062 CHEMBL4525766

CHEMBL50995
0.0690.130.157GABA C receptor rho-1 antagonist

0.097 0.066 CHEMBL4525767

0.157 0.018 CHEMBL50995

0.098 0.064 CHEMBL1093458

0.127 0.034 CHEMBL1743350

CHEMBL50995
0.0690.1310.108Electrolyte absorption antagonist

0.108 0.047 CHEMBL50995

CHEMBL50995
0.0120.0770.021Neuraminidase (Influenza B) inhibitor

0.021 0.014 CHEMBL50995

CHEMBL50995
0.0290.0950.381Alcohol oxidase inhibitor

0.381 0.004 CHEMBL50995

0.158 0.009 CHEMBL1743350

CHEMBL50995
0.0320.1030.0895 Hydroxytryptamine 2A agonist

0.089 0.02 CHEMBL1743350

CHEMBL1743350
0.0490.1230.145Adrenaline agonist

0.096 0.039 CHEMBL4525767

0.08 0.058 CHEMBL2137046

0.145 0.016 CHEMBL1093458

0.081 0.057 CHEMBL4525766

CHEMBL1093458
0.1190.1930.288Neurotrophic factor enhancer

0.159 0.125 CHEMBL2137046

0.288 0.022 CHEMBL50995

0.181 0.097 CHEMBL1093458

0.178 0.1 CHEMBL4525766

CHEMBL50995
0.010.0850.023Beta 1 adrenoreceptor agonist

0.023 0.015 CHEMBL1093458

CHEMBL1093458
0.0430.1180.059Immunoglobulin Fc receptor antagonist

0.059 0.027 CHEMBL50995

CHEMBL50995
0.0340.1110.07Sphingosine kinase 2 inhibitor

0.07 0.022 CHEMBL50995

0.059 0.033 CHEMBL1743350

CHEMBL50995
0.0680.1470.123Mucolytic

0.123 0.052 CHEMBL50995

CHEMBL50995
0.0520.1310.127Opioid kappa receptor antagonist

0.078 0.06 CHEMBL2137046

0.127 0.021 CHEMBL50995

0.088 0.047 CHEMBL1093458

CHEMBL50995
0.070.1490.145Tubulin antagonist

0.145 0.06 CHEMBL50995

0.138 0.064 CHEMBL4525766

CHEMBL50995
0.020.10.04Guanylate cyclase inhibitor

0.04 0.033 CHEMBL50995

CHEMBL50995
0.060.140.123NADH dehydrogenase inhibitor

0.123 0.027 CHEMBL50995

CHEMBL50995
0.0580.1390.131Breast cancer-resistant protein inhibitor

0.131 0.032 CHEMBL50995

CHEMBL50995
0.0770.1580.195Toll-Like receptor 2 antagonist

0.109 0.091 CHEMBL2137046

0.195 0.026 CHEMBL50995

0.138 0.061 CHEMBL1093458

0.125 0.073 CHEMBL1743350

0.126 0.072 CHEMBL4525766

CHEMBL50995
0.0310.1130.123Phosphofructokinase-1 inhibitor

0.123 0.024 CHEMBL50995

CHEMBL50995
0.0210.1030.094Beta tubulin antagonist

0.094 0.024 CHEMBL50995

0.069 0.035 CHEMBL4525766

CHEMBL50995
0.1010.1840.213Melanin inhibitor

0.134 0.107 CHEMBL2137046

0.213 0.036 CHEMBL50995

0.129 0.116 CHEMBL1093458

0.139 0.098 CHEMBL4525766

CHEMBL50995
0.1560.2390.252Insulysin inhibitor

0.252 0.095 CHEMBL50995

0.193 0.167 CHEMBL1093458

0.213 0.139 CHEMBL1743350

CHEMBL50995
0.0430.1280.064Ryanodine receptor antagonist

0.064 0.029 CHEMBL50995

CHEMBL50995
0.0160.10.036HMG CoA reductase inhibitor

0.036 0.021 CHEMBL50995

CHEMBL50995
0.0120.0970.0395-Alpha-reductase inhibitor

0.039 0.025 CHEMBL50995

CHEMBL50995
0.0290.1170.076Aconitate hydratase inhibitor

0.076 0.015 CHEMBL50995

CHEMBL50995
0.1350.2240.325Lipoxygenase inhibitor

0.207 0.133 CHEMBL2137046

0.325 0.059 CHEMBL50995

0.212 0.128 CHEMBL1093458

0.183 0.159 CHEMBL1743350

0.253 0.099 CHEMBL4525766

CHEMBL50995
0.1290.2180.197Hypoglycemic

0.178 0.136 CHEMBL2137046

0.174 0.142 CHEMBL1093458

0.197 0.115 CHEMBL1743350

0.194 0.118 CHEMBL4525766

CHEMBL1743350
0.1940.2840.545Calcium channel L-type activator

0.529 0.018 CHEMBL4525767

0.328 0.134 CHEMBL2137046

0.433 0.06 CHEMBL50995

0.545 0.014 CHEMBL1093458

CHEMBL1093458
0.0610.1520.087Nitric-oxide synthase inhibitor

0.087 0.084 CHEMBL4525767

CHEMBL4525767
0.0460.1370.084Myeloperoxidase inhibitor

0.076 0.075 CHEMBL1093458

0.084 0.059 CHEMBL1743350

CHEMBL1743350
0.0240.1170.137Opioid delta receptor antagonist

0.053 0.051 CHEMBL2137046

0.137 0.022 CHEMBL50995

0.059 0.047 CHEMBL1093458

CHEMBL50995
0.0420.1360.085Glutamate (mGluR7) antagonist

0.085 0.022 CHEMBL50995

CHEMBL50995
0.0430.1380.103Glutamate dehydrogenase inhibitor

0.103 0.029 CHEMBL50995

0.069 0.058 CHEMBL1743350

CHEMBL50995
0.0810.1760.194Protein kinase stimulant

0.194 0.044 CHEMBL50995

0.121 0.092 CHEMBL1093458

0.111 0.103 CHEMBL1743350

CHEMBL50995
0.0340.130.057Vanilloid 2 antagonist

0.053 0.034 CHEMBL50995

0.049 0.043 CHEMBL1093458

0.057 0.027 CHEMBL4525766

CHEMBL4525766
0.0120.1120.046Kainate receptor antagonist

0.046 0.024 CHEMBL50995

CHEMBL50995
0.1090.2090.137ATPase inhibitor

0.137 0.126 CHEMBL50995

CHEMBL50995
0.0180.1190.052Ornithine carbamoyltransferase inhibitor

0.052 0.038 CHEMBL50995

0.052 0.037 CHEMBL1743350

CHEMBL1743350
0.0740.1760.139Cathepsin H inhibitor

0.139 0.055 CHEMBL50995

0.118 0.078 CHEMBL1743350

CHEMBL50995
0.0270.130.082Carbamoyl phosphate synthetase inhibitor

0.082 0.028 CHEMBL50995

CHEMBL50995
0.0250.1290.0593-Hydroxyanthranilate 3,4-dioxygenase inhibitor

0.059 0.008 CHEMBL50995

CHEMBL50995
0.0510.1570.078Vanilloid 4 agonist

0.078 0.045 CHEMBL50995

CHEMBL50995
0.0070.1120.018Telomerase stimulant

0.018 0.011 CHEMBL50995

CHEMBL50995
0.0310.1390.104Catalase inhibitor

0.104 0.037 CHEMBL50995

CHEMBL50995
0.1150.2230.144Catenin beta inhibitor

0.144 0.12 CHEMBL2137046

CHEMBL2137046
0.1360.2450.251Hypoxia-inducible factor 1 alpha inhibitor

0.19 0.165 CHEMBL2137046

0.251 0.1 CHEMBL50995

0.207 0.144 CHEMBL4525766

CHEMBL50995
0.0120.1240.0281,3-Beta-glucan synthase inhibitor

0.028 0.02 CHEMBL1743350

CHEMBL1743350
0.030.1430.155Phenylalanine 4-hydroxylase inhibitor

0.155 0.011 CHEMBL50995

0.08 0.037 CHEMBL1093458

0.076 0.04 CHEMBL1743350

0.06 0.058 CHEMBL4525766

CHEMBL50995
0.0430.1580.092Glycine receptor antagonist

0.092 0.041 CHEMBL50995

CHEMBL50995
0.0440.1590.096Glycine receptor agonist

0.096 0.023 CHEMBL50995

0.074 0.047 CHEMBL1743350

CHEMBL50995
0.0980.2140.18CF transmembrane conductance regulator agonist

0.18 0.036 CHEMBL50995

CHEMBL50995
0.0410.1580.091Macrophage migration inhibitory factor inhibitor

0.091 0.041 CHEMBL50995

0.07 0.066 CHEMBL4525766

CHEMBL50995
0.0180.1350.036Glutamate (mGluR3) agonist

0.036 0.015 CHEMBL50995

CHEMBL50995
0.0220.140.093Argininosuccinate synthase inhibitor

0.093 0.021 CHEMBL50995

CHEMBL50995
0.0590.1780.113Vanilloid agonist

0.078 0.076 CHEMBL4525767

0.08 0.072 CHEMBL50995

0.09 0.047 CHEMBL1093458

0.113 0.022 CHEMBL1743350

0.092 0.043 CHEMBL4525766

CHEMBL1743350
0.0730.1920.53Peroxidase inhibitor

0.122 0.098 CHEMBL2137046

0.53 0.007 CHEMBL50995

0.122 0.098 CHEMBL1093458

0.154 0.076 CHEMBL1743350

0.132 0.089 CHEMBL4525766

CHEMBL50995
0.0330.1520.159Glutamate decarboxylase inhibitor

0.159 0.011 CHEMBL50995

0.081 0.043 CHEMBL1743350

CHEMBL50995
0.0620.1840.102Microtubule formation inhibitor

0.102 0.087 CHEMBL50995

CHEMBL50995
0.0130.1340.027Purinergic P2Y15 antagonist

0.027 0.024 CHEMBL50995

CHEMBL50995
0.0260.150.056Mannitol-1-phosphate 5-dehydrogenase inhibitor

0.056 0.039 CHEMBL50995

CHEMBL50995
0.0510.1770.219Ferrochelatase inhibitor

0.219 0.018 CHEMBL50995

CHEMBL50995
0.0480.1740.104Expectorant

0.104 0.065 CHEMBL50995

CHEMBL50995
0.0430.170.08Glutamate (mGluR6) antagonist

0.08 0.024 CHEMBL50995

0.065 0.052 CHEMBL1743350

CHEMBL50995
0.0030.1310.022Kainate receptor 1 antagonist

0.022 0.014 CHEMBL50995

CHEMBL50995
0.0240.1510.05Kainate receptor agonist

0.05 0.014 CHEMBL50995

CHEMBL50995
0.0140.1420.052Carbonic anhydrase VB inhibitor

0.052 0.043 CHEMBL50995

CHEMBL50995
0.010.140.037Fumarate hydratase inhibitor

0.037 0.021 CHEMBL50995

CHEMBL50995
0.0320.1640.06NMDA receptor agonist

0.06 0.047 CHEMBL50995

CHEMBL50995
0.0260.1580.057Dopamine beta hydroxylase inhibitor

0.057 0.019 CHEMBL50995

CHEMBL50995
0.0770.210.117Sphingosine 1-phosphate receptor 4 antagonist

0.117 0.078 CHEMBL50995

CHEMBL50995
0.0110.1450.024Thyroid hormone agonist

0.024 0.023 CHEMBL50995

CHEMBL50995
0.0160.1510.042Adenosine deaminase inhibitor

0.042 0.038 CHEMBL50995

CHEMBL50995
0.0210.1560.115Opioid mu receptor antagonist

0.115 0.026 CHEMBL50995

CHEMBL50995
0.0410.1770.122Opioid antagonist

0.122 0.035 CHEMBL50995

0.08 0.068 CHEMBL1093458

CHEMBL50995
0.1040.2410.407Streptokinase A inhibitor

0.407 0.045 CHEMBL50995

0.189 0.14 CHEMBL1093458

CHEMBL50995
0.0280.1670.216Porphobilinogen synthase inhibitor

0.216 0.01 CHEMBL50995

0.072 0.054 CHEMBL1743350

CHEMBL50995
0.0480.190.196GABA C receptor agonist

0.196 0.021 CHEMBL50995

0.137 0.039 CHEMBL1743350

CHEMBL50995
0.0290.1720.074Carbonic anhydrase XIII inhibitor

0.074 0.054 CHEMBL50995

CHEMBL50995
0.0090.1530.045Estradiol 17 beta-dehydrogenase 3 inhibitor

0.045 0.013 CHEMBL50995

CHEMBL50995
0.0360.1830.112GABA aminotransferase inhibitor

0.112 0.019 CHEMBL50995

CHEMBL50995
0.0480.1950.096GABA B receptor agonist

0.096 0.02 CHEMBL50995

0.077 0.047 CHEMBL1743350

CHEMBL50995
0.040.1910.097Carbonic anhydrase VI inhibitor

0.097 0.041 CHEMBL50995

CHEMBL50995
0.0220.1740.036Vanilloid 3 antagonist

0.036 0.034 CHEMBL50995

CHEMBL50995
0.0270.180.064Sphingosine kinase inhibitor

0.064 0.033 CHEMBL50995

CHEMBL50995
0.1190.2760.186Gastrin inhibitor

0.186 0.171 CHEMBL4525767

0.186 0.17 CHEMBL50995

CHEMBL50995
0.0230.1820.0963-Oxoacyl-[acyl-carrier-protein] synthase inhibitor

0.096 0.018 CHEMBL50995

CHEMBL50995
0.030.1890.1Purinergic P2X1 antagonist

0.1 0.017 CHEMBL50995

CHEMBL50995
0.0810.2440.235Interleukin agonist

0.235 0.09 CHEMBL50995

0.184 0.135 CHEMBL1743350

CHEMBL50995
0.0870.2520.185Interferon gamma antagonist

0.185 0.047 CHEMBL50995

CHEMBL50995
0.1040.270.183Neurotensin receptor agonist

0.183 0.046 CHEMBL50995

0.151 0.1 CHEMBL1093458

0.142 0.123 CHEMBL1743350

CHEMBL50995
0.0490.2170.111DNA polymerase I inhibitor

0.107 0.079 CHEMBL50995

0.111 0.076 CHEMBL4525766

CHEMBL4525766
0.120.2890.251RNA-directed DNA polymerase inhibitor

0.251 0.048 CHEMBL50995

CHEMBL50995
0.0440.2150.228Cystathionine beta-synthase inhibitor

0.228 0.019 CHEMBL50995

CHEMBL50995
0.0960.2680.162Calpain inhibitor

0.162 0.161 CHEMBL50995

CHEMBL50995
0.0360.2090.1685-Lipoxygenase inhibitor

0.168 0.032 CHEMBL50995

0.096 0.067 CHEMBL4525766

CHEMBL50995
0.0370.2110.091Urease inhibitor

0.091 0.078 CHEMBL50995

CHEMBL50995
0.0460.220.126UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor

0.126 0.036 CHEMBL50995

CHEMBL50995
0.0190.1960.073Biliverdin reductase inhibitor

0.073 0.03 CHEMBL50995

CHEMBL50995
0.030.2090.069Enoyl-[acyl-carrier-protein] reductase inhibitor

0.069 0.029 CHEMBL50995

CHEMBL50995
0.0340.2180.112Alcohol dehydrogenase inhibitor

0.112 0.041 CHEMBL50995

CHEMBL50995
0.0490.2340.165Lipid peroxidase inhibitor

0.126 0.087 CHEMBL2137046

0.117 0.097 CHEMBL50995

0.165 0.059 CHEMBL4525766

CHEMBL4525766
0.0470.2330.092MAP kinase kinase 7 inhibitor

0.092 0.022 CHEMBL50995

CHEMBL50995
0.0520.2410.115D-Ala-D-Ala ligase inhibitor

0.115 0.016 CHEMBL50995

CHEMBL50995
0.0280.2180.05Factor III inhibitor

0.05 0.034 CHEMBL50995

CHEMBL50995
0.0180.210.041Glutamate (mGluR8) agonist

0.041 0.021 CHEMBL50995

CHEMBL50995
0.1070.3080.201DNA synthesis inhibitor

0.201 0.122 CHEMBL50995

CHEMBL50995
0.010.2110.039Alpha 1d adrenoreceptor agonist

0.039 0.027 CHEMBL50995

CHEMBL50995
0.0090.2120.041NMDA receptor subunit 3A antagonist

0.041 0.024 CHEMBL50995

CHEMBL50995
0.0130.2180.049NMDA receptor subunit 3B antagonist

0.049 0.026 CHEMBL50995

CHEMBL50995
0.1060.310.194Transcription factor STAT3 inhibitor

0.194 0.142 CHEMBL50995

0.184 0.158 CHEMBL1743350

CHEMBL50995
0.040.2450.109Chelator

0.109 0.066 CHEMBL4525766

CHEMBL4525766
0.0770.2870.144Non-steroidal antiinflammatory agent

0.144 0.124 CHEMBL50995

CHEMBL50995
0.0120.2250.057Alpha tubulin antagonist

0.057 0.033 CHEMBL50995

CHEMBL50995
0.1440.3580.188MAP kinase kinase 3 inhibitor

0.188 0.16 CHEMBL1743350

CHEMBL1743350
0.0530.2680.198Amyloid beta aggregation inhibitor

0.198 0.079 CHEMBL4525766

CHEMBL4525766
0.0410.2610.099Bile acid receptor antagonist

0.099 0.051 CHEMBL50995

CHEMBL50995
0.0370.2590.134HIV-1 integrase (Overall Integration) inhibitor

0.134 0.032 CHEMBL50995

CHEMBL50995
0.0240.2460.08NMDA receptor antagonist

0.08 0.066 CHEMBL50995

CHEMBL50995
0.0250.2480.064Cathepsin G inhibitor

0.064 0.062 CHEMBL50995

CHEMBL50995
0.0430.2660.183Amylase inhibitor

0.183 0.05 CHEMBL50995

CHEMBL50995
0.040.2670.085Xanthine oxidase inhibitor

0.085 0.08 CHEMBL50995

CHEMBL50995
0.0180.2490.0873(or 17)beta-hydroxysteroid dehydrogenase inhibitor

0.087 0.014 CHEMBL50995

CHEMBL50995
0.0610.2920.125Mannose-6-phosphate isomerase inhibitor

0.125 0.093 CHEMBL50995

CHEMBL50995
0.0070.2390.027Nicotinic acid receptor 2 antagonist

0.027 0.017 CHEMBL50995

CHEMBL50995
0.0190.2570.124Histidine decarboxylase inhibitor

0.124 0.024 CHEMBL50995

CHEMBL50995
0.030.2690.054Adenine nucleotide translocase inhibitor

0.054 0.044 CHEMBL50995

CHEMBL50995
0.0490.2890.174DOPA decarboxylase inhibitor

0.174 0.012 CHEMBL50995

CHEMBL50995
0.0610.3020.121Transcription factor STAT6 inhibitor

0.121 0.058 CHEMBL50995

CHEMBL50995
0.0080.2590.039ATP citrate lysase inhibitor

0.039 0.014 CHEMBL50995

CHEMBL50995
0.0860.340.28412-Lipoxygenase inhibitor

0.284 0.089 CHEMBL50995

CHEMBL50995
0.0350.2920.061Transcription factor RelA inhibitor

0.061 0.051 CHEMBL50995

CHEMBL50995
0.0580.3150.379Interleukin antagonist

0.379 0.034 CHEMBL1743350

CHEMBL1743350
0.0210.2830.091Protein-tyrosine phosphatase 1B inhibitor

0.091 0.088 CHEMBL50995

CHEMBL50995
0.0030.2660.025Nicotinic acid receptor 1 antagonist

0.025 0.005 CHEMBL50995

CHEMBL50995
0.0050.2750.04Estradiol 17 beta-dehydrogenase inhibitor

0.04 0.031 CHEMBL50995

CHEMBL50995
0.0230.2950.049Parathyroid hormone antagonist

0.049 0.024 CHEMBL1743350

CHEMBL1743350
0.0260.2990.048Alpha 1b adrenoreceptor agonist

0.048 0.041 CHEMBL4525767

CHEMBL4525767
0.0160.2940.149Monophenol monooxygenase inhibitor

0.149 0.047 CHEMBL50995

CHEMBL50995
0.090.3760.27415-Lipoxygenase inhibitor

0.274 0.147 CHEMBL50995

CHEMBL50995
0.0790.3710.157MAP kinase kinase 4 inhibitor

0.157 0.049 CHEMBL50995

CHEMBL50995
0.0330.3280.091Beta glucuronidase inhibitor

0.091 0.086 CHEMBL50995

CHEMBL50995
0.0630.3580.162Growth hormone agonist

0.139 0.097 CHEMBL50995

0.162 0.078 CHEMBL1743350

CHEMBL1743350
0.030.3330.0965 Hydroxytryptamine 3A agonist

0.096 0.08 CHEMBL50995

CHEMBL50995
0.020.3660.057Dihydroorotate oxidase inhibitor

0.057 0.033 CHEMBL50995

CHEMBL50995
0.0670.4270.184Transcription factor STAT inhibitor

0.184 0.162 CHEMBL50995

CHEMBL50995
0.0690.4370.14Papain-like protease (SARS coronavirus) inhibitor

0.14 0.044 CHEMBL50995

0.117 0.09 CHEMBL1093458

CHEMBL50995
0.0270.4320.169Pyruvate kinase inhibitor

0.169 0.1 CHEMBL50995

CHEMBL50995
0.0950.5050.249Interleukin 2 agonist

0.249 0.119 CHEMBL50995

0.229 0.144 CHEMBL1743350

CHEMBL50995
0.0420.4610.143Hexokinase inhibitor

0.143 0.088 CHEMBL50995

CHEMBL50995
0.0320.4830.12Farnesoid X receptor antagonist

0.12 0.105 CHEMBL50995

CHEMBL50995
0.0350.5010.135Nitric oxide antagonist

0.135 0.111 CHEMBL50995

CHEMBL50995
0.030.6080.125Interleukin 4 antagonist

0.125 0.079 CHEMBL50995

CHEMBL50995
0.0460.6560.14Death-associated protein kinase 2 inhibitor

0.14 0.132 CHEMBL50995

CHEMBL50995
Ext Pa Pi Pmax Activity Other Results ID Pa_max