| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.93 | 0 | 0.977 | Vitamin D receptor agonist | 0.977 0 CHEMBL3351075 0.823 0 CHEMBL3544529 0.918 0 CHEMBL3542380 0.977 0 CHEMBL3542403 0.918 0 CHEMBL3542386 | CHEMBL3542403 | |
| 0.893 | 0.004 | 0.893 | Immunomodulator | 0.862 0.004 CHEMBL3351075 0.869 0.004 CHEMBL3544529 0.853 0.004 CHEMBL3542380 0.862 0.004 CHEMBL3542403 0.853 0.004 CHEMBL3542386 | ||
| 0.882 | 0.006 | 0.893 | Antiinflammatory | 0.893 0.005 CHEMBL3351075 0.858 0.009 CHEMBL3544529 0.83 0.012 CHEMBL3542380 0.893 0.005 CHEMBL3542403 0.83 0.012 CHEMBL3542386 | CHEMBL3542403 | |
| 0.866 | 0.003 | 0.904 | Non-steroidal antiinflammatory agent | 0.706 0.004 CHEMBL3351075 0.904 0.002 CHEMBL3544529 0.779 0.003 CHEMBL3542380 0.706 0.004 CHEMBL3542403 0.779 0.003 CHEMBL3542386 | CHEMBL3544529 | |
| 0.863 | 0.009 | 0.863 | Transcription factor NF kappa B inhibitor | 0.756 0.016 CHEMBL3351075 0.858 0.009 CHEMBL3544529 0.785 0.014 CHEMBL3542380 0.756 0.016 CHEMBL3542403 0.785 0.014 CHEMBL3542386 | ||
| 0.825 | 0.001 | 0.825 | Interferon gamma antagonist | 0.719 0.001 CHEMBL3351075 0.705 0.001 CHEMBL3544529 0.722 0.001 CHEMBL3542380 0.719 0.001 CHEMBL3542403 0.722 0.001 CHEMBL3542386 | ||
| 0.796 | 0.001 | 0.796 | Calcium channel activator | 0.621 0.002 CHEMBL3351075 0.642 0.002 CHEMBL3544529 0.626 0.002 CHEMBL3542380 0.621 0.002 CHEMBL3542403 0.626 0.002 CHEMBL3542386 | ||
| 0.804 | 0.01 | 0.804 | Caspase 9 stimulant | 0.515 0.054 CHEMBL3351075 0.557 0.043 CHEMBL3544529 0.533 0.049 CHEMBL3542380 0.515 0.054 CHEMBL3542403 0.533 0.049 CHEMBL3542386 | ||
| 0.782 | 0 | 0.782 | Vitamin D-like | 0.564 0 CHEMBL3351075 0.399 0 CHEMBL3544529 0.649 0 CHEMBL3542380 0.564 0 CHEMBL3542403 0.649 0 CHEMBL3542386 | ||
| 0.795 | 0.017 | 0.795 | Apoptosis agonist | 0.754 0.023 CHEMBL3351075 0.729 0.026 CHEMBL3544529 0.699 0.031 CHEMBL3542380 0.754 0.023 CHEMBL3542403 0.699 0.031 CHEMBL3542386 | ||
| 0.761 | 0 | 0.761 | Vitamin D receptor antagonist | 0.686 0 CHEMBL3351075 0.688 0 CHEMBL3544529 0.698 0 CHEMBL3542380 0.686 0 CHEMBL3542403 0.698 0 CHEMBL3542386 | ||
| 0.75 | 0 | 0.75 | Parathyroid hormone antagonist | 0.676 0 CHEMBL3351075 0.682 0 CHEMBL3544529 0.697 0 CHEMBL3542380 0.676 0 CHEMBL3542403 0.697 0 CHEMBL3542386 | ||
| 0.73 | 0.003 | 0.804 | Interleukin agonist | 0.767 0.003 CHEMBL3351075 0.804 0.002 CHEMBL3544529 0.766 0.003 CHEMBL3542380 0.767 0.003 CHEMBL3542403 0.766 0.003 CHEMBL3542386 | CHEMBL3544529 | |
| 0.724 | 0.005 | 0.724 | Immunosuppressant | 0.713 0.005 CHEMBL3351075 0.703 0.005 CHEMBL3544529 0.692 0.005 CHEMBL3542380 0.713 0.005 CHEMBL3542403 0.692 0.005 CHEMBL3542386 | ||
| 0.646 | 0.02 | 0.668 | Cyclophilin D inhibitor | 0.648 0.02 CHEMBL3351075 0.668 0.018 CHEMBL3544529 0.558 0.036 CHEMBL3542380 0.648 0.02 CHEMBL3542403 0.558 0.036 CHEMBL3542386 | CHEMBL3544529 | |
| 0.573 | 0.004 | 0.595 | Bone formation stimulant | 0.595 0.004 CHEMBL3351075 0.58 0.004 CHEMBL3544529 0.531 0.005 CHEMBL3542380 0.595 0.004 CHEMBL3542403 0.531 0.005 CHEMBL3542386 | CHEMBL3542403 | |
| 0.567 | 0.001 | 0.575 | CYP24 inhibitor | 0.541 0.001 CHEMBL3351075 0.575 0.001 CHEMBL3544529 0.53 0.001 CHEMBL3542380 0.541 0.001 CHEMBL3542403 0.53 0.001 CHEMBL3542386 | CHEMBL3544529 | |
| 0.547 | 0.002 | 0.547 | Progesterone antagonist | 0.379 0.003 CHEMBL3351075 0.403 0.003 CHEMBL3544529 0.349 0.003 CHEMBL3542380 0.379 0.003 CHEMBL3542403 0.349 0.003 CHEMBL3542386 | ||
| 0.566 | 0.023 | 0.622 | Cholesterol antagonist | 0.615 0.017 CHEMBL3351075 0.622 0.016 CHEMBL3544529 0.429 0.044 CHEMBL3542380 0.615 0.017 CHEMBL3542403 0.429 0.044 CHEMBL3542386 | CHEMBL3544529 | |
| 0.543 | 0.002 | 0.579 | Keratolytic | 0.471 0.003 CHEMBL3351075 0.579 0.002 CHEMBL3544529 0.528 0.002 CHEMBL3542380 0.471 0.003 CHEMBL3542403 0.528 0.002 CHEMBL3542386 | CHEMBL3544529 | |
| 0.516 | 0.003 | 0.516 | Sodium/bile acid cotransporter inhibitor | 0.513 0.003 CHEMBL3351075 0.513 0.003 CHEMBL3544529 0.488 0.004 CHEMBL3542380 0.513 0.003 CHEMBL3542403 0.488 0.004 CHEMBL3542386 | ||
| 0.497 | 0.016 | 0.559 | Nitric oxide antagonist | 0.559 0.012 CHEMBL3351075 0.452 0.02 CHEMBL3544529 0.467 0.018 CHEMBL3542380 0.559 0.012 CHEMBL3542403 0.467 0.018 CHEMBL3542386 | CHEMBL3542403 | |
| 0.491 | 0.013 | 0.593 | Hypolipemic | 0.491 0.013 CHEMBL3351075 0.428 0.02 CHEMBL3544529 0.593 0.007 CHEMBL3542380 0.491 0.013 CHEMBL3542403 0.593 0.007 CHEMBL3542386 | CHEMBL3542386 | |
| 0.471 | 0.004 | 0.471 | T cell inhibitor | 0.342 0.005 CHEMBL3351075 0.41 0.004 CHEMBL3544529 0.363 0.004 CHEMBL3542380 0.342 0.005 CHEMBL3542403 0.363 0.004 CHEMBL3542386 | ||
| 0.469 | 0.003 | 0.469 | Cholesterol synthesis inhibitor | 0.381 0.005 CHEMBL3351075 0.39 0.005 CHEMBL3544529 0.418 0.004 CHEMBL3542380 0.381 0.005 CHEMBL3542403 0.418 0.004 CHEMBL3542386 | ||
| 0.449 | 0.004 | 0.449 | ABCA1 expression enhancer | 0.379 0.004 CHEMBL3351075 0.405 0.004 CHEMBL3544529 0.378 0.004 CHEMBL3542380 0.379 0.004 CHEMBL3542403 0.378 0.004 CHEMBL3542386 | ||
| 0.428 | 0.004 | 0.428 | Androgen antagonist | 0.353 0.005 CHEMBL3351075 0.239 0.01 CHEMBL3544529 0.304 0.007 CHEMBL3542380 0.353 0.005 CHEMBL3542403 0.304 0.007 CHEMBL3542386 | ||
| 0.386 | 0.01 | 0.386 | Lipocortins synthesis antagonist | 0.366 0.012 CHEMBL3351075 0.383 0.01 CHEMBL3544529 0.333 0.016 CHEMBL3542380 0.366 0.012 CHEMBL3542403 0.333 0.016 CHEMBL3542386 | ||
| 0.419 | 0.044 | 0.419 | Immunostimulant | 0.418 0.045 CHEMBL3351075 0.375 0.057 CHEMBL3544529 0.387 0.053 CHEMBL3542380 0.418 0.045 CHEMBL3542403 0.387 0.053 CHEMBL3542386 | ||
| 0.375 | 0.004 | 0.375 | Farnesoid X receptor antagonist | 0.35 0.004 CHEMBL3351075 0.361 0.004 CHEMBL3544529 0.323 0.005 CHEMBL3542380 0.35 0.004 CHEMBL3542403 0.323 0.005 CHEMBL3542386 | ||
| 0.424 | 0.066 | 0.477 | Antibacterial | 0.477 0.047 CHEMBL3351075 0.434 0.063 CHEMBL3544529 0.345 0.105 CHEMBL3542380 0.477 0.047 CHEMBL3542403 0.345 0.105 CHEMBL3542386 | CHEMBL3542403 | |
| 0.397 | 0.039 | 0.472 | Apoptosis antagonist | 0.406 0.037 CHEMBL3351075 0.472 0.024 CHEMBL3544529 0.361 0.051 CHEMBL3542380 0.406 0.037 CHEMBL3542403 0.361 0.051 CHEMBL3542386 | CHEMBL3544529 | |
| 0.356 | 0.003 | 0.356 | Pregnane X receptor agonist | 0.221 0.007 CHEMBL3351075 0.241 0.005 CHEMBL3544529 0.219 0.007 CHEMBL3542380 0.221 0.007 CHEMBL3542403 0.219 0.007 CHEMBL3542386 | ||
| 0.351 | 0.001 | 0.351 | Anabolic | 0.252 0.002 CHEMBL3351075 0.255 0.002 CHEMBL3544529 0.259 0.002 CHEMBL3542380 0.252 0.002 CHEMBL3542403 0.259 0.002 CHEMBL3542386 | ||
| 0.358 | 0.023 | 0.358 | Anesthetic general | 0.21 0.069 CHEMBL3351075 0.231 0.059 CHEMBL3544529 0.295 0.034 CHEMBL3542380 0.21 0.069 CHEMBL3542403 0.295 0.034 CHEMBL3542386 | ||
| 0.353 | 0.019 | 0.358 | Hepatoprotectant | 0.358 0.018 CHEMBL3351075 0.343 0.02 CHEMBL3544529 0.309 0.027 CHEMBL3542380 0.358 0.018 CHEMBL3542403 0.309 0.027 CHEMBL3542386 | CHEMBL3542403 | |
| 0.346 | 0.034 | 0.358 | Angiogenesis stimulant | 0.319 0.042 CHEMBL3351075 0.358 0.03 CHEMBL3544529 0.318 0.043 CHEMBL3542380 0.319 0.042 CHEMBL3542403 0.318 0.043 CHEMBL3542386 | CHEMBL3544529 | |
| 0.315 | 0.012 | 0.317 | Antipruritic | 0.247 0.025 CHEMBL3351075 0.317 0.012 CHEMBL3544529 0.205 0.046 CHEMBL3542380 0.247 0.025 CHEMBL3542403 0.205 0.046 CHEMBL3542386 | CHEMBL3544529 | |
| 0.297 | 0.004 | 0.297 | CDC25A inhibitor | 0.279 0.004 CHEMBL3351075 0.295 0.004 CHEMBL3544529 0.232 0.005 CHEMBL3542380 0.279 0.004 CHEMBL3542403 0.232 0.005 CHEMBL3542386 | ||
| 0.338 | 0.05 | 0.353 | Antioxidant | 0.353 0.046 CHEMBL3351075 0.312 0.057 CHEMBL3544529 0.271 0.074 CHEMBL3542380 0.353 0.046 CHEMBL3542403 0.271 0.074 CHEMBL3542386 | CHEMBL3542403 | |
| 0.296 | 0.019 | 0.296 | Amylase inhibitor | 0.242 0.03 CHEMBL3351075 0.259 0.025 CHEMBL3544529 0.191 0.048 CHEMBL3542380 0.242 0.03 CHEMBL3542403 0.191 0.048 CHEMBL3542386 | ||
| 0.325 | 0.068 | 0.325 | Caspase 3 stimulant | 0.199 0.17 CHEMBL3351075 0.21 0.155 CHEMBL3542380 0.199 0.17 CHEMBL3542403 0.21 0.155 CHEMBL3542386 | ||
| 0.254 | 0.008 | 0.267 | Microtubule formation inhibitor | 0.267 0.005 CHEMBL3351075 0.252 0.008 CHEMBL3544529 0.262 0.006 CHEMBL3542380 0.267 0.005 CHEMBL3542403 0.262 0.006 CHEMBL3542386 | CHEMBL3542403 | |
| 0.264 | 0.026 | 0.264 | Growth factor agonist | 0.262 0.027 CHEMBL3351075 0.249 0.032 CHEMBL3544529 0.201 0.062 CHEMBL3542380 0.262 0.027 CHEMBL3542403 0.201 0.062 CHEMBL3542386 | ||
| 0.293 | 0.056 | 0.304 | Tumour necrosis factor alpha release inhibitor | 0.304 0.051 CHEMBL3351075 0.216 0.096 CHEMBL3544529 0.252 0.074 CHEMBL3542380 0.304 0.051 CHEMBL3542403 0.252 0.074 CHEMBL3542386 | CHEMBL3542403 | |
| 0.24 | 0.005 | 0.24 | Interleukin 12 antagonist | 0.15 0.012 CHEMBL3351075 0.159 0.01 CHEMBL3544529 0.154 0.011 CHEMBL3542380 0.15 0.012 CHEMBL3542403 0.154 0.011 CHEMBL3542386 | ||
| 0.221 | 0.009 | 0.221 | Antineoplastic alkaloid | 0.109 0.042 CHEMBL3351075 0.107 0.044 CHEMBL3544529 0.147 0.028 CHEMBL3542380 0.109 0.042 CHEMBL3542403 0.147 0.028 CHEMBL3542386 | ||
| 0.217 | 0.019 | 0.234 | Arachidonic acid antagonist | 0.196 0.037 CHEMBL3351075 0.234 0.01 CHEMBL3544529 0.182 0.052 CHEMBL3542380 0.196 0.037 CHEMBL3542403 0.182 0.052 CHEMBL3542386 | CHEMBL3544529 | |
| 0.308 | 0.111 | 0.328 | Antiobesity | 0.328 0.098 CHEMBL3351075 0.238 0.168 CHEMBL3544529 0.328 0.098 CHEMBL3542403 | CHEMBL3542403 | |
| 0.226 | 0.031 | 0.289 | Phospholipase C inhibitor | 0.23 0.03 CHEMBL3351075 0.289 0.019 CHEMBL3544529 0.169 0.074 CHEMBL3542380 0.23 0.03 CHEMBL3542403 0.169 0.074 CHEMBL3542386 | CHEMBL3544529 | |
| 0.214 | 0.022 | 0.214 | Neurotrophic factor | 0.179 0.038 CHEMBL3351075 0.142 0.067 CHEMBL3544529 0.14 0.069 CHEMBL3542380 0.179 0.038 CHEMBL3542403 0.14 0.069 CHEMBL3542386 | ||
| 0.185 | 0.005 | 0.287 | 5-Alpha-reductase inhibitor | 0.108 0.009 CHEMBL3351075 0.287 0.003 CHEMBL3544529 0.083 0.012 CHEMBL3542380 0.108 0.009 CHEMBL3542403 0.083 0.012 CHEMBL3542386 | CHEMBL3544529 | |
| 0.201 | 0.028 | 0.207 | DNA polymerase I inhibitor | 0.181 0.035 CHEMBL3351075 0.207 0.026 CHEMBL3544529 0.151 0.048 CHEMBL3542380 0.181 0.035 CHEMBL3542403 0.151 0.048 CHEMBL3542386 | CHEMBL3544529 | |
| 0.2 | 0.041 | 0.2 | Melanin inhibitor | 0.159 0.07 CHEMBL3351075 0.153 0.077 CHEMBL3544529 0.185 0.048 CHEMBL3542380 0.159 0.07 CHEMBL3542403 0.185 0.048 CHEMBL3542386 | ||
| 0.211 | 0.057 | 0.277 | P-glycoprotein inhibitor | 0.277 0.034 CHEMBL3351075 0.187 0.074 CHEMBL3544529 0.271 0.035 CHEMBL3542380 0.277 0.034 CHEMBL3542403 0.271 0.035 CHEMBL3542386 | CHEMBL3542403 | |
| 0.196 | 0.043 | 0.247 | Protein kinase stimulant | 0.199 0.042 CHEMBL3351075 0.247 0.027 CHEMBL3544529 0.119 0.094 CHEMBL3542380 0.199 0.042 CHEMBL3542403 0.119 0.094 CHEMBL3542386 | CHEMBL3544529 | |
| 0.155 | 0.005 | 0.16 | Na+ K+ transporting ATPase inhibitor | 0.158 0.005 CHEMBL3351075 0.16 0.004 CHEMBL3544529 0.152 0.005 CHEMBL3542380 0.158 0.005 CHEMBL3542403 0.152 0.005 CHEMBL3542386 | CHEMBL3544529 | |
| 0.23 | 0.083 | 0.23 | DNA synthesis inhibitor | 0.219 0.096 CHEMBL3544529 0.186 0.144 CHEMBL3542380 0.186 0.144 CHEMBL3542386 | ||
| 0.153 | 0.007 | 0.265 | Bile acid receptor antagonist | 0.124 0.016 CHEMBL3351075 0.265 0.003 CHEMBL3544529 0.11 0.031 CHEMBL3542380 0.124 0.016 CHEMBL3542403 0.11 0.031 CHEMBL3542386 | CHEMBL3544529 | |
| 0.251 | 0.117 | 0.33 | Interleukin 2 agonist | 0.282 0.088 CHEMBL3351075 0.33 0.055 CHEMBL3544529 0.234 0.137 CHEMBL3542380 0.282 0.088 CHEMBL3542403 0.234 0.137 CHEMBL3542386 | CHEMBL3544529 | |
| 0.204 | 0.073 | 0.204 | Neurotrophic factor enhancer | 0.147 0.142 CHEMBL3542380 0.147 0.142 CHEMBL3542386 | ||
| 0.13 | 0.01 | 0.131 | Glycine receptor agonist | 0.074 0.048 CHEMBL3351075 0.131 0.01 CHEMBL3544529 0.074 0.048 CHEMBL3542380 0.074 0.048 CHEMBL3542403 0.074 0.048 CHEMBL3542386 | CHEMBL3544529 | |
| 0.152 | 0.032 | 0.152 | Papain-like protease (SARS coronavirus) inhibitor | 0.121 0.078 CHEMBL3542380 0.121 0.078 CHEMBL3542386 | ||
| 0.16 | 0.042 | 0.186 | Protein-tyrosine phosphatase 1B inhibitor | 0.162 0.041 CHEMBL3351075 0.186 0.033 CHEMBL3544529 0.118 0.065 CHEMBL3542380 0.162 0.041 CHEMBL3542403 0.118 0.065 CHEMBL3542386 | CHEMBL3544529 | |
| 0.127 | 0.01 | 0.127 | CDC25B inhibitor | 0.096 0.017 CHEMBL3351075 0.12 0.011 CHEMBL3544529 0.076 0.032 CHEMBL3542380 0.096 0.017 CHEMBL3542403 0.076 0.032 CHEMBL3542386 | ||
| 0.142 | 0.033 | 0.172 | Antineoplastic antibiotic | 0.172 0.026 CHEMBL3351075 0.131 0.035 CHEMBL3544529 0.135 0.034 CHEMBL3542380 0.172 0.026 CHEMBL3542403 0.135 0.034 CHEMBL3542386 | CHEMBL3542403 | |
| 0.124 | 0.037 | 0.124 | Hedgehog signaling inhibitor | |||
| 0.094 | 0.008 | 0.094 | Liver X receptor agonist | 0.059 0.017 CHEMBL3351075 0.043 0.032 CHEMBL3544529 0.079 0.01 CHEMBL3542380 0.059 0.017 CHEMBL3542403 0.079 0.01 CHEMBL3542386 | ||
| 0.089 | 0.005 | 0.126 | Farnesoid X receptor agonist | 0.126 0.003 CHEMBL3351075 0.093 0.004 CHEMBL3544529 0.082 0.005 CHEMBL3542380 0.126 0.003 CHEMBL3542403 0.082 0.005 CHEMBL3542386 | CHEMBL3542403 | |
| 0.098 | 0.015 | 0.098 | Androgen agonist | 0.073 0.028 CHEMBL3351075 0.074 0.027 CHEMBL3544529 0.065 0.035 CHEMBL3542380 0.073 0.028 CHEMBL3542403 0.065 0.035 CHEMBL3542386 | ||
| 0.153 | 0.075 | 0.187 | Protein-tyrosine phosphatase inhibitor | 0.153 0.075 CHEMBL3351075 0.187 0.052 CHEMBL3544529 0.153 0.075 CHEMBL3542403 | CHEMBL3544529 | |
| 0.077 | 0.006 | 0.15 | 5-Alpha-reductase 2 inhibitor | 0.021 0.012 CHEMBL3351075 0.15 0.004 CHEMBL3544529 0.021 0.012 CHEMBL3542403 | CHEMBL3544529 | |
| 0.081 | 0.013 | 0.081 | Lipocortins synthesis agonist | 0.078 0.015 CHEMBL3351075 0.081 0.013 CHEMBL3544529 0.075 0.017 CHEMBL3542380 0.078 0.015 CHEMBL3542403 0.075 0.017 CHEMBL3542386 | ||
| 0.102 | 0.035 | 0.119 | Inducible nitric-oxide synthase inhibitor | 0.119 0.025 CHEMBL3544529 | CHEMBL3544529 | |
| 0.085 | 0.019 | 0.108 | Prostaglandin F2 alpha antagonist | 0.108 0.009 CHEMBL3351075 0.107 0.009 CHEMBL3544529 0.099 0.012 CHEMBL3542380 0.108 0.009 CHEMBL3542403 0.099 0.012 CHEMBL3542386 | CHEMBL3542403 | |
| 0.068 | 0.004 | 0.088 | HMG CoA reductase inhibitor | 0.068 0.004 CHEMBL3351075 0.067 0.004 CHEMBL3544529 0.088 0.003 CHEMBL3542380 0.068 0.004 CHEMBL3542403 0.088 0.003 CHEMBL3542386 | CHEMBL3542386 | |
| 0.063 | 0.011 | 0.063 | Liver X receptor alpha agonist | 0.05 0.019 CHEMBL3351075 0.041 0.028 CHEMBL3544529 0.056 0.015 CHEMBL3542380 0.05 0.019 CHEMBL3542403 0.056 0.015 CHEMBL3542386 | ||
| 0.071 | 0.024 | 0.075 | Heme oxygenase stimulant | 0.068 0.028 CHEMBL3351075 0.075 0.019 CHEMBL3544529 0.068 0.028 CHEMBL3542380 0.068 0.028 CHEMBL3542403 0.068 0.028 CHEMBL3542386 | CHEMBL3544529 | |
| 0.06 | 0.014 | 0.062 | Microtubule stabilization | 0.062 0.012 CHEMBL3351075 0.059 0.016 CHEMBL3544529 0.061 0.014 CHEMBL3542380 0.062 0.012 CHEMBL3542403 0.061 0.014 CHEMBL3542386 | CHEMBL3542403 | |
| 0.101 | 0.055 | 0.101 | Lanosterol 14 alpha demethylase inhibitor | |||
| 0.054 | 0.012 | 0.057 | RNA-directed RNA polymerase stimulant | 0.05 0.013 CHEMBL3351075 0.057 0.012 CHEMBL3544529 0.05 0.013 CHEMBL3542380 0.05 0.013 CHEMBL3542403 0.05 0.013 CHEMBL3542386 | CHEMBL3544529 | |
| 0.052 | 0.01 | 0.052 | 2,3-Oxidosqualene-lanosterol cyclase inhibitor | 0.041 0.02 CHEMBL3351075 0.035 0.029 CHEMBL3544529 0.034 0.03 CHEMBL3542380 0.041 0.02 CHEMBL3542403 0.034 0.03 CHEMBL3542386 | ||
| 0.111 | 0.073 | 0.115 | Estrogen antagonist | 0.115 0.064 CHEMBL3544529 | CHEMBL3544529 | |
| 0.065 | 0.027 | 0.079 | Protein 50S ribosomal subunit inhibitor | 0.079 0.02 CHEMBL3351075 0.065 0.027 CHEMBL3544529 0.062 0.029 CHEMBL3542380 0.079 0.02 CHEMBL3542403 0.062 0.029 CHEMBL3542386 | CHEMBL3542403 | |
| 0.147 | 0.109 | 0.175 | Platelet adhesion inhibitor | 0.175 0.085 CHEMBL3544529 | CHEMBL3544529 | |
| 0.107 | 0.074 | 0.13 | Interleukin 1b antagonist | 0.13 0.055 CHEMBL3351075 0.123 0.06 CHEMBL3544529 0.117 0.065 CHEMBL3542380 0.13 0.055 CHEMBL3542403 0.117 0.065 CHEMBL3542386 | CHEMBL3542403 | |
| 0.1 | 0.068 | 0.198 | Expectorant | 0.135 0.042 CHEMBL3351075 0.198 0.021 CHEMBL3544529 0.112 0.057 CHEMBL3542380 0.135 0.042 CHEMBL3542403 0.112 0.057 CHEMBL3542386 | CHEMBL3544529 | |
| 0.06 | 0.028 | 0.06 | Leukotriene B4 antagonist | 0.057 0.032 CHEMBL3544529 0.049 0.047 CHEMBL3542380 0.049 0.047 CHEMBL3542386 | ||
| 0.036 | 0.006 | 0.043 | Hedgehog signaling activator | 0.032 0.01 CHEMBL3351075 0.032 0.009 CHEMBL3544529 0.043 0.004 CHEMBL3542380 0.032 0.01 CHEMBL3542403 0.043 0.004 CHEMBL3542386 | CHEMBL3542386 | |
| 0.046 | 0.017 | 0.046 | Glucocorticoid antagonist | 0.036 0.021 CHEMBL3351075 0.03 0.024 CHEMBL3542380 0.036 0.021 CHEMBL3542403 0.03 0.024 CHEMBL3542386 | ||
| 0.044 | 0.017 | 0.047 | Glucose-6-phosphate dehydrogenase inhibitor | 0.042 0.019 CHEMBL3351075 0.047 0.014 CHEMBL3544529 0.042 0.019 CHEMBL3542380 0.042 0.019 CHEMBL3542403 0.042 0.019 CHEMBL3542386 | CHEMBL3544529 | |
| 0.027 | 0.006 | 0.027 | Progesterone receptor B antagonist | 0.025 0.007 CHEMBL3351075 0.025 0.007 CHEMBL3544529 0.025 0.007 CHEMBL3542380 0.025 0.007 CHEMBL3542403 0.025 0.007 CHEMBL3542386 | ||
| 0.117 | 0.096 | 0.132 | Vanilloid 1 agonist | 0.116 0.097 CHEMBL3351075 0.132 0.063 CHEMBL3544529 0.117 0.096 CHEMBL3542380 0.116 0.097 CHEMBL3542403 0.117 0.096 CHEMBL3542386 | CHEMBL3544529 | |
| 0.169 | 0.149 | 0.302 | Hypoglycemic | 0.268 0.066 CHEMBL3351075 0.302 0.052 CHEMBL3544529 0.268 0.066 CHEMBL3542403 | CHEMBL3544529 | |
| 0.037 | 0.019 | 0.039 | Tubulin agonist | 0.036 0.02 CHEMBL3351075 0.039 0.017 CHEMBL3544529 0.036 0.02 CHEMBL3542380 0.036 0.02 CHEMBL3542403 0.036 0.02 CHEMBL3542386 | CHEMBL3544529 | |
| 0.052 | 0.034 | 0.052 | Estrogen agonist | 0.052 0.034 CHEMBL3544529 | ||
| 0.027 | 0.011 | 0.034 | Prostaglandin F2 alpha agonist | 0.034 0.007 CHEMBL3351075 0.028 0.01 CHEMBL3544529 0.028 0.01 CHEMBL3542380 0.034 0.007 CHEMBL3542403 0.028 0.01 CHEMBL3542386 | CHEMBL3542403 | |
| 0.034 | 0.018 | 0.035 | Prostaglandin D2 agonist | 0.035 0.017 CHEMBL3351075 0.034 0.018 CHEMBL3544529 0.028 0.025 CHEMBL3542380 0.035 0.017 CHEMBL3542403 0.028 0.025 CHEMBL3542386 | CHEMBL3542403 | |
| 0.138 | 0.127 | 0.149 | Interleukin antagonist | 0.149 0.118 CHEMBL3544529 | CHEMBL3544529 | |
| 0.032 | 0.022 | 0.04 | ATP citrate lysase inhibitor | 0.04 0.013 CHEMBL3351075 0.034 0.019 CHEMBL3544529 0.04 0.013 CHEMBL3542380 0.04 0.013 CHEMBL3542403 0.04 0.013 CHEMBL3542386 | CHEMBL3542386 | |
| 0.111 | 0.103 | 0.127 | Interleukin 1 antagonist | 0.125 0.082 CHEMBL3351075 0.127 0.079 CHEMBL3544529 0.125 0.082 CHEMBL3542403 | CHEMBL3544529 | |
| 0.014 | 0.006 | 0.014 | 3 Beta-hydroxy-delta 5-steroid dehydrogenase inhibitor | 0.013 0.007 CHEMBL3351075 0.014 0.006 CHEMBL3544529 0.013 0.008 CHEMBL3542380 0.013 0.007 CHEMBL3542403 0.013 0.008 CHEMBL3542386 | ||
| 0.027 | 0.02 | 0.059 | 11-Beta-hydroxysteroid dehydrogenase 2 inhibitor | 0.059 0.007 CHEMBL3351075 0.059 0.007 CHEMBL3542403 | CHEMBL3542403 | |
| 0.019 | 0.011 | 0.088 | 5-Alpha-reductase 1 inhibitor | 0.088 0.005 CHEMBL3544529 | CHEMBL3544529 | |
| 0.071 | 0.064 | 0.071 | Estrogen receptor alpha antagonist | 0.071 0.065 CHEMBL3544529 | ||
| 0.02 | 0.017 | 0.022 | Corticosteroid-like | 0.022 0.014 CHEMBL3544529 | CHEMBL3544529 | |
| 0.018 | 0.015 | 0.018 | Steroid 17-alpha-hydroxylase/17,20 lyase inhibitor | |||
| 0.137 | 0.136 | 0.137 | Antimitotic | |||
| 0.025 | 0.026 | 0.031 | Retinoid X gamma receptor antagonist | 0.031 0.011 CHEMBL3544529 | CHEMBL3544529 | |
| 0.073 | 0.075 | 0.125 | Ornithine decarboxylase inhibitor | 0.125 0.023 CHEMBL3544529 | CHEMBL3544529 | |
| 0.076 | 0.079 | 0.093 | Transcription factor NF kappa B stimulant | 0.093 0.046 CHEMBL3544529 | CHEMBL3544529 | |
| 0.036 | 0.044 | 0.049 | 11-Beta-hydroxysteroid dehydrogenase 1 inhibitor | 0.049 0.031 CHEMBL3351075 0.049 0.031 CHEMBL3542403 | CHEMBL3542403 | |
| 0.018 | 0.03 | 0.022 | Retinoic acid gamma receptor agonist | 0.022 0.017 CHEMBL3544529 | CHEMBL3544529 | |
| 0.091 | 0.105 | 0.097 | TRPA1 agonist | 0.097 0.093 CHEMBL3351075 0.097 0.093 CHEMBL3544529 0.097 0.093 CHEMBL3542403 | CHEMBL3542403 | |
| 0.01 | 0.025 | 0.017 | Ileal bile acid transport inhibitor | 0.017 0.012 CHEMBL3544529 | CHEMBL3544529 | |
| 0.1 | 0.117 | 0.165 | Lipid peroxidase inhibitor | 0.165 0.058 CHEMBL3351075 0.165 0.058 CHEMBL3542403 | CHEMBL3542403 | |
| 0.015 | 0.04 | 0.025 | Retinoid X beta receptor antagonist | 0.025 0.007 CHEMBL3544529 | CHEMBL3544529 | |
| 0.108 | 0.134 | 0.215 | Insulin secretagoues | 0.215 0.029 CHEMBL3544529 | CHEMBL3544529 | |
| 0.154 | 0.183 | 0.197 | Peptidyltransferase inhibitor | 0.197 0.103 CHEMBL3544529 | CHEMBL3544529 | |
| 0.013 | 0.047 | 0.023 | Retinoid X gamma receptor agonist | 0.023 0.016 CHEMBL3544529 | CHEMBL3544529 | |
| 0.079 | 0.117 | 0.143 | Mucolytic | 0.099 0.078 CHEMBL3351075 0.143 0.037 CHEMBL3544529 0.099 0.078 CHEMBL3542403 | CHEMBL3544529 | |
| 0.131 | 0.175 | 0.191 | Free radical scavenger | 0.191 0.105 CHEMBL3351075 0.191 0.105 CHEMBL3542403 | CHEMBL3542403 | |
| 0.104 | 0.169 | 0.146 | Adenylate cyclase stimulant | 0.146 0.07 CHEMBL3544529 | CHEMBL3544529 | |
| 0.011 | 0.097 | 0.043 | Retinoid X receptor agonist | 0.043 0.021 CHEMBL3544529 | CHEMBL3544529 | |
| 0.145 | 0.259 | 0.2 | Antithrombotic | 0.2 0.177 CHEMBL3544529 | CHEMBL3544529 | |
| 0.098 | 0.225 | 0.22 | Platelet antagonist | 0.22 0.088 CHEMBL3544529 | CHEMBL3544529 | |
| 0.019 | 0.156 | 0.035 | Retinoid X receptor antagonist | 0.035 0.033 CHEMBL3544529 | CHEMBL3544529 | |
| 0.011 | 0.15 | 0.034 | Retinoid X alpha receptor agonist | 0.034 0.025 CHEMBL3544529 | CHEMBL3544529 | |
| 0.004 | 0.195 | 0.016 | Free fatty acid receptor 1 agonist | 0.016 0.014 CHEMBL3544529 | CHEMBL3544529 | |
| 0.043 | 0.242 | 0.096 | UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor | 0.096 0.058 CHEMBL3544529 | CHEMBL3544529 | |
| 0.138 | 0.341 | 0.19 | 5 Hydroxytryptamine uptake stimulant | 0.19 0.173 CHEMBL3544529 | CHEMBL3544529 | |
| 0.051 | 0.327 | 0.147 | Insulin sensitizer | 0.147 0.137 CHEMBL3544529 | CHEMBL3544529 | |
| 0.019 | 0.616 | 0.099 | Cell adhesion inhibitor | 0.099 0.09 CHEMBL3544529 | CHEMBL3544529 | |
| 0.004 | 0.718 | 0.015 | Integrin beta6 antagonist | 0.015 0.007 CHEMBL3544529 | CHEMBL3544529 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |