| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.88 | 0.002 | 0.979 | DNA synthesis inhibitor | 0.948 0.001 CHEMBL1232305 0.973 0.001 CHEMBL1232161 0.909 0.002 CHEMBL3638310 0.95 0.001 CHEMBL3544876 0.979 0.001 CHEMBL1201384 | CHEMBL1201384 | |
| 0.79 | 0.002 | 0.977 | RNA-directed DNA polymerase inhibitor | 0.936 0.001 CHEMBL1232305 0.968 0.001 CHEMBL1232161 0.836 0.001 CHEMBL3638310 0.917 0.001 CHEMBL3544876 0.977 0 CHEMBL1201384 | CHEMBL1201384 | |
| 0.716 | 0.032 | 0.976 | DNA directed DNA polymerase inhibitor | 0.856 0.012 CHEMBL1232305 0.958 0.004 CHEMBL1232161 0.914 0.006 CHEMBL3638310 0.796 0.02 CHEMBL3544876 0.976 0.004 CHEMBL1201384 | CHEMBL1201384 | |
| 0.631 | 0.002 | 0.631 | Peptidyltransferase inhibitor | 0.548 0.003 CHEMBL1232305 0.518 0.003 CHEMBL1232161 0.462 0.004 CHEMBL3638310 0.504 0.003 CHEMBL3544876 0.509 0.003 CHEMBL1201384 | ||
| 0.578 | 0.004 | 0.815 | Cytidine deaminase inhibitor | 0.692 0.003 CHEMBL1232305 0.782 0.002 CHEMBL1232161 0.765 0.003 CHEMBL3638310 0.567 0.005 CHEMBL3544876 0.815 0.002 CHEMBL1201384 | CHEMBL1201384 | |
| 0.572 | 0.009 | 0.626 | DNA damaging | 0.465 0.017 CHEMBL1232305 0.459 0.018 CHEMBL1232161 0.561 0.01 CHEMBL3638310 0.626 0.007 CHEMBL3544876 0.408 0.027 CHEMBL1201384 | CHEMBL3544876 | |
| 0.55 | 0.003 | 0.757 | DNA polymerase I inhibitor | 0.63 0.002 CHEMBL1232305 0.728 0.001 CHEMBL1232161 0.633 0.002 CHEMBL3638310 0.657 0.002 CHEMBL3544876 0.757 0.001 CHEMBL1201384 | CHEMBL1201384 | |
| 0.532 | 0.001 | 0.793 | Mannitol-1-phosphate 5-dehydrogenase inhibitor | 0.703 0 CHEMBL1232305 0.772 0 CHEMBL1232161 0.57 0.001 CHEMBL3638310 0.672 0 CHEMBL3544876 0.793 0 CHEMBL1201384 | CHEMBL1201384 | |
| 0.532 | 0.005 | 0.592 | DNA methylase inhibitor | 0.515 0.005 CHEMBL1232305 0.442 0.008 CHEMBL1232161 0.469 0.007 CHEMBL3638310 0.592 0.004 CHEMBL3544876 0.39 0.012 CHEMBL1201384 | CHEMBL3544876 | |
| 0.527 | 0.002 | 0.758 | Carbamoyl phosphate synthetase inhibitor | 0.708 0.001 CHEMBL1232305 0.746 0 CHEMBL1232161 0.578 0.002 CHEMBL3638310 0.676 0.001 CHEMBL3544876 0.758 0 CHEMBL1201384 | CHEMBL1201384 | |
| 0.518 | 0.005 | 0.711 | Adenylate cyclase inhibitor | 0.656 0.002 CHEMBL1232305 0.698 0.002 CHEMBL1232161 0.678 0.002 CHEMBL3638310 0.656 0.002 CHEMBL3544876 0.711 0.001 CHEMBL1201384 | CHEMBL1201384 | |
| 0.508 | 0.004 | 0.793 | DNA directed RNA polymerase inhibitor | 0.609 0.004 CHEMBL1232305 0.75 0.003 CHEMBL1232161 0.583 0.004 CHEMBL3638310 0.6 0.004 CHEMBL3544876 0.793 0.003 CHEMBL1201384 | CHEMBL1201384 | |
| 0.5 | 0.004 | 0.647 | Glyceraldehyde-3-phosphate dehydrogenase inhibitor | 0.613 0.002 CHEMBL1232305 0.647 0.002 CHEMBL1232161 0.523 0.004 CHEMBL3638310 0.58 0.003 CHEMBL3544876 0.635 0.002 CHEMBL1201384 | CHEMBL1232161 | |
| 0.497 | 0.003 | 0.909 | Antimetabolite | 0.76 0.001 CHEMBL1232305 0.853 0.001 CHEMBL1232161 0.909 0.001 CHEMBL3638310 0.856 0.001 CHEMBL3544876 0.865 0.001 CHEMBL1201384 | CHEMBL3638310 | |
| 0.49 | 0.002 | 0.81 | Phosphofructokinase-1 inhibitor | 0.706 0.001 CHEMBL1232305 0.784 0.001 CHEMBL1232161 0.555 0.002 CHEMBL3638310 0.688 0.001 CHEMBL3544876 0.81 0.001 CHEMBL1201384 | CHEMBL1201384 | |
| 0.449 | 0.004 | 0.6 | UDP-glucose 4-epimerase inhibitor | 0.551 0.002 CHEMBL1232305 0.588 0.001 CHEMBL1232161 0.465 0.003 CHEMBL3638310 0.524 0.002 CHEMBL3544876 0.6 0.001 CHEMBL1201384 | CHEMBL1201384 | |
| 0.487 | 0.044 | 0.511 | Antibacterial | 0.453 0.056 CHEMBL1232305 0.418 0.069 CHEMBL1232161 0.511 0.038 CHEMBL3638310 0.477 0.047 CHEMBL3544876 0.372 0.09 CHEMBL1201384 | CHEMBL3638310 | |
| 0.464 | 0.029 | 0.555 | Immunomodulator | 0.492 0.024 CHEMBL1232305 0.541 0.018 CHEMBL1232161 0.555 0.016 CHEMBL3638310 0.518 0.021 CHEMBL3544876 0.515 0.021 CHEMBL1201384 | CHEMBL3638310 | |
| 0.438 | 0.006 | 0.438 | DNA methyltransferase I inhibitor | |||
| 0.431 | 0.002 | 0.865 | Argininosuccinate synthase inhibitor | 0.79 0.001 CHEMBL1232305 0.847 0 CHEMBL1232161 0.479 0.002 CHEMBL3638310 0.722 0.001 CHEMBL3544876 0.865 0 CHEMBL1201384 | CHEMBL1201384 | |
| 0.446 | 0.038 | 0.629 | Immunostimulant | 0.561 0.021 CHEMBL1232305 0.563 0.021 CHEMBL1232161 0.595 0.017 CHEMBL3638310 0.629 0.014 CHEMBL3544876 0.537 0.024 CHEMBL1201384 | CHEMBL3544876 | |
| 0.404 | 0.003 | 0.512 | DNA repair enzyme inhibitor | 0.512 0.002 CHEMBL1232305 0.324 0.004 CHEMBL1232161 0.187 0.011 CHEMBL3638310 0.259 0.005 CHEMBL3544876 0.276 0.005 CHEMBL1201384 | CHEMBL1232305 | |
| 0.401 | 0.004 | 0.858 | Glutamate dehydrogenase inhibitor | 0.805 0.001 CHEMBL1232305 0.847 0.001 CHEMBL1232161 0.569 0.003 CHEMBL3638310 0.796 0.001 CHEMBL3544876 0.858 0.001 CHEMBL1201384 | CHEMBL1201384 | |
| 0.394 | 0.008 | 0.594 | Alkylator | 0.524 0.004 CHEMBL1232305 0.46 0.005 CHEMBL1232161 0.594 0.004 CHEMBL3638310 0.589 0.004 CHEMBL3544876 0.409 0.007 CHEMBL1201384 | CHEMBL3638310 | |
| 0.359 | 0.005 | 0.637 | NADH dehydrogenase inhibitor | 0.567 0.002 CHEMBL1232305 0.637 0.002 CHEMBL1232161 0.403 0.005 CHEMBL3638310 0.531 0.003 CHEMBL3544876 0.614 0.002 CHEMBL1201384 | CHEMBL1232161 | |
| 0.344 | 0.007 | 0.678 | Hexokinase inhibitor | 0.535 0.003 CHEMBL1232305 0.654 0.002 CHEMBL1232161 0.357 0.005 CHEMBL3638310 0.459 0.003 CHEMBL3544876 0.678 0.002 CHEMBL1201384 | CHEMBL1201384 | |
| 0.329 | 0.003 | 0.875 | Fumarate hydratase inhibitor | 0.808 0.001 CHEMBL1232305 0.86 0.001 CHEMBL1232161 0.391 0.002 CHEMBL3638310 0.723 0.001 CHEMBL3544876 0.875 0 CHEMBL1201384 | CHEMBL1201384 | |
| 0.327 | 0.005 | 0.617 | HIV-1 reverse transcriptase inhibitor | 0.397 0.004 CHEMBL1232305 0.571 0.003 CHEMBL1232161 0.351 0.005 CHEMBL3638310 0.382 0.004 CHEMBL3544876 0.617 0.003 CHEMBL1201384 | CHEMBL1201384 | |
| 0.291 | 0.001 | 0.291 | Thymidine phosphorylase inhibitor | 0.195 0.002 CHEMBL1232305 0.118 0.003 CHEMBL1232161 0.032 0.01 CHEMBL3638310 0.063 0.004 CHEMBL3544876 0.103 0.003 CHEMBL1201384 | ||
| 0.319 | 0.035 | 0.319 | Cyclic AMP phosphodiesterase inhibitor | |||
| 0.304 | 0.023 | 0.304 | Ca2+/calmodulin-dependent kinase IV inhibitor | 0.208 0.144 CHEMBL1232305 | ||
| 0.284 | 0.007 | 0.61 | Aminoacyl-tRNA synthetase inhibitor | 0.411 0.004 CHEMBL1232305 0.556 0.003 CHEMBL1232161 0.403 0.004 CHEMBL3638310 0.48 0.003 CHEMBL3544876 0.61 0.002 CHEMBL1201384 | CHEMBL1201384 | |
| 0.252 | 0.005 | 0.819 | Ornithine carbamoyltransferase inhibitor | 0.713 0.001 CHEMBL1232305 0.799 0.001 CHEMBL1232161 0.404 0.003 CHEMBL3638310 0.766 0.001 CHEMBL3544876 0.819 0.001 CHEMBL1201384 | CHEMBL1201384 | |
| 0.371 | 0.13 | 0.543 | Caspase 9 stimulant | 0.543 0.046 CHEMBL1232305 0.329 0.163 CHEMBL1232161 0.292 0.203 CHEMBL1201384 | CHEMBL1232305 | |
| 0.241 | 0.003 | 0.503 | Phosphoglycerate kinase inhibitor | 0.44 0.001 CHEMBL1232305 0.492 0.001 CHEMBL1232161 0.346 0.002 CHEMBL3638310 0.483 0.001 CHEMBL3544876 0.503 0.001 CHEMBL1201384 | CHEMBL1201384 | |
| 0.24 | 0.009 | 0.24 | Adenosine A1 receptor antagonist | 0.058 0.041 CHEMBL1232305 | ||
| 0.238 | 0.014 | 0.536 | Expectorant | 0.311 0.008 CHEMBL1232305 0.502 0.004 CHEMBL1232161 0.29 0.009 CHEMBL3638310 0.328 0.007 CHEMBL3544876 0.536 0.003 CHEMBL1201384 | CHEMBL1201384 | |
| 0.3 | 0.078 | 0.3 | Caspase 3 stimulant | 0.2 0.168 CHEMBL1232305 | ||
| 0.217 | 0.008 | 0.261 | Transcription factor NF kappa B stimulant | 0.22 0.008 CHEMBL1232305 0.261 0.005 CHEMBL1232161 0.194 0.01 CHEMBL3638310 0.226 0.007 CHEMBL3544876 0.252 0.005 CHEMBL1201384 | CHEMBL1232161 | |
| 0.215 | 0.007 | 0.475 | Ribonucleotide reductase inhibitor | 0.363 0.003 CHEMBL1232305 0.441 0.002 CHEMBL1232161 0.377 0.003 CHEMBL3638310 0.368 0.003 CHEMBL3544876 0.475 0.002 CHEMBL1201384 | CHEMBL1201384 | |
| 0.263 | 0.054 | 0.263 | Ca2+/calmodulin-dependent kinase I alpha inhibitor | |||
| 0.218 | 0.013 | 0.471 | UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor | 0.442 0.003 CHEMBL1232305 0.471 0.003 CHEMBL1232161 0.15 0.027 CHEMBL3638310 0.305 0.006 CHEMBL3544876 0.441 0.003 CHEMBL1201384 | CHEMBL1232161 | |
| 0.204 | 0.006 | 0.341 | Ribonucleoside-diphosphate reductase inhibitor | 0.305 0.004 CHEMBL1232305 0.341 0.003 CHEMBL1232161 0.334 0.003 CHEMBL3638310 0.305 0.004 CHEMBL3544876 0.308 0.004 CHEMBL1201384 | CHEMBL1232161 | |
| 0.341 | 0.144 | 0.355 | Apoptosis agonist | 0.355 0.136 CHEMBL1232305 0.268 0.197 CHEMBL1232161 0.348 0.14 CHEMBL3638310 0.348 0.14 CHEMBL3544876 0.24 0.225 CHEMBL1201384 | CHEMBL1232305 | |
| 0.225 | 0.029 | 0.225 | Interleukin 6 antagonist | 0.211 0.035 CHEMBL1232305 0.143 0.1 CHEMBL1232161 0.223 0.03 CHEMBL3638310 0.131 0.122 CHEMBL1201384 | ||
| 0.208 | 0.012 | 0.391 | Mucolytic | 0.231 0.008 CHEMBL1232305 0.355 0.004 CHEMBL1232161 0.215 0.01 CHEMBL3638310 0.25 0.006 CHEMBL3544876 0.391 0.003 CHEMBL1201384 | CHEMBL1201384 | |
| 0.235 | 0.048 | 0.235 | MAP kinase kinase 3 inhibitor | 0.197 0.131 CHEMBL1232305 | ||
| 0.273 | 0.086 | 0.273 | Ca2+/calmodulin-dependent kinase II alpha inhibitor | |||
| 0.197 | 0.01 | 0.197 | Adenosine A2a receptor antagonist | |||
| 0.297 | 0.117 | 0.486 | Immunosuppressant | 0.486 0.037 CHEMBL1232305 0.39 0.067 CHEMBL1232161 0.346 0.089 CHEMBL3638310 0.419 0.056 CHEMBL3544876 0.378 0.073 CHEMBL1201384 | CHEMBL1232305 | |
| 0.177 | 0.003 | 0.701 | Thymidine kinase inhibitor | 0.438 0.002 CHEMBL1232305 0.644 0.001 CHEMBL1232161 0.18 0.003 CHEMBL3638310 0.349 0.002 CHEMBL3544876 0.701 0.001 CHEMBL1201384 | CHEMBL1201384 | |
| 0.214 | 0.043 | 0.214 | Protein kinase C nu inhibitor | |||
| 0.183 | 0.018 | 0.468 | Adenylate kinase inhibitor | 0.41 0.003 CHEMBL1232305 0.455 0.002 CHEMBL1232161 0.332 0.005 CHEMBL3638310 0.416 0.003 CHEMBL3544876 0.468 0.002 CHEMBL1201384 | CHEMBL1201384 | |
| 0.176 | 0.013 | 0.176 | Adenosine A2 receptor antagonist | |||
| 0.27 | 0.113 | 0.27 | Transcription factor NF kappa B inhibitor | |||
| 0.264 | 0.117 | 0.457 | Vasodilator, peripheral | 0.203 0.172 CHEMBL1232305 0.409 0.052 CHEMBL1232161 0.262 0.118 CHEMBL3638310 0.457 0.038 CHEMBL1201384 | CHEMBL1201384 | |
| 0.147 | 0.003 | 0.151 | Adenosine deaminase inhibitor | 0.124 0.004 CHEMBL1232305 0.151 0.003 CHEMBL1232161 0.078 0.01 CHEMBL3638310 0.106 0.005 CHEMBL3544876 0.135 0.003 CHEMBL1201384 | CHEMBL1232161 | |
| 0.149 | 0.007 | 0.258 | 3-Oxoacyl-[acyl-carrier-protein] synthase inhibitor | 0.232 0.004 CHEMBL1232305 0.258 0.003 CHEMBL1232161 0.113 0.013 CHEMBL3638310 0.213 0.004 CHEMBL3544876 0.227 0.004 CHEMBL1201384 | CHEMBL1232161 | |
| 0.148 | 0.01 | 0.422 | Biliverdin reductase inhibitor | 0.398 0.002 CHEMBL1232305 0.422 0.002 CHEMBL1232161 0.281 0.004 CHEMBL3638310 0.377 0.002 CHEMBL3544876 0.398 0.002 CHEMBL1201384 | CHEMBL1232161 | |
| 0.135 | 0.014 | 0.135 | Adenosine A3 receptor antagonist | |||
| 0.117 | 0.004 | 0.266 | Thymidylate synthase inhibitor | 0.266 0.002 CHEMBL1232305 0.145 0.003 CHEMBL1232161 0.112 0.004 CHEMBL3638310 0.124 0.004 CHEMBL3544876 0.127 0.004 CHEMBL1201384 | CHEMBL1232305 | |
| 0.115 | 0.002 | 0.141 | Uridine phosphorylase inhibitor | 0.141 0.001 CHEMBL1232305 0.098 0.002 CHEMBL1232161 0.042 0.011 CHEMBL3638310 0.083 0.003 CHEMBL3544876 0.092 0.003 CHEMBL1201384 | CHEMBL1232305 | |
| 0.245 | 0.139 | 0.292 | Vasodilator, coronary | 0.268 0.117 CHEMBL1232161 0.263 0.122 CHEMBL3638310 0.241 0.144 CHEMBL3544876 0.292 0.094 CHEMBL1201384 | CHEMBL1201384 | |
| 0.16 | 0.056 | 0.16 | Cell wall synthesis inhibitor | 0.155 0.061 CHEMBL1232305 0.154 0.062 CHEMBL1232161 0.135 0.08 CHEMBL3638310 0.16 0.057 CHEMBL3544876 0.128 0.088 CHEMBL1201384 | ||
| 0.111 | 0.021 | 0.111 | Interferon agonist | 0.084 0.046 CHEMBL1232305 | ||
| 0.094 | 0.015 | 0.094 | Interferon inducer | |||
| 0.145 | 0.067 | 0.145 | MAP3K9 inhibitor | |||
| 0.173 | 0.097 | 0.865 | Psychostimulant | 0.48 0.013 CHEMBL1232305 0.445 0.016 CHEMBL1232161 0.865 0.003 CHEMBL3638310 0.603 0.006 CHEMBL3544876 0.391 0.024 CHEMBL1201384 | CHEMBL3638310 | |
| 0.094 | 0.019 | 0.094 | Phosphodiesterase VIII inhibitor | 0.071 0.051 CHEMBL1232305 | ||
| 0.095 | 0.025 | 0.095 | Protein kinase C alpha inhibitor | |||
| 0.074 | 0.005 | 0.151 | Hypoxanthine phosphoribosyltransferase inhibitor | 0.122 0.002 CHEMBL1232305 0.143 0.001 CHEMBL1232161 0.087 0.004 CHEMBL3638310 0.108 0.002 CHEMBL3544876 0.151 0.001 CHEMBL1201384 | CHEMBL1201384 | |
| 0.133 | 0.066 | 0.133 | Alpha-N-acetylglucosaminidase inhibitor | |||
| 0.221 | 0.155 | 0.221 | Interleukin 2 agonist | |||
| 0.072 | 0.007 | 0.574 | HCV NS5B polymerase inhibitor | 0.239 0.003 CHEMBL1232305 0.509 0.002 CHEMBL1232161 0.105 0.005 CHEMBL3638310 0.212 0.004 CHEMBL3544876 0.574 0.002 CHEMBL1201384 | CHEMBL1201384 | |
| 0.069 | 0.005 | 0.091 | Guanylate cyclase inhibitor | 0.084 0.002 CHEMBL1232305 0.09 0.002 CHEMBL1232161 0.067 0.006 CHEMBL3638310 0.078 0.003 CHEMBL3544876 0.091 0.001 CHEMBL1201384 | CHEMBL1201384 | |
| 0.109 | 0.049 | 0.109 | Protein kinase C mu inhibitor | |||
| 0.107 | 0.047 | 0.107 | Protein kinase C delta inhibitor | |||
| 0.077 | 0.023 | 0.247 | Acyl-CoA dehydrogenase inhibitor | 0.212 0.004 CHEMBL1232305 0.245 0.003 CHEMBL1232161 0.21 0.005 CHEMBL3638310 0.247 0.003 CHEMBL3544876 0.235 0.004 CHEMBL1201384 | CHEMBL3544876 | |
| 0.055 | 0.003 | 0.055 | Thymidine kinase (Herpes simplex virus 1) inhibitor | 0.048 0.004 CHEMBL1232305 0.032 0.009 CHEMBL1232161 0.03 0.011 CHEMBL1201384 | ||
| 0.066 | 0.017 | 0.467 | Purinergic P2Y antagonist | 0.353 0.003 CHEMBL1232305 0.441 0.002 CHEMBL1232161 0.294 0.003 CHEMBL3638310 0.377 0.003 CHEMBL3544876 0.467 0.002 CHEMBL1201384 | CHEMBL1201384 | |
| 0.075 | 0.028 | 0.26 | Purinergic P2X1 antagonist | 0.208 0.003 CHEMBL1232305 0.246 0.002 CHEMBL1232161 0.102 0.016 CHEMBL3638310 0.148 0.007 CHEMBL3544876 0.26 0.002 CHEMBL1201384 | CHEMBL1201384 | |
| 0.053 | 0.006 | 0.129 | Adenosine kinase inhibitor | 0.081 0.004 CHEMBL1232305 0.114 0.003 CHEMBL1232161 0.04 0.007 CHEMBL3638310 0.058 0.005 CHEMBL3544876 0.129 0.003 CHEMBL1201384 | CHEMBL1201384 | |
| 0.074 | 0.027 | 0.074 | Protein kinase C eta inhibitor | |||
| 0.047 | 0.002 | 0.047 | Isoleucine-tRNA ligase inhibitor | 0.026 0.009 CHEMBL1232305 | ||
| 0.135 | 0.091 | 0.135 | Adenylate cyclase stimulant | 0.128 0.106 CHEMBL1232305 | ||
| 0.134 | 0.091 | 0.134 | NOS3 expression enhancer | |||
| 0.054 | 0.011 | 0.513 | RNA-directed RNA polymerase inhibitor | 0.141 0.004 CHEMBL1232305 0.449 0.002 CHEMBL1232161 0.08 0.007 CHEMBL3638310 0.133 0.004 CHEMBL3544876 0.513 0.002 CHEMBL1201384 | CHEMBL1201384 | |
| 0.107 | 0.067 | 0.107 | Protein kinase C gamma inhibitor | |||
| 0.043 | 0.007 | 0.043 | Adenosine A1 receptor agonist | 0.038 0.008 CHEMBL1232305 0.032 0.01 CHEMBL1232161 0.027 0.014 CHEMBL3638310 0.03 0.012 CHEMBL3544876 0.031 0.011 CHEMBL1201384 | ||
| 0.06 | 0.025 | 0.238 | Phosphorylase inhibitor | 0.148 0.007 CHEMBL1232305 0.226 0.004 CHEMBL1232161 0.082 0.016 CHEMBL3638310 0.121 0.01 CHEMBL3544876 0.238 0.004 CHEMBL1201384 | CHEMBL1201384 | |
| 0.036 | 0.004 | 0.036 | Thymidine kinase (Herpes simplex virus 2) inhibitor | |||
| 0.046 | 0.016 | 0.046 | Antibiotic Aminoglycoside-like | 0.034 0.028 CHEMBL1232305 0.035 0.028 CHEMBL3544876 | ||
| 0.033 | 0.004 | 0.522 | Purinergic receptor agonist | 0.11 0.001 CHEMBL1232305 0.351 0.001 CHEMBL1232161 0.162 0.001 CHEMBL3638310 0.152 0.001 CHEMBL3544876 0.522 0.001 CHEMBL1201384 | CHEMBL1201384 | |
| 0.033 | 0.004 | 0.522 | Purinergic P2 agonist | 0.11 0.001 CHEMBL1232305 0.351 0.001 CHEMBL1232161 0.162 0.001 CHEMBL3638310 0.152 0.001 CHEMBL3544876 0.522 0.001 CHEMBL1201384 | CHEMBL1201384 | |
| 0.059 | 0.03 | 0.065 | Adenine nucleotide translocase inhibitor | 0.065 0.02 CHEMBL1232305 0.059 0.029 CHEMBL1232161 0.054 0.044 CHEMBL3544876 0.058 0.033 CHEMBL1201384 | CHEMBL1232305 | |
| 0.025 | 0.001 | 0.215 | Purinergic P2Y2 agonist | 0.083 0 CHEMBL1232305 0.169 0 CHEMBL1232161 0.04 0.001 CHEMBL3638310 0.047 0.001 CHEMBL3544876 0.215 0 CHEMBL1201384 | CHEMBL1201384 | |
| 0.063 | 0.04 | 0.14 | HIV-1 integrase (Strand Transfer) inhibitor | 0.14 0.014 CHEMBL1232305 0.082 0.03 CHEMBL1232161 0.056 0.044 CHEMBL3544876 0.074 0.034 CHEMBL1201384 | CHEMBL1232305 | |
| 0.028 | 0.004 | 0.513 | Purinergic P2Y agonist | 0.101 0.001 CHEMBL1232305 0.331 0.001 CHEMBL1232161 0.149 0.001 CHEMBL3638310 0.14 0.001 CHEMBL3544876 0.513 0.001 CHEMBL1201384 | CHEMBL1201384 | |
| 0.039 | 0.016 | 0.208 | Purinergic P2Y2 antagonist | 0.147 0.003 CHEMBL1232305 0.195 0.002 CHEMBL1232161 0.168 0.002 CHEMBL3638310 0.168 0.002 CHEMBL3544876 0.208 0.002 CHEMBL1201384 | CHEMBL1201384 | |
| 0.117 | 0.096 | 0.117 | Protein kinase stimulant | |||
| 0.132 | 0.111 | 0.361 | Heat shock protein 70 antagonist | 0.191 0.008 CHEMBL1232305 0.316 0.003 CHEMBL1232161 0.156 0.033 CHEMBL3638310 0.202 0.006 CHEMBL3544876 0.361 0.003 CHEMBL1201384 | CHEMBL1201384 | |
| 0.063 | 0.044 | 0.134 | HIV-1 integrase (3'-Processing) inhibitor | 0.134 0.016 CHEMBL1232305 0.082 0.033 CHEMBL1232161 0.058 0.049 CHEMBL3544876 0.074 0.037 CHEMBL1201384 | CHEMBL1232305 | |
| 0.023 | 0.005 | 0.133 | Purinergic P2Y1 agonist | 0.085 0.001 CHEMBL1232305 0.122 0.001 CHEMBL1232161 0.051 0.002 CHEMBL3638310 0.065 0.002 CHEMBL3544876 0.133 0.001 CHEMBL1201384 | CHEMBL1201384 | |
| 0.072 | 0.055 | 0.072 | S-adenosyl-L-methionine decarboxylase inhibitor | |||
| 0.02 | 0.008 | 0.02 | Adenosine A2 receptor agonist | |||
| 0.029 | 0.018 | 0.288 | Purinergic P2X agonist | 0.119 0.003 CHEMBL1232305 0.225 0.001 CHEMBL1232161 0.129 0.002 CHEMBL3638310 0.145 0.002 CHEMBL3544876 0.288 0.001 CHEMBL1201384 | CHEMBL1201384 | |
| 0.019 | 0.008 | 0.019 | Adenosine A2a receptor agonist | |||
| 0.017 | 0.007 | 0.017 | Adenosine A2b receptor agonist | |||
| 0.029 | 0.019 | 0.029 | Purinergic P2Y15 antagonist | |||
| 0.135 | 0.126 | 0.135 | Hepatoprotectant | |||
| 0.017 | 0.008 | 0.017 | S-adenosyl-L-homocysteine hydrolase inhibitor | |||
| 0.018 | 0.01 | 0.018 | Adenosine A3 receptor agonist | |||
| 0.007 | 0.001 | 0.085 | Purinergic P2Y6 agonist | 0.03 0 CHEMBL1232305 0.066 0 CHEMBL1232161 0.013 0.001 CHEMBL3638310 0.018 0 CHEMBL3544876 0.085 0 CHEMBL1201384 | CHEMBL1201384 | |
| 0.06 | 0.054 | 0.117 | Carbonic anhydrase V inhibitor | 0.117 0.022 CHEMBL1232305 | CHEMBL1232305 | |
| 0.064 | 0.061 | 0.064 | Protein kinase C beta inhibitor | |||
| 0.06 | 0.059 | 0.06 | Carbonic anhydrase VA inhibitor | |||
| 0.004 | 0.003 | 0.254 | Purinergic P2Y4 agonist | 0.018 0.001 CHEMBL1232305 0.101 0.001 CHEMBL1232161 0.023 0.001 CHEMBL3638310 0.03 0.001 CHEMBL3544876 0.254 0 CHEMBL1201384 | CHEMBL1201384 | |
| 0.017 | 0.016 | 0.03 | Methylmalonyl-CoA mutase inhibitor | 0.026 0.004 CHEMBL1232305 0.03 0.002 CHEMBL1232161 0.024 0.005 CHEMBL3638310 0.028 0.003 CHEMBL3544876 0.028 0.003 CHEMBL1201384 | CHEMBL1232161 | |
| 0.011 | 0.01 | 0.016 | Purine nucleoside phosphorylase inhibitor | 0.013 0.007 CHEMBL1232305 0.016 0.004 CHEMBL1232161 0.011 0.01 CHEMBL3544876 0.014 0.005 CHEMBL1201384 | CHEMBL1232161 | |
| 0.013 | 0.023 | 0.333 | Purinergic P2T antagonist | 0.09 0.005 CHEMBL1232305 0.251 0.004 CHEMBL1232161 0.131 0.004 CHEMBL3638310 0.117 0.004 CHEMBL3544876 0.333 0.003 CHEMBL1201384 | CHEMBL1201384 | |
| 0.015 | 0.028 | 0.268 | Purinergic P2Y12 antagonist | 0.083 0.004 CHEMBL1232305 0.213 0.004 CHEMBL1232161 0.088 0.004 CHEMBL3638310 0.102 0.004 CHEMBL3544876 0.268 0.003 CHEMBL1201384 | CHEMBL1201384 | |
| 0.013 | 0.026 | 0.076 | Inosine monophosphate dehydrogenase 1 inhibitor | 0.058 0.004 CHEMBL1232305 0.076 0.003 CHEMBL1232161 0.05 0.004 CHEMBL3638310 0.06 0.004 CHEMBL3544876 0.072 0.003 CHEMBL1201384 | CHEMBL1232161 | |
| 0.046 | 0.064 | 0.288 | Purinergic P2X2 antagonist | 0.221 0.004 CHEMBL1232305 0.267 0.003 CHEMBL1232161 0.214 0.004 CHEMBL3638310 0.229 0.004 CHEMBL3544876 0.288 0.002 CHEMBL1201384 | CHEMBL1201384 | |
| 0.039 | 0.056 | 0.065 | Glucose-6-phosphate isomerase inhibitor | 0.065 0.015 CHEMBL1232305 0.045 0.038 CHEMBL1232161 | CHEMBL1232305 | |
| 0.033 | 0.058 | 0.076 | AICAR transformylase inhibitor | 0.076 0.008 CHEMBL1232305 0.045 0.03 CHEMBL1232161 0.04 0.038 CHEMBL1201384 | CHEMBL1232305 | |
| 0.192 | 0.226 | 0.275 | Calcium channel activator | 0.275 0.118 CHEMBL1232305 0.24 0.159 CHEMBL1232161 0.226 0.177 CHEMBL3544876 0.208 0.201 CHEMBL1201384 | CHEMBL1232305 | |
| 0.008 | 0.045 | 0.097 | Purinergic P2Y1 antagonist | 0.08 0.003 CHEMBL1232305 0.088 0.003 CHEMBL1232161 0.061 0.003 CHEMBL3638310 0.063 0.003 CHEMBL3544876 0.097 0.003 CHEMBL1201384 | CHEMBL1201384 | |
| 0.039 | 0.078 | 0.156 | Antiviral (Hepatitis D) | 0.081 0.008 CHEMBL1232305 0.132 0.004 CHEMBL1232161 0.09 0.005 CHEMBL3638310 0.096 0.005 CHEMBL3544876 0.156 0.003 CHEMBL1201384 | CHEMBL1201384 | |
| 0.073 | 0.122 | 0.123 | Toll-Like receptor 3 antagonist | 0.123 0.027 CHEMBL3544876 | CHEMBL3544876 | |
| 0.07 | 0.122 | 0.133 | Anabolic | 0.109 0.051 CHEMBL1232305 0.127 0.033 CHEMBL1232161 0.133 0.029 CHEMBL3638310 0.11 0.05 CHEMBL3544876 0.133 0.028 CHEMBL1201384 | CHEMBL1201384 | |
| 0.064 | 0.121 | 0.274 | Phosphodiesterase I inhibitor | 0.143 0.019 CHEMBL1232305 0.246 0.007 CHEMBL1232161 0.094 0.052 CHEMBL3638310 0.118 0.028 CHEMBL3544876 0.274 0.005 CHEMBL1201384 | CHEMBL1201384 | |
| 0.067 | 0.13 | 0.092 | Hematopoietic | 0.092 0.046 CHEMBL1232305 0.083 0.064 CHEMBL3544876 | CHEMBL1232305 | |
| 0.164 | 0.229 | 0.396 | Antithrombotic | 0.28 0.103 CHEMBL1232305 0.236 0.138 CHEMBL1232161 0.396 0.05 CHEMBL3638310 0.389 0.052 CHEMBL3544876 0.203 0.174 CHEMBL1201384 | CHEMBL3638310 | |
| 0.062 | 0.127 | 0.126 | Triose-phosphate isomerase inhibitor | 0.126 0.029 CHEMBL1232305 | CHEMBL1232305 | |
| 0.076 | 0.155 | 0.324 | Aldehyde dehydrogenase inhibitor | 0.214 0.025 CHEMBL1232305 0.324 0.009 CHEMBL1232161 0.121 0.07 CHEMBL3638310 0.187 0.031 CHEMBL3544876 0.281 0.014 CHEMBL1201384 | CHEMBL1232161 | |
| 0.018 | 0.117 | 0.073 | Geranyltranstransferase inhibitor | 0.043 0.032 CHEMBL1232305 0.073 0.006 CHEMBL1232161 0.061 0.013 CHEMBL3638310 0.064 0.011 CHEMBL3544876 0.067 0.009 CHEMBL1201384 | CHEMBL1232161 | |
| 0.006 | 0.107 | 0.05 | Inosine monophosphate dehydrogenase 2 inhibitor | 0.041 0.005 CHEMBL1232305 0.05 0.004 CHEMBL1232161 0.039 0.005 CHEMBL1201384 | CHEMBL1232161 | |
| 0.116 | 0.217 | 0.322 | Vasodilator | 0.159 0.144 CHEMBL1232305 0.224 0.087 CHEMBL1232161 0.322 0.041 CHEMBL3638310 0.28 0.055 CHEMBL3544876 0.243 0.073 CHEMBL1201384 | CHEMBL3638310 | |
| 0.015 | 0.12 | 0.091 | Inosine monophosphate dehydrogenase inhibitor | 0.074 0.008 CHEMBL1232305 0.091 0.005 CHEMBL1232161 0.082 0.006 CHEMBL3544876 0.069 0.008 CHEMBL1201384 | CHEMBL1232161 | |
| 0.001 | 0.113 | 0.017 | Mannitol 2-dehydrogenase inhibitor | 0.017 0.003 CHEMBL1232305 0.009 0.005 CHEMBL1232161 0.01 0.004 CHEMBL3638310 0.012 0.004 CHEMBL3544876 0.009 0.005 CHEMBL1201384 | CHEMBL1232305 | |
| 0.071 | 0.21 | 0.21 | Acetylcholine M1 receptor antagonist | 0.125 0.102 CHEMBL1232161 0.21 0.038 CHEMBL3638310 0.139 0.085 CHEMBL1201384 | CHEMBL3638310 | |
| 0.04 | 0.185 | 0.104 | Alcohol dehydrogenase inhibitor | 0.088 0.066 CHEMBL1232305 0.104 0.048 CHEMBL1232161 0.089 0.066 CHEMBL3544876 0.089 0.065 CHEMBL1201384 | CHEMBL1232161 | |
| 0.089 | 0.3 | 0.24 | Phospholipase C inhibitor | 0.213 0.037 CHEMBL1232305 0.143 0.122 CHEMBL1232161 0.24 0.027 CHEMBL3638310 0.19 0.051 CHEMBL3544876 | CHEMBL3638310 | |
| 0.019 | 0.251 | 0.15 | Purinergic P2X4 antagonist | 0.07 0.009 CHEMBL1232305 0.119 0.004 CHEMBL1232161 0.15 0.004 CHEMBL1201384 | CHEMBL1201384 | |
| 0.065 | 0.309 | 0.229 | Platelet antagonist | 0.207 0.096 CHEMBL1232161 0.198 0.102 CHEMBL3638310 0.229 0.082 CHEMBL3544876 0.223 0.086 CHEMBL1201384 | CHEMBL3544876 | |
| 0.064 | 0.311 | 0.231 | Spasmolytic | 0.231 0.1 CHEMBL3638310 | CHEMBL3638310 | |
| 0.02 | 0.285 | 0.079 | NAD(P)H dehydrogenase (quinone) inhibitor | 0.079 0.052 CHEMBL1232161 0.067 0.064 CHEMBL1201384 | CHEMBL1232161 | |
| 0.054 | 0.326 | 0.106 | Folate antagonist | 0.106 0.054 CHEMBL1232305 0.092 0.082 CHEMBL3638310 0.101 0.063 CHEMBL3544876 | CHEMBL1232305 | |
| 0.013 | 0.31 | 0.338 | Purinergic P2 antagonist | 0.217 0.006 CHEMBL1232305 0.301 0.005 CHEMBL1232161 0.164 0.009 CHEMBL3638310 0.199 0.007 CHEMBL3544876 0.338 0.004 CHEMBL1201384 | CHEMBL1201384 | |
| 0.013 | 0.312 | 0.036 | Toll-Like receptor 4 agonist | 0.036 0.007 CHEMBL1232305 0.029 0.012 CHEMBL1232161 0.032 0.009 CHEMBL3638310 0.035 0.007 CHEMBL3544876 0.029 0.014 CHEMBL1201384 | CHEMBL1232305 | |
| 0.039 | 0.339 | 0.446 | Pyruvate kinase inhibitor | 0.316 0.044 CHEMBL1232305 0.403 0.02 CHEMBL1232161 0.194 0.084 CHEMBL3544876 0.446 0.014 CHEMBL1201384 | CHEMBL1201384 | |
| 0.024 | 0.373 | 0.08 | Telomerase inhibitor | 0.08 0.045 CHEMBL3638310 | CHEMBL3638310 | |
| 0.033 | 0.427 | 0.12 | Mannose-6-phosphate isomerase inhibitor | 0.12 0.101 CHEMBL1232305 | CHEMBL1232305 | |
| 0.031 | 0.442 | 0.081 | Thioredoxin reductase inhibitor | 0.081 0.059 CHEMBL3638310 | CHEMBL3638310 | |
| 0.035 | 0.461 | 0.157 | Antimitotic | 0.157 0.115 CHEMBL1232305 | CHEMBL1232305 | |
| 0.029 | 0.472 | 0.097 | Toll-Like receptor 4 antagonist | 0.097 0.074 CHEMBL3544876 | CHEMBL3544876 | |
| 0.027 | 0.528 | 0.164 | Platelet aggregation inhibitor | 0.164 0.112 CHEMBL3638310 | CHEMBL3638310 | |
| 0.031 | 0.532 | 0.119 | Insulin secretagoues | 0.119 0.113 CHEMBL1201384 | CHEMBL1201384 | |
| 0.005 | 0.569 | 0.043 | Purinergic P2X3 antagonist | 0.035 0.023 CHEMBL1232161 0.043 0.014 CHEMBL1201384 | CHEMBL1201384 | |
| 0.049 | 0.631 | 0.202 | Sphingosine 1-phosphate receptor 2 agonist | 0.202 0.011 CHEMBL1232305 0.117 0.06 CHEMBL1232161 0.124 0.049 CHEMBL3638310 0.141 0.031 CHEMBL3544876 0.112 0.071 CHEMBL1201384 | CHEMBL1232305 | |
| 0.005 | 0.654 | 0.037 | Growth factor receptor-bound protein 2 antagonist | 0.037 0.019 CHEMBL1232305 0.035 0.024 CHEMBL1232161 0.034 0.026 CHEMBL3544876 0.034 0.026 CHEMBL1201384 | CHEMBL1232305 | |
| 0.013 | 0.68 | 0.088 | Acetylcholine M3 receptor agonist | 0.088 0.053 CHEMBL3638310 | CHEMBL3638310 | |
| 0.01 | 0.731 | 0.06 | Autotaxin inhibitor | 0.06 0.028 CHEMBL1232305 | CHEMBL1232305 | |
| 0.005 | 0.84 | 0.062 | Sphingosine 1-phosphate receptor 5 agonist | 0.062 0.023 CHEMBL1232305 | CHEMBL1232305 | |
| 0.002 | 0.882 | 0.085 | Sphingosine 1-phosphate receptor 3 agonist | 0.085 0.008 CHEMBL1232305 0.029 0.028 CHEMBL3638310 0.055 0.014 CHEMBL3544876 | CHEMBL1232305 | |
| 0.007 | 0.901 | 0.128 | Bone formation stimulant | 0.128 0.079 CHEMBL1232305 | CHEMBL1232305 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |