Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.9680.0030.968Immunomodulator

0.779 0.005 CHEMBL731

0.906 0.004 CHEMBL87658

0.8 0.004 CHEMBL3544546

0.697 0.005 CHEMBL3706538

0.644 0.008 CHEMBL3706539

0.428 0.037 CHEMBL3706542

0.279 0.095 CHEMBL1213529

0.519 0.021 CHEMBL3706541

0.9320.0020.958DNA damaging

0.958 0.001 CHEMBL731

0.898 0.002 CHEMBL87658

0.243 0.084 CHEMBL506976

0.87 0.003 CHEMBL3544546

0.876 0.003 CHEMBL1593

0.858 0.003 CHEMBL3706538

0.93 0.002 CHEMBL3544547

0.804 0.004 CHEMBL525

0.947 0.002 CHEMBL3706540

0.938 0.002 CHEMBL3706539

0.257 0.077 CHEMBL1213529

0.608 0.008 CHEMBL913

0.307 0.054 CHEMBL3706541

CHEMBL731
0.8990.0010.96Alkylator

0.951 0.001 CHEMBL731

0.862 0.001 CHEMBL87658

0.232 0.019 CHEMBL506976

0.748 0.002 CHEMBL3544546

0.831 0.002 CHEMBL1593

0.71 0.003 CHEMBL3706538

0.875 0.001 CHEMBL3544547

0.162 0.041 CHEMBL721

0.836 0.002 CHEMBL525

0.892 0.001 CHEMBL3706540

0.96 0.001 CHEMBL3706539

0.223 0.021 CHEMBL3706542

0.159 0.042 CHEMBL1213529

0.459 0.005 CHEMBL913

0.722 0.003 CHEMBL3706541

CHEMBL3706539
0.860.0020.86P-glycoprotein inhibitor

0.64 0.004 CHEMBL731

0.658 0.004 CHEMBL87658

0.692 0.004 CHEMBL3544546

0.687 0.004 CHEMBL3706538

0.281 0.033 CHEMBL3706539

0.161 0.1 CHEMBL913

0.860.010.86Apoptosis agonist

0.646 0.04 CHEMBL731

0.545 0.061 CHEMBL87658

0.249 0.215 CHEMBL506976

0.619 0.045 CHEMBL3544546

0.492 0.077 CHEMBL1593

0.778 0.019 CHEMBL3706538

0.542 0.062 CHEMBL3544547

0.675 0.035 CHEMBL721

0.42 0.104 CHEMBL525

0.58 0.054 CHEMBL3706540

0.548 0.061 CHEMBL3706539

0.586 0.052 CHEMBL1213529

0.541 0.063 CHEMBL913

0.235 0.231 CHEMBL3706541

0.8350.0030.841Immunosuppressant

0.836 0.003 CHEMBL731

0.841 0.003 CHEMBL87658

0.764 0.004 CHEMBL3544546

0.363 0.08 CHEMBL1593

0.79 0.004 CHEMBL3706538

0.405 0.06 CHEMBL3544547

0.285 0.125 CHEMBL721

0.451 0.047 CHEMBL525

0.412 0.058 CHEMBL3706540

0.615 0.011 CHEMBL3706539

0.3 0.115 CHEMBL3706542

0.414 0.058 CHEMBL1213529

0.4 0.063 CHEMBL913

0.325 0.1 CHEMBL3706541

CHEMBL87658
0.8110.0030.854DNA synthesis inhibitor

0.808 0.003 CHEMBL731

0.743 0.004 CHEMBL87658

0.431 0.018 CHEMBL506976

0.677 0.005 CHEMBL3544546

0.354 0.029 CHEMBL1593

0.659 0.005 CHEMBL3706538

0.389 0.023 CHEMBL3544547

0.369 0.026 CHEMBL721

0.366 0.027 CHEMBL525

0.377 0.025 CHEMBL3706540

0.854 0.003 CHEMBL3706539

0.287 0.048 CHEMBL3706542

0.367 0.027 CHEMBL1213529

0.447 0.017 CHEMBL913

0.239 0.074 CHEMBL3706541

CHEMBL3706539
0.7860.0050.786Angiogenesis inhibitor

0.247 0.125 CHEMBL731

0.219 0.149 CHEMBL87658

0.326 0.081 CHEMBL3544546

0.474 0.035 CHEMBL3706538

0.302 0.091 CHEMBL721

0.266 0.112 CHEMBL1213529

0.6420.0060.642Antiamyloidogenic

0.181 0.113 CHEMBL87658

0.241 0.075 CHEMBL3544546

0.331 0.043 CHEMBL3706538

0.5740.020.699Immunostimulant

0.437 0.04 CHEMBL731

0.387 0.053 CHEMBL87658

0.21 0.114 CHEMBL506976

0.44 0.039 CHEMBL3544546

0.415 0.045 CHEMBL3706538

0.196 0.123 CHEMBL3544547

0.337 0.068 CHEMBL721

0.699 0.008 CHEMBL3706539

0.65 0.012 CHEMBL3706542

0.342 0.067 CHEMBL1213529

0.228 0.105 CHEMBL913

0.607 0.016 CHEMBL3706541

CHEMBL3706539
0.390.0040.995ErbB-2 antagonist

0.135 0.023 CHEMBL731

0.091 0.04 CHEMBL87658

0.183 0.011 CHEMBL3544546

0.989 0.002 CHEMBL1593

0.211 0.009 CHEMBL3706538

0.975 0.002 CHEMBL3544547

0.981 0.002 CHEMBL525

0.995 0.002 CHEMBL3706540

0.15 0.019 CHEMBL913

0.096 0.037 CHEMBL3706541

CHEMBL3706540
0.3150.0030.315Bcl2 antagonist

0.171 0.005 CHEMBL731

0.19 0.004 CHEMBL87658

0.203 0.004 CHEMBL3544546

0.204 0.004 CHEMBL3706538

0.136 0.007 CHEMBL3706539

0.2620.0130.654Epidermal growth factor receptor kinase inhibitor

0.132 0.061 CHEMBL3544546

0.564 0.004 CHEMBL1593

0.153 0.046 CHEMBL3706538

0.473 0.005 CHEMBL3544547

0.166 0.039 CHEMBL721

0.472 0.005 CHEMBL525

0.654 0.004 CHEMBL3706540

0.171 0.037 CHEMBL1213529

0.137 0.058 CHEMBL913

CHEMBL3706540
0.3050.2110.757Antiinflammatory

0.353 0.17 CHEMBL721

0.757 0.021 CHEMBL1213529

CHEMBL1213529
0.0790.0290.241Carbamoyl phosphate synthetase inhibitor

0.091 0.023 CHEMBL731

0.079 0.029 CHEMBL87658

0.237 0.006 CHEMBL506976

0.085 0.026 CHEMBL3544546

0.083 0.027 CHEMBL1593

0.123 0.015 CHEMBL3706538

0.231 0.006 CHEMBL3544547

0.109 0.018 CHEMBL721

0.157 0.01 CHEMBL525

0.155 0.011 CHEMBL3706540

0.116 0.017 CHEMBL3706542

0.241 0.006 CHEMBL1213529

0.228 0.006 CHEMBL913

0.102 0.02 CHEMBL3706541

CHEMBL1213529
0.090.060.546Triose-phosphate isomerase inhibitor

0.081 0.074 CHEMBL731

0.09 0.06 CHEMBL87658

0.546 0.002 CHEMBL506976

0.099 0.049 CHEMBL3544546

0.174 0.015 CHEMBL1593

0.147 0.021 CHEMBL3706538

0.272 0.006 CHEMBL3544547

0.402 0.003 CHEMBL721

0.195 0.011 CHEMBL525

0.17 0.015 CHEMBL3706540

0.466 0.003 CHEMBL1213529

0.293 0.005 CHEMBL913

CHEMBL506976
0.0660.0590.221Aminopeptidase I inhibitor

0.066 0.059 CHEMBL87658

0.141 0.014 CHEMBL506976

0.083 0.039 CHEMBL3706538

0.12 0.019 CHEMBL3544547

0.082 0.04 CHEMBL721

0.118 0.02 CHEMBL525

0.089 0.035 CHEMBL3706540

0.119 0.02 CHEMBL3706539

0.221 0.005 CHEMBL3706542

0.154 0.012 CHEMBL1213529

0.175 0.009 CHEMBL913

0.202 0.007 CHEMBL3706541

CHEMBL3706542
0.0860.0790.461UDP-glucose 4-epimerase inhibitor

0.102 0.058 CHEMBL731

0.086 0.079 CHEMBL87658

0.461 0.004 CHEMBL506976

0.105 0.055 CHEMBL3544546

0.144 0.031 CHEMBL1593

0.172 0.023 CHEMBL3706538

0.108 0.053 CHEMBL3544547

0.33 0.009 CHEMBL721

0.186 0.02 CHEMBL525

0.129 0.038 CHEMBL3706540

0.237 0.014 CHEMBL1213529

0.31 0.01 CHEMBL913

CHEMBL506976
0.0650.0680.469NAD(P)H dehydrogenase (quinone) inhibitor

0.116 0.03 CHEMBL506976

0.314 0.004 CHEMBL1593

0.11 0.033 CHEMBL3706538

0.447 0.003 CHEMBL3544547

0.453 0.003 CHEMBL525

0.469 0.003 CHEMBL3706540

0.09 0.044 CHEMBL1213529

0.128 0.026 CHEMBL913

CHEMBL3706540
0.0330.0540.136Antimetabolite

0.056 0.028 CHEMBL506976

0.041 0.039 CHEMBL1593

0.062 0.025 CHEMBL3706538

0.082 0.019 CHEMBL3544547

0.051 0.03 CHEMBL721

0.051 0.031 CHEMBL525

0.061 0.025 CHEMBL3706540

0.09 0.018 CHEMBL3706539

0.136 0.013 CHEMBL3706542

0.128 0.013 CHEMBL1213529

0.12 0.014 CHEMBL913

0.1 0.016 CHEMBL3706541

CHEMBL3706542
0.0150.0360.078Hypoxanthine phosphoribosyltransferase inhibitor

0.067 0.006 CHEMBL506976

0.035 0.014 CHEMBL1593

0.027 0.02 CHEMBL3706538

0.032 0.016 CHEMBL3544547

0.041 0.012 CHEMBL721

0.039 0.012 CHEMBL525

0.046 0.01 CHEMBL3706540

0.034 0.015 CHEMBL1213529

0.078 0.005 CHEMBL913

CHEMBL913
0.0570.0840.509Glutamate dehydrogenase inhibitor

0.212 0.009 CHEMBL506976

0.094 0.034 CHEMBL3706538

0.169 0.013 CHEMBL3544547

0.175 0.012 CHEMBL721

0.127 0.021 CHEMBL525

0.085 0.04 CHEMBL3706540

0.093 0.035 CHEMBL3706539

0.296 0.006 CHEMBL3706542

0.509 0.003 CHEMBL1213529

0.203 0.01 CHEMBL913

0.22 0.009 CHEMBL3706541

CHEMBL1213529
0.0120.0490.029Purinergic P2X agonist

0.029 0.018 CHEMBL525

CHEMBL525
0.0330.080.171Glucose-6-phosphate isomerase inhibitor

0.117 0.004 CHEMBL506976

0.051 0.028 CHEMBL1593

0.047 0.034 CHEMBL3706538

0.067 0.014 CHEMBL3544547

0.127 0.003 CHEMBL721

0.051 0.028 CHEMBL525

0.052 0.027 CHEMBL3706540

0.171 0.002 CHEMBL1213529

0.061 0.018 CHEMBL913

CHEMBL1213529
0.0250.0780.152Ribonucleoside-diphosphate reductase inhibitor

0.061 0.034 CHEMBL506976

0.045 0.044 CHEMBL3706538

0.047 0.043 CHEMBL3544547

0.05 0.041 CHEMBL721

0.081 0.024 CHEMBL3706539

0.152 0.011 CHEMBL3706542

0.092 0.021 CHEMBL1213529

0.069 0.029 CHEMBL913

0.084 0.023 CHEMBL3706541

CHEMBL3706542
0.0240.0780.148Ribonucleotide reductase inhibitor

0.062 0.035 CHEMBL506976

0.046 0.045 CHEMBL3706538

0.048 0.044 CHEMBL3544547

0.049 0.043 CHEMBL721

0.082 0.026 CHEMBL3706539

0.148 0.012 CHEMBL3706542

0.092 0.023 CHEMBL1213529

0.071 0.031 CHEMBL913

0.089 0.024 CHEMBL3706541

CHEMBL3706542
0.2180.2730.575MAP kinase 1 inhibitor

0.575 0.027 CHEMBL731

0.246 0.239 CHEMBL3706538

CHEMBL731
0.1010.1570.253Arachidonic acid antagonist

0.226 0.014 CHEMBL506976

0.176 0.059 CHEMBL3706538

0.177 0.057 CHEMBL3544547

0.209 0.025 CHEMBL721

0.158 0.079 CHEMBL525

0.159 0.078 CHEMBL3706540

0.253 0.005 CHEMBL1213529

0.214 0.021 CHEMBL913

CHEMBL1213529
0.0740.1320.41GABA C receptor antagonist

0.149 0.03 CHEMBL506976

0.137 0.038 CHEMBL3706538

0.257 0.006 CHEMBL721

0.125 0.048 CHEMBL525

0.41 0.003 CHEMBL1213529

0.208 0.011 CHEMBL913

CHEMBL1213529
0.0770.140.322Bone formation stimulant

0.187 0.039 CHEMBL3706538

0.146 0.062 CHEMBL3544547

0.156 0.054 CHEMBL721

0.322 0.015 CHEMBL525

0.168 0.047 CHEMBL3706540

0.138 0.069 CHEMBL3706539

0.197 0.037 CHEMBL3706542

0.122 0.084 CHEMBL1213529

0.316 0.015 CHEMBL3706541

CHEMBL525
0.1190.1840.724Succinate dehydrogenase inhibitor

0.564 0.003 CHEMBL506976

0.189 0.059 CHEMBL1593

0.173 0.076 CHEMBL3706538

0.249 0.023 CHEMBL3544547

0.471 0.003 CHEMBL721

0.168 0.083 CHEMBL525

0.188 0.059 CHEMBL3706540

0.156 0.101 CHEMBL3706542

0.724 0.002 CHEMBL1213529

0.32 0.008 CHEMBL913

CHEMBL1213529
0.0640.130.742GABA C receptor agonist

0.283 0.01 CHEMBL506976

0.114 0.054 CHEMBL3706538

0.164 0.029 CHEMBL3544547

0.355 0.007 CHEMBL721

0.11 0.057 CHEMBL525

0.093 0.075 CHEMBL3706542

0.742 0.002 CHEMBL1213529

0.374 0.006 CHEMBL913

CHEMBL1213529
0.0580.1260.552Glutathione S-transferase inhibitor

0.125 0.02 CHEMBL506976

0.212 0.005 CHEMBL1593

0.1 0.038 CHEMBL3706538

0.311 0.003 CHEMBL3544547

0.13 0.018 CHEMBL721

0.209 0.005 CHEMBL525

0.32 0.003 CHEMBL3706540

0.27 0.003 CHEMBL3706539

0.498 0.002 CHEMBL3706542

0.245 0.004 CHEMBL1213529

0.161 0.01 CHEMBL913

0.552 0.001 CHEMBL3706541

CHEMBL3706541
0.0610.1360.246NADH dehydrogenase inhibitor

0.148 0.018 CHEMBL506976

0.088 0.06 CHEMBL3706538

0.085 0.064 CHEMBL3544547

0.134 0.022 CHEMBL721

0.112 0.033 CHEMBL525

0.08 0.074 CHEMBL3706540

0.246 0.008 CHEMBL1213529

0.156 0.016 CHEMBL913

CHEMBL1213529
0.0030.0990.022Lysophosphatidic acid receptor 3 agonist

0.012 0.011 CHEMBL721

0.022 0.005 CHEMBL1213529

CHEMBL1213529
0.0070.1060.015Purinergic P2Y1 agonist

0.015 0.011 CHEMBL1213529

CHEMBL1213529
0.0110.110.024Methylmalonyl-CoA mutase inhibitor

0.022 0.006 CHEMBL506976

0.023 0.005 CHEMBL721

0.022 0.006 CHEMBL3706542

0.024 0.004 CHEMBL1213529

0.02 0.009 CHEMBL913

CHEMBL1213529
0.0230.1230.233Acyl-CoA dehydrogenase inhibitor

0.096 0.017 CHEMBL506976

0.055 0.037 CHEMBL3544547

0.153 0.009 CHEMBL721

0.063 0.031 CHEMBL525

0.093 0.018 CHEMBL3706542

0.233 0.004 CHEMBL1213529

0.123 0.012 CHEMBL913

0.08 0.022 CHEMBL3706541

CHEMBL1213529
0.0460.1510.648Aminopeptidase B inhibitor

0.24 0.014 CHEMBL506976

0.082 0.08 CHEMBL1593

0.089 0.073 CHEMBL3706538

0.143 0.041 CHEMBL3544547

0.155 0.035 CHEMBL721

0.148 0.039 CHEMBL525

0.095 0.068 CHEMBL3706540

0.243 0.014 CHEMBL3706539

0.648 0.002 CHEMBL3706542

0.196 0.022 CHEMBL1213529

0.217 0.018 CHEMBL913

0.354 0.006 CHEMBL3706541

CHEMBL3706542
0.0090.1170.027Antibiotic Anthracycline-like

0.021 0.01 CHEMBL506976

0.019 0.013 CHEMBL1213529

0.027 0.004 CHEMBL913

CHEMBL913
0.0650.180.713Alpha-N-acetylglucosaminidase inhibitor

0.655 0.003 CHEMBL506976

0.106 0.093 CHEMBL1593

0.133 0.066 CHEMBL3544547

0.638 0.004 CHEMBL721

0.11 0.088 CHEMBL525

0.105 0.095 CHEMBL3706540

0.235 0.026 CHEMBL3706542

0.713 0.003 CHEMBL1213529

0.414 0.008 CHEMBL913

CHEMBL1213529
0.0250.1420.394Phosphofructokinase-1 inhibitor

0.211 0.01 CHEMBL506976

0.059 0.058 CHEMBL1593

0.109 0.029 CHEMBL3544547

0.291 0.006 CHEMBL721

0.064 0.053 CHEMBL525

0.06 0.057 CHEMBL3706540

0.13 0.022 CHEMBL3706542

0.394 0.003 CHEMBL1213529

0.103 0.031 CHEMBL913

CHEMBL1213529
0.0490.170.258Prolactin inhibitor

0.197 0.009 CHEMBL506976

0.1 0.055 CHEMBL3706538

0.182 0.012 CHEMBL721

0.199 0.009 CHEMBL1213529

0.258 0.004 CHEMBL913

CHEMBL913
0.0170.1420.116Membrane dipeptidase inhibitor

0.049 0.016 CHEMBL506976

0.053 0.014 CHEMBL721

0.116 0.003 CHEMBL3706542

0.101 0.004 CHEMBL1213529

0.067 0.008 CHEMBL913

0.1 0.004 CHEMBL3706541

CHEMBL3706542
0.0110.140.041Vanilloid 2 agonist

0.024 0.021 CHEMBL506976

0.032 0.008 CHEMBL721

0.041 0.004 CHEMBL1213529

0.025 0.018 CHEMBL913

CHEMBL1213529
0.0520.1830.165Anabolic

0.144 0.021 CHEMBL506976

0.088 0.081 CHEMBL3706538

0.146 0.02 CHEMBL721

0.087 0.084 CHEMBL525

0.09 0.079 CHEMBL3706542

0.165 0.011 CHEMBL1213529

0.14 0.024 CHEMBL913

CHEMBL1213529
0.0140.1450.491Ornithine carbamoyltransferase inhibitor

0.104 0.015 CHEMBL506976

0.052 0.038 CHEMBL3544547

0.192 0.007 CHEMBL721

0.051 0.038 CHEMBL3706540

0.491 0.003 CHEMBL3706542

0.258 0.005 CHEMBL1213529

0.092 0.018 CHEMBL913

0.178 0.008 CHEMBL3706541

CHEMBL3706542
0.010.1440.345Fumarate hydratase inhibitor

0.047 0.015 CHEMBL506976

0.036 0.022 CHEMBL3544547

0.055 0.012 CHEMBL721

0.345 0.002 CHEMBL1213529

0.039 0.02 CHEMBL913

CHEMBL1213529
0.0020.1390.035Glutamate (mGluR6) agonist

0.035 0.003 CHEMBL1213529

CHEMBL1213529
0.0390.1770.072Lipocortins synthesis agonist

0.072 0.019 CHEMBL506976

0.064 0.029 CHEMBL913

CHEMBL506976
0.0060.1440.022Telomerase stimulant

0.017 0.013 CHEMBL506976

0.016 0.015 CHEMBL721

0.022 0.006 CHEMBL1213529

CHEMBL1213529
0.0230.170.222Mannitol-1-phosphate 5-dehydrogenase inhibitor

0.15 0.009 CHEMBL506976

0.052 0.046 CHEMBL3706538

0.222 0.006 CHEMBL721

0.055 0.041 CHEMBL525

0.205 0.006 CHEMBL1213529

0.076 0.022 CHEMBL913

CHEMBL721
0.010.1590.04Lysophosphatidic acid receptor 1 agonist

0.024 0.019 CHEMBL721

0.04 0.005 CHEMBL1213529

0.025 0.017 CHEMBL913

CHEMBL1213529
0.0210.1720.079Alpha-mannosidase inhibitor

0.079 0.012 CHEMBL506976

0.075 0.014 CHEMBL721

0.053 0.038 CHEMBL3706542

0.078 0.012 CHEMBL1213529

0.066 0.02 CHEMBL913

CHEMBL506976
0.1390.2910.44Tyrosine 3 hydroxylase inhibitor

0.294 0.036 CHEMBL506976

0.2 0.135 CHEMBL3544547

0.295 0.036 CHEMBL721

0.213 0.113 CHEMBL3706542

0.44 0.005 CHEMBL1213529

0.346 0.017 CHEMBL913

CHEMBL1213529
0.0610.2160.382Adenylate kinase inhibitor

0.263 0.009 CHEMBL506976

0.092 0.082 CHEMBL1593

0.12 0.043 CHEMBL3544547

0.355 0.004 CHEMBL721

0.112 0.052 CHEMBL525

0.303 0.007 CHEMBL3706542

0.382 0.004 CHEMBL1213529

0.159 0.023 CHEMBL913

0.192 0.016 CHEMBL3706541

CHEMBL1213529
0.0190.1810.113Glutamate (mGluR8) agonist

0.047 0.014 CHEMBL506976

0.051 0.011 CHEMBL721

0.041 0.02 CHEMBL3706542

0.113 0.003 CHEMBL1213529

0.04 0.023 CHEMBL913

0.036 0.03 CHEMBL3706541

CHEMBL1213529
0.0170.190.198Argininosuccinate synthase inhibitor

0.176 0.009 CHEMBL506976

0.051 0.046 CHEMBL3544547

0.168 0.01 CHEMBL721

0.149 0.011 CHEMBL3706542

0.198 0.008 CHEMBL1213529

0.08 0.025 CHEMBL913

0.05 0.047 CHEMBL3706541

CHEMBL1213529
0.0390.2130.14Glutamate (mGluR6) antagonist

0.079 0.026 CHEMBL506976

0.066 0.048 CHEMBL3544547

0.08 0.024 CHEMBL721

0.064 0.054 CHEMBL3706542

0.14 0.004 CHEMBL1213529

0.072 0.036 CHEMBL913

CHEMBL1213529
0.0110.1880.036Growth factor receptor-bound protein 2 antagonist

0.036 0.022 CHEMBL3706541

CHEMBL3706541
0.0120.190.059Dopamine D5 agonist

0.042 0.025 CHEMBL506976

0.039 0.029 CHEMBL721

0.049 0.018 CHEMBL1213529

0.059 0.012 CHEMBL913

CHEMBL913
0.0130.2030.067Mannosidase inhibitor

0.066 0.014 CHEMBL506976

0.063 0.015 CHEMBL721

0.067 0.013 CHEMBL1213529

0.053 0.023 CHEMBL913

CHEMBL1213529
0.1310.3230.2765 Hydroxytryptamine 3E antagonist

0.226 0.031 CHEMBL506976

0.177 0.113 CHEMBL3706538

0.234 0.025 CHEMBL721

0.187 0.088 CHEMBL1213529

0.276 0.008 CHEMBL913

CHEMBL913
0.0120.2150.063Metalloproteinase-3 inhibitor

0.063 0.022 CHEMBL3706542

CHEMBL3706542
0.0360.2430.2Creatine kinase inhibitor

0.13 0.034 CHEMBL506976

0.117 0.043 CHEMBL721

0.2 0.01 CHEMBL1213529

0.135 0.031 CHEMBL913

CHEMBL1213529
0.0430.2540.336GABA C receptor rho-1 antagonist

0.124 0.036 CHEMBL506976

0.232 0.005 CHEMBL721

0.099 0.063 CHEMBL525

0.336 0.003 CHEMBL1213529

0.173 0.014 CHEMBL913

CHEMBL1213529
0.0160.2280.335Biliverdin reductase inhibitor

0.096 0.02 CHEMBL506976

0.055 0.046 CHEMBL3544547

0.161 0.008 CHEMBL721

0.335 0.003 CHEMBL1213529

0.082 0.025 CHEMBL913

CHEMBL1213529
0.0030.2150.015Melatonin 2 antagonist

0.015 0.005 CHEMBL913

CHEMBL913
0.0030.2160.031Carbonic anhydrase VIII inhibitor

0.017 0.011 CHEMBL506976

0.016 0.013 CHEMBL721

0.031 0.004 CHEMBL1213529

0.018 0.01 CHEMBL913

CHEMBL1213529
0.0030.2160.031Carbonic anhydrase X inhibitor

0.017 0.011 CHEMBL506976

0.016 0.013 CHEMBL721

0.031 0.004 CHEMBL1213529

0.018 0.01 CHEMBL913

CHEMBL1213529
0.1040.3220.192Ca2+-transporting ATPase inhibitor

0.165 0.018 CHEMBL506976

0.17 0.013 CHEMBL721

0.192 0.004 CHEMBL1213529

0.156 0.03 CHEMBL913

CHEMBL1213529
0.0020.2250.05Aminopeptidase A inhibitor

0.05 0.004 CHEMBL3706542

0.017 0.013 CHEMBL1213529

0.034 0.005 CHEMBL3706541

CHEMBL3706542
0.0670.2980.354Hepatoprotectant

0.164 0.096 CHEMBL721

0.194 0.069 CHEMBL3706539

0.354 0.018 CHEMBL3706542

0.302 0.029 CHEMBL1213529

0.244 0.045 CHEMBL3706541

CHEMBL3706542
0.0080.240.065Guanylate cyclase inhibitor

0.041 0.032 CHEMBL721

0.065 0.008 CHEMBL1213529

CHEMBL1213529
0.0190.2570.567Porphobilinogen synthase inhibitor

0.153 0.02 CHEMBL506976

0.065 0.061 CHEMBL3544547

0.241 0.008 CHEMBL721

0.567 0.003 CHEMBL1213529

0.118 0.029 CHEMBL913

CHEMBL1213529
0.0060.2460.017O6-alkylguanine-DNA alkyltransferase inhibitor

0.017 0.012 CHEMBL913

CHEMBL913
0.0080.250.044Fructose-1,6-bisphosphatase inhibitor

0.043 0.035 CHEMBL506976

0.044 0.033 CHEMBL913

CHEMBL913
0.0050.250.129Lysine carboxypeptidase inhibitor

0.129 0.003 CHEMBL3706542

0.043 0.009 CHEMBL1213529

0.026 0.019 CHEMBL913

0.044 0.009 CHEMBL3706541

CHEMBL3706542
0.0490.30.125Glutamate (mGluR7) agonist

0.098 0.064 CHEMBL1213529

0.125 0.026 CHEMBL913

CHEMBL913
0.0010.2560.007DNA topoisomerase III inhibitor

0.007 0.006 CHEMBL506976

0.007 0.005 CHEMBL913

CHEMBL913
0.0020.2610.021N-Acetylated alpha-linked acidic dipeptidase inhibitor

0.02 0.007 CHEMBL3706542

0.021 0.007 CHEMBL3706541

CHEMBL3706541
0.0050.2660.042Phosphoglycerate kinase inhibitor

0.042 0.018 CHEMBL1213529

0.032 0.028 CHEMBL913

CHEMBL1213529
0.0380.30.347Thioredoxin inhibitor

0.179 0.011 CHEMBL506976

0.09 0.062 CHEMBL3706538

0.096 0.053 CHEMBL1213529

0.347 0.002 CHEMBL913

CHEMBL913
0.0180.2820.894Glutamate decarboxylase inhibitor

0.168 0.01 CHEMBL506976

0.067 0.059 CHEMBL3544547

0.245 0.004 CHEMBL721

0.066 0.06 CHEMBL3706539

0.894 0.001 CHEMBL3706542

0.459 0.003 CHEMBL1213529

0.093 0.034 CHEMBL913

0.473 0.003 CHEMBL3706541

CHEMBL3706542
0.0020.2670.0121-Deoxy-D-xylulose-5-phosphate reductoisomerase inhibitor

0.012 0.011 CHEMBL1213529

CHEMBL1213529
0.0080.2730.039Acid ceramidase inhibitor

0.027 0.015 CHEMBL506976

0.039 0.004 CHEMBL913

CHEMBL913
0.0160.2840.123Na+ K+ transporting ATPase inhibitor

0.1 0.032 CHEMBL506976

0.123 0.015 CHEMBL721

0.116 0.019 CHEMBL1213529

0.07 0.06 CHEMBL913

CHEMBL721
0.0980.3680.274RNA-directed DNA polymerase inhibitor

0.213 0.082 CHEMBL506976

0.235 0.06 CHEMBL721

0.274 0.038 CHEMBL1213529

0.196 0.105 CHEMBL913

CHEMBL1213529
0.050.3230.513Anesthetic general

0.295 0.034 CHEMBL506976

0.143 0.121 CHEMBL3706538

0.24 0.055 CHEMBL3544547

0.266 0.044 CHEMBL721

0.168 0.096 CHEMBL3706540

0.513 0.007 CHEMBL1213529

0.293 0.035 CHEMBL913

CHEMBL1213529
0.0670.3410.187Vanilloid 1 agonist

0.144 0.045 CHEMBL721

0.12 0.089 CHEMBL3706540

0.141 0.048 CHEMBL3706542

0.187 0.016 CHEMBL1213529

0.112 0.107 CHEMBL913

0.137 0.055 CHEMBL3706541

CHEMBL1213529
0.0360.3130.39UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor

0.146 0.028 CHEMBL506976

0.178 0.02 CHEMBL721

0.164 0.023 CHEMBL3706542

0.39 0.004 CHEMBL1213529

0.129 0.034 CHEMBL913

0.136 0.031 CHEMBL3706541

CHEMBL1213529
0.0070.2860.108Carbonic anhydrase VB inhibitor

0.108 0.014 CHEMBL1213529

0.057 0.038 CHEMBL913

CHEMBL1213529
0.0230.3030.302GABA aminotransferase inhibitor

0.136 0.011 CHEMBL506976

0.144 0.009 CHEMBL721

0.302 0.003 CHEMBL1213529

0.162 0.006 CHEMBL913

CHEMBL1213529
0.0040.2880.028Isoleucine-tRNA ligase inhibitor

0.023 0.014 CHEMBL506976

0.028 0.007 CHEMBL1213529

0.022 0.016 CHEMBL913

CHEMBL1213529
0.0150.2990.354Aconitate hydratase inhibitor

0.078 0.014 CHEMBL506976

0.097 0.009 CHEMBL721

0.354 0.002 CHEMBL1213529

0.063 0.023 CHEMBL913

CHEMBL1213529
0.0070.2920.039Purinergic P2Y15 antagonist

0.032 0.014 CHEMBL506976

0.029 0.02 CHEMBL721

0.029 0.018 CHEMBL1213529

0.039 0.007 CHEMBL913

CHEMBL913
0.0150.3020.081Androgen agonist

0.067 0.033 CHEMBL506976

0.055 0.049 CHEMBL721

0.074 0.028 CHEMBL1213529

0.081 0.023 CHEMBL913

CHEMBL913
0.0260.3140.18Ornithine decarboxylase inhibitor

0.116 0.028 CHEMBL506976

0.151 0.011 CHEMBL721

0.101 0.043 CHEMBL3706542

0.18 0.006 CHEMBL1213529

0.11 0.034 CHEMBL913

CHEMBL1213529
0.010.30.049Carboxypeptidase B inhibitor

0.046 0.008 CHEMBL3706542

0.033 0.022 CHEMBL1213529

0.049 0.007 CHEMBL3706541

CHEMBL3706541
0.0080.2990.107Thymidylate synthase inhibitor

0.053 0.024 CHEMBL506976

0.046 0.032 CHEMBL721

0.107 0.004 CHEMBL3706542

0.08 0.007 CHEMBL1213529

0.06 0.017 CHEMBL913

0.063 0.015 CHEMBL3706541

CHEMBL3706542
0.0070.2990.08Matrix metalloproteinase 1 inhibitor

0.08 0.021 CHEMBL3706542

0.048 0.04 CHEMBL3706541

CHEMBL3706542
0.0970.3890.362Vasodilator, coronary

0.276 0.109 CHEMBL506976

0.223 0.161 CHEMBL3706538

0.237 0.148 CHEMBL721

0.305 0.083 CHEMBL1213529

0.362 0.05 CHEMBL913

CHEMBL913
0.0110.3070.525Alcohol oxidase inhibitor

0.394 0.004 CHEMBL506976

0.386 0.004 CHEMBL721

0.525 0.004 CHEMBL1213529

0.088 0.021 CHEMBL913

CHEMBL1213529
0.0150.3110.074HCV NS3/NS4A protease inhibitor

0.067 0.016 CHEMBL721

0.074 0.013 CHEMBL3706542

0.066 0.017 CHEMBL1213529

CHEMBL3706542
0.0390.3350.222Microtubule formation inhibitor

0.17 0.029 CHEMBL506976

0.191 0.022 CHEMBL721

0.222 0.015 CHEMBL1213529

0.18 0.025 CHEMBL913

CHEMBL1213529
0.0040.3030.022Fructose-1,6-bisphosphatase 1 inhibitor

0.022 0.02 CHEMBL1213529

CHEMBL1213529
0.0060.3060.058Prostaglandin F2 alpha agonist

0.027 0.011 CHEMBL721

0.058 0.004 CHEMBL1213529

CHEMBL1213529
0.0280.3290.285Cystathionine beta-synthase inhibitor

0.259 0.014 CHEMBL506976

0.135 0.048 CHEMBL721

0.285 0.011 CHEMBL1213529

0.21 0.022 CHEMBL913

CHEMBL1213529
0.0280.3340.091Sphingomyelinase inhibitor

0.088 0.075 CHEMBL1213529

0.091 0.071 CHEMBL913

CHEMBL913
0.0170.3260.075Dopamine beta hydroxylase inhibitor

0.062 0.014 CHEMBL506976

0.069 0.008 CHEMBL721

0.075 0.006 CHEMBL1213529

0.069 0.009 CHEMBL913

CHEMBL1213529
0.0350.3480.314Amylase inhibitor

0.314 0.017 CHEMBL506976

0.27 0.023 CHEMBL721

0.271 0.023 CHEMBL1213529

0.162 0.059 CHEMBL913

CHEMBL506976
0.0590.3740.261Adenylate cyclase stimulant

0.142 0.078 CHEMBL506976

0.201 0.013 CHEMBL721

0.261 0.004 CHEMBL1213529

0.171 0.034 CHEMBL913

CHEMBL1213529
0.0110.3260.071Adenosine deaminase inhibitor

0.071 0.013 CHEMBL506976

0.063 0.018 CHEMBL721

0.061 0.02 CHEMBL3706542

0.065 0.016 CHEMBL1213529

0.062 0.019 CHEMBL913

CHEMBL506976
0.0210.3420.145Glycine receptor antagonist

0.082 0.054 CHEMBL506976

0.117 0.02 CHEMBL721

0.145 0.009 CHEMBL1213529

0.094 0.038 CHEMBL913

CHEMBL1213529
0.0110.3340.056Prolyl endopeptidase inhibitor

0.049 0.037 CHEMBL506976

0.047 0.041 CHEMBL721

0.056 0.029 CHEMBL3706542

CHEMBL3706542
0.0990.4230.667GABA C receptor rho-3 antagonist

0.477 0.032 CHEMBL506976

0.21 0.195 CHEMBL3706538

0.646 0.004 CHEMBL721

0.667 0.004 CHEMBL1213529

0.556 0.014 CHEMBL913

CHEMBL1213529
0.0020.3270.026Thromboxane A2 agonist

0.015 0.013 CHEMBL506976

0.014 0.013 CHEMBL721

0.026 0.004 CHEMBL1213529

CHEMBL1213529
0.0080.3340.025Thymidine phosphorylase inhibitor

0.025 0.02 CHEMBL1213529

CHEMBL1213529
0.0350.360.26Cathepsin H inhibitor

0.26 0.013 CHEMBL506976

0.181 0.029 CHEMBL721

0.159 0.04 CHEMBL3706542

0.143 0.051 CHEMBL1213529

0.205 0.021 CHEMBL913

CHEMBL506976
0.0210.3470.102Purinergic P2X1 antagonist

0.077 0.027 CHEMBL506976

0.071 0.031 CHEMBL721

0.102 0.016 CHEMBL1213529

0.056 0.051 CHEMBL913

CHEMBL1213529
0.0030.3290.021Nicotinic alpha4 receptor agonist

0.021 0.006 CHEMBL721

CHEMBL721
0.0150.3430.154Kainate receptor agonist

0.044 0.023 CHEMBL506976

0.07 0.004 CHEMBL721

0.154 0.002 CHEMBL1213529

0.042 0.027 CHEMBL913

CHEMBL1213529
0.0270.3560.193Glycine receptor agonist

0.078 0.041 CHEMBL506976

0.11 0.016 CHEMBL721

0.193 0.004 CHEMBL1213529

0.072 0.052 CHEMBL913

CHEMBL1213529
0.0020.3360.122Arginase inhibitor

0.122 0.003 CHEMBL3706542

0.055 0.012 CHEMBL1213529

0.035 0.027 CHEMBL913

0.053 0.014 CHEMBL3706541

CHEMBL3706542
0.0040.340.032Nicotinic alpha4beta2 receptor agonist

0.032 0.015 CHEMBL721

CHEMBL721
0.0240.3620.081Ryanodine receptor antagonist

0.063 0.029 CHEMBL721

0.081 0.008 CHEMBL1213529

0.059 0.04 CHEMBL913

CHEMBL1213529
0.0380.3770.181DOPA decarboxylase inhibitor

0.134 0.032 CHEMBL506976

0.128 0.037 CHEMBL721

0.181 0.01 CHEMBL1213529

0.11 0.058 CHEMBL913

CHEMBL1213529
0.0070.3460.053Calcitonin receptor agonist

0.053 0.016 CHEMBL3706542

CHEMBL3706542
0.0110.350.116Matrix metalloproteinase inhibitor

0.116 0.021 CHEMBL3706542

0.08 0.037 CHEMBL3706541

CHEMBL3706542
0.0070.3470.08GABA uptake inhibitor

0.044 0.022 CHEMBL506976

0.068 0.008 CHEMBL721

0.08 0.005 CHEMBL1213529

CHEMBL1213529
0.0030.3490.062Uridine phosphorylase inhibitor

0.038 0.013 CHEMBL721

0.062 0.005 CHEMBL1213529

CHEMBL1213529
0.0050.3520.024Alpha 2b adrenoreceptor agonist

0.024 0.006 CHEMBL721

CHEMBL721
0.0360.3840.304Thioredoxin reductase inhibitor

0.202 0.004 CHEMBL506976

0.128 0.014 CHEMBL721

0.08 0.061 CHEMBL1213529

0.304 0.003 CHEMBL913

CHEMBL913
0.0110.3590.133Lysophosphatidic acid 3 receptor antagonist

0.07 0.015 CHEMBL721

0.058 0.024 CHEMBL3706542

0.133 0.003 CHEMBL1213529

CHEMBL1213529
0.0150.3630.0623-Hydroxyanthranilate 3,4-dioxygenase inhibitor

0.05 0.015 CHEMBL506976

0.045 0.021 CHEMBL721

0.062 0.007 CHEMBL1213529

0.049 0.015 CHEMBL913

CHEMBL1213529
0.0060.3560.035Neuraminidase (Influenza B) inhibitor

0.026 0.007 CHEMBL721

0.035 0.004 CHEMBL1213529

CHEMBL1213529
0.0190.370.156Cathepsin G inhibitor

0.156 0.02 CHEMBL506976

0.085 0.04 CHEMBL721

0.082 0.042 CHEMBL3706542

0.111 0.03 CHEMBL1213529

0.091 0.037 CHEMBL913

CHEMBL506976
0.0040.3550.028Nicotinic alpha3beta4 receptor agonist

0.028 0.024 CHEMBL913

CHEMBL913
0.060.4130.548Phospholipase C inhibitor

0.14 0.129 CHEMBL506976

0.142 0.124 CHEMBL3544547

0.202 0.042 CHEMBL721

0.139 0.131 CHEMBL3706540

0.548 0.005 CHEMBL3706542

0.375 0.012 CHEMBL1213529

0.17 0.073 CHEMBL913

0.454 0.008 CHEMBL3706541

CHEMBL3706542
0.0040.3580.056Geranyltranstransferase inhibitor

0.048 0.025 CHEMBL506976

0.056 0.017 CHEMBL721

0.053 0.019 CHEMBL1213529

0.055 0.017 CHEMBL913

CHEMBL721
0.0140.3680.114Carbonic anhydrase VA inhibitor

0.114 0.02 CHEMBL1213529

0.061 0.058 CHEMBL913

CHEMBL1213529
0.0080.3650.274Toll-Like receptor 2 agonist

0.274 0.003 CHEMBL3706542

0.044 0.027 CHEMBL1213529

0.038 0.031 CHEMBL913

0.254 0.004 CHEMBL3706541

CHEMBL3706542
0.0120.3730.12Carbonic anhydrase V inhibitor

0.12 0.021 CHEMBL1213529

CHEMBL1213529
0.0030.3650.019Neurokinin 1 agonist

0.019 0.015 CHEMBL3706542

CHEMBL3706542
0.0310.3960.101Vanilloid 4 agonist

0.078 0.045 CHEMBL506976

0.089 0.027 CHEMBL721

0.101 0.016 CHEMBL1213529

0.096 0.02 CHEMBL913

CHEMBL1213529
0.0490.4150.349GABA C receptor rho-2 antagonist

0.175 0.046 CHEMBL506976

0.294 0.006 CHEMBL721

0.349 0.004 CHEMBL1213529

0.222 0.019 CHEMBL913

CHEMBL1213529
0.0780.4440.5575 Hydroxytryptamine release stimulant

0.245 0.091 CHEMBL506976

0.401 0.046 CHEMBL721

0.484 0.03 CHEMBL1213529

0.557 0.019 CHEMBL913

CHEMBL913
0.0120.3840.502Histidine decarboxylase inhibitor

0.084 0.04 CHEMBL506976

0.084 0.04 CHEMBL721

0.502 0.003 CHEMBL3706542

0.333 0.005 CHEMBL1213529

0.082 0.041 CHEMBL913

0.365 0.004 CHEMBL3706541

CHEMBL3706542
0.0040.3770.026Sodium/glucose cotransporter 2 inhibitor

0.026 0.018 CHEMBL913

CHEMBL913
0.0210.3950.326Mucolytic

0.118 0.057 CHEMBL721

0.326 0.004 CHEMBL3706542

0.209 0.011 CHEMBL1213529

0.11 0.065 CHEMBL913

0.236 0.008 CHEMBL3706541

CHEMBL3706542
0.1090.4840.4385 Hydroxytryptamine uptake stimulant

0.289 0.051 CHEMBL506976

0.346 0.027 CHEMBL721

0.438 0.009 CHEMBL1213529

0.355 0.024 CHEMBL913

CHEMBL1213529
0.0010.3770.013Carbonic anhydrase XI inhibitor

0.013 0.009 CHEMBL1213529

CHEMBL1213529
0.0090.3860.048Glutamate (mGluR3) agonist

0.031 0.026 CHEMBL3706542

0.048 0.005 CHEMBL1213529

CHEMBL1213529
0.0090.3850.063Histamine H1 receptor agonist

0.063 0.007 CHEMBL913

CHEMBL913
0.0160.3940.095Phospholipase D inhibitor

0.068 0.057 CHEMBL506976

0.072 0.048 CHEMBL721

0.091 0.021 CHEMBL1213529

0.095 0.018 CHEMBL913

CHEMBL913
0.0070.3870.065Oxytocin agonist

0.065 0.013 CHEMBL3706542

0.049 0.025 CHEMBL913

CHEMBL3706542
0.0320.4120.243Protein kinase stimulant

0.133 0.081 CHEMBL721

0.243 0.028 CHEMBL1213529

CHEMBL1213529
0.0010.3810.006Integrin alpha5beta6 antagonist

0.006 0.005 CHEMBL1213529

CHEMBL1213529
0.020.4050.046Heme oxygenase inhibitor

0.041 0.04 CHEMBL506976

0.042 0.031 CHEMBL721

0.046 0.021 CHEMBL1213529

CHEMBL1213529
0.0510.4390.174DNA repair enzyme inhibitor

0.132 0.052 CHEMBL506976

0.118 0.077 CHEMBL1213529

0.174 0.016 CHEMBL913

CHEMBL913
0.0370.4270.103D-Ala-D-Ala ligase inhibitor

0.085 0.054 CHEMBL506976

0.079 0.071 CHEMBL721

0.103 0.026 CHEMBL1213529

0.088 0.048 CHEMBL913

CHEMBL1213529
0.0120.4020.054Thymidine kinase inhibitor

0.04 0.03 CHEMBL721

0.054 0.017 CHEMBL1213529

0.039 0.031 CHEMBL913

CHEMBL1213529
0.0080.3980.033Dipeptidyl peptidase II inhibitor

0.033 0.022 CHEMBL913

CHEMBL913
0.0320.4240.114Granulocyte macrophage colony stimulating factor agonist

0.104 0.03 CHEMBL506976

0.105 0.029 CHEMBL721

0.114 0.02 CHEMBL1213529

0.099 0.036 CHEMBL913

CHEMBL1213529
0.040.4350.103Estrogen-related receptor beta agonist

0.083 0.056 CHEMBL506976

0.082 0.061 CHEMBL721

0.103 0.022 CHEMBL1213529

0.097 0.028 CHEMBL913

CHEMBL1213529
0.0010.4010.015Thromboxane agonist

0.015 0.005 CHEMBL1213529

CHEMBL1213529
0.0110.4120.317Phenylalanine 4-hydroxylase inhibitor

0.069 0.048 CHEMBL506976

0.107 0.023 CHEMBL721

0.101 0.025 CHEMBL3706542

0.317 0.004 CHEMBL1213529

0.085 0.034 CHEMBL913

CHEMBL1213529
0.0210.4260.523Ferrochelatase inhibitor

0.248 0.013 CHEMBL506976

0.331 0.005 CHEMBL721

0.523 0.002 CHEMBL1213529

0.237 0.015 CHEMBL913

CHEMBL1213529
0.0140.420.344Expectorant

0.095 0.075 CHEMBL721

0.344 0.006 CHEMBL3706542

0.239 0.014 CHEMBL1213529

0.241 0.014 CHEMBL3706541

CHEMBL3706542
0.0060.4120.15Lysophosphatidic acid 2 receptor antagonist

0.033 0.018 CHEMBL721

0.15 0.004 CHEMBL1213529

CHEMBL1213529
0.0030.410.018Vitamin D receptor agonist

0.018 0.008 CHEMBL1213529

CHEMBL1213529
0.0060.4170.024Caspase 8 inhibitor

0.019 0.014 CHEMBL506976

0.024 0.008 CHEMBL3706542

CHEMBL3706542
0.090.5020.273Nitric-oxide synthase stimulant

0.223 0.057 CHEMBL506976

0.204 0.082 CHEMBL721

0.231 0.047 CHEMBL1213529

0.273 0.02 CHEMBL913

CHEMBL913
0.0030.4160.138Retinoid X receptor agonist

0.049 0.018 CHEMBL721

0.138 0.003 CHEMBL1213529

CHEMBL1213529
0.0140.430.073Calcium antagonist

0.073 0.07 CHEMBL913

CHEMBL913
0.0040.4220.071Retinoid X beta receptor antagonist

0.026 0.006 CHEMBL721

0.071 0.002 CHEMBL1213529

CHEMBL1213529
0.0060.4240.026Factor XIII inhibitor

0.026 0.006 CHEMBL721

0.022 0.011 CHEMBL1213529

CHEMBL721
0.0050.4270.03Thyroid hormone agonist

0.03 0.013 CHEMBL1213529

CHEMBL1213529
0.0130.4370.108S-adenosyl-L-methionine decarboxylase inhibitor

0.084 0.03 CHEMBL506976

0.091 0.021 CHEMBL721

0.094 0.018 CHEMBL1213529

0.108 0.009 CHEMBL913

CHEMBL913
0.0020.4330.02Alpha 2c adrenoreceptor agonist

0.02 0.011 CHEMBL721

CHEMBL721
0.010.4410.103Metalloproteinase-9 inhibitor

0.103 0.031 CHEMBL3706542

CHEMBL3706542
0.0350.4680.174Sphingosine 1-phosphate receptor 4 antagonist

0.151 0.033 CHEMBL506976

0.14 0.044 CHEMBL1213529

0.174 0.017 CHEMBL913

CHEMBL913
0.0090.4470.03Thymidine kinase (Herpes simplex virus 1) inhibitor

0.027 0.017 CHEMBL721

0.03 0.011 CHEMBL1213529

0.026 0.02 CHEMBL913

CHEMBL1213529
0.0030.4410.019Imidazoline I1 receptor antagonist

0.019 0.017 CHEMBL721

CHEMBL721
0.0030.4420.039Glutamate (mGluR1a) agonist

0.029 0.009 CHEMBL506976

0.039 0.006 CHEMBL1213529

0.025 0.012 CHEMBL913

CHEMBL1213529
0.0160.4560.284Cholesterol synthesis inhibitor

0.128 0.058 CHEMBL506976

0.187 0.03 CHEMBL721

0.284 0.013 CHEMBL1213529

CHEMBL1213529
0.0060.4470.039Integrin alpha2beta1 antagonist

0.039 0.006 CHEMBL1213529

CHEMBL1213529
0.020.4620.1645 Hydroxytryptamine 3A agonist

0.109 0.066 CHEMBL506976

0.09 0.089 CHEMBL721

0.164 0.028 CHEMBL913

CHEMBL913
0.0290.4730.174Toll-Like receptor 4 antagonist

0.09 0.089 CHEMBL721

0.174 0.011 CHEMBL1213529

CHEMBL1213529
0.0140.4610.115Alpha 2 adrenoreceptor antagonist

0.115 0.038 CHEMBL913

CHEMBL913
0.1260.5730.459Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.456 0.058 CHEMBL506976

0.436 0.071 CHEMBL721

0.388 0.112 CHEMBL1213529

0.459 0.056 CHEMBL913

CHEMBL913
0.0270.4750.224Mannose-6-phosphate isomerase inhibitor

0.224 0.02 CHEMBL506976

0.206 0.027 CHEMBL721

0.209 0.026 CHEMBL1213529

CHEMBL506976
0.0090.4590.42Catalase inhibitor

0.167 0.022 CHEMBL506976

0.177 0.02 CHEMBL721

0.42 0.003 CHEMBL3706542

0.255 0.008 CHEMBL1213529

0.071 0.054 CHEMBL913

0.08 0.048 CHEMBL3706541

CHEMBL3706542
0.010.4610.026Hedgehog signaling activator

0.026 0.024 CHEMBL913

CHEMBL913
0.0050.4560.046Alpha 1d adrenoreceptor agonist

0.035 0.032 CHEMBL506976

0.046 0.02 CHEMBL913

CHEMBL913
0.0040.4620.151Retinoid X alpha receptor agonist

0.04 0.02 CHEMBL721

0.151 0.003 CHEMBL1213529

CHEMBL1213529
0.0070.4660.058Histamine H2 receptor agonist

0.058 0.015 CHEMBL913

CHEMBL913
0.020.4810.467Neurotrophic factor

0.467 0.004 CHEMBL721

0.115 0.104 CHEMBL3706542

CHEMBL721
0.0250.4870.363Toll-Like receptor 2 antagonist

0.162 0.045 CHEMBL721

0.363 0.004 CHEMBL3706542

0.216 0.017 CHEMBL1213529

0.104 0.098 CHEMBL913

0.281 0.005 CHEMBL3706541

CHEMBL3706542
0.020.4820.202Keratolytic

0.07 0.065 CHEMBL721

0.202 0.008 CHEMBL1213529

CHEMBL1213529
0.0040.4660.024Sodium/glucose cotransporter inhibitor

0.024 0.021 CHEMBL913

CHEMBL913
0.030.4920.431TRPA1 agonist

0.235 0.006 CHEMBL506976

0.431 0.004 CHEMBL721

0.209 0.009 CHEMBL1213529

0.151 0.03 CHEMBL913

CHEMBL721
0.0120.480.084Sphingosine 1-phosphate receptor 1 antagonist

0.084 0.013 CHEMBL913

CHEMBL913
0.010.4820.048Squalene epoxidase inhibitor

0.047 0.04 CHEMBL721

0.046 0.042 CHEMBL1213529

0.048 0.038 CHEMBL913

CHEMBL913
0.0090.4840.136Sphingosine 1-phosphate receptor 4 agonist

0.061 0.053 CHEMBL721

0.136 0.011 CHEMBL1213529

CHEMBL1213529
0.0060.4820.052Matrix metalloproteinase (membrane-type) inhibitor

0.052 0.042 CHEMBL3706542

CHEMBL3706542
0.0150.4950.099Histamine N-methyltransferase inhibitor

0.099 0.047 CHEMBL913

CHEMBL913
0.0050.4850.014S-adenosyl-L-homocysteine hydrolase inhibitor

0.014 0.011 CHEMBL506976

CHEMBL506976
0.010.4950.066Sphingosine 1-phosphate receptor 3 antagonist

0.066 0.029 CHEMBL913

CHEMBL913
0.0230.5080.284Electrolyte absorption antagonist

0.142 0.023 CHEMBL506976

0.177 0.012 CHEMBL721

0.284 0.004 CHEMBL1213529

0.154 0.018 CHEMBL913

CHEMBL1213529
0.0070.4930.053Integrin alpha2 antagonist

0.053 0.01 CHEMBL1213529

CHEMBL1213529
0.010.4960.094AICAR transformylase inhibitor

0.049 0.023 CHEMBL506976

0.049 0.024 CHEMBL721

0.094 0.005 CHEMBL3706542

0.055 0.017 CHEMBL1213529

CHEMBL3706542
0.0110.5010.25Alcohol dehydrogenase inhibitor

0.25 0.008 CHEMBL506976

0.116 0.038 CHEMBL721

0.122 0.034 CHEMBL3706542

0.135 0.026 CHEMBL1213529

0.127 0.03 CHEMBL913

CHEMBL506976
0.0020.4920.022NMDA receptor glycine site antagonist

0.022 0.019 CHEMBL1213529

CHEMBL1213529
0.0040.50.025Thymidine kinase (Herpes simplex virus 2) inhibitor

0.021 0.013 CHEMBL721

0.025 0.007 CHEMBL1213529

0.021 0.013 CHEMBL913

CHEMBL1213529
0.030.5260.646Peroxidase inhibitor

0.25 0.047 CHEMBL506976

0.22 0.054 CHEMBL721

0.646 0.004 CHEMBL3706542

0.47 0.012 CHEMBL1213529

0.323 0.033 CHEMBL913

0.38 0.023 CHEMBL3706541

CHEMBL3706542
0.0080.5090.041Melatonin receptor 1A agonist

0.041 0.013 CHEMBL721

0.04 0.014 CHEMBL1213529

CHEMBL721
0.0280.5360.189Cyclooxygenase 3 inhibitor

0.118 0.08 CHEMBL721

0.156 0.043 CHEMBL3706542

0.189 0.023 CHEMBL1213529

0.102 0.101 CHEMBL913

CHEMBL1213529
0.0090.5170.1Adenylate cyclase 1 inhibitor

0.09 0.005 CHEMBL721

0.1 0.004 CHEMBL1213529

0.076 0.009 CHEMBL913

CHEMBL1213529
0.0010.510.018Ileal bile acid transport inhibitor

0.018 0.011 CHEMBL3706542

CHEMBL3706542
0.0230.5340.102MAP kinase kinase 7 inhibitor

0.09 0.024 CHEMBL721

0.102 0.012 CHEMBL1213529

0.082 0.04 CHEMBL913

CHEMBL1213529
0.0150.5260.049Nicotinic alpha3beta2 receptor antagonist

0.049 0.046 CHEMBL1213529

CHEMBL1213529
0.0170.5310.102GABA B receptor agonist

0.071 0.064 CHEMBL506976

0.102 0.015 CHEMBL1213529

0.086 0.032 CHEMBL913

CHEMBL1213529
0.0090.5250.069Retinoid X alpha receptor antagonist

0.037 0.018 CHEMBL721

0.069 0.003 CHEMBL1213529

CHEMBL1213529
0.0370.5520.3773C-like protease (Human coronavirus) inhibitor

0.377 0.004 CHEMBL506976

0.257 0.024 CHEMBL721

0.15 0.1 CHEMBL1213529

0.27 0.019 CHEMBL913

CHEMBL506976
0.0410.5610.262Neurotrophic factor enhancer

0.147 0.143 CHEMBL506976

0.169 0.111 CHEMBL721

0.262 0.032 CHEMBL1213529

CHEMBL1213529
0.0080.5290.05Sphingosine kinase 2 inhibitor

0.05 0.048 CHEMBL1213529

CHEMBL1213529
0.0040.5280.043Carbonic anhydrase VII inhibitor

0.043 0.036 CHEMBL1213529

CHEMBL1213529
0.0050.5290.105NMDA receptor glycine site agonist

0.105 0.014 CHEMBL1213529

0.075 0.032 CHEMBL913

CHEMBL1213529
0.0010.5270.039Prostaglandin H2 antagonist

0.039 0.006 CHEMBL1213529

CHEMBL1213529
0.0050.5320.039Nerve growth factor antagonist

0.039 0.038 CHEMBL506976

CHEMBL506976
0.0050.5330.041Nicotinic receptor alpha3 subunit antagonist

0.041 0.034 CHEMBL913

CHEMBL913
0.0090.540.079Retinoid X receptor antagonist

0.042 0.021 CHEMBL721

0.079 0.003 CHEMBL1213529

CHEMBL1213529
0.0140.5470.098Dihydroorotate oxidase inhibitor

0.055 0.038 CHEMBL506976

0.084 0.009 CHEMBL721

0.098 0.005 CHEMBL1213529

CHEMBL1213529
0.0110.5480.04Vanilloid 3 antagonist

0.04 0.023 CHEMBL1213529

CHEMBL1213529
0.0040.5420.022CXC chemokine 5 receptor antagonist

0.022 0.007 CHEMBL1213529

CHEMBL1213529
0.0620.5990.37Calcium channel activator

0.255 0.142 CHEMBL506976

0.311 0.081 CHEMBL721

0.37 0.038 CHEMBL1213529

0.327 0.067 CHEMBL913

CHEMBL1213529
0.0030.5410.064Dihydropteroate synthase inhibitor

0.039 0.028 CHEMBL721

0.064 0.01 CHEMBL1213529

CHEMBL1213529
0.0040.5410.027MAP3K8 inhibitor

0.027 0.025 CHEMBL913

CHEMBL913
0.0010.540.044Prostaglandin EP4 agonist

0.044 0.005 CHEMBL1213529

CHEMBL1213529
0.0150.5560.038Glucose-6-phosphate dehydrogenase inhibitor

0.038 0.026 CHEMBL913

CHEMBL913
0.0040.5490.032Lysophosphatidic acid 1 receptor antagonist

0.032 0.006 CHEMBL1213529

CHEMBL1213529
0.0040.550.058ATP citrate lysase inhibitor

0.058 0.005 CHEMBL1213529

CHEMBL1213529
0.0040.5540.0412,3-Oxidosqualene-lanosterol cyclase inhibitor

0.041 0.02 CHEMBL721

0.039 0.022 CHEMBL1213529

CHEMBL721
0.0080.5590.878Epidermal growth factor antagonist

0.833 0.003 CHEMBL1593

0.738 0.004 CHEMBL3544547

0.115 0.035 CHEMBL721

0.75 0.004 CHEMBL525

0.878 0.003 CHEMBL3706540

0.143 0.025 CHEMBL1213529

0.101 0.044 CHEMBL913

CHEMBL3706540
0.0110.5630.078Interferon agonist

0.078 0.056 CHEMBL1213529

0.073 0.065 CHEMBL913

CHEMBL1213529
0.0180.570.151Exportin-1 inhibitor

0.091 0.014 CHEMBL506976

0.142 0.004 CHEMBL721

0.151 0.003 CHEMBL1213529

0.074 0.035 CHEMBL913

CHEMBL1213529
0.0570.6090.157Catenin beta inhibitor

0.157 0.091 CHEMBL1213529

CHEMBL1213529
0.0110.5640.071Pregnane X receptor antagonist

0.065 0.022 CHEMBL506976

0.066 0.02 CHEMBL721

0.071 0.013 CHEMBL1213529

0.055 0.045 CHEMBL913

CHEMBL1213529
0.0160.5690.064Bombesin 2 receptor antagonist

0.064 0.022 CHEMBL3706542

CHEMBL3706542
0.0070.5620.031Complement factor 1s inhibitor

0.031 0.007 CHEMBL721

0.027 0.014 CHEMBL1213529

CHEMBL721
0.0090.5650.146NMDA receptor agonist

0.089 0.024 CHEMBL3706542

0.146 0.009 CHEMBL1213529

0.079 0.029 CHEMBL913

CHEMBL1213529
0.0150.5730.057Corticotropin releasing factor 2 receptor antagonist

0.057 0.054 CHEMBL913

CHEMBL913
0.0020.5630.0695-Alpha-reductase inhibitor

0.069 0.014 CHEMBL1213529

CHEMBL1213529
0.0030.5640.047Nicotinic acid receptor 2 antagonist

0.035 0.008 CHEMBL721

0.047 0.004 CHEMBL1213529

CHEMBL1213529
0.0170.5790.243Telomerase inhibitor

0.243 0.01 CHEMBL913

CHEMBL913
0.0120.5750.063Interferon inducer

0.063 0.047 CHEMBL1213529

0.061 0.051 CHEMBL913

CHEMBL1213529
0.0060.5690.0365 Hydroxytryptamine 2B agonist

0.036 0.034 CHEMBL721

CHEMBL721
0.010.5740.041Potassium channel Kv1.1 blocker

0.041 0.021 CHEMBL721

0.035 0.033 CHEMBL913

CHEMBL721
0.0110.5770.069Glutamate (mGluR4) antagonist

0.069 0.01 CHEMBL1213529

0.04 0.038 CHEMBL913

CHEMBL1213529
0.0210.5870.196Adenylate cyclase inhibitor

0.109 0.077 CHEMBL721

0.196 0.026 CHEMBL1213529

CHEMBL1213529
0.0040.5720.088Caspase 2 inhibitor

0.088 0.005 CHEMBL506976

0.05 0.012 CHEMBL3706542

CHEMBL506976
0.0240.5920.555Aldehyde oxidase inhibitor

0.34 0.057 CHEMBL506976

0.279 0.072 CHEMBL721

0.555 0.025 CHEMBL1213529

0.295 0.068 CHEMBL913

CHEMBL1213529
0.020.5890.095Phosphodiesterase I inhibitor

0.095 0.052 CHEMBL913

CHEMBL913
0.0690.6390.731Caspase 9 stimulant

0.296 0.198 CHEMBL506976

0.491 0.063 CHEMBL721

0.731 0.02 CHEMBL1213529

0.284 0.212 CHEMBL913

CHEMBL1213529
0.0040.5740.046Peptide deformylase inhibitor

0.046 0.012 CHEMBL3706542

CHEMBL3706542
0.0380.6080.559Superoxide dismutase inhibitor

0.407 0.025 CHEMBL506976

0.519 0.011 CHEMBL721

0.559 0.009 CHEMBL3706542

0.498 0.013 CHEMBL1213529

0.358 0.035 CHEMBL913

CHEMBL3706542
0.0140.5840.243Caspase 3 inhibitor

0.152 0.027 CHEMBL506976

0.139 0.037 CHEMBL1593

0.143 0.033 CHEMBL3544547

0.135 0.041 CHEMBL721

0.104 0.085 CHEMBL3706540

0.243 0.005 CHEMBL3706542

0.147 0.03 CHEMBL1213529

0.119 0.061 CHEMBL913

CHEMBL3706542
0.0060.5760.11Nicotinic alpha4beta2 receptor antagonist

0.09 0.04 CHEMBL506976

0.11 0.024 CHEMBL721

0.086 0.044 CHEMBL1213529

0.096 0.035 CHEMBL913

CHEMBL721
0.0270.6030.339Melanin inhibitor

0.156 0.073 CHEMBL506976

0.339 0.017 CHEMBL721

0.259 0.027 CHEMBL1213529

CHEMBL721
0.0090.5860.0623(or 17)beta-hydroxysteroid dehydrogenase inhibitor

0.056 0.034 CHEMBL721

0.062 0.028 CHEMBL1213529

CHEMBL1213529
0.0360.6150.105Glutamate release inhibitor

0.093 0.056 CHEMBL506976

0.105 0.036 CHEMBL1213529

0.099 0.043 CHEMBL913

CHEMBL1213529
0.010.590.147Protease 3C (Human rhinovirus) inhibitor

0.079 0.028 CHEMBL506976

0.095 0.018 CHEMBL721

0.147 0.007 CHEMBL3706542

0.068 0.04 CHEMBL1213529

CHEMBL3706542
0.0230.6060.124Carbonic anhydrase XV inhibitor

0.102 0.064 CHEMBL1213529

0.124 0.043 CHEMBL913

CHEMBL913
0.0110.5940.0875 Hydroxytryptamine 3 agonist

0.087 0.022 CHEMBL721

0.066 0.04 CHEMBL1213529

CHEMBL721
0.0050.5910.125Angiotensin-converting enzyme inhibitor

0.073 0.017 CHEMBL3706539

0.125 0.006 CHEMBL3706542

0.095 0.01 CHEMBL3706541

CHEMBL3706542
0.0170.6060.197Proteasome inhibitor

0.173 0.035 CHEMBL506976

0.167 0.037 CHEMBL721

0.197 0.026 CHEMBL3706542

0.116 0.069 CHEMBL1213529

0.133 0.056 CHEMBL913

CHEMBL3706542
0.0350.6280.577Cholesterol antagonist

0.25 0.125 CHEMBL506976

0.32 0.079 CHEMBL721

0.577 0.022 CHEMBL1213529

0.241 0.132 CHEMBL913

CHEMBL1213529
0.0010.5950.0165-Alpha-reductase 1 inhibitor

0.016 0.013 CHEMBL1213529

CHEMBL1213529
0.0030.5970.0275-Alpha-reductase 2 inhibitor

0.027 0.01 CHEMBL1213529

CHEMBL1213529
0.0010.5990.045Prostaglandin EP2 agonist

0.045 0.007 CHEMBL1213529

CHEMBL1213529
0.0040.6020.045GABA B receptor antagonist

0.045 0.026 CHEMBL1213529

CHEMBL1213529
0.0080.6070.135CYP2A6 inhibitor

0.069 0.06 CHEMBL506976

0.135 0.021 CHEMBL721

0.089 0.042 CHEMBL1213529

0.075 0.053 CHEMBL913

CHEMBL721
0.0020.6030.017Angiotensin-converting enzyme 2 inhibitor

0.016 0.014 CHEMBL3706542

0.017 0.012 CHEMBL3706541

CHEMBL3706541
0.0050.6060.05Leukotriene C4 antagonist

0.05 0.011 CHEMBL1213529

CHEMBL1213529
0.0070.6090.059Epithelial sodium channel blocker

0.052 0.045 CHEMBL1213529

0.059 0.03 CHEMBL913

CHEMBL913
0.0050.6080.053AMPA 4 receptor antagonist

0.039 0.028 CHEMBL3706542

0.053 0.013 CHEMBL1213529

CHEMBL1213529
0.0180.6210.259HIV-1 integrase (Overall Integration) inhibitor

0.129 0.035 CHEMBL721

0.259 0.005 CHEMBL1213529

CHEMBL1213529
0.0080.6130.06Glutamate (mGluR group III) agonist

0.06 0.018 CHEMBL1213529

CHEMBL1213529
0.0140.620.074CD45 antagonist

0.051 0.033 CHEMBL3706542

0.074 0.014 CHEMBL1213529

CHEMBL1213529
0.0250.6340.284Glyceraldehyde-3-phosphate dehydrogenase inhibitor

0.156 0.136 CHEMBL506976

0.155 0.138 CHEMBL721

0.284 0.029 CHEMBL1213529

0.168 0.112 CHEMBL913

CHEMBL1213529
0.0110.620.123Carbonic anhydrase XIII inhibitor

0.067 0.062 CHEMBL506976

0.088 0.044 CHEMBL721

0.123 0.028 CHEMBL1213529

CHEMBL1213529
0.0020.6110.11Kainate receptor 2 antagonist

0.04 0.022 CHEMBL721

0.11 0.004 CHEMBL1213529

CHEMBL1213529
0.0080.6180.091Carbonic anhydrase stimulant

0.091 0.021 CHEMBL3706542

0.069 0.032 CHEMBL1213529

0.055 0.046 CHEMBL913

CHEMBL3706542
0.0180.6320.056Immunoglobulin Fc receptor antagonist

0.056 0.036 CHEMBL913

CHEMBL913
0.0050.6210.094Glutamate (mGluR1) agonist

0.03 0.01 CHEMBL721

0.094 0.004 CHEMBL1213529

CHEMBL1213529
0.0210.6380.067Transcription factor RelA inhibitor

0.067 0.036 CHEMBL721

0.064 0.042 CHEMBL1213529

CHEMBL721
0.0130.630.149Sphingosine 1-phosphate receptor 2 antagonist

0.148 0.043 CHEMBL1213529

0.149 0.043 CHEMBL913

CHEMBL913
0.0050.6220.054Carbonic anhydrase XIV inhibitor

0.054 0.029 CHEMBL1213529

CHEMBL1213529
0.0170.6350.616Thioredoxin glutathione reductase inhibitor

0.616 0.014 CHEMBL506976

0.51 0.027 CHEMBL913

CHEMBL506976
0.0040.6220.0953-Oxoacyl-[acyl-carrier-protein] synthase inhibitor

0.095 0.018 CHEMBL1213529

CHEMBL1213529
0.0190.6380.2855 Hydroxytryptamine 1E antagonist

0.285 0.04 CHEMBL721

0.251 0.074 CHEMBL1213529

0.211 0.118 CHEMBL913

CHEMBL721
0.0050.6250.072Endothelin-converting enzyme inhibitor

0.059 0.025 CHEMBL3706542

0.072 0.02 CHEMBL3706541

CHEMBL3706541
0.0330.6530.084CC chemokine 5 receptor agonist

0.082 0.057 CHEMBL721

0.08 0.066 CHEMBL1213529

0.084 0.052 CHEMBL913

CHEMBL913
0.0090.630.062Glutamate (mGluR group III) antagonist

0.062 0.012 CHEMBL1213529

CHEMBL1213529
0.0180.6410.17Carbonic anhydrase III inhibitor

0.17 0.022 CHEMBL1213529

CHEMBL1213529
0.0010.6240.018G-protein-coupled receptor 120 agonist

0.018 0.011 CHEMBL1213529

CHEMBL1213529
0.0060.630.073Leukotriene C antagonist

0.073 0.012 CHEMBL1213529

CHEMBL1213529
0.0280.6580.308Interleukin agonist

0.164 0.154 CHEMBL721

0.239 0.087 CHEMBL3706542

0.308 0.044 CHEMBL1213529

0.2 0.121 CHEMBL913

CHEMBL1213529
0.0020.6330.046Diamine oxidase inhibitor

0.046 0.017 CHEMBL1213529

CHEMBL1213529
0.0010.6310.065Kainate receptor 1 antagonist

0.065 0.005 CHEMBL1213529

CHEMBL1213529
0.0050.6360.038Glutamate (mGluR4) agonist

0.038 0.018 CHEMBL1213529

CHEMBL1213529
0.0230.6560.218Cyclic AMP phosphodiesterase inhibitor

0.202 0.092 CHEMBL1213529

0.218 0.081 CHEMBL913

CHEMBL913
0.0080.640.096Sphingosine 1-phosphate receptor antagonist

0.096 0.024 CHEMBL913

CHEMBL913
0.0040.6370.125Neutrophil collagenase inhibitor

0.125 0.016 CHEMBL3706542

0.082 0.03 CHEMBL3706541

CHEMBL3706542
0.0050.640.101Metalloproteinase-2 inhibitor

0.101 0.038 CHEMBL3706542

0.071 0.064 CHEMBL1213529

CHEMBL3706542
0.0250.6610.158Sphingosine 1-phosphate receptor 5 antagonist

0.158 0.049 CHEMBL1213529

0.132 0.096 CHEMBL913

CHEMBL1213529
0.0080.6450.099Glutamate (mGluR7) antagonist

0.073 0.037 CHEMBL506976

0.073 0.038 CHEMBL721

0.099 0.011 CHEMBL1213529

CHEMBL1213529
0.0030.6410.054Glutamate (mGluR3) antagonist

0.054 0.01 CHEMBL1213529

CHEMBL1213529
0.010.6490.193Prostaglandin dehydrogenase inhibitor

0.193 0.161 CHEMBL1213529

CHEMBL1213529
0.0090.6510.073Potassium channel (Tandem pore domain) blocker

0.073 0.054 CHEMBL913

CHEMBL913
0.0030.6480.032Calcium-sensing receptor agonist

0.032 0.012 CHEMBL3706542

CHEMBL3706542
0.0110.6570.316DNA intercalator

0.316 0.011 CHEMBL913

CHEMBL913
0.0210.670.217Photosensitizer

0.102 0.085 CHEMBL506976

0.15 0.031 CHEMBL721

0.217 0.01 CHEMBL1213529

0.097 0.094 CHEMBL913

CHEMBL1213529
0.0130.6630.366Spasmolytic

0.366 0.048 CHEMBL1213529

0.314 0.065 CHEMBL913

CHEMBL1213529
0.0130.6690.113Alpha 2b adrenoreceptor antagonist

0.113 0.064 CHEMBL913

CHEMBL913
0.0140.6710.134Carbonic anhydrase VI inhibitor

0.134 0.025 CHEMBL1213529

0.073 0.068 CHEMBL913

CHEMBL1213529
0.0120.6690.086Estrogen receptor alpha antagonist

0.086 0.04 CHEMBL1213529

CHEMBL1213529
0.0020.6620.063Oleamide hydrolase inhibitor

0.045 0.032 CHEMBL506976

0.043 0.034 CHEMBL721

0.063 0.019 CHEMBL913

CHEMBL913
0.0160.6760.316Aldehyde dehydrogenase inhibitor

0.195 0.029 CHEMBL506976

0.312 0.01 CHEMBL721

0.316 0.01 CHEMBL3706542

0.27 0.015 CHEMBL1213529

CHEMBL3706542
0.0020.6660.112Kainate receptor antagonist

0.112 0.006 CHEMBL1213529

CHEMBL1213529
0.0290.6940.2Neurotensin receptor agonist

0.159 0.081 CHEMBL506976

0.14 0.129 CHEMBL721

0.191 0.04 CHEMBL3706542

0.2 0.034 CHEMBL1213529

0.2 0.035 CHEMBL913

CHEMBL913
0.0030.6680.096NMDA 2C receptor antagonist

0.096 0.017 CHEMBL1213529

CHEMBL1213529
0.0020.6680.03HCV NS5B polymerase inhibitor

0.03 0.023 CHEMBL1213529

CHEMBL1213529
0.0020.6710.04Free fatty acid receptor 1 antagonist

0.04 0.016 CHEMBL1213529

CHEMBL1213529
0.0030.6720.055NMDA receptor subunit 3B antagonist

0.055 0.022 CHEMBL1213529

CHEMBL1213529
0.0240.6940.272Interferon gamma antagonist

0.135 0.101 CHEMBL506976

0.18 0.05 CHEMBL721

0.272 0.024 CHEMBL1213529

CHEMBL1213529
0.0010.6710.011Integrin beta2 antagonist

0.011 0.01 CHEMBL1213529

CHEMBL1213529
0.0020.6730.045NMDA receptor subunit 3A antagonist

0.045 0.022 CHEMBL1213529

CHEMBL1213529
0.0190.6910.135Lanosterol 14 alpha demethylase inhibitor

0.111 0.04 CHEMBL721

0.135 0.018 CHEMBL1213529

0.094 0.066 CHEMBL913

CHEMBL1213529
0.0120.6870.134Acetylcholine M1 receptor antagonist

0.134 0.091 CHEMBL913

CHEMBL913
0.0090.6860.064Beta 3 adrenoreceptor antagonist

0.064 0.046 CHEMBL913

CHEMBL913
0.0040.6810.092Amidase inhibitor

0.079 0.038 CHEMBL506976

0.092 0.029 CHEMBL721

CHEMBL721
0.0050.6820.063Beta 2 adrenoreceptor agonist

0.063 0.039 CHEMBL913

CHEMBL913
0.0070.6850.061Heparanase inhibitor

0.061 0.021 CHEMBL1213529

CHEMBL1213529
0.0020.6810.057Kynurenine 3 monooxygenase inhibitor

0.057 0.005 CHEMBL1213529

CHEMBL1213529
0.0030.6840.096Leukotriene B4 antagonist

0.096 0.011 CHEMBL1213529

CHEMBL1213529
0.0070.6880.041CF transmembrane conductance regulator antagonist

0.041 0.023 CHEMBL1213529

CHEMBL1213529
0.0030.6860.053NMDA 2A receptor antagonist

0.053 0.035 CHEMBL1213529

CHEMBL1213529
0.0020.6860.041AMPA 3 receptor antagonist

0.041 0.013 CHEMBL1213529

CHEMBL1213529
0.0160.7030.121Vanilloid agonist

0.121 0.018 CHEMBL1213529

0.079 0.072 CHEMBL3706541

CHEMBL1213529
0.0050.6940.117Acetylcholine M2 receptor agonist

0.117 0.005 CHEMBL3544546

CHEMBL3544546
0.0580.7480.277Heat shock protein 70 antagonist

0.157 0.032 CHEMBL721

0.277 0.004 CHEMBL1213529

0.13 0.123 CHEMBL913

CHEMBL1213529
0.040.7310.4415 Hydroxytryptamine release inhibitor

0.327 0.136 CHEMBL506976

0.295 0.17 CHEMBL721

0.441 0.056 CHEMBL1213529

0.344 0.121 CHEMBL913

CHEMBL1213529
0.0150.7060.523Transcription factor NF kappa B inhibitor

0.289 0.1 CHEMBL506976

0.468 0.049 CHEMBL721

0.303 0.092 CHEMBL3706542

0.523 0.041 CHEMBL1213529

0.263 0.118 CHEMBL913

CHEMBL1213529
0.0020.6940.041Methionyl aminopeptidase 1 inhibitor

0.03 0.026 CHEMBL721

0.029 0.028 CHEMBL3706542

0.041 0.011 CHEMBL1213529

CHEMBL1213529
0.0030.6960.065Aromatase inhibitor

0.065 0.038 CHEMBL721

CHEMBL721
0.0050.70.042Tryptophan 5 hydroxylase inhibitor

0.042 0.013 CHEMBL1213529

CHEMBL1213529
0.0030.70.077Nicotinic acid receptor agonist

0.077 0.007 CHEMBL1213529

CHEMBL1213529
0.0050.7020.076Alpha adrenoreceptor antagonist

0.076 0.075 CHEMBL913

CHEMBL913
0.0030.70.041Dihydrofolate reductase inhibitor

0.041 0.036 CHEMBL1213529

CHEMBL1213529
0.0080.7050.158Falcipain 3 inhibitor

0.14 0.041 CHEMBL506976

0.156 0.034 CHEMBL721

0.158 0.033 CHEMBL3706542

0.094 0.077 CHEMBL913

CHEMBL3706542
0.0010.6980.046Prostaglandin E2 agonist

0.046 0.006 CHEMBL1213529

CHEMBL1213529
0.0020.7010.079Prostaglandin agonist

0.079 0.007 CHEMBL1213529

CHEMBL1213529
0.0030.7030.06Potassium channel Kv1.3 blocker

0.06 0.021 CHEMBL721

0.059 0.022 CHEMBL1213529

CHEMBL721
0.0020.7030.056Phosphorylase inhibitor

0.056 0.027 CHEMBL1213529

CHEMBL1213529
0.0040.7070.031Trypsin II inhibitor

0.031 0.019 CHEMBL506976

0.027 0.025 CHEMBL3706542

CHEMBL506976
0.0070.710.291Calpain inhibitor

0.279 0.042 CHEMBL506976

0.236 0.078 CHEMBL721

0.291 0.035 CHEMBL3706542

0.22 0.094 CHEMBL913

CHEMBL3706542
0.0040.7090.048Factor XIIIa inhibitor

0.04 0.023 CHEMBL721

0.034 0.031 CHEMBL3706542

0.048 0.017 CHEMBL1213529

CHEMBL1213529
0.0140.7250.107Acetylcholine release stimulant

0.106 0.074 CHEMBL721

0.107 0.071 CHEMBL1213529

CHEMBL1213529
0.0050.7180.18Cytidine deaminase inhibitor

0.155 0.071 CHEMBL721

0.18 0.057 CHEMBL1213529

CHEMBL1213529
0.0030.720.0321-Alkyl-2-acetylglycerophosphocholine esterase inhibitor

0.032 0.027 CHEMBL1213529

CHEMBL1213529
0.0020.7230.061Neutral endopeptidase inhibitor

0.061 0.006 CHEMBL3706542

0.033 0.011 CHEMBL3706541

CHEMBL3706542
0.0010.7270.054Peroxisome proliferator-activated receptor delta agonist

0.054 0.011 CHEMBL1213529

CHEMBL1213529
0.0030.730.076NMDA receptor antagonist

0.076 0.07 CHEMBL1213529

CHEMBL1213529
0.0010.7290.027AMPA 1 receptor antagonist

0.027 0.022 CHEMBL1213529

CHEMBL1213529
0.0020.7320.079Thromboxane A2 antagonist

0.079 0.015 CHEMBL1213529

CHEMBL1213529
0.0030.7330.141Glycine transporter 2 inhibitor

0.141 0.008 CHEMBL3706542

CHEMBL3706542
0.0050.7380.145Anesthetic local

0.145 0.051 CHEMBL721

0.132 0.058 CHEMBL1213529

CHEMBL721
0.0040.740.184Psychostimulant

0.184 0.09 CHEMBL1213529

CHEMBL1213529
0.0050.7410.091Androgen antagonist

0.091 0.054 CHEMBL506976

0.077 0.069 CHEMBL1213529

0.089 0.056 CHEMBL913

CHEMBL506976
0.0020.7410.03Liver X receptor beta antagonist

0.03 0.019 CHEMBL1213529

CHEMBL1213529
0.0060.7450.419Calpain 2 inhibitor

0.419 0.051 CHEMBL506976

0.318 0.103 CHEMBL721

0.334 0.095 CHEMBL3706542

0.282 0.126 CHEMBL913

CHEMBL506976
0.0080.7470.077Myeloperoxidase inhibitor

0.077 0.073 CHEMBL913

CHEMBL913
0.0150.7570.075Antineoplastic alkaloid

0.075 0.073 CHEMBL1213529

CHEMBL1213529
0.0110.7520.417Thiol protease inhibitor

0.189 0.043 CHEMBL506976

0.203 0.038 CHEMBL721

0.417 0.013 CHEMBL3706542

0.165 0.057 CHEMBL1213529

0.137 0.085 CHEMBL913

0.133 0.091 CHEMBL3706541

CHEMBL3706542
0.0220.7640.185CF transmembrane conductance regulator agonist

0.134 0.108 CHEMBL506976

0.184 0.033 CHEMBL721

0.185 0.032 CHEMBL1213529

0.135 0.106 CHEMBL913

CHEMBL1213529
0.0050.7480.051Glucosylceramidase inhibitor

0.051 0.045 CHEMBL721

CHEMBL721
0.0030.7510.093Cathepsin L inhibitor

0.058 0.041 CHEMBL506976

0.093 0.022 CHEMBL3706542

CHEMBL3706542
0.0080.7570.099AMP-activated protein kinase stimulant

0.099 0.072 CHEMBL1213529

CHEMBL1213529
0.0030.7530.085Thromboxane antagonist

0.085 0.017 CHEMBL1213529

CHEMBL1213529
0.0120.7630.112Bile acid receptor antagonist

0.112 0.028 CHEMBL1213529

CHEMBL1213529
0.0030.7550.074Cannabinoid CB2 receptor antagonist

0.074 0.022 CHEMBL913

CHEMBL913
0.0020.7550.032LFA antagonist

0.032 0.013 CHEMBL1213529

CHEMBL1213529
0.0030.7570.045RNA-directed RNA polymerase inhibitor

0.045 0.015 CHEMBL1213529

CHEMBL1213529
0.010.7640.134Pregnane X receptor agonist

0.127 0.107 CHEMBL721

0.134 0.089 CHEMBL1213529

CHEMBL1213529
0.0040.7610.415Phospholipase A2 inhibitor

0.415 0.005 CHEMBL3706542

0.209 0.038 CHEMBL1213529

0.16 0.065 CHEMBL3706541

CHEMBL3706542
0.0020.7630.09Squalene synthetase inhibitor

0.09 0.007 CHEMBL1213529

CHEMBL1213529
0.0020.7630.068Peroxisome proliferator-activated receptor alpha agonist

0.068 0.023 CHEMBL1213529

CHEMBL1213529
0.0030.7670.21Monophenol monooxygenase inhibitor

0.095 0.08 CHEMBL721

0.21 0.031 CHEMBL1213529

CHEMBL1213529
0.0060.7730.063Botulinum neurotoxin type A inhibitor

0.063 0.033 CHEMBL3706542

0.06 0.038 CHEMBL1213529

CHEMBL3706542
0.0030.7710.032Angiotensin II receptor antagonist

0.032 0.027 CHEMBL1213529

CHEMBL1213529
0.0020.7710.052Cannabinoid CB1 receptor agonist

0.052 0.051 CHEMBL913

CHEMBL913
0.0010.7710.036Progesterone antagonist

0.036 0.025 CHEMBL1213529

CHEMBL1213529
0.0060.7770.193Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase inhibitor

0.193 0.104 CHEMBL1213529

CHEMBL1213529
0.0030.7750.029ICAM 1 antagonist

0.029 0.007 CHEMBL1213529

CHEMBL1213529
0.010.7850.154Interleukin 8 antagonist

0.154 0.032 CHEMBL1213529

CHEMBL1213529
0.0040.7790.041Melatonin 2 agonist

0.041 0.015 CHEMBL913

CHEMBL913
0.020.7950.394Insulysin inhibitor

0.192 0.169 CHEMBL506976

0.284 0.069 CHEMBL721

0.394 0.023 CHEMBL3706542

0.357 0.032 CHEMBL1213529

0.228 0.119 CHEMBL913

0.238 0.108 CHEMBL3706541

CHEMBL3706542
0.0020.7790.04Leukocyte elastase inhibitor

0.04 0.033 CHEMBL1213529

CHEMBL1213529
0.0050.7830.095Caspase 7 inhibitor

0.095 0.034 CHEMBL506976

0.092 0.038 CHEMBL721

0.081 0.058 CHEMBL1213529

CHEMBL506976
0.0020.7810.044Angiotensin AT1 receptor antagonist

0.044 0.026 CHEMBL1213529

CHEMBL1213529
0.0190.7990.297Cyclophilin D inhibitor

0.297 0.166 CHEMBL1213529

CHEMBL1213529
0.010.7910.16Antibacterial (Helicobacter pylori)

0.133 0.063 CHEMBL1213529

0.16 0.039 CHEMBL913

CHEMBL913
0.0180.8010.162Hexokinase inhibitor

0.143 0.087 CHEMBL506976

0.162 0.065 CHEMBL721

0.158 0.07 CHEMBL1213529

CHEMBL721
0.0110.7930.467Antithrombotic

0.276 0.106 CHEMBL506976

0.326 0.074 CHEMBL721

0.446 0.039 CHEMBL3706542

0.467 0.034 CHEMBL1213529

0.191 0.189 CHEMBL913

CHEMBL1213529
0.0130.7990.261Hypoxia-inducible factor 1 alpha inhibitor

0.261 0.09 CHEMBL506976

0.209 0.141 CHEMBL721

0.23 0.119 CHEMBL1213529

0.209 0.142 CHEMBL913

CHEMBL506976
0.0050.7910.126Alkaline phosphatase inhibitor

0.126 0.079 CHEMBL1213529

CHEMBL1213529
0.0050.7950.052Fatty acid synthase inhibitor

0.052 0.048 CHEMBL1213529

CHEMBL1213529
0.0060.7960.063Cyclin D1 inhibitor

0.063 0.039 CHEMBL721

CHEMBL721
0.0010.7960.042Urate transporter 1 inhibitor

0.042 0.024 CHEMBL1213529

CHEMBL1213529
0.0090.8050.154Xanthine oxidase inhibitor

0.095 0.064 CHEMBL721

0.154 0.033 CHEMBL1213529

CHEMBL1213529
0.0050.8020.102Plasminogen activator inhibitor

0.064 0.036 CHEMBL731

0.102 0.015 CHEMBL506976

0.069 0.033 CHEMBL3706542

CHEMBL506976
0.0130.8110.113Phosphodiesterase 6D inhibitor

0.089 0.077 CHEMBL721

0.113 0.032 CHEMBL1213529

CHEMBL1213529
0.0190.8170.145MAP kinase 3 inhibitor

0.129 0.109 CHEMBL721

0.145 0.076 CHEMBL1213529

CHEMBL1213529
0.0030.8010.079Thromboxane synthase inhibitor

0.079 0.012 CHEMBL1213529

CHEMBL1213529
0.0080.8080.086MDM2 inhibitor

0.086 0.014 CHEMBL1213529

CHEMBL1213529
0.0050.8110.173Interleukin 1 beta converting enzyme inhibitor

0.126 0.031 CHEMBL506976

0.136 0.024 CHEMBL721

0.173 0.01 CHEMBL3706542

0.136 0.024 CHEMBL1213529

0.084 0.083 CHEMBL913

CHEMBL3706542
0.0040.810.035Caspase 6 inhibitor

0.035 0.013 CHEMBL506976

0.03 0.023 CHEMBL3706542

CHEMBL506976
0.0130.8190.167NADPH oxidase inhibitor

0.163 0.047 CHEMBL506976

0.167 0.045 CHEMBL721

0.114 0.091 CHEMBL1213529

CHEMBL721
0.0220.8290.518Histamine release inhibitor

0.255 0.152 CHEMBL721

0.407 0.072 CHEMBL3706542

0.518 0.023 CHEMBL1213529

0.217 0.183 CHEMBL3706541

CHEMBL1213529
0.010.8190.055Sodium/calcium exchanger inhibitor

0.055 0.025 CHEMBL913

CHEMBL913
0.0040.8130.132Macrophage migration inhibitory factor inhibitor

0.132 0.021 CHEMBL1213529

CHEMBL1213529
0.0070.8180.103Beta glucuronidase inhibitor

0.103 0.066 CHEMBL721

0.09 0.088 CHEMBL1213529

CHEMBL721
0.0020.8140.093Xanthine dehydrogenase inhibitor

0.093 0.018 CHEMBL721

0.093 0.018 CHEMBL1213529

CHEMBL1213529
0.0030.8160.072Adrenaline agonist

0.072 0.068 CHEMBL913

CHEMBL913
0.0020.8150.106Leukotriene antagonist

0.106 0.019 CHEMBL1213529

CHEMBL1213529
0.0030.8180.341TRPA1 antagonist

0.077 0.027 CHEMBL506976

0.341 0.004 CHEMBL721

CHEMBL721
0.0020.8210.041Cathepsin L1 inhibitor

0.041 0.026 CHEMBL3706542

CHEMBL3706542
0.0040.8240.112Beta amyloid protein antagonist

0.112 0.076 CHEMBL1213529

CHEMBL1213529
0.020.8410.144Transcription factor NF kappa B stimulant

0.082 0.066 CHEMBL721

0.08 0.069 CHEMBL3706539

0.142 0.018 CHEMBL3706542

0.144 0.017 CHEMBL1213529

0.121 0.024 CHEMBL3706541

CHEMBL1213529
0.0030.8280.059Cannabinoid CB1 receptor antagonist

0.059 0.046 CHEMBL913

CHEMBL913
0.0040.8320.297Pyruvate kinase inhibitor

0.201 0.08 CHEMBL721

0.297 0.048 CHEMBL1213529

CHEMBL1213529
0.010.8380.058Factor III inhibitor

0.058 0.02 CHEMBL1213529

CHEMBL1213529
0.0010.8320.036Prostaglandin EP4 antagonist

0.036 0.012 CHEMBL1213529

CHEMBL1213529
0.0160.8470.349Gastrin inhibitor

0.22 0.119 CHEMBL721

0.182 0.176 CHEMBL3706542

0.349 0.011 CHEMBL1213529

0.204 0.143 CHEMBL913

CHEMBL1213529
0.0050.8380.14Neuropeptide Y1 antagonist

0.14 0.082 CHEMBL913

CHEMBL913
0.0130.8470.484Vasodilator, peripheral

0.207 0.168 CHEMBL721

0.484 0.031 CHEMBL1213529

0.199 0.177 CHEMBL913

CHEMBL1213529
0.0110.8460.273ATPase inhibitor

0.177 0.062 CHEMBL506976

0.273 0.009 CHEMBL721

0.241 0.016 CHEMBL1213529

0.141 0.118 CHEMBL913

CHEMBL721
0.0150.8490.182DNA polymerase I inhibitor

0.182 0.034 CHEMBL1213529

CHEMBL1213529
0.0030.8430.064Cannabinoid receptor antagonist

0.064 0.057 CHEMBL913

CHEMBL913
0.0040.8440.112MAP kinase kinase 1 inhibitor

0.112 0.043 CHEMBL1213529

CHEMBL1213529
0.0030.8450.083Peroxisome proliferator-activated receptor gamma antagonist

0.083 0.03 CHEMBL1213529

CHEMBL1213529
0.0130.8590.201Histone acetyltransferase inhibitor

0.169 0.114 CHEMBL506976

0.201 0.068 CHEMBL913

CHEMBL913
0.0030.8550.113Inducible nitric-oxide synthase inhibitor

0.113 0.028 CHEMBL3706542

0.095 0.041 CHEMBL1213529

0.079 0.064 CHEMBL913

CHEMBL3706542
0.0010.8550.028Aminopeptidase P inhibitor

0.028 0.011 CHEMBL3706542

0.021 0.019 CHEMBL3706541

CHEMBL3706542
0.0050.8640.235Transcription factor STAT3 inhibitor

0.235 0.096 CHEMBL721

0.217 0.114 CHEMBL1213529

CHEMBL721
0.0030.8640.082Antineoplastic antibiotic

0.078 0.058 CHEMBL721

0.082 0.056 CHEMBL1213529

CHEMBL1213529
0.0020.8630.049Liver X receptor alpha agonist

0.049 0.02 CHEMBL1213529

CHEMBL1213529
0.0020.8650.039Renin inhibitor

0.039 0.024 CHEMBL3706542

CHEMBL3706542
0.0070.8740.232Cell wall synthesis inhibitor

0.137 0.078 CHEMBL721

0.168 0.049 CHEMBL3706542

0.232 0.02 CHEMBL1213529

CHEMBL1213529
0.0090.8770.272Chymotrypsin inhibitor

0.272 0.005 CHEMBL506976

0.116 0.027 CHEMBL721

0.085 0.048 CHEMBL3706539

0.108 0.031 CHEMBL3706542

0.094 0.04 CHEMBL913

CHEMBL506976
0.0080.8830.249DNA methylase inhibitor

0.249 0.049 CHEMBL3706542

0.247 0.05 CHEMBL1213529

CHEMBL3706542
0.0050.880.565Topoisomerase II alpha inhibitor

0.17 0.02 CHEMBL506976

0.565 0.004 CHEMBL913

CHEMBL913
00.8780.012Immunosuppressant Cyclosporine-like

0.011 0.008 CHEMBL721

0.012 0.008 CHEMBL3706542

CHEMBL3706542
0.0090.890.122CDK3/cyclin E inhibitor

0.122 0.053 CHEMBL913

CHEMBL913
0.0030.8840.11MAP kinase kinase inhibitor

0.11 0.084 CHEMBL1213529

CHEMBL1213529
0.0040.8860.294Insulin sensitizer

0.158 0.123 CHEMBL721

0.228 0.049 CHEMBL3706542

0.294 0.017 CHEMBL1213529

CHEMBL1213529
0.0030.8860.156Nitric-oxide synthase inhibitor

0.099 0.061 CHEMBL721

0.156 0.02 CHEMBL3706542

0.09 0.078 CHEMBL1213529

0.091 0.076 CHEMBL913

CHEMBL3706542
0.0050.8910.203Transcription factor STAT inhibitor

0.203 0.134 CHEMBL721

0.194 0.148 CHEMBL1213529

CHEMBL721
0.0030.8940.23112-Lipoxygenase inhibitor

0.19 0.162 CHEMBL721

0.231 0.121 CHEMBL1213529

CHEMBL1213529
0.0040.8940.141Mediator release inhibitor

0.141 0.033 CHEMBL1213529

CHEMBL1213529
0.0030.9020.274Cyclin-dependent kinase 5 inhibitor

0.201 0.022 CHEMBL506976

0.274 0.012 CHEMBL913

CHEMBL913
0.0060.9060.266DNA methyltransferase I inhibitor

0.139 0.117 CHEMBL721

0.163 0.091 CHEMBL3706542

0.266 0.04 CHEMBL1213529

CHEMBL1213529
0.0070.9170.05Glutamate (mGluR8) antagonist

0.048 0.009 CHEMBL3706542

0.05 0.008 CHEMBL1213529

0.045 0.012 CHEMBL3706541

CHEMBL1213529
0.0040.9150.238Non-steroidal antiinflammatory agent

0.177 0.09 CHEMBL721

0.238 0.048 CHEMBL1213529

CHEMBL1213529
0.010.9260.101Adenine nucleotide translocase inhibitor

0.054 0.042 CHEMBL3706539

0.101 0.004 CHEMBL3706542

0.091 0.005 CHEMBL3706541

CHEMBL3706542
0.0040.9250.38Antibacterial

0.219 0.208 CHEMBL506976

0.375 0.088 CHEMBL721

0.373 0.089 CHEMBL3706542

0.38 0.086 CHEMBL1213529

CHEMBL1213529
0.0030.9240.179Diuretic

0.179 0.054 CHEMBL1213529

CHEMBL1213529
0.0030.9290.27215-Lipoxygenase inhibitor

0.272 0.148 CHEMBL1213529

CHEMBL1213529
0.0050.9340.061Neurokinin 2 agonist

0.061 0.012 CHEMBL3706542

0.038 0.034 CHEMBL3706541

CHEMBL3706542
0.0030.9320.109Gastric antisecretory

0.109 0.055 CHEMBL1213529

CHEMBL1213529
0.0040.9340.518Growth factor antagonist

0.348 0.022 CHEMBL1593

0.243 0.036 CHEMBL3544547

0.194 0.048 CHEMBL525

0.518 0.01 CHEMBL3706540

CHEMBL3706540
0.0050.9360.122Hemostatic

0.122 0.11 CHEMBL1213529

CHEMBL1213529
0.0060.9420.133Tumour necrosis factor antagonist

0.133 0.122 CHEMBL721

CHEMBL721
0.0020.9410.253Lipoxygenase inhibitor

0.253 0.098 CHEMBL1213529

CHEMBL1213529
0.0030.9460.098Aminopeptidase N inhibitor

0.098 0.014 CHEMBL3706542

0.086 0.016 CHEMBL3706541

CHEMBL3706542
0.0350.9830.349Peptidyltransferase inhibitor

0.215 0.081 CHEMBL721

0.198 0.102 CHEMBL3706539

0.307 0.022 CHEMBL3706542

0.329 0.016 CHEMBL1213529

0.349 0.012 CHEMBL913

0.253 0.049 CHEMBL3706541

CHEMBL913
0.0080.9610.061Integrin alpha1beta1 antagonist

0.037 0.029 CHEMBL3706542

0.061 0.004 CHEMBL1213529

CHEMBL1213529
0.0030.9560.118Plasmin inhibitor

0.118 0.014 CHEMBL506976

0.088 0.02 CHEMBL721

0.079 0.022 CHEMBL3706542

CHEMBL506976
0.0040.9580.132Antipruritic

0.132 0.118 CHEMBL1213529

CHEMBL1213529
0.0020.9570.0361,3-Beta-glucan synthase inhibitor

0.036 0.005 CHEMBL731

CHEMBL731
0.0030.9620.117Aminopeptidase microsomal inhibitor

0.117 0.013 CHEMBL3706542

0.105 0.016 CHEMBL3706541

CHEMBL3706542
0.0190.9780.182Lipocortins synthesis antagonist

0.182 0.069 CHEMBL1213529

CHEMBL1213529
00.960.012Calcineurin inhibitor

0.012 0.007 CHEMBL1213529

CHEMBL1213529
0.0290.990.172ErbB-1 antagonist

0.172 0.13 CHEMBL721

0.166 0.141 CHEMBL1213529

CHEMBL721
0.0020.9650.037Bradykinin B2 receptor agonist

0.037 0.013 CHEMBL3706542

0.027 0.021 CHEMBL3706541

CHEMBL3706542
0.010.9740.3953C-Like protease (SARS coronavirus) inhibitor

0.395 0.003 CHEMBL506976

0.08 0.069 CHEMBL1593

0.324 0.003 CHEMBL721

0.117 0.021 CHEMBL3706542

CHEMBL506976
0.0080.9740.056Cathepsin E inhibitor

0.056 0.047 CHEMBL3706542

0.056 0.047 CHEMBL1213529

CHEMBL1213529
0.0040.970.144Estrogen antagonist

0.144 0.026 CHEMBL1213529

CHEMBL1213529
0.0060.9750.169Acetylcholine M3 receptor agonist

0.169 0.011 CHEMBL3544546

CHEMBL3544546
0.0140.9820.139Folate antagonist

0.139 0.027 CHEMBL3706542

0.09 0.086 CHEMBL1213529

0.128 0.033 CHEMBL3706541

CHEMBL3706542
0.0040.9730.143Aminoacyl-tRNA synthetase inhibitor

0.143 0.021 CHEMBL3706542

0.08 0.078 CHEMBL1213529

0.105 0.04 CHEMBL3706541

CHEMBL3706542
0.0020.9720.056Collagenase inhibitor

0.056 0.022 CHEMBL3706542

0.053 0.026 CHEMBL3706541

CHEMBL3706542
0.020.9920.359Interleukin 2 agonist

0.224 0.151 CHEMBL3706539

0.359 0.042 CHEMBL3706542

0.331 0.055 CHEMBL1213529

0.294 0.078 CHEMBL3706541

CHEMBL3706542
0.0020.9760.15Leukotriene A4 hydrolase inhibitor

0.094 0.006 CHEMBL3706539

0.15 0.005 CHEMBL3706542

0.062 0.014 CHEMBL3706541

CHEMBL3706542
0.0060.9810.035Calcium-independent phospholipase A2 inhibitor

0.035 0.02 CHEMBL3706542

0.033 0.027 CHEMBL1213529

CHEMBL3706542
0.0030.9790.057Neuraminidase inhibitor

0.057 0.047 CHEMBL1213529

CHEMBL1213529
0.0090.9880.061Prolactin release inhibitor

0.061 0.049 CHEMBL1213529

CHEMBL1213529
0.0030.9830.116Protein 50S ribosomal subunit inhibitor

0.095 0.014 CHEMBL506976

0.116 0.01 CHEMBL721

CHEMBL721
0.0040.9830.073Human rhinovirus A protease inhibitor

0.06 0.035 CHEMBL506976

0.073 0.027 CHEMBL3706542

CHEMBL3706542
0.0010.9810.024Integrin beta3 antagonist

0.024 0.011 CHEMBL1213529

CHEMBL1213529
0.0020.9820.243Bruton tyrosine kinase inhibitor

0.243 0.005 CHEMBL721

0.133 0.009 CHEMBL1213529

CHEMBL721
0.0020.9820.045HMG CoA reductase inhibitor

0.045 0.01 CHEMBL1213529

CHEMBL1213529
0.0120.9930.358Factor V inhibitor

0.358 0.001 CHEMBL506976

0.176 0.01 CHEMBL1593

0.332 0.001 CHEMBL721

0.116 0.043 CHEMBL3706539

0.235 0.003 CHEMBL3706542

0.139 0.024 CHEMBL3706541

CHEMBL506976
0.0040.9840.06Cholecystokinin B agonist

0.06 0.012 CHEMBL3706542

0.041 0.022 CHEMBL3706541

CHEMBL3706542
0.0070.9880.055Gonadotropin-releasing hormone receptor agonist

0.055 0.05 CHEMBL913

CHEMBL913
0.0040.9870.093Somatostatin 1 agonist

0.093 0.039 CHEMBL3706542

CHEMBL3706542
0.0030.9860.246Antiadrenergic

0.246 0.018 CHEMBL913

CHEMBL913
0.0020.9850.276Calpain 1 inhibitor

0.276 0.002 CHEMBL506976

0.2 0.003 CHEMBL721

0.049 0.005 CHEMBL3706542

CHEMBL506976
0.0040.9870.443Topoisomerase II inhibitor

0.443 0.008 CHEMBL913

CHEMBL913
0.0030.9870.22Adrenaline antagonist

0.22 0.02 CHEMBL913

CHEMBL913
0.0040.9880.393Antioxidant

0.235 0.092 CHEMBL3544547

0.256 0.08 CHEMBL721

0.169 0.144 CHEMBL3706540

0.28 0.07 CHEMBL3706542

0.393 0.036 CHEMBL1213529

0.278 0.07 CHEMBL3706541

CHEMBL1213529
0.0090.9930.389ABCA1 expression enhancer

0.191 0.01 CHEMBL506976

0.128 0.026 CHEMBL721

0.096 0.056 CHEMBL3706542

0.389 0.004 CHEMBL1213529

CHEMBL1213529
0.0120.9960.134Papain-like protease (SARS coronavirus) inhibitor

0.134 0.053 CHEMBL721

0.124 0.072 CHEMBL1213529

CHEMBL721
0.010.9960.393Growth hormone agonist

0.15 0.087 CHEMBL3706539

0.393 0.017 CHEMBL3706542

0.336 0.025 CHEMBL1213529

0.262 0.04 CHEMBL3706541

CHEMBL3706542
0.0040.9890.052Cathepsin F inhibitor

0.052 0.011 CHEMBL3706542

0.041 0.031 CHEMBL3706541

CHEMBL3706542
0.0090.9950.431Sodium/bile acid cotransporter inhibitor

0.343 0.044 CHEMBL3706539

0.431 0.01 CHEMBL3706542

0.339 0.047 CHEMBL1213529

0.395 0.018 CHEMBL3706541

CHEMBL3706542
0.0040.990.092Bombesin 1 receptor agonist

0.092 0.02 CHEMBL3706542

0.053 0.051 CHEMBL3706541

CHEMBL3706542
0.0050.9920.057Kallikrein 1 inhibitor

0.057 0.039 CHEMBL3706542

CHEMBL3706542
0.0070.9950.086Ca(v)3.1 blocker

0.086 0.044 CHEMBL721

CHEMBL721
0.0040.9910.207Chelator

0.207 0.023 CHEMBL3706542

0.155 0.034 CHEMBL1213529

0.129 0.046 CHEMBL3706541

CHEMBL3706542
0.0030.9910.051Bombesin antagonist

0.051 0.028 CHEMBL3706542

CHEMBL3706542
0.0030.9920.193Tubulin antagonist

0.193 0.039 CHEMBL913

CHEMBL913
0.0020.9910.137CDK4/cyclin D1 inhibitor

0.137 0.008 CHEMBL721

CHEMBL721
0.0040.9930.238Insulin secretagoues

0.238 0.022 CHEMBL1213529

CHEMBL1213529
0.0010.990.191ErbB-4 antagonist

0.149 0.021 CHEMBL721

0.191 0.014 CHEMBL1213529

CHEMBL1213529
0.0030.9920.445MAP3K7 inhibitor

0.065 0.063 CHEMBL721

0.445 0.003 CHEMBL1213529

CHEMBL1213529
0.0020.9910.077CDK4/cyclin D inhibitor

0.077 0.023 CHEMBL721

CHEMBL721
0.0040.9930.238Vasodilator

0.238 0.076 CHEMBL721

0.23 0.082 CHEMBL1213529

CHEMBL721
0.0060.9950.435Hematopoietic

0.091 0.048 CHEMBL3706539

0.435 0.004 CHEMBL3706542

0.278 0.005 CHEMBL3706541

CHEMBL3706542
0.0030.9920.099ATPase (Vacuolar H+) inhibitor

0.099 0.041 CHEMBL1213529

CHEMBL1213529
0.0020.9920.047Growth hormone release inhibitor

0.047 0.024 CHEMBL3706542

CHEMBL3706542
0.0040.9930.33Free radical scavenger

0.221 0.082 CHEMBL721

0.209 0.09 CHEMBL3706542

0.33 0.044 CHEMBL1213529

CHEMBL1213529
0.0030.9930.067Analgesic, opioid

0.067 0.066 CHEMBL3706542

CHEMBL3706542
0.0040.9940.446Angiogenesis stimulant

0.238 0.076 CHEMBL3706539

0.446 0.016 CHEMBL3706542

0.281 0.056 CHEMBL1213529

0.358 0.03 CHEMBL3706541

CHEMBL3706542
0.0050.9950.069Vanilloid 2 antagonist

0.069 0.015 CHEMBL3706542

0.048 0.047 CHEMBL3706541

CHEMBL3706542
00.9910.009Phosphoribosylglycinamide formyltransferase inhibitor

0.009 0.004 CHEMBL3706542

CHEMBL3706542
0.0010.9920.038Leukotriene B4 receptor 2 antagonist

0.038 0.005 CHEMBL1213529

CHEMBL1213529
0.0050.9960.87Caspase 3 stimulant

0.252 0.11 CHEMBL506976

0.87 0.003 CHEMBL721

0.378 0.051 CHEMBL1213529

0.277 0.091 CHEMBL913

CHEMBL721
0.0050.9960.083DNA helicase inhibitor

0.083 0.01 CHEMBL1213529

CHEMBL1213529
0.0040.9950.186ErbB-3 antagonist

0.128 0.026 CHEMBL721

0.186 0.011 CHEMBL1213529

CHEMBL1213529
0.0020.9930.056Carbonic anhydrase I stimulant

0.056 0.013 CHEMBL3706542

0.035 0.029 CHEMBL3706541

CHEMBL3706542
0.0030.9940.089Estrogen receptor beta antagonist

0.089 0.085 CHEMBL1213529

CHEMBL1213529
0.0060.9980.585NOS3 expression enhancer

0.205 0.039 CHEMBL721

0.585 0.004 CHEMBL1213529

CHEMBL1213529
00.9920.014Carbonic anhydrase IV stimulant

0.014 0.013 CHEMBL3706542

CHEMBL3706542
0.0040.9960.064Carbonic anhydrase II stimulant

0.064 0.019 CHEMBL3706542

0.049 0.041 CHEMBL3706541

CHEMBL3706542
0.0030.9950.111Thrombin inhibitor

0.098 0.027 CHEMBL506976

0.111 0.021 CHEMBL3706542

CHEMBL3706542
0.0030.9950.372Antimitotic

0.372 0.028 CHEMBL913

CHEMBL913
0.0040.9960.478Platelet adhesion inhibitor

0.478 0.006 CHEMBL721

0.167 0.09 CHEMBL3706542

0.325 0.026 CHEMBL1213529

CHEMBL721
0.0030.9950.42Thrombolytic

0.164 0.072 CHEMBL3706539

0.42 0.009 CHEMBL3706542

0.19 0.057 CHEMBL1213529

0.341 0.018 CHEMBL3706541

CHEMBL3706542
0.0030.9950.055Cathepsin D inhibitor

0.055 0.037 CHEMBL3706542

CHEMBL3706542
0.0030.9950.349Hypolipemic

0.349 0.035 CHEMBL1213529

CHEMBL1213529
0.0030.9950.135Factor XII inhibitor

0.121 0.023 CHEMBL506976

0.078 0.07 CHEMBL721

0.135 0.017 CHEMBL3706542

0.078 0.071 CHEMBL3706541

CHEMBL3706542
0.0030.9950.183Protease inhibitor

0.113 0.054 CHEMBL506976

0.096 0.069 CHEMBL721

0.183 0.018 CHEMBL3706542

0.101 0.065 CHEMBL3706541

CHEMBL3706542
0.0030.9950.043DNA gyrase subunit A inhibitor

0.043 0.027 CHEMBL3544546

CHEMBL3544546
0.0030.9950.193VCAM-1 antagonist

0.044 0.016 CHEMBL3706542

0.193 0.004 CHEMBL1213529

CHEMBL1213529
0.0030.9950.193VCAM antagonist

0.044 0.016 CHEMBL3706542

0.193 0.004 CHEMBL1213529

CHEMBL1213529
0.0010.9940.06Prostaglandin D2 agonist

0.06 0.005 CHEMBL1213529

CHEMBL1213529
0.0030.9950.153Histone deacetylase class III inhibitor

0.153 0.042 CHEMBL3706542

CHEMBL3706542
0.0030.9960.388Hypoglycemic

0.198 0.115 CHEMBL721

0.388 0.03 CHEMBL1213529

CHEMBL1213529
0.0030.9960.246Histone deacetylase SIRT1 inhibitor

0.246 0.018 CHEMBL3706542

0.158 0.055 CHEMBL3706541

CHEMBL3706542
0.0020.9950.057Farnesyltransferase inhibitor

0.057 0.022 CHEMBL3706542

CHEMBL3706542
0.0020.9950.228Cathepsin B inhibitor

0.228 0.004 CHEMBL506976

0.188 0.005 CHEMBL721

0.157 0.006 CHEMBL3706542

CHEMBL506976
0.0030.9950.091Nitric oxide donor

0.091 0.014 CHEMBL3706542

0.059 0.05 CHEMBL3706541

CHEMBL3706542
0.0030.9960.089Prostaglandin F2 alpha antagonist

0.089 0.016 CHEMBL1213529

CHEMBL1213529
0.0020.9950.058Neurotensin receptor antagonist

0.058 0.024 CHEMBL3706542

0.039 0.038 CHEMBL3706541

CHEMBL3706542
0.0030.9960.479EphB2 antagonist

0.479 0.008 CHEMBL1213529

CHEMBL1213529
0.0020.9950.094Lipase inhibitor

0.094 0.031 CHEMBL721

CHEMBL721
0.0020.9950.265Protein-tyrosine phosphatase 1B inhibitor

0.265 0.014 CHEMBL1213529

CHEMBL1213529
0.0030.9970.111Caspase 9 inhibitor

0.107 0.012 CHEMBL506976

0.111 0.011 CHEMBL721

0.097 0.015 CHEMBL3706542

0.063 0.041 CHEMBL1213529

CHEMBL721
0.0020.9950.074Erythropoietin receptor agonist

0.074 0.014 CHEMBL3706542

0.045 0.024 CHEMBL3706541

CHEMBL3706542
0.0020.9950.434Prostaglandin EP2 antagonist

0.434 0.004 CHEMBL1213529

CHEMBL1213529
0.0020.9950.107Glucagon-like peptide 1 agonist

0.057 0.05 CHEMBL3706539

0.107 0.018 CHEMBL3706542

0.075 0.038 CHEMBL3706541

CHEMBL3706542
0.0030.9960.443Apoptosis antagonist

0.316 0.075 CHEMBL721

0.443 0.029 CHEMBL3706542

0.372 0.047 CHEMBL1213529

0.198 0.181 CHEMBL3706541

CHEMBL3706542
0.0020.9960.087Trypsin inhibitor

0.061 0.045 CHEMBL721

0.087 0.023 CHEMBL3706542

CHEMBL3706542
0.0020.9960.369Anticoagulant

0.369 0.019 CHEMBL3706542

0.127 0.103 CHEMBL3706541

CHEMBL3706542
0.0010.9950.074Retinoic acid gamma receptor agonist

0.074 0.003 CHEMBL1213529

CHEMBL1213529
0.0030.9960.114Nav1.4 sodium channel blocker

0.114 0.058 CHEMBL3706542

CHEMBL3706542
00.9940.014Antibiotic Macrolide-like

0.014 0.01 CHEMBL721

CHEMBL721
0.0030.9960.454Platelet antagonist

0.346 0.039 CHEMBL3706542

0.454 0.019 CHEMBL1213529

CHEMBL1213529
0.0010.9950.077GP IIb/IIIa receptor antagonist

0.077 0.022 CHEMBL3706542

0.047 0.035 CHEMBL1213529

CHEMBL3706542
0.0020.9960.493Nitric oxide antagonist

0.493 0.016 CHEMBL721

0.42 0.023 CHEMBL1213529

CHEMBL721
0.0020.9960.146Retinoic acid alpha receptor agonist

0.146 0.003 CHEMBL1213529

CHEMBL1213529
0.0030.9970.373Interleukin 6 antagonist

0.373 0.009 CHEMBL1213529

CHEMBL1213529
0.0030.9970.041HCV polyprotein inhibitor

0.041 0.011 CHEMBL1213529

CHEMBL1213529
0.0020.9970.234Tumour necrosis factor alpha release inhibitor

0.234 0.083 CHEMBL1213529

CHEMBL1213529
00.9950.0373C-Like protease (MERS coronavirus) inhibitor

0.037 0.002 CHEMBL506976

0.036 0.002 CHEMBL721

CHEMBL506976
0.0010.9950.077Complement C3a chemotactic receptor antagonist

0.077 0.015 CHEMBL3706542

0.05 0.026 CHEMBL3706541

CHEMBL3706542
0.0020.9960.122HIV-1 integrase inhibitor

0.122 0.014 CHEMBL1213529

CHEMBL1213529
0.0020.9970.096Elastase 1 inhibitor

0.096 0.023 CHEMBL721

CHEMBL721
0.0020.9960.323Protein-tyrosine phosphatase inhibitor

0.323 0.015 CHEMBL1213529

CHEMBL1213529
0.0010.9960.041Protocollagen prolyl hydroxylase inhibitor

0.041 0.007 CHEMBL3706542

0.025 0.023 CHEMBL3706541

CHEMBL3706542
0.0020.9960.12Sirtuin 1 inhibitor

0.12 0.014 CHEMBL3706542

0.061 0.058 CHEMBL1213529

0.066 0.05 CHEMBL3706541

CHEMBL3706542
0.0010.9950.104Retinoic acid beta receptor agonist

0.104 0.003 CHEMBL1213529

CHEMBL1213529
0.0010.9950.185Retinoid X gamma receptor agonist

0.185 0.002 CHEMBL1213529

CHEMBL1213529
0.0010.9950.293Retinoid X beta receptor agonist

0.293 0.002 CHEMBL1213529

CHEMBL1213529
0.0020.9960.134CDC25A inhibitor

0.134 0.015 CHEMBL1213529

CHEMBL1213529
0.0020.9960.112Cell adhesion molecule inhibitor

0.112 0.027 CHEMBL1213529

CHEMBL1213529
0.0020.9960.099Aldose reductase inhibitor

0.099 0.018 CHEMBL1213529

CHEMBL1213529
0.0010.9960.044Trypsin I inhibitor

0.044 0.015 CHEMBL3706542

CHEMBL3706542
0.0020.9960.055Neuropeptide agonist

0.055 0.04 CHEMBL3706542

CHEMBL3706542
0.0020.9970.546Interleukin antagonist

0.546 0.016 CHEMBL3706542

0.295 0.049 CHEMBL1213529

0.336 0.041 CHEMBL3706541

CHEMBL3706542
0.0010.9960.053Opioid delta receptor antagonist

0.053 0.052 CHEMBL3706542

CHEMBL3706542
0.0010.9960.104Fibroblast growth factor 4 antagonist

0.104 0.008 CHEMBL721

0.074 0.023 CHEMBL1213529

CHEMBL721
0.0020.9970.229Interleukin 1 antagonist

0.229 0.023 CHEMBL1213529

CHEMBL1213529
0.0010.9960.026Cathepsin K inhibitor

0.025 0.021 CHEMBL506976

0.026 0.019 CHEMBL3706542

CHEMBL3706542
0.0010.9960.053Kinesin antagonist

0.034 0.031 CHEMBL3706542

0.053 0.015 CHEMBL3706541

CHEMBL3706541
0.0010.9960.053Kinesin-like protein 1 inhibitor

0.034 0.031 CHEMBL3706542

0.053 0.015 CHEMBL3706541

CHEMBL3706541
0.0010.9960.057Integrin alpha5beta1 antagonist

0.057 0.013 CHEMBL3706542

0.038 0.033 CHEMBL3706541

CHEMBL3706542
0.0010.9960.02Prostaglandin EP1 antagonist

0.02 0.014 CHEMBL1213529

CHEMBL1213529
0.0010.9960.083Integrin antagonist

0.049 0.027 CHEMBL3706542

0.083 0.019 CHEMBL1213529

CHEMBL1213529
0.0010.9960.033Integrin beta5 antagonist

0.033 0.008 CHEMBL1213529

CHEMBL1213529
0.0010.9960.141Selectin antagonist

0.141 0.019 CHEMBL3706542

0.105 0.026 CHEMBL1213529

0.07 0.042 CHEMBL3706541

CHEMBL3706542
0.0010.9960.128Retinoic acid receptor agonist

0.128 0.004 CHEMBL1213529

CHEMBL1213529
0.0020.9970.093Falcipain inhibitor

0.093 0.06 CHEMBL721

CHEMBL721
0.0010.9960.106Retinoid X gamma receptor antagonist

0.106 0.001 CHEMBL1213529

CHEMBL1213529
0.0020.9970.239Cell adhesion inhibitor

0.239 0.016 CHEMBL1213529

CHEMBL1213529
0.0010.9970.034Cyclophilin A inhibitor

0.034 0.017 CHEMBL3706539

CHEMBL3706539
0.0020.9970.13Lipid peroxidase inhibitor

0.13 0.083 CHEMBL1213529

CHEMBL1213529
0.0020.9980.158Interleukin 4 antagonist

0.122 0.083 CHEMBL721

0.158 0.043 CHEMBL1213529

CHEMBL1213529
0.0010.9960.026Vitronectin receptor antagonist

0.026 0.012 CHEMBL1213529

CHEMBL1213529
0.0010.9970.111HIV-1 integrase (3'-Processing) inhibitor

0.111 0.022 CHEMBL1213529

CHEMBL1213529
0.0010.9970.088CDC25B inhibitor

0.076 0.031 CHEMBL721

0.088 0.022 CHEMBL1213529

CHEMBL1213529
0.0010.9970.097Prostaglandin E2 antagonist

0.097 0.015 CHEMBL1213529

CHEMBL1213529
00.9960.086Retinoic acid alpha receptor antagonist

0.086 0.003 CHEMBL1213529

CHEMBL1213529
0.0010.9970.095Transcription factor AP-1 inhibitor

0.095 0.014 CHEMBL1213529

CHEMBL1213529
0.0010.9970.133HIV-1 integrase (Strand Transfer) inhibitor

0.068 0.037 CHEMBL721

0.133 0.014 CHEMBL1213529

CHEMBL1213529
0.0010.9960.033Prostacyclin agonist

0.033 0.005 CHEMBL1213529

CHEMBL1213529
0.0010.9960.05VLA-4 antagonist

0.032 0.017 CHEMBL3706542

0.05 0.013 CHEMBL1213529

CHEMBL1213529
0.0010.9970.173Peroxisome proliferator-activated receptor gamma agonist

0.173 0.009 CHEMBL1213529

CHEMBL1213529
0.0010.9970.213Prostaglandin antagonist

0.213 0.006 CHEMBL1213529

CHEMBL1213529
00.9960.035Retinoic acid receptor gamma antagonist

0.035 0.004 CHEMBL1213529

CHEMBL1213529
0.0010.9970.183Uric acid excretion stimulant

0.09 0.065 CHEMBL721

0.183 0.016 CHEMBL1213529

CHEMBL1213529
0.0010.9970.042Macrophage elastase inhibitor

0.042 0.032 CHEMBL3706542

CHEMBL3706542
0.0010.9970.109Leukotriene B4 receptor 1 antagonist

0.109 0.004 CHEMBL1213529

CHEMBL1213529
0.0010.9970.075Prostacyclin antagonist

0.075 0.006 CHEMBL1213529

CHEMBL1213529
0.0010.9970.026NMDA 2D receptor antagonist

0.026 0.02 CHEMBL1213529

CHEMBL1213529
0.0020.9980.218Interleukin 1b antagonist

0.218 0.016 CHEMBL1213529

CHEMBL1213529
00.9960.04Retinoic acid beta receptor antagonist

0.04 0.004 CHEMBL1213529

CHEMBL1213529
0.0010.9970.091Leukotriene synthesis inhibitor

0.091 0.031 CHEMBL1213529

CHEMBL1213529
0.0010.9970.036Peroxisome proliferator-activated receptor delta antagonist

0.036 0.019 CHEMBL1213529

CHEMBL1213529
0.0010.9970.082Retinoic acid receptor antagonist

0.082 0.003 CHEMBL1213529

CHEMBL1213529
0.0010.9970.06Plasminogen activator inhibitor antagonist

0.06 0.024 CHEMBL1213529

CHEMBL1213529
0.0010.9970.058Prostaglandin D2 antagonist

0.058 0.006 CHEMBL1213529

CHEMBL1213529
0.0010.9980.163Amyloid beta precursor protein antagonist

0.163 0.087 CHEMBL721

CHEMBL721
0.0010.9970.024Free fatty acid receptor 1 agonist

0.024 0.008 CHEMBL1213529

CHEMBL1213529
0.0010.9970.161Prostaglandin EP3 antagonist

0.161 0.004 CHEMBL1213529

CHEMBL1213529
0.0010.9980.0965-Lipoxygenase inhibitor

0.096 0.067 CHEMBL1213529

CHEMBL1213529
Ext Pa Pi Pmax Activity Other Results ID Pa_max