| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.529 | 0.003 | 0.567 | Gastric antisecretory | 0.486 0.003 CID_19369784 0.318 0.004 CID_154700079 0.567 0.003 CID_154699560 | CID_154699560 | |
| 0.302 | 0.045 | 0.326 | Potassium channel blocker | 0.257 0.063 CID_19369784 0.326 0.039 CID_154700079 0.29 0.05 CID_154699560 | CID_154700079 | |
| 0.312 | 0.06 | 0.315 | Hypoxia-inducible factor 1 alpha inhibitor | 0.315 0.059 CID_19369784 0.204 0.148 CID_154700079 0.282 0.075 CID_154699560 | CID_19369784 | |
| 0.298 | 0.052 | 0.302 | Antiamyloidogenic | 0.297 0.053 CID_19369784 0.302 0.051 CID_154700079 0.218 0.088 CID_154699560 | CID_154700079 | |
| 0.239 | 0.004 | 0.245 | H+/K+-transporting ATPase inhibitor | 0.234 0.004 CID_19369784 0.233 0.004 CID_154700079 0.245 0.004 CID_154699560 | CID_154699560 | |
| 0.202 | 0.008 | 0.202 | Phosphodiesterase 4B inhibitor | 0.084 0.033 CID_19369784 0.141 0.014 CID_154700079 0.094 0.028 CID_154699560 | ||
| 0.197 | 0.004 | 0.227 | Potassium channel (ATP-sensitive) blocker | 0.168 0.004 CID_19369784 0.148 0.005 CID_154700079 0.227 0.004 CID_154699560 | CID_154699560 | |
| 0.204 | 0.027 | 0.281 | Protein-tyrosine kinase (PTK, not ETK, WZC) inhibitor | 0.207 0.026 CID_19369784 0.281 0.013 CID_154700079 0.161 0.042 CID_154699560 | CID_154700079 | |
| 0.203 | 0.027 | 0.28 | Abl kinase inhibitor | 0.206 0.027 CID_19369784 0.28 0.013 CID_154700079 0.161 0.042 CID_154699560 | CID_154700079 | |
| 0.198 | 0.039 | 0.206 | ATPase inhibitor | 0.206 0.032 CID_19369784 0.157 0.091 CID_154700079 0.141 0.118 CID_154699560 | CID_19369784 | |
| 0.161 | 0.004 | 0.161 | Potassium channel (Inward rectifier) blocker | 0.128 0.005 CID_19369784 0.104 0.006 CID_154700079 0.105 0.006 CID_154699560 | ||
| 0.174 | 0.02 | 0.23 | Pim-1 kinase inhibitor | 0.201 0.014 CID_19369784 0.221 0.012 CID_154700079 0.23 0.011 CID_154699560 | CID_154699560 | |
| 0.26 | 0.107 | 0.3 | Immunomodulator | 0.3 0.082 CID_19369784 0.281 0.093 CID_154700079 0.244 0.12 CID_154699560 | CID_19369784 | |
| 0.22 | 0.067 | 0.22 | Platelet aggregation inhibitor | 0.166 0.111 CID_19369784 0.2 0.081 CID_154700079 | ||
| 0.176 | 0.058 | 0.188 | Catenin beta inhibitor | 0.188 0.043 CID_19369784 0.145 0.117 CID_154700079 0.183 0.048 CID_154699560 | CID_19369784 | |
| 0.163 | 0.055 | 0.163 | Toll-Like receptor 9 antagonist | 0.133 0.075 CID_19369784 | ||
| 0.301 | 0.193 | 0.316 | Caspase 9 stimulant | 0.274 0.224 CID_19369784 0.301 0.193 CID_154700079 0.316 0.176 CID_154699560 | CID_154699560 | |
| 0.152 | 0.048 | 0.179 | Interleukin 4 antagonist | 0.179 0.03 CID_19369784 0.153 0.047 CID_154699560 | CID_19369784 | |
| 0.144 | 0.04 | 0.199 | Platelet activating factor beta antagonist | 0.107 0.058 CID_19369784 0.199 0.025 CID_154700079 | CID_154700079 | |
| 0.125 | 0.026 | 0.14 | Phosphodiesterase 4D inhibitor | 0.087 0.043 CID_19369784 0.14 0.021 CID_154700079 0.106 0.035 CID_154699560 | CID_154700079 | |
| 0.152 | 0.055 | 0.152 | Toll-Like receptor antagonist | 0.151 0.055 CID_19369784 | ||
| 0.172 | 0.075 | 0.267 | Tumour necrosis factor antagonist | 0.166 0.081 CID_154700079 0.267 0.026 CID_154699560 | CID_154699560 | |
| 0.113 | 0.023 | 0.127 | Phosphodiesterase 11A inhibitor | 0.096 0.036 CID_19369784 0.113 0.024 CID_154700079 0.127 0.017 CID_154699560 | CID_154699560 | |
| 0.113 | 0.023 | 0.127 | Phosphodiesterase XI inhibitor | 0.096 0.036 CID_19369784 0.113 0.024 CID_154700079 0.127 0.017 CID_154699560 | CID_154699560 | |
| 0.227 | 0.139 | 0.256 | Ca(v)3.3 blocker | 0.205 0.182 CID_19369784 0.256 0.092 CID_154700079 0.238 0.119 CID_154699560 | CID_154700079 | |
| 0.113 | 0.046 | 0.134 | Hedgehog signaling inhibitor | 0.119 0.04 CID_19369784 0.113 0.047 CID_154700079 0.134 0.031 CID_154699560 | CID_154699560 | |
| 0.087 | 0.025 | 0.098 | MAP kinase 7 inhibitor | 0.08 0.044 CID_19369784 0.098 0.009 CID_154700079 0.088 0.022 CID_154699560 | CID_154700079 | |
| 0.158 | 0.097 | 0.163 | Platelet adhesion inhibitor | 0.163 0.093 CID_19369784 | CID_19369784 | |
| 0.211 | 0.154 | 0.261 | Caspase 3 stimulant | 0.2 0.17 CID_19369784 0.21 0.155 CID_154700079 0.261 0.103 CID_154699560 | CID_154699560 | |
| 0.115 | 0.066 | 0.123 | Interleukin 1b antagonist | 0.123 0.06 CID_154700079 0.096 0.086 CID_154699560 | CID_154700079 | |
| 0.115 | 0.067 | 0.148 | Platelet activating factor antagonist | 0.148 0.045 CID_154700079 | CID_154700079 | |
| 0.095 | 0.049 | 0.154 | 5 Hydroxytryptamine 2C antagonist | 0.154 0.026 CID_154700079 | CID_154700079 | |
| 0.113 | 0.069 | 0.115 | Sphingosine 1-phosphate receptor 2 agonist | 0.115 0.063 CID_19369784 0.108 0.078 CID_154699560 | CID_19369784 | |
| 0.122 | 0.08 | 0.122 | Phosphodiesterase inhibitor | 0.106 0.098 CID_154700079 0.122 0.08 CID_154699560 | ||
| 0.091 | 0.052 | 0.091 | Phosphodiesterase IV inhibitor | 0.08 0.062 CID_154700079 | ||
| 0.101 | 0.065 | 0.113 | Nav1.1 sodium channel blocker | 0.109 0.057 CID_19369784 0.113 0.053 CID_154700079 | CID_154700079 | |
| 0.132 | 0.096 | 0.143 | Sphingosine 1-phosphate receptor 5 antagonist | 0.143 0.074 CID_19369784 | CID_19369784 | |
| 0.2 | 0.167 | 0.279 | Ca2+/calmodulin-dependent kinase IV inhibitor | 0.206 0.149 CID_19369784 0.279 0.037 CID_154700079 | CID_154700079 | |
| 0.069 | 0.038 | 0.069 | Aryl hydrocarbon receptor antagonist | 0.069 0.039 CID_19369784 0.061 0.052 CID_154699560 | ||
| 0.213 | 0.186 | 0.215 | Toll-Like receptor agonist | 0.215 0.184 CID_19369784 0.207 0.193 CID_154699560 | CID_19369784 | |
| 0.117 | 0.093 | 0.246 | Ribosomal protein S6 kinase inhibitor | 0.134 0.077 CID_19369784 0.246 0.022 CID_154700079 | CID_154700079 | |
| 0.057 | 0.034 | 0.114 | Pim-2 kinase inhibitor | 0.074 0.023 CID_19369784 0.08 0.02 CID_154700079 0.114 0.012 CID_154699560 | CID_154699560 | |
| 0.055 | 0.034 | 0.055 | Melanin-concentrating hormone receptor 1 antagonist | 0.053 0.037 CID_154699560 | ||
| 0.054 | 0.033 | 0.055 | Phosphodiesterase 4A inhibitor | 0.055 0.032 CID_154700079 0.052 0.034 CID_154699560 | CID_154700079 | |
| 0.06 | 0.041 | 0.073 | Potassium channel (Ca-activated) blocker | 0.066 0.032 CID_154700079 0.073 0.024 CID_154699560 | CID_154699560 | |
| 0.137 | 0.119 | 0.169 | Amyloid beta aggregation inhibitor | 0.155 0.104 CID_19369784 0.169 0.095 CID_154699560 | CID_154699560 | |
| 0.085 | 0.066 | 0.134 | Pim-3 kinase inhibitor | 0.098 0.047 CID_19369784 0.134 0.024 CID_154700079 0.111 0.036 CID_154699560 | CID_154700079 | |
| 0.054 | 0.04 | 0.059 | Phosphodiesterase II inhibitor | 0.059 0.034 CID_154700079 0.056 0.038 CID_154699560 | CID_154700079 | |
| 0.054 | 0.04 | 0.068 | Phosphodiesterase 4C inhibitor | 0.068 0.028 CID_154700079 | CID_154700079 | |
| 0.152 | 0.138 | 0.193 | Growth factor agonist | 0.157 0.127 CID_19369784 0.193 0.07 CID_154699560 | CID_154699560 | |
| 0.081 | 0.071 | 0.159 | Alpha adrenoreceptor antagonist | 0.159 0.035 CID_154700079 | CID_154700079 | |
| 0.043 | 0.033 | 0.064 | 5 Hydroxytryptamine 2C agonist | 0.043 0.034 CID_19369784 0.064 0.018 CID_154700079 | CID_154700079 | |
| 0.144 | 0.135 | 0.299 | Ca2+/calmodulin-dependent kinase II beta inhibitor | 0.158 0.117 CID_19369784 0.181 0.093 CID_154700079 0.299 0.037 CID_154699560 | CID_154699560 | |
| 0.047 | 0.039 | 0.051 | Phosphodiesterase 2A inhibitor | 0.051 0.033 CID_154700079 0.048 0.037 CID_154699560 | CID_154700079 | |
| 0.077 | 0.074 | 0.097 | Antiadrenergic | 0.097 0.058 CID_154700079 | CID_154700079 | |
| 0.065 | 0.063 | 0.129 | Nav1.8 sodium channel blocker | 0.129 0.018 CID_154700079 0.068 0.059 CID_154699560 | CID_154700079 | |
| 0.075 | 0.073 | 0.094 | Adrenaline antagonist | 0.094 0.057 CID_154700079 | CID_154700079 | |
| 0.009 | 0.008 | 0.013 | Corticotropin releasing factor antagonist | 0.013 0.005 CID_154700079 | CID_154700079 | |
| 0.076 | 0.082 | 0.083 | T cell inhibitor | 0.083 0.054 CID_154699560 | CID_154699560 | |
| 0.012 | 0.018 | 0.017 | Purinergic P2Y1 antagonist | 0.017 0.01 CID_154700079 | CID_154700079 | |
| 0.046 | 0.056 | 0.052 | Alpha 1L adrenoreceptor antagonist | 0.052 0.037 CID_154700079 | CID_154700079 | |
| 0.115 | 0.125 | 0.121 | MAP3K9 inhibitor | 0.121 0.113 CID_154700079 | CID_154700079 | |
| 0.09 | 0.104 | 0.171 | Beta amyloid protein antagonist | 0.171 0.028 CID_154700079 | CID_154700079 | |
| 0.086 | 0.1 | 0.111 | Topoisomerase II inhibitor | 0.111 0.075 CID_19369784 0.109 0.077 CID_154699560 | CID_19369784 | |
| 0.069 | 0.086 | 0.094 | MAP kinase kinase 7 inhibitor | 0.094 0.018 CID_19369784 | CID_19369784 | |
| 0.042 | 0.064 | 0.063 | NMDA 2B receptor antagonist | 0.063 0.029 CID_19369784 | CID_19369784 | |
| 0.104 | 0.13 | 0.121 | Thrombolytic | 0.121 0.109 CID_19369784 | CID_19369784 | |
| 0.099 | 0.126 | 0.183 | Nav1.6 sodium channel blocker | 0.183 0.026 CID_154700079 | CID_154700079 | |
| 0.107 | 0.135 | 0.287 | Ca2+/calmodulin-dependent kinase II gamma inhibitor | 0.152 0.087 CID_154700079 0.287 0.037 CID_154699560 | CID_154699560 | |
| 0.169 | 0.203 | 0.212 | Transcription factor NF kappa B inhibitor | 0.212 0.158 CID_19369784 0.194 0.175 CID_154699560 | CID_19369784 | |
| 0.085 | 0.12 | 0.123 | CDC-like kinase 3 inhibitor | 0.123 0.039 CID_154699560 | CID_154699560 | |
| 0.029 | 0.066 | 0.039 | 5 Hydroxytryptamine 2B agonist | 0.039 0.026 CID_154700079 | CID_154700079 | |
| 0.034 | 0.071 | 0.053 | 5 Hydroxytryptamine 2 agonist | 0.053 0.035 CID_154700079 | CID_154700079 | |
| 0.068 | 0.105 | 0.088 | Aminoacyl-tRNA synthetase inhibitor | 0.088 0.062 CID_154699560 | CID_154699560 | |
| 0.048 | 0.087 | 0.072 | Vanilloid antagonist | 0.072 0.054 CID_19369784 | CID_19369784 | |
| 0.05 | 0.094 | 0.067 | Topoisomerase II alpha inhibitor | 0.067 0.064 CID_154699560 | CID_154699560 | |
| 0.014 | 0.059 | 0.018 | Granulocyte colony stimulating factor receptor agonist | 0.018 0.015 CID_154700079 | CID_154700079 | |
| 0.072 | 0.119 | 0.102 | DNA intercalator | 0.102 0.071 CID_154699560 | CID_154699560 | |
| 0.103 | 0.151 | 0.121 | Aurora-C kinase inhibitor | 0.121 0.104 CID_154699560 | CID_154699560 | |
| 0.034 | 0.089 | 0.089 | Alpha 1a adrenoreceptor antagonist | 0.089 0.04 CID_154700079 | CID_154700079 | |
| 0.084 | 0.14 | 0.223 | Sodium channel (voltage-gated) blocker | 0.223 0.022 CID_154700079 | CID_154700079 | |
| 0.044 | 0.101 | 0.059 | Corticotropin releasing factor 2 receptor antagonist | 0.059 0.048 CID_154700079 | CID_154700079 | |
| 0.04 | 0.096 | 0.098 | Alpha 1 adrenoreceptor antagonist | 0.098 0.044 CID_154700079 | CID_154700079 | |
| 0.051 | 0.112 | 0.097 | Bcr-Abl kinase inhibitor | 0.097 0.044 CID_154699560 | CID_154699560 | |
| 0.067 | 0.13 | 0.082 | Transforming growth factor beta 3 antagonist | 0.082 0.058 CID_154700079 | CID_154700079 | |
| 0.114 | 0.177 | 0.132 | MAP kinase kinase 4 inhibitor | 0.132 0.106 CID_19369784 | CID_19369784 | |
| 0.08 | 0.144 | 0.194 | Cytokine production inhibitor | 0.194 0.038 CID_154699560 | CID_154699560 | |
| 0.033 | 0.098 | 0.071 | Factor IXa inhibitor | 0.071 0.02 CID_154700079 | CID_154700079 | |
| 0.047 | 0.112 | 0.065 | I kappa B kinase 1 inhibitor | 0.065 0.056 CID_154699560 | CID_154699560 | |
| 0.079 | 0.152 | 0.269 | Sodium channel blocker | 0.269 0.015 CID_154700079 | CID_154700079 | |
| 0.075 | 0.15 | 0.203 | Nav1.5 sodium channel blocker | 0.203 0.012 CID_154700079 0.1 0.085 CID_154699560 | CID_154700079 | |
| 0.122 | 0.198 | 0.155 | Proto-oncogene tyrosine-protein kinase Fyn inhibitor | 0.155 0.125 CID_154700079 | CID_154700079 | |
| 0.009 | 0.084 | 0.017 | Factor IX inhibitor | 0.017 0.015 CID_154700079 | CID_154700079 | |
| 0.183 | 0.259 | 0.243 | Analgesic | 0.243 0.189 CID_19369784 | CID_19369784 | |
| 0.151 | 0.235 | 0.275 | Ca2+/calmodulin-dependent kinase II alpha inhibitor | 0.275 0.084 CID_154699560 | CID_154699560 | |
| 0.049 | 0.134 | 0.061 | Calcium channel P-type blocker | 0.061 0.056 CID_154700079 | CID_154700079 | |
| 0.107 | 0.192 | 0.146 | Potassium channel (Voltage-sensitive) blocker | 0.146 0.14 CID_154700079 | CID_154700079 | |
| 0.038 | 0.124 | 0.071 | Protein kinase C beta inhibitor | 0.071 0.045 CID_19369784 | CID_19369784 | |
| 0.148 | 0.241 | 0.192 | Nootropic | 0.192 0.169 CID_154700079 | CID_154700079 | |
| 0.052 | 0.152 | 0.096 | 5 Hydroxytryptamine 2 antagonist | 0.096 0.075 CID_154700079 | CID_154700079 | |
| 0.097 | 0.2 | 0.162 | HERG channel blocker | 0.162 0.118 CID_154700079 | CID_154700079 | |
| 0.052 | 0.155 | 0.07 | Estrogen receptor alpha antagonist | 0.07 0.067 CID_19369784 | CID_19369784 | |
| 0.035 | 0.139 | 0.087 | Nav1.7 sodium channel blocker | 0.087 0.029 CID_154700079 | CID_154700079 | |
| 0.186 | 0.298 | 0.248 | Calcium channel L-type activator | 0.248 0.207 CID_19369784 | CID_19369784 | |
| 0.041 | 0.153 | 0.113 | Alpha 2 adrenoreceptor antagonist | 0.113 0.04 CID_154700079 | CID_154700079 | |
| 0.071 | 0.184 | 0.115 | Estrogen antagonist | 0.115 0.065 CID_19369784 | CID_19369784 | |
| 0.082 | 0.196 | 0.254 | Clk dual-specificity kinase inhibitor | 0.254 0.053 CID_154699560 | CID_154699560 | |
| 0.04 | 0.163 | 0.075 | Insulin like growth factor 1 antagonist | 0.075 0.069 CID_154700079 | CID_154700079 | |
| 0.038 | 0.165 | 0.077 | Insulin growth factor antagonist | 0.077 0.071 CID_154700079 | CID_154700079 | |
| 0.056 | 0.185 | 0.097 | Granulocyte macrophage colony stimulating factor agonist | 0.097 0.039 CID_154700079 | CID_154700079 | |
| 0.064 | 0.197 | 0.192 | CDC-like kinase 2 inhibitor | 0.192 0.071 CID_154699560 | CID_154699560 | |
| 0.043 | 0.177 | 0.092 | 5 Hydroxytryptamine antagonist | 0.092 0.087 CID_154700079 | CID_154700079 | |
| 0.071 | 0.205 | 0.213 | CDC-like kinase 4 inhibitor | 0.213 0.061 CID_154699560 | CID_154699560 | |
| 0.061 | 0.196 | 0.094 | mTOR complex 1 inhibitor | 0.094 0.077 CID_154700079 | CID_154700079 | |
| 0.063 | 0.2 | 0.188 | Ca2+/calmodulin-dependent kinase II delta inhibitor | 0.188 0.049 CID_154699560 | CID_154699560 | |
| 0.018 | 0.161 | 0.063 | Dihydrofolate reductase inhibitor | 0.063 0.009 CID_154700079 | CID_154700079 | |
| 0.082 | 0.228 | 0.16 | Polo-like kinase-3 inhibitor | 0.16 0.074 CID_154700079 0.133 0.105 CID_154699560 | CID_154700079 | |
| 0.051 | 0.196 | 0.105 | Proto-oncogene tyrosine-protein kinase Yes inhibitor | 0.105 0.095 CID_154700079 | CID_154700079 | |
| 0.091 | 0.241 | 0.131 | CF transmembrane conductance regulator agonist | 0.131 0.115 CID_154700079 | CID_154700079 | |
| 0.046 | 0.197 | 0.115 | Glycogen synthase kinase-3 alpha inhibitor | 0.115 0.089 CID_154699560 | CID_154699560 | |
| 0.088 | 0.246 | 0.178 | Ca2+/calmodulin-dependent protein kinase inhibitor | 0.178 0.089 CID_154699560 | CID_154699560 | |
| 0.059 | 0.222 | 0.135 | Glutamate release inhibitor | 0.135 0.014 CID_154700079 | CID_154700079 | |
| 0.059 | 0.226 | 0.111 | Protein kinase C nu inhibitor | 0.111 0.103 CID_154699560 | CID_154699560 | |
| 0.049 | 0.217 | 0.094 | Protein kinase C gamma inhibitor | 0.094 0.088 CID_154699560 | CID_154699560 | |
| 0.07 | 0.245 | 0.21 | Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor | 0.21 0.086 CID_154699560 | CID_154699560 | |
| 0.054 | 0.229 | 0.157 | CDC-like kinase 1 inhibitor | 0.157 0.065 CID_154699560 | CID_154699560 | |
| 0.028 | 0.204 | 0.094 | Alpha 2a adrenoreceptor antagonist | 0.094 0.04 CID_154700079 | CID_154700079 | |
| 0.022 | 0.2 | 0.073 | Fibroblast growth factor 3 antagonist | 0.073 0.06 CID_154699560 | CID_154699560 | |
| 0.073 | 0.254 | 0.218 | Dyrk kinase inhibitor | 0.218 0.088 CID_154699560 | CID_154699560 | |
| 0.067 | 0.25 | 0.138 | Interleukin-1 receptor-associated protein kinase 1 inhibitor | 0.138 0.106 CID_154699560 | CID_154699560 | |
| 0.014 | 0.2 | 0.049 | Bruton tyrosine kinase inhibitor | 0.049 0.048 CID_154700079 | CID_154700079 | |
| 0.025 | 0.22 | 0.07 | TIE-2 antagonist | 0.07 0.068 CID_154700079 | CID_154700079 | |
| 0.056 | 0.251 | 0.195 | Dual specificity tyrosine-phosphorylation regulated kinase 3 inhibitor | 0.195 0.08 CID_154699560 | CID_154699560 | |
| 0.059 | 0.263 | 0.161 | TRKC antagonist | 0.161 0.093 CID_154700079 | CID_154700079 | |
| 0.044 | 0.273 | 0.092 | mTOR complex 2 inhibitor | 0.092 0.044 CID_154700079 | CID_154700079 | |
| 0.035 | 0.27 | 0.103 | TRKB antagonist | 0.103 0.096 CID_154700079 | CID_154700079 | |
| 0.074 | 0.341 | 0.162 | DNA damaging | 0.162 0.155 CID_154699560 | CID_154699560 | |
| 0.033 | 0.311 | 0.136 | Dual specificity tyrosine-phosphorylation-regulated kinase 4 inhibitor | 0.136 0.088 CID_154699560 | CID_154699560 | |
| 0.033 | 0.367 | 0.118 | Protein kinase (CK1) gamma 1 inhibitor | 0.118 0.1 CID_154700079 | CID_154700079 | |
| 0.053 | 0.387 | 0.138 | Interleukin 6 antagonist | 0.138 0.11 CID_154699560 | CID_154699560 | |
| 0.062 | 0.4 | 0.217 | Ca2+/calmodulin-dependent kinase I alpha inhibitor | 0.217 0.079 CID_154700079 | CID_154700079 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |