Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.7120.0030.712Histamine H1 receptor antagonist

0.453 0.004 CID_40584683

0.560.0030.594Poly(ADP-ribose) polymerase inhibitor

0.594 0.003 CID_40584683

CID_40584683
0.5550.0040.555Antihistaminic

0.376 0.007 CID_40584683

0.5520.0040.552Histamine antagonist

0.374 0.007 CID_40584683

0.5310.0030.56Poly(ADP-ribose) polymerase 1 inhibitor

0.56 0.003 CID_40584683

CID_40584683
0.5120.0250.512Histamine release inhibitor

0.469 0.041 CID_40584683

0.4520.0050.452Phosphodiesterase inhibitor

0.445 0.005 CID_40584683

0.4570.0630.457Analgesic

0.406 0.082 CID_40584683

0.4250.0510.426Toll-Like receptor 7 agonist

0.426 0.05 CID_40584683

CID_40584683
0.4180.0530.419Toll-Like receptor agonist

0.419 0.053 CID_40584683

CID_40584683
0.3510.0060.351Alpha 1b adrenoreceptor antagonist

0.245 0.01 CID_40584683

0.3380.0040.338Phosphodiesterase I inhibitor

0.241 0.007 CID_40584683

0.3350.0050.341Phosphodiesterase 4D inhibitor

0.341 0.005 CID_40584683

CID_40584683
0.3280.0050.384Phosphodiesterase IV inhibitor

0.384 0.004 CID_40584683

CID_40584683
0.3140.0040.314Histamine H3 receptor antagonist

0.264 0.004 CID_40584683

0.2630.0050.268Phosphodiesterase 4A inhibitor

0.268 0.005 CID_40584683

CID_40584683
0.3140.0650.314Spasmolytic

0.197 0.122 CID_40584683

0.250.0050.255 Hydroxytryptamine 3A agonist

0.219 0.01 CID_40584683

0.3350.0950.435Antiobesity

0.435 0.054 CID_40584683

CID_40584683
0.250.0150.25Alpha 1 adrenoreceptor antagonist

0.188 0.022 CID_40584683

0.2360.0050.274Phosphodiesterase 4B inhibitor

0.274 0.005 CID_40584683

CID_40584683
0.2350.0130.235Alpha 1a adrenoreceptor antagonist

0.186 0.018 CID_40584683

0.240.0210.24Alpha adrenoreceptor antagonist

0.187 0.029 CID_40584683

0.2140.0050.22Phosphodiesterase 4C inhibitor

0.22 0.005 CID_40584683

CID_40584683
0.2720.0650.287Tumour necrosis factor alpha release inhibitor

0.287 0.059 CID_40584683

CID_40584683
0.2260.0230.233Cyclin-dependent kinase 8 inhibitor

0.233 0.02 CID_40584683

CID_40584683
0.210.0090.222Phosphodiesterase 7B inhibitor

0.222 0.008 CID_40584683

CID_40584683
0.190.0050.19Phosphodiesterase 1B inhibitor

0.105 0.013 CID_40584683

0.2440.0690.244HERG channel blocker

0.22 0.079 CID_40584683

0.2640.0960.264Nootropic

0.225 0.13 CID_40584683

0.1630.0040.163Phosphodiesterase VII inhibitor

0.159 0.004 CID_40584683

0.2320.0760.232Potassium channel (Voltage-sensitive) blocker

0.214 0.087 CID_40584683

0.1580.0040.158Phosphodiesterase 1A inhibitor

0.098 0.01 CID_40584683

0.160.0080.165 Hydroxytryptamine 3 antagonist

0.093 0.019 CID_40584683

0.2360.090.2365 Hydroxytryptamine 1E antagonist
0.2080.0650.208Non-steroidal antiinflammatory agent

0.201 0.07 CID_40584683

0.1670.0260.167Bronchodilator

0.166 0.026 CID_40584683

0.2490.1080.249Ca2+/calmodulin-dependent kinase II alpha inhibitor

0.228 0.128 CID_40584683

0.1430.0110.143Bromodomain-containing protein 2 inhibitor

0.126 0.019 CID_40584683

0.1830.0620.183Antipruritic

0.139 0.108 CID_40584683

0.1240.0040.124Phosphodiesterase 7A inhibitor

0.122 0.004 CID_40584683

0.1580.0590.184Hemostatic

0.184 0.04 CID_40584683

CID_40584683
0.1020.010.102Phosphodiesterase 1C inhibitor

0.081 0.019 CID_40584683

0.1130.0210.113Phosphodiesterase 5A inhibitor

0.096 0.029 CID_40584683

0.1140.0230.114Phosphodiesterase XI inhibitor

0.099 0.033 CID_40584683

0.1140.0230.114Phosphodiesterase 11A inhibitor

0.099 0.033 CID_40584683

0.1120.0220.112Phosphodiesterase V inhibitor

0.096 0.03 CID_40584683

0.210.1330.2665 Hydroxytryptamine uptake stimulant

0.266 0.066 CID_40584683

CID_40584683
0.1830.1080.183Cyclic AMP phosphodiesterase inhibitor

0.155 0.144 CID_40584683

0.1090.040.109Acetylcholine M3 receptor agonist

0.1 0.045 CID_40584683

0.0740.010.074Bromodomain-containing protein 3 inhibitor

0.068 0.014 CID_40584683

0.0950.0310.095Cannabinoid receptor antagonist

0.093 0.032 CID_40584683

0.1690.1080.169Anticonvulsant
0.1630.1050.178MAP kinase kinase 5 inhibitor

0.178 0.066 CID_40584683

CID_40584683
0.0810.0260.084Cannabinoid CB1 receptor antagonist

0.084 0.024 CID_40584683

CID_40584683
0.110.060.11Vascular endothelial growth factor 1 antagonist

0.102 0.064 CID_40584683

0.1120.0620.112Acetylcholine release stimulant
0.0650.0170.065Smo receptor antagonist

0.058 0.02 CID_40584683

0.0970.0490.097Acetylcholine agonist

0.079 0.067 CID_40584683

0.0830.0360.083MAP3K7 inhibitor

0.068 0.058 CID_40584683

0.0740.0290.075MDM2 inhibitor

0.075 0.027 CID_40584683

CID_40584683
0.1560.1110.156Psychostimulant

0.147 0.119 CID_40584683

0.1670.1220.182Ca2+/calmodulin-dependent kinase I alpha inhibitor

0.182 0.106 CID_40584683

CID_40584683
0.0740.0320.0745 Hydroxytryptamine 3 agonist

0.057 0.055 CID_40584683

0.0540.0140.054Nerve growth factor antagonist
0.1320.0930.132Acetylcholine M1 receptor antagonist
0.120.0860.12Toll-Like receptor 9 antagonist
0.0440.010.082Poly(ADP-ribose) polymerase 2 inhibitor

0.082 0.005 CID_40584683

CID_40584683
0.0760.0420.076Phosphodiesterase VIII inhibitor

0.075 0.043 CID_40584683

0.20.1670.239Ca2+/calmodulin-dependent kinase IV inhibitor

0.239 0.08 CID_40584683

CID_40584683
0.0640.0310.064Acetylcholine muscarinic agonist
0.0550.0240.055Acetylcholine M1 receptor agonist
0.1980.1670.198Immunomodulator
0.0780.0490.078Acetylcholine M4 receptor antagonist
0.0450.0180.1255 Hydroxytryptamine 2B agonist

0.125 0.004 CID_40584683

CID_40584683
0.0520.0260.052Neurokinin 3 antagonist

0.05 0.028 CID_40584683

0.0670.0450.0675 Hydroxytryptamine 3A antagonist
0.0610.040.061Alpha 1d adrenoreceptor antagonist
0.2680.2470.268Antiinflammatory
0.0680.0470.076Cyclin B3 inhibitor

0.076 0.041 CID_40584683

CID_40584683
0.0860.0650.086Antiadrenergic

0.081 0.07 CID_40584683

0.060.0410.06Acetylcholine M5 receptor antagonist
0.0280.010.032Phosphodiesterase IX inhibitor

0.032 0.007 CID_40584683

CID_40584683
0.0930.0750.093Nav1.1 sodium channel blocker
0.0490.0330.049Histamine H4 receptor antagonist

0.046 0.038 CID_40584683

0.0820.0660.082Adrenaline antagonist

0.077 0.071 CID_40584683

0.0270.0130.03Phosphodiesterase 9A inhibitor

0.03 0.009 CID_40584683

CID_40584683
0.1680.1540.168Cardiotonic
0.1120.0980.112Toll-Like receptor antagonist
0.0510.0370.0855 Hydroxytryptamine 2 agonist

0.085 0.013 CID_40584683

CID_40584683
0.0430.030.069GABA B receptor antagonist

0.069 0.009 CID_40584683

CID_40584683
0.0630.0510.063Acetylcholine M5 receptor agonist
0.1480.1370.148Potassium channel blocker
0.0460.0360.046Dopamine transporter inhibitor
0.1220.1120.122Sigma receptor agonist
0.0470.0390.047Cannabinoid CB2 receptor antagonist
0.0580.050.058Corticotropin releasing factor 2 receptor antagonist
0.0340.0260.034Adenosine uptake inhibitor
0.10.0930.1Interleukin 2 antagonist
0.1130.1070.113Neurotrophic factor
0.0460.040.072Topoisomerase II beta inhibitor

0.072 0.016 CID_40584683

CID_40584683
0.050.0440.053Nicotinic alpha3beta2 receptor antagonist

0.053 0.038 CID_40584683

CID_40584683
0.0580.0530.058Dopamine D1 antagonist
0.0720.0680.087Acetylcholine nicotinic agonist

0.087 0.048 CID_40584683

CID_40584683
0.0680.0650.077Nicotinic alpha4beta2 receptor antagonist

0.077 0.054 CID_40584683

CID_40584683
0.0730.070.073ALK inhibitor
0.1240.1220.143MAP kinase 3 inhibitor

0.143 0.08 CID_40584683

CID_40584683
0.0540.0520.0685 Hydroxytryptamine uptake inhibitor

0.068 0.04 CID_40584683

CID_40584683
0.0830.080.089Protein kinase C zeta inhibitor

0.089 0.067 CID_40584683

CID_40584683
0.0510.0480.051Dopamine uptake inhibitor
0.0110.0080.011CD80 antagonist
0.0360.0350.036Neurokinin 2 antagonist
0.0480.0470.048Dipeptidyl peptidase inhibitor
0.0310.0380.048Somatostatin 4 agonist

0.048 0.016 CID_40584683

CID_40584683
0.0530.060.056Potassium channel (Ca-activated) blocker

0.056 0.05 CID_40584683

CID_40584683
0.1850.1940.197Vasodilator, peripheral

0.197 0.18 CID_40584683

CID_40584683
0.040.0520.044Neurokinin antagonist

0.044 0.043 CID_40584683

CID_40584683
0.0470.0640.061Adrenaline uptake inhibitor

0.061 0.043 CID_40584683

CID_40584683
0.0660.0880.105NMDA receptor antagonist

0.105 0.044 CID_40584683

CID_40584683
0.0390.0620.053Nicotinic neuronal receptor agonist

0.053 0.043 CID_40584683

CID_40584683
0.0280.0520.0965 Hydroxytryptamine 2C agonist

0.096 0.008 CID_40584683

CID_40584683
0.090.1250.116Cytokine production inhibitor

0.116 0.093 CID_40584683

CID_40584683
0.0370.0790.045Nicotinic receptor alpha4 subunit antagonist

0.045 0.044 CID_40584683

CID_40584683
0.2430.30.279Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.279 0.243 CID_40584683

CID_40584683
0.0320.1020.0755 Hydroxytryptamine 2A agonist

0.075 0.032 CID_40584683

CID_40584683
0.10.1770.122Neuropeptide Y1 antagonist

0.122 0.119 CID_40584683

CID_40584683
0.030.110.041Alpha 1L adrenoreceptor agonist

0.041 0.036 CID_40584683

CID_40584683
0.1380.4330.248Calcium channel L-type activator

0.248 0.207 CID_40584683

CID_40584683
Ext Pa Pi Pmax Activity Other Results ID Pa_max