| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.79 | 0.002 | 0.943 | Phosphodiesterase 5A inhibitor | 0.579 0.003 CID_154699828 0.72 0.002 CID_154699990 0.686 0.003 CID_154699935 0.58 0.003 CID_154699749 0.693 0.003 CID_154699748 0.688 0.003 CID_154699578 0.732 0.002 CID_154699573 0.943 0.002 CID_135499879 | CID_135499879 | |
| 0.775 | 0.002 | 0.942 | Phosphodiesterase V inhibitor | 0.563 0.003 CID_154699828 0.694 0.002 CID_154699990 0.657 0.003 CID_154699935 0.563 0.003 CID_154699749 0.666 0.003 CID_154699748 0.658 0.003 CID_154699578 0.709 0.002 CID_154699573 0.942 0.002 CID_135499879 | CID_135499879 | |
| 0.634 | 0.004 | 0.797 | Phosphodiesterase inhibitor | 0.441 0.005 CID_154699828 0.558 0.005 CID_154699990 0.534 0.005 CID_154699935 0.389 0.008 CID_154699749 0.531 0.005 CID_154699748 0.451 0.005 CID_154699578 0.58 0.004 CID_154699573 0.797 0.004 CID_135499879 | CID_135499879 | |
| 0.412 | 0.003 | 0.678 | Phosphodiesterase I inhibitor | 0.134 0.021 CID_154699828 0.309 0.004 CID_154699990 0.241 0.007 CID_154699935 0.126 0.024 CID_154699749 0.202 0.01 CID_154699748 0.124 0.025 CID_154699578 0.307 0.005 CID_154699573 0.678 0.002 CID_135499879 | CID_135499879 | |
| 0.428 | 0.024 | 0.455 | Cardiotonic | 0.385 0.031 CID_154699828 0.395 0.03 CID_154699990 0.455 0.02 CID_154699935 0.312 0.051 CID_154699749 0.401 0.029 CID_154699748 0.3 0.056 CID_154699578 0.398 0.029 CID_154699573 0.321 0.048 CID_135499879 | CID_154699935 | |
| 0.404 | 0.002 | 0.82 | Phosphodiesterase VI inhibitor | 0.148 0.007 CID_154699828 0.325 0.003 CID_154699990 0.345 0.003 CID_154699935 0.17 0.005 CID_154699749 0.303 0.003 CID_154699748 0.165 0.005 CID_154699578 0.34 0.003 CID_154699573 0.82 0.001 CID_135499879 | CID_135499879 | |
| 0.42 | 0.02 | 0.446 | Vasodilator | 0.333 0.038 CID_154699828 0.387 0.025 CID_154699990 0.446 0.017 CID_154699935 0.347 0.034 CID_154699749 0.398 0.023 CID_154699748 0.329 0.039 CID_154699578 0.411 0.021 CID_154699573 0.421 0.02 CID_135499879 | CID_154699935 | |
| 0.289 | 0.003 | 0.722 | Phosphodiesterase 6D inhibitor | 0.119 0.026 CID_154699828 0.226 0.004 CID_154699990 0.301 0.003 CID_154699935 0.199 0.005 CID_154699749 0.287 0.003 CID_154699748 0.144 0.011 CID_154699578 0.242 0.004 CID_154699573 0.722 0.001 CID_135499879 | CID_135499879 | |
| 0.32 | 0.034 | 0.517 | Cyclic AMP phosphodiesterase inhibitor | 0.198 0.095 CID_154699828 0.203 0.091 CID_154699990 0.283 0.049 CID_154699935 0.252 0.063 CID_154699749 0.246 0.066 CID_154699748 0.22 0.08 CID_154699573 0.517 0.006 CID_135499879 | CID_135499879 | |
| 0.288 | 0.003 | 0.565 | Phosphodiesterase 1A inhibitor | 0.087 0.013 CID_154699828 0.167 0.004 CID_154699990 0.081 0.016 CID_154699935 0.068 0.026 CID_154699749 0.075 0.019 CID_154699748 0.071 0.023 CID_154699578 0.166 0.004 CID_154699573 0.565 0.001 CID_135499879 | CID_135499879 | |
| 0.272 | 0.004 | 0.645 | Phosphodiesterase 1B inhibitor | 0.08 0.023 CID_154699828 0.14 0.008 CID_154699990 0.079 0.023 CID_154699935 0.066 0.035 CID_154699748 0.14 0.008 CID_154699573 0.645 0.002 CID_135499879 | CID_135499879 | |
| 0.31 | 0.05 | 0.322 | Platelet antagonist | 0.228 0.083 CID_154699828 0.306 0.051 CID_154699990 0.287 0.057 CID_154699935 0.28 0.06 CID_154699749 0.322 0.046 CID_154699748 0.287 0.057 CID_154699578 0.321 0.046 CID_154699573 | CID_154699748 | |
| 0.192 | 0.019 | 0.225 | Bronchodilator | 0.147 0.032 CID_154699828 0.172 0.024 CID_154699990 0.153 0.031 CID_154699935 0.225 0.015 CID_154699749 0.168 0.026 CID_154699748 0.112 0.05 CID_154699578 0.212 0.017 CID_154699573 0.204 0.018 CID_135499879 | CID_154699749 | |
| 0.16 | 0.002 | 0.291 | Phosphodiesterase 6C inhibitor | 0.085 0.003 CID_154699828 0.123 0.003 CID_154699990 0.11 0.003 CID_154699935 0.09 0.003 CID_154699749 0.111 0.003 CID_154699748 0.109 0.003 CID_154699578 0.127 0.002 CID_154699573 0.291 0.002 CID_135499879 | CID_135499879 | |
| 0.163 | 0.013 | 0.285 | Phosphodiesterase 3A inhibitor | 0.099 0.033 CID_154699828 0.116 0.024 CID_154699990 0.13 0.02 CID_154699935 0.076 0.062 CID_154699749 0.104 0.03 CID_154699748 0.091 0.041 CID_154699578 0.117 0.023 CID_154699573 0.285 0.005 CID_135499879 | CID_135499879 | |
| 0.139 | 0.005 | 0.641 | Phosphodiesterase 1C inhibitor | 0.085 0.016 CID_154699990 0.057 0.056 CID_154699935 0.087 0.015 CID_154699573 0.641 0.001 CID_135499879 | CID_135499879 | |
| 0.161 | 0.041 | 0.189 | Nav1.3 sodium channel blocker | 0.11 0.086 CID_154699828 0.107 0.089 CID_154699990 0.189 0.028 CID_154699935 0.125 0.069 CID_154699749 0.174 0.035 CID_154699748 0.176 0.034 CID_154699573 | CID_154699935 | |
| 0.123 | 0.007 | 0.228 | Phosphodiesterase II inhibitor | 0.119 0.008 CID_154699990 0.12 0.008 CID_154699935 0.1 0.011 CID_154699749 0.103 0.01 CID_154699748 0.081 0.017 CID_154699578 0.121 0.008 CID_154699573 0.228 0.004 CID_135499879 | CID_135499879 | |
| 0.129 | 0.016 | 0.162 | Phosphodiesterase XI inhibitor | 0.108 0.026 CID_154699990 0.093 0.039 CID_154699935 0.091 0.041 CID_154699748 0.09 0.042 CID_154699578 0.107 0.027 CID_154699573 0.162 0.008 CID_135499879 | CID_135499879 | |
| 0.129 | 0.016 | 0.162 | Phosphodiesterase 11A inhibitor | 0.108 0.026 CID_154699990 0.093 0.039 CID_154699935 0.091 0.041 CID_154699748 0.09 0.042 CID_154699578 0.107 0.027 CID_154699573 0.162 0.008 CID_135499879 | CID_135499879 | |
| 0.1 | 0.009 | 0.195 | Phosphodiesterase 2A inhibitor | 0.098 0.009 CID_154699990 0.099 0.009 CID_154699935 0.085 0.012 CID_154699749 0.084 0.012 CID_154699748 0.065 0.021 CID_154699578 0.099 0.009 CID_154699573 0.195 0.004 CID_135499879 | CID_135499879 | |
| 0.109 | 0.018 | 0.299 | Sirtuin 1 inhibitor | 0.109 0.018 CID_154699990 0.107 0.019 CID_154699935 0.07 0.045 CID_154699749 0.1 0.023 CID_154699748 0.299 0.003 CID_154699578 0.105 0.02 CID_154699573 0.122 0.014 CID_135499879 | CID_154699578 | |
| 0.094 | 0.003 | 0.134 | Phosphodiesterase 6B inhibitor | 0.06 0.005 CID_154699828 0.078 0.004 CID_154699990 0.072 0.004 CID_154699935 0.068 0.004 CID_154699749 0.078 0.004 CID_154699748 0.069 0.004 CID_154699578 0.082 0.004 CID_154699573 0.134 0.002 CID_135499879 | CID_135499879 | |
| 0.106 | 0.02 | 0.172 | Phosphodiesterase III inhibitor | 0.09 0.028 CID_154699828 0.106 0.02 CID_154699990 0.091 0.027 CID_154699935 0.079 0.036 CID_154699748 0.106 0.02 CID_154699573 0.172 0.008 CID_135499879 | CID_135499879 | |
| 0.088 | 0.014 | 0.138 | Phosphodiesterase 3B inhibitor | 0.055 0.022 CID_154699828 0.087 0.014 CID_154699990 0.06 0.019 CID_154699935 0.051 0.024 CID_154699748 0.089 0.013 CID_154699573 0.138 0.006 CID_135499879 | CID_135499879 | |
| 0.115 | 0.042 | 0.181 | Phosphodiesterase 7B inhibitor | 0.124 0.035 CID_154699828 0.092 0.067 CID_154699990 0.085 0.078 CID_154699749 0.095 0.063 CID_154699573 0.181 0.013 CID_135499879 | CID_135499879 | |
| 0.098 | 0.027 | 0.098 | Polo-like kinase-2 inhibitor | 0.097 0.028 CID_154699990 0.086 0.038 CID_154699935 0.088 0.037 CID_154699749 0.086 0.038 CID_154699748 0.08 0.044 CID_154699578 0.097 0.028 CID_154699573 0.07 0.053 CID_135499879 | ||
| 0.228 | 0.169 | 0.29 | Toll-Like receptor 7 agonist | 0.245 0.152 CID_154699990 0.236 0.16 CID_154699935 0.29 0.117 CID_154699749 0.248 0.15 CID_154699573 0.221 0.176 CID_135499879 | CID_154699749 | |
| 0.055 | 0.004 | 0.109 | Phosphodiesterase 6A inhibitor | 0.042 0.004 CID_154699828 0.04 0.004 CID_154699990 0.036 0.005 CID_154699935 0.037 0.004 CID_154699749 0.043 0.004 CID_154699748 0.033 0.005 CID_154699578 0.048 0.004 CID_154699573 0.109 0.003 CID_135499879 | CID_135499879 | |
| 0.224 | 0.175 | 0.292 | Toll-Like receptor agonist | 0.244 0.154 CID_154699990 0.234 0.163 CID_154699935 0.292 0.116 CID_154699749 0.246 0.152 CID_154699573 0.218 0.181 CID_135499879 | CID_154699749 | |
| 0.142 | 0.093 | 0.159 | Polo-like kinase-3 inhibitor | 0.156 0.078 CID_154699990 0.131 0.108 CID_154699935 0.133 0.106 CID_154699749 0.128 0.112 CID_154699748 0.159 0.075 CID_154699573 | CID_154699573 | |
| 0.077 | 0.028 | 0.119 | Phosphodiesterase VII inhibitor | 0.063 0.043 CID_154699990 0.067 0.038 CID_154699573 0.119 0.006 CID_135499879 | CID_135499879 | |
| 0.047 | 0.003 | 0.067 | Phosphodiesterase 6G inhibitor | 0.033 0.005 CID_154699828 0.041 0.004 CID_154699990 0.039 0.004 CID_154699935 0.036 0.005 CID_154699749 0.04 0.004 CID_154699748 0.037 0.004 CID_154699578 0.042 0.004 CID_154699573 0.067 0.002 CID_135499879 | CID_135499879 | |
| 0.047 | 0.003 | 0.067 | Phosphodiesterase 6H inhibitor | 0.033 0.005 CID_154699828 0.041 0.004 CID_154699990 0.039 0.004 CID_154699935 0.036 0.005 CID_154699749 0.04 0.004 CID_154699748 0.037 0.004 CID_154699578 0.042 0.004 CID_154699573 0.067 0.002 CID_135499879 | CID_135499879 | |
| 0.16 | 0.117 | 0.172 | Platelet aggregation inhibitor | 0.162 0.115 CID_154699828 0.172 0.105 CID_154699990 0.144 0.136 CID_154699935 0.142 0.14 CID_154699749 0.172 0.105 CID_154699748 0.171 0.106 CID_154699573 | CID_154699748 | |
| 0.069 | 0.044 | 0.069 | Bcl2 antagonist | 0.06 0.054 CID_154699828 0.06 0.055 CID_154699990 0.069 0.043 CID_154699573 | ||
| 0.053 | 0.033 | 0.075 | Phosphodiesterase 7A inhibitor | 0.049 0.042 CID_154699573 0.075 0.009 CID_135499879 | CID_135499879 | |
| 0.03 | 0.014 | 0.03 | Myristoyl transferase inhibitor | 0.028 0.016 CID_154699573 | ||
| 0.059 | 0.045 | 0.059 | Bcl-xL inhibitor | 0.057 0.051 CID_154699828 0.059 0.044 CID_154699990 0.059 0.044 CID_154699573 | ||
| 0.028 | 0.016 | 0.038 | Histone deacetylase class IIb inhibitor | 0.026 0.018 CID_154699990 0.025 0.019 CID_154699573 0.038 0.013 CID_135499879 | CID_135499879 | |
| 0.028 | 0.016 | 0.038 | Histone deacetylase 6 inhibitor | 0.026 0.018 CID_154699990 0.024 0.019 CID_154699573 0.038 0.013 CID_135499879 | CID_135499879 | |
| 0.026 | 0.014 | 0.032 | Phosphodiesterase 9A inhibitor | 0.026 0.014 CID_154699828 0.023 0.021 CID_154699990 0.023 0.021 CID_154699573 0.032 0.008 CID_135499879 | CID_135499879 | |
| 0.033 | 0.024 | 0.04 | Histone deacetylase 2 inhibitor | 0.04 0.018 CID_135499879 | CID_135499879 | |
| 0.023 | 0.016 | 0.031 | Phosphodiesterase IX inhibitor | 0.023 0.017 CID_154699828 0.031 0.008 CID_135499879 | CID_135499879 | |
| 0.028 | 0.021 | 0.034 | Histone deacetylase class II inhibitor | 0.026 0.023 CID_154699990 0.034 0.015 CID_135499879 | CID_135499879 | |
| 0.052 | 0.046 | 0.098 | Adenosine A1 receptor antagonist | 0.098 0.024 CID_135499879 | CID_135499879 | |
| 0.235 | 0.23 | 0.407 | Cyclophilin D inhibitor | 0.29 0.171 CID_154699990 0.338 0.131 CID_154699935 0.277 0.184 CID_154699749 0.407 0.087 CID_154699748 0.291 0.17 CID_154699573 | CID_154699748 | |
| 0.039 | 0.04 | 0.049 | Guanylate cyclase stimulant | 0.049 0.022 CID_135499879 | CID_135499879 | |
| 0.113 | 0.121 | 0.155 | Anticoagulant | 0.155 0.075 CID_154699748 | CID_154699748 | |
| 0.017 | 0.026 | 0.024 | Histone deacetylase 1 inhibitor | 0.024 0.017 CID_135499879 | CID_135499879 | |
| 0.043 | 0.06 | 0.053 | Carbonic anhydrase II stimulant | 0.053 0.034 CID_135499879 | CID_135499879 | |
| 0.013 | 0.041 | 0.019 | Guanylate cyclase 1 stimulant | 0.019 0.014 CID_135499879 | CID_135499879 | |
| 0.049 | 0.083 | 0.061 | ZAP-70 protein tyrosine kinase inhibitor | 0.061 0.06 CID_135499879 | CID_135499879 | |
| 0.05 | 0.096 | 0.076 | I kappa B kinase 1 inhibitor | 0.076 0.041 CID_135499879 | CID_135499879 | |
| 0.06 | 0.118 | 0.107 | Check point kinase 2 inhibitor | 0.086 0.078 CID_154699828 0.107 0.059 CID_135499879 | CID_135499879 | |
| 0.023 | 0.092 | 0.072 | Phosphodiesterase 4A inhibitor | 0.072 0.024 CID_135499879 | CID_135499879 | |
| 0.023 | 0.095 | 0.039 | Nicotinic acid receptor 1 agonist | 0.039 0.03 CID_135499879 | CID_135499879 | |
| 0.143 | 0.216 | 0.2 | Peptidyltransferase inhibitor | 0.174 0.139 CID_154699990 0.178 0.132 CID_154699935 0.186 0.119 CID_154699749 0.163 0.162 CID_154699748 0.2 0.099 CID_135499879 | CID_135499879 | |
| 0.111 | 0.19 | 0.136 | MAP kinase kinase 4 inhibitor | 0.136 0.096 CID_154699828 0.135 0.099 CID_135499879 | CID_154699828 | |
| 0.052 | 0.14 | 0.104 | CDK2/cyclin A inhibitor | 0.104 0.055 CID_135499879 | CID_135499879 | |
| 0.16 | 0.249 | 0.269 | Sodium/bile acid cotransporter inhibitor | 0.214 0.17 CID_154699828 0.229 0.152 CID_154699935 0.217 0.165 CID_154699749 0.205 0.181 CID_154699748 0.269 0.109 CID_135499879 | CID_135499879 | |
| 0.026 | 0.117 | 0.056 | Phosphodiesterase 4C inhibitor | 0.056 0.039 CID_135499879 | CID_135499879 | |
| 0.058 | 0.153 | 0.161 | Cyclin-dependent kinase 2 inhibitor | 0.161 0.034 CID_154699828 0.126 0.049 CID_135499879 | CID_154699828 | |
| 0.081 | 0.183 | 0.132 | Mcl-1 antagonist | 0.132 0.11 CID_154699573 | CID_154699573 | |
| 0.101 | 0.207 | 0.16 | Antipruritic | 0.16 0.084 CID_135499879 | CID_135499879 | |
| 0.031 | 0.154 | 0.065 | CDK2/cyclin E2 inhibitor | 0.065 0.054 CID_135499879 | CID_135499879 | |
| 0.025 | 0.164 | 0.063 | Cyclin B1 inhibitor | 0.063 0.04 CID_135499879 | CID_135499879 | |
| 0.027 | 0.173 | 0.054 | Cyclin H inhibitor | 0.054 0.048 CID_135499879 | CID_135499879 | |
| 0.051 | 0.203 | 0.133 | Cyclin-dependent kinase inhibitor | 0.133 0.065 CID_154699828 | CID_154699828 | |
| 0.032 | 0.192 | 0.097 | CDK/cyclin complex inhibitor | 0.097 0.054 CID_154699828 | CID_154699828 | |
| 0.144 | 0.313 | 0.212 | Interleukin 2 agonist | 0.199 0.192 CID_154699990 0.212 0.169 CID_154699573 | CID_154699573 | |
| 0.016 | 0.197 | 0.051 | Cyclin B2 inhibitor | 0.051 0.046 CID_135499879 | CID_135499879 | |
| 0.073 | 0.256 | 0.214 | Insulin sensitizer | 0.15 0.133 CID_154699935 0.214 0.06 CID_135499879 | CID_135499879 | |
| 0.021 | 0.206 | 0.065 | Phosphodiesterase 4D inhibitor | 0.065 0.06 CID_135499879 | CID_135499879 | |
| 0.031 | 0.227 | 0.082 | I kappa B kinase inhibitor | 0.082 0.058 CID_135499879 | CID_135499879 | |
| 0.019 | 0.225 | 0.109 | Phosphodiesterase 4B inhibitor | 0.109 0.021 CID_135499879 | CID_135499879 | |
| 0.008 | 0.218 | 0.096 | CDK2/cyclin E inhibitor | 0.096 0.024 CID_154699828 | CID_154699828 | |
| 0.024 | 0.237 | 0.106 | Cyclin-dependent kinase 1 inhibitor | 0.106 0.062 CID_135499879 | CID_135499879 | |
| 0.155 | 0.375 | 0.23 | MAP kinase kinase 6 inhibitor | 0.23 0.219 CID_154699828 | CID_154699828 | |
| 0.095 | 0.323 | 0.146 | Catenin beta inhibitor | 0.146 0.116 CID_154699748 | CID_154699748 | |
| 0.009 | 0.242 | 0.086 | Cyclin E1 inhibitor | 0.086 0.023 CID_154699828 | CID_154699828 | |
| 0.009 | 0.243 | 0.103 | Cyclin E inhibitor | 0.103 0.023 CID_154699828 | CID_154699828 | |
| 0.095 | 0.348 | 0.255 | Cyclin-dependent kinase 3 inhibitor | 0.255 0.015 CID_135499879 | CID_135499879 | |
| 0.013 | 0.329 | 0.134 | Phosphodiesterase IV inhibitor | 0.134 0.028 CID_135499879 | CID_135499879 | |
| 0.07 | 0.409 | 0.221 | Hypoglycemic | 0.194 0.118 CID_154699749 0.221 0.096 CID_154699748 | CID_154699748 | |
| 0.003 | 0.354 | 0.049 | Carbonic anhydrase IX inhibitor | 0.049 0.043 CID_135499879 | CID_135499879 | |
| 0.032 | 0.395 | 0.161 | EphB2 antagonist | 0.161 0.119 CID_135499879 | CID_135499879 | |
| 0.003 | 0.373 | 0.045 | Carbonic anhydrase XII inhibitor | 0.045 0.042 CID_135499879 | CID_135499879 | |
| 0.037 | 0.407 | 0.093 | Carbonic anhydrase XV inhibitor | 0.093 0.078 CID_135499879 | CID_135499879 | |
| 0.02 | 0.399 | 0.047 | Antiviral (Hepatitis D) | 0.047 0.042 CID_154699748 | CID_154699748 | |
| 0.02 | 0.451 | 0.189 | Cyclooxygenase 2 inhibitor | 0.189 0.034 CID_135499879 | CID_135499879 | |
| 0.024 | 0.468 | 0.203 | Cyclooxygenase inhibitor | 0.203 0.041 CID_135499879 | CID_135499879 | |
| 0.025 | 0.482 | 0.121 | Electrolyte absorption antagonist | 0.121 0.035 CID_135499879 | CID_135499879 | |
| 0.011 | 0.599 | 0.122 | Cyclooxygenase 1 inhibitor | 0.122 0.078 CID_135499879 | CID_135499879 | |
| 0.025 | 0.617 | 0.27 | Histone deacetylase SIRT1 inhibitor | 0.27 0.013 CID_154699578 | CID_154699578 | |
| 0.012 | 0.689 | 0.15 | Histone deacetylase class III inhibitor | 0.15 0.044 CID_154699578 | CID_154699578 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |