| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.734 | 0.004 | 0.734 | MAP kinase kinase 6 inhibitor | 0.637 0.005 CID_67181 | ||
| 0.594 | 0.01 | 0.594 | Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase inhibitor | 0.584 0.011 CID_67181 | ||
| 0.396 | 0.005 | 0.396 | Sodium channel blocker | 0.329 0.008 CID_67181 | ||
| 0.447 | 0.055 | 0.447 | 15-Lipoxygenase inhibitor | 0.358 0.095 CID_67181 | ||
| 0.385 | 0.025 | 0.385 | Ca2+/calmodulin-dependent kinase II alpha inhibitor | 0.335 0.043 CID_67181 | ||
| 0.373 | 0.016 | 0.373 | MAP kinase kinase 2 inhibitor | 0.285 0.04 CID_67181 | ||
| 0.345 | 0.006 | 0.391 | Nav1.3 sodium channel blocker | 0.391 0.005 CID_67181 | CID_67181 | |
| 0.344 | 0.005 | 0.344 | Sodium channel (voltage-gated) blocker | 0.301 0.008 CID_67181 | ||
| 0.322 | 0.009 | 0.322 | Alkaline phosphatase inhibitor | 0.283 0.014 CID_67181 | ||
| 0.356 | 0.055 | 0.356 | 12-Lipoxygenase inhibitor | 0.345 0.059 CID_67181 | ||
| 0.3 | 0.005 | 0.3 | Nav1.5 sodium channel blocker | 0.223 0.01 CID_67181 | ||
| 0.301 | 0.008 | 0.301 | Carbonic anhydrase XV inhibitor | 0.179 0.023 CID_67181 | ||
| 0.294 | 0.015 | 0.294 | Histone acetyltransferase inhibitor | 0.216 0.048 CID_67181 | ||
| 0.335 | 0.065 | 0.335 | Immunomodulator | 0.254 0.112 CID_67181 | ||
| 0.269 | 0.002 | 0.269 | Dihydropteroate synthase inhibitor | 0.216 0.002 CID_67181 | ||
| 0.286 | 0.02 | 0.286 | Focal adhesion kinase 2 inhibitor | 0.254 0.035 CID_67181 | ||
| 0.268 | 0.008 | 0.268 | Nav1.6 sodium channel blocker | 0.16 0.043 CID_67181 | ||
| 0.274 | 0.032 | 0.274 | Dual specificity tyrosine-phosphorylation-regulated kinase 4 inhibitor | 0.195 0.053 CID_67181 | ||
| 0.27 | 0.029 | 0.27 | LIM domain kinase 1 inhibitor | 0.227 0.05 CID_67181 | ||
| 0.258 | 0.022 | 0.258 | Antipruritic | 0.237 0.029 CID_67181 | ||
| 0.359 | 0.131 | 0.373 | MAP kinase 1 inhibitor | 0.373 0.122 CID_67181 | CID_67181 | |
| 0.255 | 0.027 | 0.255 | MAP kinase kinase 3 inhibitor | 0.193 0.144 CID_67181 | ||
| 0.226 | 0.003 | 0.226 | Glutamate (mGluR4) agonist | 0.112 0.004 CID_67181 | ||
| 0.219 | 0.005 | 0.219 | Nav1.7 sodium channel blocker | 0.176 0.008 CID_67181 | ||
| 0.264 | 0.053 | 0.264 | Ca2+/calmodulin-dependent protein kinase inhibitor | 0.154 0.108 CID_67181 | ||
| 0.225 | 0.018 | 0.225 | Cyclin-dependent kinase 9 inhibitor | 0.13 0.041 CID_67181 | ||
| 0.25 | 0.047 | 0.25 | DNA methyltransferase I inhibitor | 0.245 0.049 CID_67181 | ||
| 0.212 | 0.009 | 0.212 | HIV-1 integrase (3'-Processing) inhibitor | 0.167 0.012 CID_67181 | ||
| 0.211 | 0.009 | 0.211 | HIV-1 integrase (Strand Transfer) inhibitor | 0.151 0.013 CID_67181 | ||
| 0.204 | 0.008 | 0.204 | Carbonic anhydrase IX inhibitor | 0.179 0.01 CID_67181 | ||
| 0.216 | 0.023 | 0.216 | MAP kinase kinase inhibitor | 0.137 0.059 CID_67181 | ||
| 0.195 | 0.004 | 0.195 | Glutamate (mGluR group III) agonist | 0.159 0.004 CID_67181 | ||
| 0.195 | 0.017 | 0.195 | Carbonic anhydrase III inhibitor | 0.162 0.024 CID_67181 | ||
| 0.232 | 0.059 | 0.232 | DNA methylase inhibitor | 0.215 0.069 CID_67181 | ||
| 0.184 | 0.011 | 0.188 | Carbonic anhydrase inhibitor | 0.188 0.011 CID_67181 | CID_67181 | |
| 0.206 | 0.042 | 0.206 | Polo-like kinase-3 inhibitor | 0.159 0.075 CID_67181 | ||
| 0.179 | 0.016 | 0.179 | Carbonic anhydrase VI inhibitor | 0.089 0.048 CID_67181 | ||
| 0.195 | 0.035 | 0.195 | Cyclin-dependent kinase 7 inhibitor | 0.17 0.047 CID_67181 | ||
| 0.197 | 0.037 | 0.217 | Hexokinase inhibitor | 0.217 0.027 CID_67181 | CID_67181 | |
| 0.159 | 0.009 | 0.166 | Carbonic anhydrase II inhibitor | 0.166 0.008 CID_67181 | CID_67181 | |
| 0.161 | 0.012 | 0.161 | CC chemokine 6 receptor antagonist | 0.153 0.018 CID_67181 | ||
| 0.187 | 0.038 | 0.187 | Mannose-6-phosphate isomerase inhibitor | |||
| 0.158 | 0.014 | 0.158 | MAP kinase kinase 1 inhibitor | 0.112 0.043 CID_67181 | ||
| 0.186 | 0.043 | 0.229 | Cyclin-dependent kinase 3 inhibitor | 0.229 0.021 CID_67181 | CID_67181 | |
| 0.159 | 0.02 | 0.159 | Carbonic anhydrase XIII inhibitor | 0.086 0.045 CID_67181 | ||
| 0.141 | 0.013 | 0.141 | Purinergic P2X2 antagonist | 0.086 0.037 CID_67181 | ||
| 0.141 | 0.014 | 0.141 | Carbonic anhydrase XII inhibitor | 0.13 0.015 CID_67181 | ||
| 0.143 | 0.018 | 0.143 | I kappa B kinase inhibitor | 0.101 0.038 CID_67181 | ||
| 0.131 | 0.011 | 0.131 | Carbonic anhydrase VB inhibitor | 0.075 0.025 CID_67181 | ||
| 0.127 | 0.009 | 0.128 | Phosphatidylinositol 3-kinase beta inhibitor | 0.128 0.009 CID_67181 | CID_67181 | |
| 0.19 | 0.073 | 0.19 | TRKC antagonist | |||
| 0.232 | 0.115 | 0.268 | Insulysin inhibitor | 0.268 0.081 CID_67181 | CID_67181 | |
| 0.281 | 0.166 | 0.416 | Transcription factor inhibitor | 0.416 0.103 CID_67181 | CID_67181 | |
| 0.128 | 0.013 | 0.141 | Carbonic anhydrase I inhibitor | 0.141 0.011 CID_67181 | CID_67181 | |
| 0.116 | 0.004 | 0.116 | Transcription factor RelA inhibitor | 0.084 0.014 CID_67181 | ||
| 0.129 | 0.019 | 0.129 | Carbonic anhydrase V inhibitor | 0.122 0.021 CID_67181 | ||
| 0.125 | 0.016 | 0.125 | Carbonic anhydrase VA inhibitor | 0.122 0.017 CID_67181 | ||
| 0.115 | 0.008 | 0.115 | Bombesin 3 receptor antagonist | 0.104 0.011 CID_67181 | ||
| 0.114 | 0.011 | 0.114 | 5 Hydroxytryptamine 6 antagonist | |||
| 0.173 | 0.072 | 0.173 | Mcl-1 antagonist | 0.154 0.086 CID_67181 | ||
| 0.108 | 0.017 | 0.108 | CDK9/cyclin T1 inhibitor | 0.072 0.03 CID_67181 | ||
| 0.103 | 0.012 | 0.103 | I kappa B kinase 2 inhibitor | 0.076 0.026 CID_67181 | ||
| 0.124 | 0.033 | 0.124 | Electrolyte absorption antagonist | 0.111 0.045 CID_67181 | ||
| 0.146 | 0.057 | 0.146 | Cyclooxygenase 2 inhibitor | 0.114 0.086 CID_67181 | ||
| 0.155 | 0.066 | 0.155 | Cyclooxygenase inhibitor | |||
| 0.144 | 0.058 | 0.163 | Aurora-C kinase inhibitor | 0.163 0.038 CID_67181 | CID_67181 | |
| 0.149 | 0.064 | 0.149 | MAP kinase kinase 4 inhibitor | |||
| 0.092 | 0.008 | 0.103 | Carbonic anhydrase IV inhibitor | 0.103 0.006 CID_67181 | CID_67181 | |
| 0.26 | 0.182 | 0.365 | Alpha-glucosidase inhibitor | 0.365 0.129 CID_67181 | CID_67181 | |
| 0.15 | 0.075 | 0.15 | CF transmembrane conductance regulator agonist | 0.129 0.12 CID_67181 | ||
| 0.118 | 0.044 | 0.118 | CDK2/cyclin A inhibitor | 0.09 0.068 CID_67181 | ||
| 0.097 | 0.024 | 0.097 | I kappa B kinase 1 inhibitor | 0.069 0.049 CID_67181 | ||
| 0.114 | 0.041 | 0.114 | Ca(v)2.2 blocker | |||
| 0.192 | 0.12 | 0.192 | Hypoglycemic | |||
| 0.09 | 0.019 | 0.09 | Phosphatidylinositol 3-kinase alpha inhibitor | 0.082 0.021 CID_67181 | ||
| 0.117 | 0.045 | 0.117 | MAP kinase 8 inhibitor | 0.097 0.063 CID_67181 | ||
| 0.084 | 0.016 | 0.084 | Cyclin H inhibitor | 0.067 0.031 CID_67181 | ||
| 0.168 | 0.101 | 0.168 | I kappa B kinase epsilon inhibitor | |||
| 0.165 | 0.099 | 0.165 | Non-steroidal antiinflammatory agent | |||
| 0.131 | 0.07 | 0.164 | Interleukin 4 antagonist | 0.164 0.039 CID_67181 | CID_67181 | |
| 0.084 | 0.024 | 0.084 | Carbonic anhydrase stimulant | 0.078 0.026 CID_67181 | ||
| 0.076 | 0.017 | 0.076 | MAP kinase kinase 9 inhibitor | 0.071 0.02 CID_67181 | ||
| 0.144 | 0.085 | 0.144 | Cyclin-dependent kinase 8 inhibitor | 0.132 0.1 CID_67181 | ||
| 0.128 | 0.074 | 0.128 | Nav1.2 sodium channel blocker | 0.109 0.097 CID_67181 | ||
| 0.08 | 0.026 | 0.08 | Phosphodiesterase VII inhibitor | |||
| 0.083 | 0.031 | 0.083 | ZAP-70 protein tyrosine kinase inhibitor | 0.072 0.046 CID_67181 | ||
| 0.191 | 0.141 | 0.234 | 5 Hydroxytryptamine 1E antagonist | 0.234 0.093 CID_67181 | CID_67181 | |
| 0.055 | 0.004 | 0.055 | 5 Hydroxytryptamine 6 agonist | |||
| 0.135 | 0.085 | 0.157 | Pregnane X receptor agonist | 0.157 0.041 CID_67181 | CID_67181 | |
| 0.079 | 0.029 | 0.079 | Phosphatidylinositol kinase inhibitor | 0.078 0.029 CID_67181 | ||
| 0.1 | 0.05 | 0.1 | Toll-Like receptor 3 antagonist | |||
| 0.141 | 0.091 | 0.141 | Ca2+/calmodulin-dependent protein kinase kinase B inhibitor | |||
| 0.063 | 0.016 | 0.063 | Fructose-1,6-bisphosphatase inhibitor | |||
| 0.055 | 0.009 | 0.055 | Integrin alpha2 antagonist | 0.035 0.03 CID_67181 | ||
| 0.067 | 0.021 | 0.067 | Carbonic anhydrase XIV inhibitor | 0.052 0.031 CID_67181 | ||
| 0.057 | 0.016 | 0.057 | AICAR transformylase inhibitor | 0.048 0.024 CID_67181 | ||
| 0.104 | 0.063 | 0.104 | Aurora-A kinase inhibitor | 0.089 0.076 CID_67181 | ||
| 0.05 | 0.01 | 0.05 | Endothelin receptor antagonist | 0.034 0.015 CID_67181 | ||
| 0.043 | 0.003 | 0.043 | CC chemokine 9 receptor antagonist | 0.024 0.005 CID_67181 | ||
| 0.082 | 0.042 | 0.085 | Polo-like kinase-2 inhibitor | 0.085 0.039 CID_67181 | CID_67181 | |
| 0.044 | 0.005 | 0.044 | Integrin alpha2beta1 antagonist | 0.025 0.02 CID_67181 | ||
| 0.057 | 0.018 | 0.057 | CDK7/cyclin H inhibitor | 0.053 0.021 CID_67181 | ||
| 0.084 | 0.047 | 0.084 | MAP kinase 10 inhibitor | 0.073 0.06 CID_67181 | ||
| 0.109 | 0.073 | 0.109 | Aurora-B kinase inhibitor | 0.107 0.075 CID_67181 | ||
| 0.073 | 0.038 | 0.073 | Bcl2 antagonist | 0.06 0.056 CID_67181 | ||
| 0.109 | 0.077 | 0.109 | Interleukin 8 antagonist | |||
| 0.06 | 0.028 | 0.06 | mTOR inhibitor | 0.057 0.031 CID_67181 | ||
| 0.04 | 0.009 | 0.04 | Methionyl aminopeptidase 2 inhibitor | |||
| 0.076 | 0.046 | 0.076 | S-adenosyl-L-methionine decarboxylase inhibitor | |||
| 0.033 | 0.005 | 0.033 | CC chemokine 8 receptor antagonist | 0.027 0.008 CID_67181 | ||
| 0.115 | 0.088 | 0.115 | Glycogen synthase kinase-3 alpha inhibitor | |||
| 0.054 | 0.027 | 0.054 | Alpha 1b adrenoreceptor agonist | |||
| 0.097 | 0.07 | 0.097 | Folate antagonist | |||
| 0.055 | 0.029 | 0.055 | Phosphodiesterase 7A inhibitor | |||
| 0.032 | 0.007 | 0.032 | Fructose-1,6-bisphosphatase 1 inhibitor | |||
| 0.034 | 0.009 | 0.034 | Endothelin A receptor antagonist | 0.025 0.012 CID_67181 | ||
| 0.147 | 0.122 | 0.147 | Dual specificity tyrosine-phosphorylation regulated kinase 3 inhibitor | |||
| 0.068 | 0.043 | 0.068 | MAP kinase kinase 10 inhibitor | 0.068 0.043 CID_67181 | ||
| 0.149 | 0.124 | 0.149 | Death-associated protein kinase 3 inhibitor | |||
| 0.06 | 0.036 | 0.081 | Potassium channel Kv1.5 blocker | 0.081 0.025 CID_67181 | CID_67181 | |
| 0.033 | 0.01 | 0.033 | Myristoyl transferase inhibitor | 0.03 0.014 CID_67181 | ||
| 0.098 | 0.076 | 0.098 | Alpha 2b adrenoreceptor antagonist | |||
| 0.06 | 0.04 | 0.06 | Bcl-xL inhibitor | |||
| 0.086 | 0.066 | 0.086 | Protein kinase (Mos, Mil/Raf, MEKK, RIPK, TESK, LIMK, IRAK, ILK, Activin/TGF-beta) inhibitor | 0.082 0.07 CID_67181 | ||
| 0.026 | 0.006 | 0.029 | Factor XIII inhibitor | 0.029 0.005 CID_67181 | CID_67181 | |
| 0.09 | 0.071 | 0.09 | MAP kinase 9 inhibitor | |||
| 0.117 | 0.099 | 0.117 | CDC-like kinase 1 inhibitor | |||
| 0.225 | 0.207 | 0.384 | DNA polymerase beta inhibitor | 0.384 0.126 CID_67181 | CID_67181 | |
| 0.141 | 0.124 | 0.141 | Anesthetic general | |||
| 0.201 | 0.185 | 0.433 | Beta lactamase inhibitor | 0.433 0.09 CID_67181 | CID_67181 | |
| 0.135 | 0.12 | 0.135 | Tumour necrosis factor antagonist | |||
| 0.154 | 0.139 | 0.154 | Ca2+/calmodulin-dependent kinase I alpha inhibitor | |||
| 0.097 | 0.087 | 0.109 | CDC-like kinase 3 inhibitor | 0.109 0.06 CID_67181 | CID_67181 | |
| 0.044 | 0.036 | 0.044 | Thymidylate synthase inhibitor | |||
| 0.076 | 0.068 | 0.076 | AXL receptor tyrosine kinase inhibitor | |||
| 0.063 | 0.056 | 0.063 | CDK1/cyclin B1 inhibitor | |||
| 0.017 | 0.01 | 0.017 | CDK2/cyclin A3 inhibitor | |||
| 0.09 | 0.084 | 0.09 | Granulocyte macrophage colony stimulating factor antagonist | |||
| 0.135 | 0.13 | 0.135 | Lipocortins synthesis antagonist | |||
| 0.098 | 0.093 | 0.146 | CDK3/cyclin E inhibitor | 0.146 0.029 CID_67181 | CID_67181 | |
| 0.048 | 0.044 | 0.048 | Carbonic anhydrase II stimulant | |||
| 0.025 | 0.02 | 0.025 | Kynurenine 3 monooxygenase inhibitor | |||
| 0.085 | 0.082 | 0.085 | Lanosterol 14 alpha demethylase inhibitor | |||
| 0.015 | 0.012 | 0.015 | CC chemokine 10 receptor antagonist | |||
| 0.043 | 0.04 | 0.048 | CC chemokine 4 receptor antagonist | 0.048 0.031 CID_67181 | CID_67181 | |
| 0.111 | 0.108 | 0.111 | Protein kinase (CK1) gamma 1 inhibitor | |||
| 0.082 | 0.079 | 0.082 | Polo-like kinase-1 inhibitor | |||
| 0.059 | 0.058 | 0.059 | CDC7 inhibitor | |||
| 0.026 | 0.036 | 0.032 | LIM domain kinase 2 inhibitor | 0.032 0.02 CID_67181 | CID_67181 | |
| 0.203 | 0.226 | 0.325 | DNA directed DNA polymerase inhibitor | 0.325 0.15 CID_67181 | CID_67181 | |
| 0.065 | 0.095 | 0.09 | Neuropeptide Y antagonist | 0.09 0.047 CID_67181 | CID_67181 | |
| 0.155 | 0.193 | 0.17 | 5 Hydroxytryptamine 3E antagonist | 0.17 0.136 CID_67181 | CID_67181 | |
| 0.166 | 0.214 | 0.215 | Angiogenesis inhibitor | 0.215 0.153 CID_67181 | CID_67181 | |
| 0.144 | 0.212 | 0.298 | Thyroid hormone beta antagonist | 0.298 0.089 CID_67181 | CID_67181 | |
| 0.144 | 0.217 | 0.293 | Thyroid hormone antagonist | 0.293 0.097 CID_67181 | CID_67181 | |
| 0.152 | 0.235 | 0.269 | Transcription factor STAT inhibitor | 0.269 0.074 CID_67181 | CID_67181 | |
| 0.164 | 0.263 | 0.228 | Interleukin 2 agonist | 0.228 0.145 CID_67181 | CID_67181 | |
| 0.126 | 0.258 | 0.241 | Transcription factor STAT3 inhibitor | 0.241 0.091 CID_67181 | CID_67181 | |
| 0.106 | 0.253 | 0.192 | Death-associated protein kinase 2 inhibitor | 0.192 0.041 CID_67181 | CID_67181 | |
| 0.054 | 0.212 | 0.109 | M17 leucyl aminopeptidase inhibitor | 0.109 0.089 CID_67181 | CID_67181 | |
| 0.123 | 0.293 | 0.18 | Neuropeptide Y2 antagonist | 0.18 0.161 CID_67181 | CID_67181 | |
| 0.046 | 0.253 | 0.098 | Caspase 3 inhibitor | 0.098 0.096 CID_67181 | CID_67181 | |
| 0.108 | 0.376 | 0.184 | Peptidyltransferase inhibitor | 0.184 0.122 CID_67181 | CID_67181 | |
| 0.007 | 0.445 | 0.059 | Neuraminidase inhibitor | 0.059 0.044 CID_67181 | CID_67181 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |