| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.598 | 0.055 | 0.823 | Beta lactamase inhibitor | 0.823 0.02 CID_65280 | CID_65280 | |
| 0.503 | 0.004 | 0.503 | Histone acetyltransferase inhibitor | 0.286 0.016 CID_114821 0.378 0.005 CID_65280 0.151 0.138 CID_154699808 | ||
| 0.548 | 0.073 | 0.705 | DNA polymerase beta inhibitor | 0.227 0.206 CID_114821 0.705 0.037 CID_65280 | CID_65280 | |
| 0.447 | 0.001 | 0.447 | Dihydropteroate synthase inhibitor | 0.2 0.002 CID_114821 0.385 0.001 CID_65280 0.099 0.005 CID_154699808 | ||
| 0.516 | 0.076 | 0.625 | Alpha-glucosidase inhibitor | 0.335 0.143 CID_114821 0.625 0.049 CID_65280 0.517 0.076 CID_154699808 | CID_65280 | |
| 0.422 | 0.004 | 0.422 | Sodium channel blocker | 0.154 0.056 CID_114821 0.357 0.006 CID_65280 | ||
| 0.489 | 0.086 | 0.619 | DNA directed DNA polymerase inhibitor | 0.309 0.157 CID_114821 0.619 0.051 CID_65280 | CID_65280 | |
| 0.407 | 0.004 | 0.407 | Carbonic anhydrase XV inhibitor | 0.118 0.048 CID_114821 0.286 0.009 CID_65280 | ||
| 0.381 | 0.019 | 0.381 | EphB2 antagonist | 0.215 0.078 CID_114821 0.373 0.02 CID_65280 | ||
| 0.414 | 0.068 | 0.414 | 15-Lipoxygenase inhibitor | 0.324 0.115 CID_65280 | ||
| 0.355 | 0.019 | 0.355 | Non-steroidal antiinflammatory agent | 0.247 0.044 CID_114821 0.27 0.036 CID_65280 0.201 0.07 CID_154699808 | ||
| 0.338 | 0.005 | 0.338 | Sodium channel (voltage-gated) blocker | 0.146 0.057 CID_114821 0.295 0.009 CID_65280 | ||
| 0.294 | 0.017 | 0.294 | Focal adhesion kinase 2 inhibitor | 0.223 0.053 CID_114821 0.264 0.03 CID_65280 | ||
| 0.309 | 0.032 | 0.309 | MAP kinase kinase 2 inhibitor | 0.212 0.074 CID_65280 | ||
| 0.278 | 0.005 | 0.323 | Carbonic anhydrase IX inhibitor | 0.097 0.021 CID_114821 0.25 0.005 CID_65280 0.323 0.004 CID_154699808 | CID_154699808 | |
| 0.311 | 0.052 | 0.338 | Insulysin inhibitor | 0.306 0.055 CID_114821 0.338 0.039 CID_65280 | CID_65280 | |
| 0.258 | 0.008 | 0.258 | Nav1.5 sodium channel blocker | 0.098 0.09 CID_114821 0.191 0.014 CID_65280 | ||
| 0.366 | 0.123 | 0.501 | Transcription factor inhibitor | 0.326 0.141 CID_114821 0.501 0.074 CID_65280 | CID_65280 | |
| 0.245 | 0.006 | 0.333 | Carbonic anhydrase XII inhibitor | 0.069 0.029 CID_114821 0.228 0.007 CID_65280 0.333 0.004 CID_154699808 | CID_154699808 | |
| 0.244 | 0.009 | 0.244 | Carbonic anhydrase VI inhibitor | 0.082 0.055 CID_114821 0.122 0.029 CID_65280 | ||
| 0.247 | 0.018 | 0.282 | Hexokinase inhibitor | 0.282 0.013 CID_65280 0.187 0.044 CID_154699808 | CID_65280 | |
| 0.227 | 0.005 | 0.227 | Nav1.7 sodium channel blocker | 0.094 0.025 CID_114821 0.185 0.007 CID_65280 | ||
| 0.289 | 0.068 | 0.289 | Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase inhibitor | 0.271 0.072 CID_65280 | ||
| 0.225 | 0.013 | 0.225 | Nav1.6 sodium channel blocker | 0.137 0.071 CID_65280 | ||
| 0.217 | 0.008 | 0.428 | Carbonic anhydrase inhibitor | 0.097 0.028 CID_114821 0.222 0.008 CID_65280 0.428 0.004 CID_154699808 | CID_154699808 | |
| 0.204 | 0.004 | 0.204 | Endothelin receptor antagonist | 0.12 0.005 CID_114821 0.16 0.004 CID_65280 0.03 0.017 CID_154699808 | ||
| 0.223 | 0.031 | 0.223 | Tyrosine-protein kinase receptor FLT3 inhibitor | 0.137 0.058 CID_65280 | ||
| 0.201 | 0.014 | 0.201 | Carbonic anhydrase XIII inhibitor | 0.112 0.032 CID_65280 0.136 0.025 CID_154699808 | ||
| 0.221 | 0.036 | 0.221 | Antipruritic | 0.137 0.11 CID_114821 0.202 0.047 CID_65280 | ||
| 0.186 | 0.003 | 0.186 | Cyclophilin A inhibitor | 0.143 0.003 CID_114821 0.184 0.003 CID_65280 0.06 0.005 CID_154699808 | ||
| 0.197 | 0.017 | 0.197 | Carbonic anhydrase III inhibitor | 0.106 0.056 CID_114821 0.163 0.024 CID_65280 | ||
| 0.182 | 0.005 | 0.182 | Bromodomain-containing protein 4 inhibitor | 0.099 0.013 CID_114821 0.144 0.007 CID_65280 | ||
| 0.164 | 0.004 | 0.164 | Endothelin A receptor antagonist | 0.088 0.005 CID_114821 0.126 0.004 CID_65280 0.02 0.016 CID_154699808 | ||
| 0.225 | 0.065 | 0.225 | MAP kinase kinase 3 inhibitor | |||
| 0.193 | 0.037 | 0.193 | Cyclooxygenase 1 inhibitor | 0.17 0.048 CID_114821 0.115 0.085 CID_65280 | ||
| 0.158 | 0.008 | 0.158 | Carbonic anhydrase VB inhibitor | 0.052 0.043 CID_114821 0.091 0.018 CID_65280 | ||
| 0.179 | 0.033 | 0.204 | Nav1.3 sodium channel blocker | 0.204 0.023 CID_65280 | CID_65280 | |
| 0.184 | 0.044 | 0.184 | Ribosomal protein S6 kinase inhibitor | |||
| 0.179 | 0.051 | 0.179 | Cyclooxygenase inhibitor | 0.15 0.07 CID_114821 0.126 0.092 CID_65280 | ||
| 0.15 | 0.022 | 0.163 | CC chemokine 6 receptor antagonist | 0.138 0.045 CID_114821 0.144 0.032 CID_65280 0.163 0.01 CID_154699808 | CID_154699808 | |
| 0.139 | 0.012 | 0.29 | Carbonic anhydrase II inhibitor | 0.056 0.038 CID_114821 0.145 0.011 CID_65280 0.29 0.004 CID_154699808 | CID_154699808 | |
| 0.317 | 0.191 | 0.359 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.359 0.141 CID_65280 | CID_65280 | |
| 0.139 | 0.017 | 0.139 | Carbonic anhydrase V inhibitor | 0.132 0.019 CID_65280 | ||
| 0.132 | 0.015 | 0.132 | Carbonic anhydrase VA inhibitor | 0.129 0.016 CID_65280 | ||
| 0.161 | 0.047 | 0.161 | Cyclooxygenase 2 inhibitor | 0.154 0.051 CID_114821 0.126 0.074 CID_65280 | ||
| 0.139 | 0.032 | 0.139 | Ca(v)2.2 blocker | 0.074 0.071 CID_65280 | ||
| 0.209 | 0.104 | 0.304 | Hypoglycemic | 0.304 0.051 CID_154699808 | CID_154699808 | |
| 0.129 | 0.03 | 0.129 | Electrolyte absorption antagonist | 0.115 0.04 CID_65280 | ||
| 0.14 | 0.042 | 0.184 | Falcipain 3 inhibitor | 0.184 0.023 CID_65280 | CID_65280 | |
| 0.219 | 0.131 | 0.219 | 12-Lipoxygenase inhibitor | 0.211 0.14 CID_65280 | ||
| 0.113 | 0.028 | 0.115 | Bromodomain-containing protein 2 inhibitor | 0.115 0.027 CID_65280 | CID_65280 | |
| 0.081 | 0.004 | 0.081 | Endothelin B receptor antagonist | 0.037 0.008 CID_114821 0.057 0.005 CID_65280 | ||
| 0.086 | 0.012 | 0.086 | Transcription factor RelA inhibitor | 0.064 0.044 CID_65280 | ||
| 0.141 | 0.071 | 0.163 | Pregnane X receptor agonist | 0.163 0.034 CID_65280 | CID_65280 | |
| 0.237 | 0.167 | 0.237 | GABA C receptor rho-3 antagonist | |||
| 0.076 | 0.01 | 0.076 | Bromodomain-containing protein 3 inhibitor | 0.058 0.023 CID_114821 0.066 0.015 CID_65280 | ||
| 0.158 | 0.094 | 0.158 | Lipocortins synthesis antagonist | |||
| 0.132 | 0.074 | 0.132 | Alkaline phosphatase inhibitor | 0.111 0.099 CID_65280 | ||
| 0.063 | 0.005 | 0.063 | Methionyl aminopeptidase 2 inhibitor | 0.034 0.012 CID_65280 | ||
| 0.224 | 0.168 | 0.398 | Calpain 2 inhibitor | 0.398 0.062 CID_65280 | CID_65280 | |
| 0.067 | 0.01 | 0.067 | Benzodiazepine inverse agonist | 0.053 0.021 CID_114821 0.058 0.016 CID_65280 | ||
| 0.105 | 0.049 | 0.105 | Protein kinase (Mos, Mil/Raf, MEKK, RIPK, TESK, LIMK, IRAK, ILK, Activin/TGF-beta) inhibitor | 0.094 0.058 CID_114821 0.098 0.055 CID_65280 | ||
| 0.065 | 0.015 | 0.065 | Fructose-1,6-bisphosphatase inhibitor | |||
| 0.216 | 0.166 | 0.254 | Sodium/bile acid cotransporter inhibitor | 0.254 0.124 CID_65280 0.249 0.129 CID_154699808 | CID_65280 | |
| 0.143 | 0.096 | 0.143 | Mcl-1 antagonist | 0.131 0.11 CID_65280 | ||
| 0.129 | 0.087 | 0.129 | Mannose-6-phosphate isomerase inhibitor | |||
| 0.184 | 0.144 | 0.193 | Streptokinase A inhibitor | 0.193 0.138 CID_65280 | CID_65280 | |
| 0.198 | 0.158 | 0.198 | Prostaglandin dehydrogenase inhibitor | |||
| 0.154 | 0.116 | 0.154 | Dual specificity tyrosine-phosphorylation regulated kinase 3 inhibitor | |||
| 0.057 | 0.021 | 0.066 | Carbonic anhydrase IV inhibitor | 0.066 0.016 CID_65280 | CID_65280 | |
| 0.066 | 0.032 | 0.089 | Potassium channel Kv1.5 blocker | 0.089 0.022 CID_65280 | CID_65280 | |
| 0.04 | 0.006 | 0.04 | Myristoyl transferase inhibitor | 0.035 0.008 CID_65280 | ||
| 0.099 | 0.064 | 0.099 | Cyclin-dependent kinase 9 inhibitor | |||
| 0.059 | 0.025 | 0.108 | Carbonic anhydrase XIV inhibitor | 0.047 0.036 CID_65280 0.108 0.009 CID_154699808 | CID_154699808 | |
| 0.051 | 0.019 | 0.051 | GHS receptor agonist | 0.041 0.032 CID_65280 | ||
| 0.068 | 0.037 | 0.068 | Raf kinase C inhibitor | 0.067 0.037 CID_65280 | ||
| 0.139 | 0.109 | 0.139 | LIM domain kinase 1 inhibitor | |||
| 0.058 | 0.028 | 0.1 | Factor IXa inhibitor | 0.065 0.023 CID_65280 0.1 0.01 CID_154699808 | CID_154699808 | |
| 0.071 | 0.042 | 0.071 | Bcl2 antagonist | |||
| 0.062 | 0.034 | 0.151 | Carbonic anhydrase I inhibitor | 0.069 0.029 CID_65280 0.151 0.01 CID_154699808 | CID_154699808 | |
| 0.11 | 0.084 | 0.144 | MAP kinase kinase inhibitor | 0.144 0.055 CID_114821 | CID_114821 | |
| 0.062 | 0.036 | 0.062 | Bcl-xL inhibitor | |||
| 0.032 | 0.007 | 0.032 | Fructose-1,6-bisphosphatase 1 inhibitor | |||
| 0.036 | 0.012 | 0.036 | Kynurenine 3 monooxygenase inhibitor | |||
| 0.059 | 0.037 | 0.059 | 5 Hydroxytryptamine 6 antagonist | |||
| 0.072 | 0.052 | 0.076 | Raf kinase inhibitor | 0.076 0.049 CID_65280 | CID_65280 | |
| 0.032 | 0.014 | 0.032 | 5 Hydroxytryptamine 6 agonist | |||
| 0.194 | 0.177 | 0.265 | Thioredoxin glutathione reductase inhibitor | 0.265 0.125 CID_65280 | CID_65280 | |
| 0.045 | 0.028 | 0.045 | Glutamate (mGluR group III) agonist | |||
| 0.037 | 0.021 | 0.037 | AMPA receptor agonist | |||
| 0.021 | 0.006 | 0.021 | CC chemokine 9 receptor antagonist | |||
| 0.044 | 0.031 | 0.044 | AICAR transformylase inhibitor | |||
| 0.018 | 0.005 | 0.018 | CC chemokine 10 receptor antagonist | |||
| 0.031 | 0.02 | 0.037 | LIM domain kinase 2 inhibitor | 0.037 0.012 CID_65280 | CID_65280 | |
| 0.09 | 0.079 | 0.09 | GABA C receptor agonist | |||
| 0.014 | 0.005 | 0.014 | 2-Acylglycerol O-acyltransferase 2 inhibitor | 0.009 0.008 CID_114821 0.013 0.005 CID_65280 | ||
| 0.024 | 0.014 | 0.024 | CC chemokine 8 receptor antagonist | |||
| 0.033 | 0.025 | 0.033 | Glutamate (mGluR4) agonist | |||
| 0.042 | 0.038 | 0.054 | Carbonic anhydrase VII inhibitor | 0.054 0.024 CID_65280 | CID_65280 | |
| 0.016 | 0.012 | 0.016 | CDK2/cyclin A3 inhibitor | |||
| 0.05 | 0.047 | 0.05 | Bombesin 3 receptor antagonist | |||
| 0.047 | 0.045 | 0.047 | Alpha 1b adrenoreceptor agonist | |||
| 0.049 | 0.052 | 0.051 | Raf kinase B inhibitor | 0.051 0.05 CID_65280 | CID_65280 | |
| 0.018 | 0.022 | 0.02 | Factor XIII inhibitor | 0.02 0.015 CID_65280 | CID_65280 | |
| 0.169 | 0.183 | 0.22 | Neuropeptide Y2 antagonist | 0.22 0.089 CID_65280 | CID_65280 | |
| 0.112 | 0.128 | 0.137 | Aurora-C kinase inhibitor | 0.137 0.069 CID_65280 | CID_65280 | |
| 0.039 | 0.057 | 0.046 | Phosphatidylinositol 3-kinase beta inhibitor | 0.046 0.04 CID_65280 | CID_65280 | |
| 0.055 | 0.073 | 0.063 | Beta 3 adrenoreceptor antagonist | 0.063 0.048 CID_65280 | CID_65280 | |
| 0.057 | 0.078 | 0.096 | Epoxide hydrolase inhibitor | 0.096 0.028 CID_65280 | CID_65280 | |
| 0.04 | 0.063 | 0.048 | CXC chemokine 1 receptor antagonist | 0.048 0.042 CID_65280 | CID_65280 | |
| 0.031 | 0.055 | 0.049 | Aggrecanase 1 inhibitor | 0.049 0.014 CID_114821 | CID_114821 | |
| 0.174 | 0.203 | 0.268 | Angiogenesis inhibitor | 0.223 0.145 CID_65280 0.268 0.11 CID_154699808 | CID_154699808 | |
| 0.043 | 0.073 | 0.085 | Glucosylceramidase inhibitor | 0.085 0.013 CID_154699808 | CID_154699808 | |
| 0.032 | 0.083 | 0.045 | Purinergic P2X4 antagonist | 0.045 0.033 CID_65280 | CID_65280 | |
| 0.02 | 0.073 | 0.031 | Carnitine palmitoyltransferase 1 inhibitor | 0.031 0.029 CID_65280 | CID_65280 | |
| 0.152 | 0.209 | 0.166 | 5 Hydroxytryptamine 3E antagonist | 0.166 0.149 CID_65280 | CID_65280 | |
| 0.05 | 0.113 | 0.075 | Metalloproteinase-2 inhibitor | 0.075 0.058 CID_114821 | CID_114821 | |
| 0.048 | 0.115 | 0.062 | Kallikrein 7 inhibitor | 0.062 0.048 CID_65280 | CID_65280 | |
| 0.116 | 0.193 | 0.437 | Immunostimulant | 0.175 0.136 CID_114821 0.437 0.04 CID_154699808 | CID_154699808 | |
| 0.019 | 0.096 | 0.039 | Macrophage elastase inhibitor | 0.039 0.034 CID_114821 | CID_114821 | |
| 0.142 | 0.22 | 0.289 | Thyroid hormone antagonist | 0.289 0.099 CID_65280 | CID_65280 | |
| 0.136 | 0.222 | 0.286 | Thyroid hormone beta antagonist | 0.286 0.095 CID_65280 | CID_65280 | |
| 0.115 | 0.221 | 0.241 | Catenin beta inhibitor | 0.241 0.013 CID_154699808 | CID_154699808 | |
| 0.027 | 0.17 | 0.06 | Heparanase inhibitor | 0.06 0.023 CID_154699808 | CID_154699808 | |
| 0.149 | 0.3 | 0.486 | Antibacterial | 0.486 0.045 CID_154699808 | CID_154699808 | |
| 0.008 | 0.159 | 0.047 | Histone deacetylase class IIa inhibitor | 0.047 0.015 CID_114821 | CID_114821 | |
| 0.056 | 0.208 | 0.112 | M17 leucyl aminopeptidase inhibitor | 0.112 0.086 CID_65280 | CID_65280 | |
| 0.147 | 0.306 | 0.217 | Interleukin 2 agonist | 0.217 0.161 CID_65280 | CID_65280 | |
| 0.095 | 0.269 | 0.178 | Calpain inhibitor | 0.178 0.137 CID_65280 | CID_65280 | |
| 0.062 | 0.24 | 0.12 | CDK3/cyclin E inhibitor | 0.12 0.055 CID_65280 | CID_65280 | |
| 0.049 | 0.233 | 0.104 | Caspase 3 inhibitor | 0.104 0.085 CID_65280 | CID_65280 | |
| 0.013 | 0.202 | 0.047 | Collagenase inhibitor | 0.047 0.039 CID_114821 | CID_114821 | |
| 0.006 | 0.225 | 0.052 | Histone deacetylase 5 inhibitor | 0.052 0.016 CID_114821 | CID_114821 | |
| 0.055 | 0.297 | 0.148 | Diuretic | 0.148 0.079 CID_154699808 | CID_154699808 | |
| 0.094 | 0.338 | 0.199 | Transcription factor STAT3 inhibitor | 0.199 0.135 CID_65280 | CID_65280 | |
| 0.006 | 0.256 | 0.05 | Histone deacetylase class II inhibitor | 0.05 0.011 CID_114821 | CID_114821 | |
| 0.006 | 0.266 | 0.034 | Histone deacetylase 4 inhibitor | 0.034 0.021 CID_114821 | CID_114821 | |
| 0.092 | 0.368 | 0.149 | Cyclin-dependent kinase 3 inhibitor | 0.149 0.097 CID_65280 | CID_65280 | |
| 0.031 | 0.345 | 0.123 | Beta glucuronidase inhibitor | 0.123 0.043 CID_154699808 | CID_154699808 | |
| 0.067 | 0.468 | 0.167 | Death-associated protein kinase 2 inhibitor | 0.167 0.072 CID_65280 | CID_65280 | |
| 0.098 | 0.536 | 0.383 | Antiinflammatory | 0.383 0.15 CID_154699808 | CID_154699808 | |
| 0.087 | 0.537 | 0.256 | Peptidyltransferase inhibitor | 0.256 0.046 CID_154699808 | CID_154699808 | |
| 0.029 | 0.548 | 0.177 | DNA synthesis inhibitor | 0.177 0.159 CID_154699808 | CID_154699808 | |
| 0.004 | 0.546 | 0.035 | Histone deacetylase class IIb inhibitor | 0.035 0.014 CID_114821 | CID_114821 | |
| 0.004 | 0.55 | 0.034 | Histone deacetylase 6 inhibitor | 0.034 0.014 CID_114821 | CID_114821 | |
| 0.014 | 0.682 | 0.229 | Angiogenesis stimulant | 0.229 0.08 CID_154699808 | CID_154699808 | |
| 0.009 | 0.686 | 0.031 | ADAM10 endopeptidase inhibitor | 0.031 0.029 CID_114821 | CID_114821 | |
| 0.023 | 0.802 | 0.14 | Hepatoprotectant | 0.14 0.121 CID_154699808 | CID_154699808 | |
| 0.018 | 0.805 | 0.512 | Cyclophilin D inhibitor | 0.512 0.047 CID_154699808 | CID_154699808 | |
| 0.014 | 0.84 | 0.209 | Immunosuppressant | 0.209 0.187 CID_154699808 | CID_154699808 | |
| 0.004 | 0.899 | 0.23 | Lipid peroxidase inhibitor | 0.23 0.031 CID_154699808 | CID_154699808 | |
| 0.003 | 0.918 | 0.099 | Selectin antagonist | 0.099 0.028 CID_154699808 | CID_154699808 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |