Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.970.0040.97Antiobesity

0.914 0.004 CID_10199199

0.7490.0030.95 Hydroxytryptamine uptake inhibitor

0.9 0.002 CID_10199199

CID_10199199
0.6810.0020.847Adrenaline uptake inhibitor

0.847 0.002 CID_10199199

CID_10199199
0.6440.0050.644Potassium channel (Voltage-sensitive) blocker

0.336 0.04 CID_10199199

0.5980.0080.598HERG channel blocker

0.255 0.064 CID_10199199

0.5630.0230.563Cholesterol antagonist

0.378 0.054 CID_10199199

0.5420.0080.542Potassium channel blocker

0.309 0.043 CID_10199199

0.5210.0030.521Dopamine uptake inhibitor

0.493 0.003 CID_10199199

0.5330.0280.533Aldehyde oxidase inhibitor

0.334 0.058 CID_10199199

0.5020.0020.546Dopamine transporter inhibitor

0.546 0.002 CID_10199199

CID_10199199
0.4320.040.565 Hydroxytryptamine release stimulant

0.56 0.019 CID_10199199

CID_10199199
0.3920.0170.392Anesthetic general

0.353 0.023 CID_10199199

0.3530.030.353Sigma receptor agonist

0.242 0.05 CID_10199199

0.3310.0320.3375 Hydroxytryptamine uptake stimulant

0.337 0.029 CID_10199199

CID_10199199
0.3450.0540.345Spasmolytic

0.246 0.093 CID_10199199

0.2810.0480.3Gastrin inhibitor

0.3 0.033 CID_10199199

CID_10199199
0.2760.050.297Psychostimulant

0.297 0.044 CID_10199199

CID_10199199
0.2790.0620.285Tumour necrosis factor alpha release inhibitor

0.285 0.059 CID_10199199

CID_10199199
0.330.120.33Analgesic

0.287 0.152 CID_10199199

0.2180.020.218Alpha 2b adrenoreceptor antagonist

0.102 0.073 CID_10199199

0.2110.030.24Neurotensin receptor agonist

0.24 0.023 CID_10199199

CID_10199199
0.2040.0310.204Anesthetic local

0.116 0.07 CID_10199199

0.2090.0510.209Lipocortins synthesis antagonist

0.191 0.062 CID_10199199

0.2320.0750.232Neuropeptide Y2 antagonist

0.214 0.097 CID_10199199

0.1580.0090.158Lanosterol 14 alpha demethylase inhibitor

0.146 0.013 CID_10199199

0.1890.0440.189Arachidonic acid antagonist

0.165 0.071 CID_10199199

0.2460.1070.246Ca(v)3.3 blocker

0.245 0.109 CID_10199199

0.2270.0930.235Tyrosine 3 hydroxylase inhibitor

0.235 0.084 CID_10199199

CID_10199199
0.1650.0370.172Cathepsin H inhibitor

0.172 0.033 CID_10199199

CID_10199199
0.2270.1010.2275 Hydroxytryptamine 1E antagonist

0.215 0.114 CID_10199199

0.1640.0380.164Cholesterol synthesis inhibitor

0.113 0.072 CID_10199199

0.1260.0050.126Prostaglandin EP3 antagonist

0.109 0.005 CID_10199199

0.1320.0150.133Glutamate release inhibitor

0.133 0.015 CID_10199199

CID_10199199
0.290.1760.2955 Hydroxytryptamine release inhibitor

0.295 0.17 CID_10199199

CID_10199199
0.1210.0070.126Vanilloid 4 agonist

0.126 0.005 CID_10199199

CID_10199199
0.2390.1310.248Interleukin 2 agonist

0.248 0.12 CID_10199199

CID_10199199
0.1770.070.177Tumour necrosis factor antagonist

0.147 0.104 CID_10199199

0.1540.0470.154Pregnane X receptor agonist

0.142 0.069 CID_10199199

0.1740.070.174Antipruritic

0.169 0.075 CID_10199199

0.180.0870.18Non-steroidal antiinflammatory agent

0.173 0.093 CID_10199199

0.1270.0360.127Sphingomyelinase inhibitor

0.122 0.039 CID_10199199

0.1020.0140.102Prostaglandin E2 antagonist

0.091 0.017 CID_10199199

0.1670.0840.167Succinate dehydrogenase inhibitor

0.161 0.094 CID_10199199

0.1010.0230.101Estrogen-related receptor beta agonist

0.09 0.04 CID_10199199

0.0860.0150.086Glycine transporter inhibitor

0.048 0.033 CID_10199199

0.1320.0640.132CC chemokine 6 receptor antagonist

0.122 0.107 CID_10199199

0.130.0640.131Nav1.3 sodium channel blocker

0.131 0.063 CID_10199199

CID_10199199
0.2340.1690.25GABA C receptor rho-3 antagonist

0.25 0.154 CID_10199199

CID_10199199
0.10.0350.129Opioid kappa receptor antagonist

0.129 0.021 CID_10199199

CID_10199199
0.1170.0560.117Falcipain 3 inhibitor

0.099 0.071 CID_10199199

0.140.080.14Thiol protease inhibitor

0.128 0.099 CID_10199199

0.1090.0490.109Falcipain inhibitor

0.098 0.056 CID_10199199

0.1070.0480.107Falcipain 2 inhibitor

0.095 0.055 CID_10199199

0.0940.0390.094Glycine receptor antagonist

0.083 0.053 CID_10199199

0.2220.170.222Calpain 2 inhibitor
0.0890.0380.089Analgesic, opioid

0.077 0.052 CID_10199199

0.150.1020.156ATPase inhibitor

0.156 0.091 CID_10199199

CID_10199199
0.1290.0820.129Nav1.6 sodium channel blocker
0.1250.0780.125Nav1.2 sodium channel blocker

0.124 0.079 CID_10199199

0.1150.0690.131Calcium channel N-type blocker

0.131 0.051 CID_10199199

CID_10199199
0.0650.020.066Purinergic P2X antagonist

0.066 0.02 CID_10199199

CID_10199199
0.1360.0910.136Ca2+-transporting ATPase inhibitor
0.090.0460.093C-Like protease (SARS coronavirus) inhibitor

0.09 0.047 CID_10199199

0.1750.1360.175Immunostimulant
0.050.0120.052,3-Oxidosqualene-lanosterol cyclase inhibitor
0.0520.0140.052GABA uptake inhibitor

0.036 0.033 CID_10199199

0.0810.0440.081Sphingosine 1-phosphate receptor antagonist

0.078 0.05 CID_10199199

0.170.1340.1715 Hydroxytryptamine 3E antagonist

0.171 0.132 CID_10199199

CID_10199199
0.060.0240.072Immunoglobulin Fc receptor antagonist

0.072 0.009 CID_10199199

CID_10199199
0.0580.0230.058Squalene epoxidase inhibitor
0.1770.1420.203Interleukin agonist

0.203 0.118 CID_10199199

CID_10199199
0.0390.0050.039Hedgehog signaling activator

0.034 0.008 CID_10199199

0.1580.1260.179Neurotrophic factor enhancer

0.179 0.099 CID_10199199

CID_10199199
0.0980.0660.098Anabolic

0.092 0.075 CID_10199199

0.0640.0330.064Calcium channel T-type blocker

0.055 0.045 CID_10199199

0.0630.0350.072Cathepsin L inhibitor

0.072 0.028 CID_10199199

CID_10199199
0.050.0220.051Parathyroid hormone antagonist

0.051 0.019 CID_10199199

CID_10199199
0.0690.0420.069MDM2 inhibitor

0.065 0.056 CID_10199199

0.0540.0290.054Neurokinin antagonist
0.0460.0220.047Alpha 1L adrenoreceptor agonist

0.047 0.021 CID_10199199

CID_10199199
0.0860.0620.101Opioid antagonist

0.101 0.047 CID_10199199

CID_10199199
0.0450.0220.059Cathepsin L1 inhibitor

0.059 0.016 CID_10199199

CID_10199199
0.120.0970.125Sphingosine 1-phosphate receptor 2 antagonist

0.125 0.084 CID_10199199

CID_10199199
0.0470.0250.05Melanocortin 4 antagonist

0.05 0.023 CID_10199199

CID_10199199
0.0510.0280.053Melanocortin antagonist

0.053 0.027 CID_10199199

CID_10199199
0.0440.0220.046Cathepsin F inhibitor

0.046 0.018 CID_10199199

CID_10199199
0.0420.020.042Glycine transporter 1 inhibitor
0.0620.040.066Neuraminidase inhibitor

0.066 0.037 CID_10199199

CID_10199199
0.0840.0620.084Alpha 2 adrenoreceptor antagonist
0.1280.1060.14Adenylate cyclase stimulant

0.14 0.08 CID_10199199

CID_10199199
0.0730.0520.116Rho-associated kinase II inhibitor

0.116 0.026 CID_10199199

CID_10199199
0.0890.0680.089ABCA1 expression enhancer

0.083 0.08 CID_10199199

0.0830.0620.083Antineoplastic alkaloid
0.0720.0520.072Glycine receptor agonist
0.0420.0240.051NMDA receptor subunit 3A antagonist

0.051 0.019 CID_10199199

CID_10199199
0.0430.0240.043Kainate receptor agonist

0.041 0.028 CID_10199199

0.0620.0430.062Corticotropin releasing factor 2 receptor antagonist

0.057 0.054 CID_10199199

0.0460.0270.046Opioid kappa receptor agonist
0.1130.0950.113Calcium channel blocker

0.112 0.097 CID_10199199

0.1010.0830.107Calcium channel (voltage-sensitive) blocker

0.107 0.075 CID_10199199

CID_10199199
0.0470.0290.047Neuraminidase (Influenza A) inhibitor

0.047 0.028 CID_10199199

0.0310.0140.031HCV NS5A inhibitor
0.0870.0710.087Prolactin inhibitor
0.0560.040.056Pregnane X receptor antagonist
0.1260.110.126Sphingosine 1-phosphate receptor 5 antagonist
0.0620.0470.062Dopamine D1 antagonist
0.0370.0230.037p53 inhibitor
0.1310.1180.131Heat shock protein 70 antagonist
0.0510.0390.051Opioid agonist
0.0240.0120.024Protease (Human cytomegalovirus) inhibitor

0.021 0.017 CID_10199199

0.0520.040.052Nicotinic alpha3beta2 receptor antagonist

0.051 0.041 CID_10199199

0.0810.070.081Antiadrenergic
0.0770.0670.077Calcium antagonist
0.1050.0960.105Cyclooxygenase 3 inhibitor

0.103 0.099 CID_10199199

0.0770.0690.077Ca(v)3.1 blocker

0.077 0.071 CID_10199199

0.060.0530.062Neuraminidase (influenza) inhibitor

0.062 0.049 CID_10199199

CID_10199199
0.1360.1290.1513C-like protease (Human coronavirus) inhibitor

0.151 0.099 CID_10199199

CID_10199199
0.2540.2480.269Caspase 9 stimulant

0.269 0.229 CID_10199199

CID_10199199
0.0570.0510.058Purinergic P2 antagonist

0.058 0.05 CID_10199199

CID_10199199
0.0380.0330.038Neurokinin 2 antagonist
0.0260.0210.02611-Beta-hydroxysteroid dehydrogenase 2 inhibitor
0.0150.0110.023NMDA receptor phencyclidine site antagonist

0.023 0.006 CID_10199199

CID_10199199
0.0760.0720.076Adrenaline antagonist
0.1060.1030.106Sphingosine 1-phosphate receptor 4 antagonist
0.0680.0650.068GABA aminotransferase inhibitor
0.0320.0290.033Purinergic P2X7 antagonist

0.033 0.027 CID_10199199

CID_10199199
0.0510.0480.061Cathepsin B inhibitor

0.061 0.035 CID_10199199

CID_10199199
0.0240.0220.024Urotensin II agonist
0.0980.0950.103Microtubule formation inhibitor

0.103 0.086 CID_10199199

CID_10199199
0.0660.0640.066Na+ K+ transporting ATPase inhibitor
0.1080.1070.109Protein kinase stimulant

0.109 0.106 CID_10199199

CID_10199199
0.0320.0330.0435-Alpha-reductase inhibitor

0.043 0.022 CID_10199199

CID_10199199
0.0230.0250.024Cathepsin K inhibitor

0.024 0.023 CID_10199199

CID_10199199
0.0190.0220.023CC chemokine 1 receptor antagonist

0.023 0.017 CID_10199199

CID_10199199
0.030.0360.033Bombesin 1 receptor antagonist

0.033 0.031 CID_10199199

CID_10199199
0.1130.1240.122Insulin secretagoues

0.122 0.108 CID_10199199

CID_10199199
0.0490.0610.059Cannabinoid CB1 receptor antagonist

0.059 0.046 CID_10199199

CID_10199199
0.0510.0650.065Matrix metalloproteinase inhibitor

0.065 0.049 CID_10199199

CID_10199199
0.0510.0650.069Opioid mu receptor antagonist

0.069 0.046 CID_10199199

CID_10199199
0.0410.0560.047Collagenase inhibitor

0.047 0.038 CID_10199199

CID_10199199
0.1060.1240.156Cell wall synthesis inhibitor

0.156 0.06 CID_10199199

CID_10199199
0.0540.0720.062Cannabinoid receptor antagonist

0.062 0.059 CID_10199199

CID_10199199
0.0340.0540.051NMDA 2A receptor antagonist

0.051 0.036 CID_10199199

CID_10199199
0.0490.070.059NMDA receptor agonist

0.059 0.049 CID_10199199

CID_10199199
0.0650.0890.081NMDA receptor antagonist

0.081 0.065 CID_10199199

CID_10199199
0.0410.0690.051Matrix metalloproteinase (membrane-type) inhibitor

0.051 0.045 CID_10199199

CID_10199199
0.0370.0660.047Potassium channel (ATP-sensitive) activator

0.047 0.037 CID_10199199

CID_10199199
0.0390.0680.049Potassium channel (Inward rectifier) activator

0.049 0.038 CID_10199199

CID_10199199
0.0290.0580.036Potassium channel Kv1.1 blocker

0.036 0.031 CID_10199199

CID_10199199
0.030.0620.049Matrix metalloproteinase 1 inhibitor

0.049 0.039 CID_10199199

CID_10199199
0.0320.0670.038VCAM-1 antagonist

0.038 0.033 CID_10199199

CID_10199199
0.0320.0670.038VCAM antagonist

0.038 0.033 CID_10199199

CID_10199199
0.0480.0850.057Caspase 9 inhibitor

0.057 0.055 CID_10199199

CID_10199199
0.0490.0870.071Rho-associated kinase inhibitor

0.071 0.054 CID_10199199

CID_10199199
0.0290.080.066Beta tubulin antagonist

0.066 0.036 CID_10199199

CID_10199199
0.0340.0860.051Baculoviral IAP repeat-containing protein inhibitor

0.051 0.019 CID_10199199

CID_10199199
0.2380.3070.292Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.292 0.224 CID_10199199

CID_10199199
0.0490.1220.085Ca(v)2.2 blocker

0.085 0.06 CID_10199199

CID_10199199
0.0570.1320.086Potassium channel activator

0.086 0.066 CID_10199199

CID_10199199
0.1720.2620.217Calcium channel activator

0.217 0.189 CID_10199199

CID_10199199
0.1010.2020.17Anticonvulsant

0.17 0.108 CID_10199199

CID_10199199
0.0180.1970.038Antibiotic Aminoglycoside-like

0.038 0.023 CID_10199199

CID_10199199
Ext Pa Pi Pmax Activity Other Results ID Pa_max