Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.6940.0050.694Amyloid beta aggregation inhibitor

0.419 0.022 CID_7515

0.6080.0040.608Amyloid beta precursor protein antagonist

0.431 0.005 CID_7515

0.5690.0110.569GABA C receptor rho-3 antagonist

0.569 0.011 CID_7515

0.5620.0130.637Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.637 0.004 CID_7515

CID_7515
0.5680.0230.568Aldehyde oxidase inhibitor

0.503 0.032 CID_7515

0.5530.0250.553Cholesterol antagonist

0.322 0.078 CID_7515

0.5140.0080.514Sigma receptor agonist

0.216 0.057 CID_7515

0.5280.0230.5285 Hydroxytryptamine release stimulant

0.497 0.028 CID_7515

0.5070.0040.507Lipocortins synthesis antagonist

0.153 0.1 CID_7515

0.4960.0340.5225 Hydroxytryptamine release inhibitor

0.522 0.026 CID_7515

CID_7515
0.4620.010.462Anesthetic general

0.409 0.015 CID_7515

0.430.0170.503Peroxidase inhibitor

0.503 0.009 CID_7515

CID_7515
0.4260.0320.426Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase inhibitor

0.326 0.057 CID_7515

0.3870.0050.394Gastrin inhibitor

0.394 0.005 CID_7515

CID_7515
0.4310.0590.534Histamine release inhibitor

0.534 0.019 CID_7515

CID_7515
0.4050.0540.405Vasodilator, peripheral

0.322 0.086 CID_7515

0.440.0880.447Caspase 9 stimulant

0.447 0.085 CID_7515

CID_7515
0.3620.0110.402Alpha-N-acetylglucosaminidase inhibitor

0.402 0.009 CID_7515

CID_7515
0.370.020.3715 Hydroxytryptamine uptake stimulant

0.371 0.02 CID_7515

CID_7515
0.3540.0120.354Glyceraldehyde-3-phosphate dehydrogenase inhibitor

0.273 0.033 CID_7515

0.3690.0290.369Sodium/bile acid cotransporter inhibitor
0.3460.0070.346NADPH oxidase inhibitor

0.155 0.051 CID_7515

0.3360.0050.383Ferrochelatase inhibitor

0.383 0.004 CID_7515

CID_7515
0.3450.0170.345Tyrosine 3 hydroxylase inhibitor

0.331 0.021 CID_7515

0.3850.0680.758MAP kinase kinase 6 inhibitor

0.758 0.004 CID_7515

CID_7515
0.3150.0050.3155 Hydroxytryptamine 1F antagonist
0.3380.0290.338Cyclic AMP phosphodiesterase inhibitor

0.238 0.07 CID_7515

0.3110.0050.311Mannose-6-phosphate isomerase inhibitor

0.224 0.019 CID_7515

0.3430.0430.343DNA damaging

0.297 0.058 CID_7515

0.3360.040.336Insulysin inhibitor

0.294 0.062 CID_7515

0.3270.0350.327DNA synthesis inhibitor

0.275 0.053 CID_7515

0.3420.0550.424Calcium channel activator

0.424 0.017 CID_7515

CID_7515
0.2990.0130.299Toll-Like receptor 9 antagonist

0.238 0.023 CID_7515

0.290.0060.295 Hydroxytryptamine 3E antagonist

0.287 0.006 CID_7515

0.3240.0420.324Pyruvate kinase inhibitor

0.167 0.102 CID_7515

0.2840.010.305GABA C receptor agonist

0.305 0.009 CID_7515

CID_7515
0.3140.0480.35Transcription factor STAT inhibitor

0.35 0.034 CID_7515

CID_7515
0.3550.0960.35515-Lipoxygenase inhibitor

0.355 0.097 CID_7515

0.3150.0580.315Hypoxia-inducible factor 1 alpha inhibitor

0.185 0.171 CID_7515

0.3060.050.306Antiamyloidogenic

0.289 0.055 CID_7515

0.2620.0090.287Ca(v)2.2 blocker

0.287 0.006 CID_7515

CID_7515
0.3090.0580.309Ca2+/calmodulin-dependent kinase II alpha inhibitor

0.286 0.074 CID_7515

0.2730.0240.273Cytidine deaminase inhibitor

0.174 0.06 CID_7515

0.2580.010.267GABA C receptor rho-2 antagonist

0.267 0.009 CID_7515

CID_7515
0.2860.040.31MAP kinase kinase 2 inhibitor

0.31 0.032 CID_7515

CID_7515
0.2680.0220.28Nitric-oxide synthase stimulant

0.28 0.017 CID_7515

CID_7515
0.2830.0430.3595 Hydroxytryptamine 1E antagonist

0.359 0.008 CID_7515

CID_7515
0.2930.0530.293Superoxide dismutase inhibitor

0.279 0.059 CID_7515

0.240.0080.24CF transmembrane conductance regulator agonist

0.235 0.009 CID_7515

0.2380.0070.238Photosensitizer

0.143 0.035 CID_7515

0.2520.0220.252Succinate dehydrogenase inhibitor

0.242 0.025 CID_7515

0.2680.040.268Neuropeptide Y2 antagonist

0.256 0.051 CID_7515

0.2770.0490.277Psychostimulant

0.236 0.064 CID_7515

0.260.0320.293I kappa B kinase epsilon inhibitor

0.293 0.017 CID_7515

CID_7515
0.250.0250.25Phospholipase C inhibitor

0.204 0.041 CID_7515

0.2610.0430.365RNA-directed DNA polymerase inhibitor

0.365 0.022 CID_7515

CID_7515
0.2330.0190.233Chelator
0.2510.0370.268Focal adhesion kinase 2 inhibitor

0.268 0.028 CID_7515

CID_7515
0.2570.0460.279Peptidyltransferase inhibitor

0.279 0.034 CID_7515

CID_7515
0.2990.0880.299Vasodilator, coronary

0.265 0.12 CID_7515

0.2150.0050.215Tyrosine-protein kinase EMT inhibitor

0.121 0.013 CID_7515

0.2120.0060.212Transcription factor STAT6 inhibitor

0.139 0.034 CID_7515

0.2110.0080.211Multidrug resistance-associated protein 1 inhibitor
0.2680.0660.29Interleukin agonist

0.29 0.053 CID_7515

CID_7515
0.2210.0230.221ATPase inhibitor

0.204 0.034 CID_7515

0.2280.0330.228Protein kinase stimulant

0.182 0.049 CID_7515

0.2120.0170.212UDP-glucose 4-epimerase inhibitor

0.184 0.02 CID_7515

0.2070.0130.2295 Hydroxytryptamine 3A agonist

0.229 0.008 CID_7515

CID_7515
0.2380.0440.46MAP kinase kinase 3 inhibitor

0.46 0.002 CID_7515

CID_7515
0.2030.0120.316GABA C receptor antagonist

0.316 0.004 CID_7515

CID_7515
0.2050.0140.205Adenylate kinase inhibitor

0.172 0.02 CID_7515

0.2340.0440.234Insulin sensitizer

0.174 0.102 CID_7515

0.2280.0380.228Histone acetyltransferase inhibitor

0.22 0.044 CID_7515

0.2050.0160.205Ca2+/calmodulin-dependent protein kinase kinase B inhibitor

0.16 0.056 CID_7515

0.2120.0230.212Arachidonic acid antagonist

0.189 0.044 CID_7515

0.2150.0290.215Neurotensin receptor agonist

0.168 0.066 CID_7515

0.1930.0090.291GABA C receptor rho-1 antagonist

0.291 0.004 CID_7515

CID_7515
0.2990.1150.299Calpain 2 inhibitor

0.26 0.142 CID_7515

0.1990.0170.212Beta amyloid protein antagonist

0.212 0.013 CID_7515

CID_7515
0.3210.140.422Calcium channel L-type activator

0.422 0.067 CID_7515

CID_7515
0.1890.0110.189Prolactin inhibitor

0.158 0.019 CID_7515

0.1870.0090.187CYP2A6 inhibitor

0.135 0.021 CID_7515

0.2550.0770.266Aryl hydrocarbon receptor agonist

0.266 0.072 CID_7515

CID_7515
0.1820.0050.182Glutamate (mGluR7) agonist

0.165 0.008 CID_7515

0.2270.050.227LIM domain kinase 1 inhibitor

0.224 0.052 CID_7515

0.3050.1310.305Antibacterial

0.294 0.14 CID_7515

0.2030.030.203Toll-Like receptor antagonist

0.163 0.047 CID_7515

0.2260.0540.262Neurotrophic factor enhancer

0.262 0.032 CID_7515

CID_7515
0.1840.0130.184Triose-phosphate isomerase inhibitor

0.166 0.016 CID_7515

0.1850.0140.185Porphobilinogen synthase inhibitor

0.144 0.022 CID_7515

0.2040.0330.204Hexokinase inhibitor

0.189 0.042 CID_7515

0.1960.0270.196Glutamate receptor antagonist

0.139 0.059 CID_7515

0.2510.0820.337Transcription factor STAT3 inhibitor

0.337 0.037 CID_7515

CID_7515
0.20.0320.2Catenin beta inhibitor

0.181 0.051 CID_7515

0.1980.0310.198Cell wall synthesis inhibitor

0.196 0.032 CID_7515

0.1810.0140.181Creatine kinase inhibitor

0.153 0.023 CID_7515

0.1950.0280.195Alkylator

0.168 0.038 CID_7515

0.1690.0020.169Glutamate (mGluR7) antagonist

0.104 0.009 CID_7515

0.1790.0140.179Sphingomyelinase inhibitor

0.145 0.027 CID_7515

0.210.0460.213C-like protease (Human coronavirus) inhibitor

0.18 0.065 CID_7515

0.1740.010.174Glutamate (mGluR group I) antagonist

0.078 0.04 CID_7515

0.1780.0140.178Nitric-oxide synthase inhibitor

0.16 0.019 CID_7515

0.2730.1110.273Transcription factor NF kappa B inhibitor

0.262 0.119 CID_7515

0.1970.0360.197Nav1.2 sodium channel blocker

0.144 0.061 CID_7515

0.1750.0150.175Folate antagonist
0.1720.0110.172Ca2+-transporting ATPase inhibitor

0.162 0.021 CID_7515

0.1740.0130.174NADH dehydrogenase inhibitor

0.152 0.017 CID_7515

0.2150.0550.215P-glycoprotein inhibitor
0.1770.0170.18Gastric antisecretory

0.18 0.016 CID_7515

CID_7515
0.1670.0090.167Histamine N-methyltransferase inhibitor

0.155 0.012 CID_7515

0.1710.0170.171Heat shock protein 70 antagonist

0.163 0.025 CID_7515

0.3160.1630.316MAP kinase 1 inhibitor

0.289 0.193 CID_7515

0.1710.0190.171HIV-1 integrase (Overall Integration) inhibitor

0.154 0.024 CID_7515

0.1810.0290.181Cystathionine beta-synthase inhibitor

0.163 0.035 CID_7515

0.1720.0210.172UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor

0.159 0.024 CID_7515

0.1840.0330.184MAO A inhibitor

0.145 0.042 CID_7515

0.1740.0250.174Calcium channel N-type blocker

0.145 0.041 CID_7515

0.1680.0190.168DNA repair enzyme inhibitor

0.145 0.036 CID_7515

0.180.0330.18Aldehyde dehydrogenase inhibitor

0.111 0.082 CID_7515

0.1550.0090.155Glutamate release inhibitor

0.13 0.016 CID_7515

0.2340.0880.272Ca2+/calmodulin-dependent kinase IV inhibitor

0.272 0.043 CID_7515

CID_7515
0.1630.0180.163Urease inhibitor

0.139 0.029 CID_7515

0.1520.0080.152GABA aminotransferase inhibitor

0.113 0.019 CID_7515

0.1820.0390.182Acetylcholinesterase inhibitor
0.1470.0040.147GABA B receptor agonist

0.088 0.028 CID_7515

0.1520.010.152Alcohol oxidase inhibitor

0.127 0.013 CID_7515

0.1520.0160.152Inducible nitric-oxide synthase inhibitor

0.111 0.029 CID_7515

0.2350.0980.235Spasmolytic

0.195 0.124 CID_7515

0.170.0350.184Adenylate cyclase stimulant

0.184 0.023 CID_7515

CID_7515
0.1680.0350.168MAP kinase kinase 4 inhibitor

0.138 0.089 CID_7515

0.1680.0350.168Cathepsin H inhibitor

0.16 0.039 CID_7515

0.150.0170.15Glutamate (mGluR) antagonist
0.1590.0270.159Protein kinase C gamma inhibitor

0.15 0.031 CID_7515

0.1480.0160.148Glutamate dehydrogenase inhibitor

0.115 0.024 CID_7515

0.1790.0480.179MAO inhibitor

0.146 0.062 CID_7515

0.1740.0420.174Calcium channel blocker

0.142 0.066 CID_7515

0.1350.0050.135CC chemokine 5 receptor agonist

0.108 0.014 CID_7515

0.1810.0510.181Acetylcholine M1 receptor antagonist

0.159 0.067 CID_7515

0.1650.0360.168Antibacterial (Helicobacter pylori)

0.168 0.034 CID_7515

CID_7515
0.150.020.15Telomerase inhibitor

0.128 0.024 CID_7515

0.1750.0460.226Cytokine production inhibitor

0.226 0.029 CID_7515

CID_7515
0.1690.0410.17Anesthetic local

0.17 0.041 CID_7515

CID_7515
0.1380.010.138Acyl-CoA dehydrogenase inhibitor

0.111 0.014 CID_7515

0.1660.0390.166Nav1.6 sodium channel blocker

0.15 0.054 CID_7515

0.1650.0380.204Interleukin 4 antagonist

0.204 0.021 CID_7515

CID_7515
0.1330.0060.133Estrogen-related receptor beta agonist

0.109 0.016 CID_7515

0.2070.0830.232EphB2 antagonist

0.232 0.067 CID_7515

CID_7515
0.1470.0230.147Calcium antagonist

0.111 0.04 CID_7515

0.1430.0190.143Thioredoxin inhibitor
0.1440.020.144NAD(P)H dehydrogenase (quinone) inhibitor

0.088 0.044 CID_7515

0.1370.0140.138Phosphodiesterase 6D inhibitor

0.138 0.014 CID_7515

CID_7515
0.1580.0350.185Alpha 2b adrenoreceptor antagonist

0.185 0.027 CID_7515

CID_7515
0.1330.0110.133Biliverdin reductase inhibitor

0.111 0.016 CID_7515

0.1290.0090.129Glutamate (mGluR1) antagonist

0.114 0.012 CID_7515

0.1420.0230.145Electrolyte absorption antagonist

0.145 0.021 CID_7515

CID_7515
0.1590.0410.16Cyclooxygenase 3 inhibitor

0.16 0.04 CID_7515

CID_7515
0.1520.0350.173Falcipain 3 inhibitor

0.173 0.027 CID_7515

CID_7515
0.1370.0210.142Phosphofructokinase-1 inhibitor

0.142 0.02 CID_7515

CID_7515
0.160.0460.175Sphingosine 1-phosphate receptor 5 antagonist

0.175 0.029 CID_7515

CID_7515
0.1510.0370.151Aminopeptidase B inhibitor

0.139 0.043 CID_7515

0.1390.0250.139Acetylcholine release stimulant

0.121 0.046 CID_7515

0.1180.0040.118Corticotropin releasing factor 2 receptor antagonist

0.074 0.023 CID_7515

0.1720.0590.191Cyclin-dependent kinase 8 inhibitor

0.191 0.042 CID_7515

CID_7515
0.170.0570.17Interferon gamma antagonist

0.143 0.088 CID_7515

0.1380.0260.138Androgen antagonist

0.123 0.032 CID_7515

0.1790.0680.179Mcl-1 antagonist
0.1710.0610.171Cholinergic
0.1450.0350.145Mucolytic

0.118 0.057 CID_7515

0.1330.0250.15MAP kinase kinase 1 inhibitor

0.15 0.016 CID_7515

CID_7515
0.1120.0040.112Squalene epoxidase inhibitor

0.058 0.023 CID_7515

0.1150.010.144Potassium channel (ATP-sensitive) blocker

0.144 0.005 CID_7515

CID_7515
0.140.0350.16Carbonic anhydrase XV inhibitor

0.16 0.027 CID_7515

CID_7515
0.1110.0060.111MAP kinase kinase 7 inhibitor

0.104 0.01 CID_7515

0.1860.0820.186Non-steroidal antiinflammatory agent
0.1390.0350.139Nav1.5 sodium channel blocker
0.1520.0490.18Pregnane X receptor agonist

0.18 0.019 CID_7515

CID_7515
0.1070.0040.107Motilin receptor agonist
0.1210.0190.121Bile acid receptor antagonist

0.104 0.04 CID_7515

0.1220.0190.122Myeloperoxidase inhibitor

0.097 0.039 CID_7515

0.1420.040.142GABA receptor agonist
0.1170.0160.117Carbamoyl phosphate synthetase inhibitor

0.099 0.021 CID_7515

0.1110.0110.146NMDA 2A receptor antagonist

0.146 0.007 CID_7515

CID_7515
0.2720.1720.272Transcription factor inhibitor

0.261 0.179 CID_7515

0.1420.0420.142Microtubule formation inhibitor

0.127 0.053 CID_7515

0.1390.040.139Calcium channel (voltage-sensitive) blocker

0.114 0.064 CID_7515

0.1410.0420.163Sphingosine 1-phosphate receptor 4 antagonist

0.163 0.024 CID_7515

CID_7515
0.1250.0270.125Potassium channel (Voltage-sensitive) activator

0.103 0.049 CID_7515

0.1720.0750.172Tumour necrosis factor antagonist

0.154 0.095 CID_7515

0.1060.010.106S-adenosyl-L-methionine decarboxylase inhibitor

0.106 0.01 CID_7515

0.1380.0420.138MAO B inhibitor

0.092 0.064 CID_7515

0.1480.0520.172MAP kinase kinase inhibitor

0.172 0.04 CID_7515

CID_7515
0.110.0140.11Carbonic anhydrase VB inhibitor

0.079 0.023 CID_7515

0.1150.020.115Phenylalanine 4-hydroxylase inhibitor

0.106 0.023 CID_7515

0.1320.0370.195Carbonic anhydrase III inhibitor

0.195 0.017 CID_7515

CID_7515
0.2710.1750.271Alpha-glucosidase inhibitor
0.1440.0490.163Sphingosine 1-phosphate receptor 2 antagonist

0.163 0.027 CID_7515

CID_7515
0.1160.0210.1163C-Like protease (SARS coronavirus) inhibitor
0.1440.0490.22Adenylate cyclase inhibitor

0.22 0.023 CID_7515

CID_7515
0.1750.0810.175CDC-like kinase 4 inhibitor
0.1660.0720.166Heat shock protein 90 alpha antagonist

0.149 0.088 CID_7515

0.1220.0290.122Lanosterol 14 alpha demethylase inhibitor

0.113 0.039 CID_7515

0.1060.0130.106Alpha 2 adrenoreceptor agonist

0.099 0.015 CID_7515

0.1170.0250.149NMDA 2 receptor antagonist

0.149 0.017 CID_7515

CID_7515
0.1140.0220.114Glycine receptor antagonist

0.108 0.025 CID_7515

0.1420.0510.142Histone deacetylase class III inhibitor

0.111 0.079 CID_7515

0.1520.0610.155Neuropeptide Y1 antagonist

0.155 0.058 CID_7515

CID_7515
0.110.0190.138D-Ala-D-Ala ligase inhibitor

0.138 0.008 CID_7515

CID_7515
0.1040.0130.104Mannitol-1-phosphate 5-dehydrogenase inhibitor

0.084 0.018 CID_7515

0.1120.0220.112Granulocyte macrophage colony stimulating factor agonist

0.11 0.023 CID_7515

0.1320.0420.132Alpha 2c adrenoreceptor antagonist

0.109 0.058 CID_7515

0.0960.0070.096Alpha-mannosidase inhibitor

0.076 0.013 CID_7515

0.1570.0680.157Heat shock protein 90 antagonist

0.121 0.112 CID_7515

0.1150.0260.115Glutathione S-transferase inhibitor

0.095 0.042 CID_7515

0.1150.0260.131Bromodomain-containing protein 2 inhibitor

0.131 0.017 CID_7515

CID_7515
0.1330.0450.133TRPA1 agonist

0.133 0.045 CID_7515

0.1030.0150.103Vanilloid 4 agonist

0.095 0.021 CID_7515

0.0930.0050.093Glutamate (mGluR group III) antagonist

0.043 0.032 CID_7515

0.1530.0660.153Thiol protease inhibitor

0.124 0.108 CID_7515

0.1080.0210.108Caspase 7 inhibitor

0.102 0.026 CID_7515

0.1020.0140.1025 Hydroxytryptamine 3 agonist

0.099 0.016 CID_7515

0.1260.0390.126DOPA decarboxylase inhibitor

0.118 0.048 CID_7515

0.1030.0160.132Purinergic P2X1 antagonist

0.132 0.009 CID_7515

CID_7515
0.2290.1440.229Antithrombotic

0.221 0.152 CID_7515

0.1820.0970.182Anticonvulsant

0.175 0.103 CID_7515

0.0990.0150.099Androgen agonist

0.083 0.022 CID_7515

0.1090.0240.112mTOR complex 2 inhibitor

0.112 0.022 CID_7515

CID_7515
0.0930.0090.093Transcription factor RelA inhibitor

0.068 0.034 CID_7515

0.1320.0480.207Interleukin 8 antagonist

0.207 0.011 CID_7515

CID_7515
0.1330.050.1335 Hydroxytryptamine 2B antagonist

0.113 0.068 CID_7515

0.2240.1410.224Thyroid hormone antagonist
0.0860.0030.086Protease (Human cytomegalovirus) inhibitor

0.045 0.005 CID_7515

0.110.0270.11Histamine H2 receptor antagonist

0.106 0.03 CID_7515

0.1210.0390.121Anabolic

0.116 0.044 CID_7515

0.0860.0050.114Diamine oxidase inhibitor

0.114 0.004 CID_7515

CID_7515
0.1350.0540.135Acetylcholine muscarinic antagonist

0.108 0.081 CID_7515

0.1060.0250.106Alpha adrenoreceptor agonist

0.097 0.029 CID_7515

0.0890.0090.089Calcium channel P-type blocker

0.063 0.047 CID_7515

0.1070.0260.107Glutamate decarboxylase inhibitor

0.096 0.032 CID_7515

0.0910.010.091Aconitate hydratase inhibitor

0.078 0.014 CID_7515

0.0840.0050.095Alpha 1d adrenoreceptor agonist

0.095 0.004 CID_7515

CID_7515
0.0920.0120.096Histone deacetylase SIRT3 inhibitor

0.096 0.011 CID_7515

CID_7515
0.1030.0240.115Carbonic anhydrase VA inhibitor

0.115 0.019 CID_7515

CID_7515
0.1150.0360.135Protein kinase C zeta inhibitor

0.135 0.025 CID_7515

CID_7515
0.1610.0830.161Dual specificity phosphatase inhibitor

0.131 0.119 CID_7515

0.0840.0060.146Dihydropteroate synthase inhibitor

0.146 0.004 CID_7515

CID_7515
0.1220.0440.122Beta glucuronidase inhibitor

0.106 0.062 CID_7515

0.1160.0390.117Interleukin 1 beta converting enzyme inhibitor

0.117 0.038 CID_7515

CID_7515
0.0910.0140.091Exportin-1 inhibitor

0.077 0.03 CID_7515

0.0920.0150.092Potassium channel (Tandem pore domain) blocker

0.085 0.024 CID_7515

0.0940.0170.094Protein kinase C beta inhibitor

0.086 0.023 CID_7515

0.0840.0080.084Mannosidase inhibitor

0.067 0.013 CID_7515

0.0940.0180.094Phospholipase D inhibitor

0.086 0.026 CID_7515

0.2130.1370.22812-Lipoxygenase inhibitor

0.228 0.124 CID_7515

CID_7515
0.080.0050.08Endothelial nitric-oxide synthase inhibitor

0.069 0.006 CID_7515

0.1010.0270.119Carbonic anhydrase V inhibitor

0.119 0.022 CID_7515

CID_7515
0.0850.010.085Histone deacetylase 7 inhibitor

0.039 0.024 CID_7515

0.0850.010.085Progesterone antagonist
0.0810.0070.081Cholesterol esterase inhibitor

0.048 0.033 CID_7515

0.1670.0930.251MAP kinase kinase 5 inhibitor

0.251 0.006 CID_7515

CID_7515
0.0840.0110.092Potassium channel (Inward rectifier) blocker

0.092 0.009 CID_7515

CID_7515
0.0870.0150.087Fatty acid synthase inhibitor

0.051 0.05 CID_7515

0.2150.1420.215Thyroid hormone beta antagonist
0.10.0290.1Interferon agonist

0.081 0.051 CID_7515

0.0850.0130.085Glucosylceramidase inhibitor

0.062 0.029 CID_7515

0.0790.0080.079Thymidylate synthase inhibitor

0.055 0.021 CID_7515

0.0940.0240.094Acetylcholine M5 receptor agonist

0.071 0.043 CID_7515

0.090.020.135NMDA 2C receptor antagonist

0.135 0.008 CID_7515

CID_7515
0.1150.0460.115Insulin receptor antagonist

0.097 0.066 CID_7515

0.0840.0150.084Phosphodiesterase 1A inhibitor

0.076 0.019 CID_7515

0.0730.0050.073Alpha 1L adrenoreceptor agonist
0.1170.0490.117Butyrylcholinesterase inhibitor
0.0790.0110.095Dihydroorotate oxidase inhibitor

0.095 0.005 CID_7515

CID_7515
0.0720.0050.072Integrin alpha2 antagonist

0.051 0.011 CID_7515

0.0720.0040.072Kainate receptor agonist

0.056 0.009 CID_7515

0.0970.030.097Aminopeptidase I inhibitor

0.088 0.035 CID_7515

0.0920.0250.1035 Hydroxytryptamine 1D antagonist

0.103 0.021 CID_7515

CID_7515
0.0720.0050.072Vascular adhesion protein 1 inhibitor
0.0750.0080.075Immunoglobulin Fc receptor antagonist

0.075 0.008 CID_7515

0.0790.0130.0795 Hydroxytryptamine 7 agonist

0.057 0.037 CID_7515

0.0880.0230.088Orexin receptor 1 antagonist
0.0880.0230.088Argininosuccinate synthase inhibitor

0.079 0.026 CID_7515

0.0760.0110.076Potassium channel small-conductance Ca-activated blocker

0.045 0.03 CID_7515

0.1550.0920.155Dual specificity phosphatase 3 inhibitor
0.0960.0320.096Histone deacetylase SIRT2 inhibitor

0.087 0.039 CID_7515

0.0860.0220.0863-Oxoacyl-[acyl-carrier-protein] synthase inhibitor

0.054 0.047 CID_7515

0.0950.0320.095Acetylcholine M4 receptor antagonist
0.1580.0960.247DNA methyltransferase I inhibitor

0.247 0.048 CID_7515

CID_7515
0.1280.0660.128Nav1.3 sodium channel blocker

0.107 0.089 CID_7515

0.1290.0670.132Vanilloid 1 agonist

0.132 0.063 CID_7515

CID_7515
0.10.0380.11Carbonic anhydrase XIII inhibitor

0.11 0.033 CID_7515

CID_7515
0.0950.0330.095Thioredoxin reductase inhibitor
0.1160.0540.116Expectorant

0.092 0.078 CID_7515

0.0860.0240.167NMDA receptor glycine site agonist

0.167 0.004 CID_7515

CID_7515
0.0720.0110.072Glucose-6-phosphate isomerase inhibitor

0.068 0.013 CID_7515

0.090.0290.095 Hydroxytryptamine 1B antagonist

0.073 0.038 CID_7515

0.1550.0940.271Death-associated protein kinase 2 inhibitor

0.271 0.01 CID_7515

CID_7515
0.0790.0180.117Potassium channel intermediate-conductance Ca-activated blocker

0.117 0.005 CID_7515

CID_7515
0.0820.0220.0965 Hydroxytryptamine 6 antagonist

0.096 0.016 CID_7515

CID_7515
0.0930.0330.093Transforming growth factor beta 3 antagonist
0.1670.1070.262Growth factor agonist

0.262 0.027 CID_7515

CID_7515
0.070.0110.07Glutamate (mGluR1a) antagonist

0.062 0.014 CID_7515

0.0650.0060.065Histamine H1 receptor agonist

0.06 0.008 CID_7515

0.20.140.2Lipoxygenase inhibitor

0.183 0.159 CID_7515

0.0890.0290.089Glycine receptor agonist

0.077 0.043 CID_7515

0.0680.0090.068Estradiol 17 beta-dehydrogenase 2 inhibitor
0.0980.040.134Carbonic anhydrase VI inhibitor

0.134 0.025 CID_7515

CID_7515
0.0680.010.068Histone deacetylase 9 inhibitor

0.042 0.023 CID_7515

0.0940.0360.106Nicotinic alpha4beta2 receptor antagonist

0.106 0.027 CID_7515

CID_7515
0.1030.0450.107Alpha 2 adrenoreceptor antagonist

0.107 0.043 CID_7515

CID_7515
0.0810.0230.081Interferon inducer

0.065 0.042 CID_7515

0.0650.0080.065Dihydrofolate reductase inhibitor

0.05 0.018 CID_7515

0.0940.0370.094Na+ K+ transporting ATPase inhibitor

0.082 0.049 CID_7515

0.090.0330.116Adenosine A3 receptor antagonist

0.116 0.019 CID_7515

CID_7515
0.0920.0350.117Histidine decarboxylase inhibitor

0.117 0.026 CID_7515

CID_7515
0.0660.0090.066Benzodiazepine antagonist

0.054 0.02 CID_7515

0.0820.0250.105Aryl hydrocarbon receptor antagonist

0.105 0.012 CID_7515

CID_7515
0.1210.0640.121Cholesterol synthesis inhibitor
0.1850.1290.185Calpain inhibitor

0.182 0.132 CID_7515

0.0690.0130.069Histamine H4 receptor antagonist

0.067 0.014 CID_7515

0.070.0140.093NMDA receptor subunit 3A antagonist

0.093 0.009 CID_7515

CID_7515
0.1350.080.135Activin receptor-like kinase 2 inhibitor

0.127 0.089 CID_7515

0.1330.0780.136Aurora-C kinase inhibitor

0.136 0.071 CID_7515

CID_7515
0.210.1550.21Caspase 3 stimulant
0.140.0860.175MAP kinase 3 inhibitor

0.175 0.038 CID_7515

CID_7515
0.1490.0950.149Antipruritic

0.136 0.112 CID_7515

0.0590.0050.059LIM domain kinase 2 inhibitor

0.041 0.009 CID_7515

0.0580.0040.058Integrin alpha2beta1 antagonist

0.036 0.008 CID_7515

0.1150.0610.115DNA intercalator
0.0720.0180.082Histamine agonist

0.082 0.013 CID_7515

CID_7515
0.1240.070.124Cholinergic antagonist

0.102 0.093 CID_7515

0.0990.0450.099Phosphodiesterase I inhibitor

0.097 0.048 CID_7515

0.080.0270.08Orexin receptor antagonist
0.0590.0060.059Liver X receptor beta antagonist

0.032 0.017 CID_7515

0.0630.010.063Cytokine production stimulant

0.051 0.027 CID_7515

0.0620.0090.062GABA uptake inhibitor

0.05 0.016 CID_7515

0.080.0270.08Protease 3C (Human rhinovirus) inhibitor

0.064 0.045 CID_7515

0.0850.0330.086Phosphodiesterase VI inhibitor

0.086 0.033 CID_7515

CID_7515
0.0810.0290.081Histone deacetylase inhibitor

0.062 0.05 CID_7515

0.0930.0410.116Catalase inhibitor

0.116 0.034 CID_7515

CID_7515
0.0760.0250.081Cyclin-dependent kinase 6 inhibitor

0.081 0.021 CID_7515

CID_7515
0.0660.0140.066Histone deacetylase 8 inhibitor

0.047 0.024 CID_7515

0.0730.0220.073Botulinum neurotoxin type A inhibitor

0.062 0.035 CID_7515

0.0560.0050.056CF transmembrane conductance regulator antagonist

0.041 0.023 CID_7515

0.1040.0520.165Potassium channel (Ca-activated) activator

0.165 0.023 CID_7515

CID_7515
0.1210.070.121Acetylcholine antagonist

0.101 0.092 CID_7515

0.0570.0070.057Protein 30S ribosomal subunit inhibitor
0.0780.0270.078Glutamate (mGluR6) antagonist

0.078 0.027 CID_7515

0.060.010.06Farnesoid X receptor agonist
0.0960.0450.107Bcr-Abl kinase inhibitor

0.107 0.035 CID_7515

CID_7515
0.1160.0660.12Caspase 3 inhibitor

0.12 0.061 CID_7515

CID_7515
0.0790.030.079MAP kinase kinase 10 inhibitor
0.0670.0170.067Estradiol 17 beta-dehydrogenase inhibitor
0.0620.0130.062Dopamine beta hydroxylase inhibitor

0.054 0.023 CID_7515

0.0670.0180.067Pregnane X receptor antagonist

0.057 0.038 CID_7515

0.0670.0180.067Topoisomerase II beta inhibitor

0.065 0.019 CID_7515

0.0550.0060.055CDK4/cyclin D3 inhibitor

0.029 0.019 CID_7515

0.060.0110.06Guanylate cyclase inhibitor

0.041 0.032 CID_7515

0.0620.0130.062Glutamate (mGluR4) antagonist

0.045 0.027 CID_7515

0.0560.0080.056Heme oxygenase inhibitor

0.041 0.038 CID_7515

0.0920.0440.111Acetylcholine nicotinic agonist

0.111 0.03 CID_7515

CID_7515
0.0820.0340.085Secretase beta inhibitor

0.085 0.03 CID_7515

CID_7515
0.0830.0370.083Benzodiazepine agonist

0.066 0.057 CID_7515

0.060.0140.06AICAR transformylase inhibitor

0.052 0.02 CID_7515

0.0720.0260.106Cyclin H inhibitor

0.106 0.006 CID_7515

CID_7515
0.0550.010.0813-Hydroxyanthranilate 3,4-dioxygenase inhibitor

0.081 0.004 CID_7515

CID_7515
0.0510.0060.051Methionyl aminopeptidase 1 inhibitor

0.041 0.011 CID_7515

0.0990.0540.117Alcohol dehydrogenase inhibitor

0.117 0.037 CID_7515

CID_7515
0.0650.020.071H+/K+-transporting ATPase inhibitor

0.071 0.017 CID_7515

CID_7515
0.1780.1340.178Immunostimulant

0.178 0.134 CID_7515

0.2540.210.254Apoptosis agonist
0.0940.0510.094Ornithine decarboxylase inhibitor

0.077 0.071 CID_7515

0.0720.0290.072Acetylcholine M5 receptor antagonist

0.059 0.043 CID_7515

0.0470.0040.047Glucosylceramidase stimulant

0.045 0.004 CID_7515

0.0560.0120.058Nerve growth factor antagonist

0.058 0.011 CID_7515

CID_7515
0.0460.0040.046Estrogen-related receptor gamma antagonist

0.036 0.008 CID_7515

0.0570.0140.057Liver X receptor alpha agonist
0.0520.010.094Potassium channel small-conductance Ca-activated activator

0.094 0.004 CID_7515

CID_7515
0.1050.0620.105Toll-Like receptor 4 antagonist
0.0620.0190.07CXC chemokine 1 receptor antagonist

0.07 0.013 CID_7515

CID_7515
0.0950.0530.148Potassium channel activator

0.148 0.021 CID_7515

CID_7515
0.070.0280.07Calcium channel T-type blocker
0.0790.0370.084Sphingosine 1-phosphate receptor 4 agonist

0.084 0.034 CID_7515

CID_7515
0.0570.0160.061Geranyltranstransferase inhibitor

0.061 0.013 CID_7515

CID_7515
0.1050.0640.105AMP-activated protein kinase stimulant
0.0590.0180.073Adenylate cyclase 1 inhibitor

0.073 0.011 CID_7515

CID_7515
0.0490.0080.059Protein kinase (CK2) beta inhibitor

0.059 0.005 CID_7515

CID_7515
0.0640.0240.064Acetyl-CoA transferase 2 inhibitor
0.0920.0520.168Stem cell growth factor agonist

0.168 0.015 CID_7515

CID_7515
0.1120.0720.112Proteasome inhibitor
0.0650.0250.065Ryanodine receptor antagonist

0.062 0.032 CID_7515

0.1270.0880.127Farnesoid X receptor antagonist
0.0730.0330.196NMDA receptor agonist

0.196 0.005 CID_7515

CID_7515
0.0990.060.099Platelet activating factor alpha antagonist
0.0640.0240.064Epithelial sodium channel blocker

0.058 0.031 CID_7515

0.0560.0170.062Histamine H2 receptor agonist

0.062 0.014 CID_7515

CID_7515
0.0690.0290.069Heat shock protein 90 beta antagonist

0.057 0.046 CID_7515

0.1530.1140.234DNA methylase inhibitor

0.234 0.058 CID_7515

CID_7515
0.0530.0140.053Potassium channel KCNQ activator

0.034 0.029 CID_7515

0.0530.0140.053Delayed rectifier potassium channel activator

0.034 0.029 CID_7515

0.0470.0090.047Bradykinin B2 receptor antagonist
0.070.0320.07Acetylcholine M3 receptor antagonist
0.090.0520.095 Hydroxytryptamine 2C antagonist

0.084 0.057 CID_7515

0.0420.0040.042Ileal bile acid transport inhibitor

0.015 0.014 CID_7515

0.0690.0310.069Dopamine uptake inhibitor

0.056 0.042 CID_7515

0.0620.0240.073Nicotinic alpha3beta2 receptor antagonist

0.073 0.016 CID_7515

CID_7515
0.0530.0150.054Dopamine D5 agonist

0.054 0.015 CID_7515

CID_7515
0.0640.0270.064Acetyl-CoA transferase inhibitor
0.0630.0260.075Nicotinic receptor alpha7 subunit antagonist

0.075 0.019 CID_7515

CID_7515
0.1460.110.146Platelet adhesion inhibitor
0.0440.0080.044Liver X receptor alpha antagonist
0.0710.0350.071MDM2 inhibitor

0.065 0.055 CID_7515

0.040.0040.04Alpha 2a adrenoreceptor agonist

0.038 0.004 CID_7515

0.070.0350.07Adrenaline uptake inhibitor
0.0850.0490.11T cell inhibitor

0.11 0.018 CID_7515

CID_7515
0.0460.0110.046Liver X receptor antagonist
0.0630.0280.063MAP kinase kinase 9 inhibitor

0.057 0.037 CID_7515

0.0430.0080.045Adenosine uptake inhibitor

0.045 0.006 CID_7515

CID_7515
0.0550.0210.057Fructose-1,6-bisphosphatase inhibitor

0.057 0.019 CID_7515

CID_7515
0.0470.0130.049Glutamate (mGluR8) agonist

0.049 0.012 CID_7515

CID_7515
0.1160.0820.123Toll-Like receptor 2 antagonist

0.123 0.075 CID_7515

CID_7515
0.0410.0070.046Nicotinic alpha4beta2 receptor agonist

0.046 0.005 CID_7515

CID_7515
0.0810.0470.081Alpha 2a adrenoreceptor antagonist

0.07 0.057 CID_7515

0.0410.0070.041Adenosine kinase inhibitor

0.023 0.014 CID_7515

0.0940.0610.102Toll-Like receptor 3 antagonist

0.102 0.048 CID_7515

CID_7515
0.0670.0340.0975 Hydroxytryptamine 5A antagonist

0.097 0.017 CID_7515

CID_7515
0.1280.0960.128Diuretic

0.119 0.106 CID_7515

0.0660.0340.08Cyclin D1 inhibitor

0.08 0.018 CID_7515

CID_7515
0.1180.0860.25Protein-tyrosine kinase Lyn inhibitor

0.25 0.029 CID_7515

CID_7515
0.080.0480.08Estrogen receptor alpha antagonist
0.0440.0120.044Ceramide glucosyltransferase inhibitor
0.0410.010.041Nicotinic alpha3beta4 receptor agonist

0.035 0.014 CID_7515

0.0530.0220.089CDK7/cyclin H inhibitor

0.089 0.007 CID_7515

CID_7515
0.0870.0570.123NMDA receptor antagonist

0.123 0.034 CID_7515

CID_7515
0.0750.0450.075Calcium channel L-type blocker
0.0430.0130.043Liver X receptor beta agonist
0.0560.0260.056Antiviral (Hepatitis D)
0.070.040.07Dopamine D1 antagonist

0.058 0.052 CID_7515

0.0380.0080.042MAP3K8 inhibitor

0.042 0.006 CID_7515

CID_7515
0.0820.0530.085Acetylcholine nicotinic antagonist

0.085 0.049 CID_7515

CID_7515
0.0450.0160.045Fumarate hydratase inhibitor

0.035 0.023 CID_7515

0.090.0610.119Polo-like kinase-1 inhibitor

0.119 0.031 CID_7515

CID_7515
0.0470.0180.047Membrane dipeptidase inhibitor

0.041 0.026 CID_7515

0.0510.0230.075Glutamate (mGluR group III) agonist

0.075 0.014 CID_7515

CID_7515
0.0950.0680.128Cyclin-dependent kinase 9 inhibitor

0.128 0.042 CID_7515

CID_7515
0.0310.0040.031Estrogen-related receptor gamma agonist

0.019 0.012 CID_7515

0.0650.0380.065Phosphodiesterase 1C inhibitor
0.0360.0090.036Purinergic P2Y15 antagonist

0.036 0.009 CID_7515

0.0440.0170.044Retinoid X alpha receptor agonist

0.034 0.025 CID_7515

0.0310.0050.031Alpha 2c adrenoreceptor agonist

0.028 0.005 CID_7515

0.0420.0160.042Sirtuin 2 inhibitor

0.03 0.026 CID_7515

0.0570.0320.067Lysine-specific demethylase 1A inhibitor

0.067 0.02 CID_7515

CID_7515
0.1150.0890.179Cyclin-dependent kinase 7 inhibitor

0.179 0.043 CID_7515

CID_7515
0.0780.0530.078Viral attachment inhibitor
0.0340.0080.039Hedgehog signaling activator

0.039 0.005 CID_7515

CID_7515
0.0610.0350.07Alpha 1 adrenoreceptor agonist

0.07 0.028 CID_7515

CID_7515
0.0630.0380.092Enoyl-[acyl-carrier-protein] reductase inhibitor

0.092 0.013 CID_7515

CID_7515
0.0740.0490.074Cathepsin G inhibitor
0.0570.0330.057Ornithine carbamoyltransferase inhibitor

0.054 0.036 CID_7515

0.0580.0340.058Sphingosine kinase 2 inhibitor

0.056 0.037 CID_7515

0.0460.0220.046Thymidine kinase inhibitor

0.044 0.024 CID_7515

0.0340.010.0345 Hydroxytryptamine 1F agonist
0.0620.0380.074Carbonic anhydrase stimulant

0.074 0.029 CID_7515

CID_7515
0.0260.0030.026Antibiotic Tetracycline-like
0.0370.0140.042Epoxide hydrolase 1 inhibitor

0.042 0.01 CID_7515

CID_7515
0.0620.040.062Beta 2 adrenoreceptor agonist

0.061 0.045 CID_7515

0.0490.0260.091Purinergic P2X4 antagonist

0.091 0.005 CID_7515

CID_7515
0.070.0480.079ZAP-70 protein tyrosine kinase inhibitor

0.079 0.036 CID_7515

CID_7515
0.0430.0210.043Retinoid X receptor agonist
0.0420.020.042Retinoid X receptor antagonist
0.0760.0540.087Keratolytic

0.087 0.041 CID_7515

CID_7515
0.0560.0340.0563(or 17)beta-hydroxysteroid dehydrogenase inhibitor

0.051 0.041 CID_7515

0.0310.0090.031Vanilloid 2 agonist

0.028 0.013 CID_7515

0.0590.0380.0915 Hydroxytryptamine 5 antagonist

0.091 0.017 CID_7515

CID_7515
0.1030.0810.123Interleukin 2 antagonist

0.123 0.041 CID_7515

CID_7515
0.070.0490.07CXC chemokine receptor antagonist
0.0490.0280.049CC chemokine 4 receptor antagonist

0.046 0.034 CID_7515

0.0330.0130.0355 Hydroxytryptamine 6 agonist

0.035 0.011 CID_7515

CID_7515
0.030.0090.038Acid ceramidase inhibitor

0.038 0.005 CID_7515

CID_7515
0.0550.0350.055Protein 50S ribosomal subunit inhibitor
0.0550.0350.055GABA A receptor antagonist
0.040.0190.04Glucocorticoid antagonist
0.0350.0150.035Cyclin E2 inhibitor
0.0470.0270.108NMDA receptor subunit 3B antagonist

0.108 0.01 CID_7515

CID_7515
0.0860.0650.093Pim-3 kinase inhibitor

0.093 0.054 CID_7515

CID_7515
0.0440.0230.044Histone deacetylase class I inhibitor
0.0790.0590.216TIE-2 antagonist

0.216 0.013 CID_7515

CID_7515
0.0380.0180.038Retinoid X alpha receptor antagonist
0.0760.0560.076Macrophage migration inhibitory factor inhibitor
0.0530.0330.0535 Hydroxytryptamine 4 antagonist

0.048 0.041 CID_7515

0.0790.060.222TIE antagonist

0.222 0.013 CID_7515

CID_7515
0.0420.0220.042Protein kinase (CK1) epsilon inhibitor

0.042 0.022 CID_7515

0.0450.0250.045Angiotensin AT1 receptor antagonist
0.1410.1210.141Ca2+/calmodulin-dependent protein kinase inhibitor
0.0820.0630.085Acetylcholine agonist

0.085 0.06 CID_7515

CID_7515
0.0230.0040.023Human herpes virus 5 capsid protein P40 inhibitor

0.013 0.009 CID_7515

0.0840.0650.086Interleukin-1 receptor-associated protein kinase 4 inhibitor

0.086 0.062 CID_7515

CID_7515
0.0410.0230.0425 Hydroxytryptamine 2B agonist

0.042 0.022 CID_7515

CID_7515
0.0270.0080.027Glutaminyl-peptide cyclotransferase inhibitor

0.025 0.01 CID_7515

0.0390.020.048Phosphoglycerate kinase inhibitor

0.048 0.015 CID_7515

CID_7515
0.0490.0310.067Adenosine deaminase inhibitor

0.067 0.016 CID_7515

CID_7515
0.0410.0220.041Factor XIIIa inhibitor

0.036 0.028 CID_7515

0.0360.0180.036Histone deacetylase 10 inhibitor
0.0310.0120.031Myristoyl transferase inhibitor

0.025 0.023 CID_7515

0.0690.050.069Amidase inhibitor
0.0550.0370.055GABA receptor antagonist
0.090.0720.128Protein kinase (CK2) inhibitor

0.128 0.043 CID_7515

CID_7515
0.0610.0430.061Acetylcholine M2 receptor antagonist
0.0580.040.058Adenosine A1 receptor antagonist

0.053 0.045 CID_7515

0.0640.0460.064Neutrophil collagenase inhibitor
0.0360.0180.036Estradiol 17 beta-dehydrogenase 3 inhibitor
0.0510.0330.078Potassium channel (Inward rectifier) activator

0.078 0.008 CID_7515

CID_7515
0.0280.0110.028Complement factor 1s inhibitor

0.028 0.01 CID_7515

0.0550.0380.055Maillard reaction inhibitor
0.0660.0480.072Neuronal nicotinic receptor antagonist

0.072 0.043 CID_7515

CID_7515
0.0390.0220.0392,3-Oxidosqualene-lanosterol cyclase inhibitor
0.0370.020.037Free fatty acid receptor 1 antagonist
0.0510.0340.059Lysophosphatidic acid 3 receptor antagonist

0.059 0.023 CID_7515

CID_7515
0.0410.0240.049MAP3K5 inhibitor

0.049 0.013 CID_7515

CID_7515
0.0390.0230.057Inosine monophosphate dehydrogenase inhibitor

0.057 0.011 CID_7515

CID_7515
0.0390.0220.039Orexin receptor 2 antagonist
0.0390.0230.039Delayed rectifier potassium channel blocker

0.038 0.024 CID_7515

0.0490.0320.075Potassium channel (ATP-sensitive) activator

0.075 0.008 CID_7515

CID_7515
0.0630.0470.071Beta 3 adrenoreceptor antagonist

0.071 0.032 CID_7515

CID_7515
0.0290.0130.029Thymidine kinase (Herpes simplex virus 1) inhibitor

0.028 0.016 CID_7515

0.0240.0090.024Histamine H4 receptor agonist

0.02 0.012 CID_7515

0.0530.0370.058Heparanase inhibitor

0.058 0.026 CID_7515

CID_7515
0.140.1240.14Clk dual-specificity kinase inhibitor
0.0350.020.035Melatonin receptor 1A agonist
0.0240.0090.024Thymidine kinase (Herpes simplex virus 2) inhibitor

0.022 0.01 CID_7515

0.0810.0660.081Insulin growth factor antagonist
0.0540.0390.054Acetylcholine muscarinic agonist
0.020.0050.02CDK2/cyclin A3 inhibitor

0.016 0.013 CID_7515

0.0670.0520.067Syk tyrosine kinase inhibitor

0.064 0.055 CID_7515

0.0640.050.0955 Hydroxytryptamine 3A antagonist

0.095 0.019 CID_7515

CID_7515
0.0310.0170.031Hypoxanthine phosphoribosyltransferase inhibitor

0.028 0.019 CID_7515

0.0720.0580.072Analgesic, opioid
0.0430.0290.043Leukocyte elastase inhibitor
0.0540.040.057Carbonic anhydrase IX inhibitor

0.057 0.039 CID_7515

CID_7515
0.0470.0340.047Antimetabolite
0.0760.0630.082Adrenaline agonist

0.082 0.055 CID_7515

CID_7515
0.0420.0290.042Cholecystokinin antagonist

0.035 0.032 CID_7515

0.0230.010.027Factor XIII inhibitor

0.027 0.005 CID_7515

CID_7515
0.0230.010.023Retinoid X beta receptor antagonist
0.0770.0650.077Insulin like growth factor 1 antagonist
0.0430.030.043Liver X receptor agonist
0.0490.0370.049Prolyl endopeptidase inhibitor
0.0230.0110.023Apolipoprotein B inhibitor

0.018 0.016 CID_7515

0.1110.0990.117Alkaline phosphatase inhibitor

0.117 0.09 CID_7515

CID_7515
0.0850.0730.085Protein kinase C mu inhibitor

0.081 0.079 CID_7515

0.0530.0410.059Carbonic anhydrase II inhibitor

0.059 0.035 CID_7515

CID_7515
0.0210.0090.021Antibiotic Anthracycline-like

0.02 0.01 CID_7515

0.0420.030.042Oxytocin agonist

0.041 0.03 CID_7515

0.0320.020.032Cholesterol ester transfer protein antagonist
0.0350.0230.035Angiotensin II receptor antagonist
0.0170.0050.0171-Deoxy-D-xylulose-5-phosphate reductoisomerase inhibitor

0.016 0.006 CID_7515

0.1040.0930.104Amylase inhibitor

0.104 0.093 CID_7515

0.0210.010.026Cyclin T1 inhibitor

0.026 0.007 CID_7515

CID_7515
0.0460.0350.046Aldosterone antagonist

0.046 0.036 CID_7515

0.0870.0760.087Xanthine oxidase inhibitor
0.040.030.04Acetyl-CoA transferase 1 inhibitor
0.0270.0170.034CXC chemokine 2 receptor antagonist

0.034 0.011 CID_7515

CID_7515
0.1280.1180.131Melanin inhibitor

0.131 0.112 CID_7515

CID_7515
0.0180.0080.025NMDA receptor phencyclidine site antagonist

0.025 0.005 CID_7515

CID_7515
0.0220.0120.029Imidazoline I1 receptor antagonist

0.029 0.008 CID_7515

CID_7515
0.0370.0270.06Potassium channel Kv1.1 blocker

0.06 0.009 CID_7515

CID_7515
0.0290.0190.045 Hydroxytryptamine 1D agonist

0.04 0.014 CID_7515

CID_7515
0.0880.0780.134MAP kinase kinase kinase inhibitor

0.134 0.043 CID_7515

CID_7515
0.0440.0340.044Glutamate (mGluR5) agonist
0.1030.0930.132Epidermal growth factor receptor kinase inhibitor

0.132 0.062 CID_7515

CID_7515
0.0750.0660.075Neuropeptide Y antagonist

0.074 0.07 CID_7515

0.0570.0480.066Carbonic anhydrase inhibitor

0.066 0.042 CID_7515

CID_7515
0.0240.0150.024Estradiol 17 beta-dehydrogenase 1 inhibitor
0.0340.0250.034Benzodiazepine receptor peripheral-type antagonist
0.0280.0190.028Motilin receptor antagonist
0.0770.0690.077GABA A receptor agonist
0.1220.1140.122Phospholipase A2 inhibitor
0.0190.0110.019Apolipoprotein B-100 inhibitor
0.0670.0580.092MAP kinase 11 inhibitor

0.092 0.04 CID_7515

CID_7515
0.0670.0580.112Epoxide hydrolase inhibitor

0.112 0.019 CID_7515

CID_7515
0.0920.0840.116Protein kinase (CK2) alpha inhibitor

0.116 0.065 CID_7515

CID_7515
0.030.0230.03Histone deacetylase 11 inhibitor
0.030.0230.03Histone deacetylase class IV inhibitor
0.0640.0560.064Elastase 1 inhibitor
0.0480.040.048Carbonic anhydrase XII inhibitor

0.048 0.04 CID_7515

0.0430.0360.067Glycine transporter 2 inhibitor

0.067 0.022 CID_7515

CID_7515
0.0350.0270.036Tryptophan 5 hydroxylase inhibitor

0.036 0.023 CID_7515

CID_7515
0.0170.0090.017Purinergic P2Y1 agonist

0.016 0.009 CID_7515

0.0290.0220.029Peptide deformylase inhibitor

0.027 0.025 CID_7515

0.050.0430.05Carbonic anhydrase I inhibitor

0.048 0.045 CID_7515

0.0480.0410.0485 Hydroxytryptamine 2 agonist

0.045 0.044 CID_7515

0.0260.0190.026Nicotinic acid receptor 2 antagonist

0.026 0.019 CID_7515

0.0290.0230.029Acetylcholine M4 receptor agonist
0.0140.0080.014Cyclin D2 inhibitor

0.013 0.011 CID_7515

0.090.0840.09Monophenol monooxygenase inhibitor
0.0180.0120.018Methylmalonyl-CoA mutase inhibitor
0.0270.0210.027Uridine phosphorylase inhibitor
0.0240.0190.025Lysophosphatidic acid receptor 1 agonist

0.025 0.017 CID_7515

CID_7515
0.0230.0170.023ICAM 1 antagonist
0.0110.0050.011Progesterone receptor A antagonist
0.0560.050.088Potassium channel (Ca-activated) blocker

0.088 0.014 CID_7515

CID_7515
0.0430.0380.043Sigma receptor antagonist
0.0390.0340.039Acetylcholine M1 receptor agonist
0.0370.0320.037CC chemokine 3 receptor antagonist
0.0430.0380.043AMPA receptor antagonist
0.0160.0110.016Nicotinic alpha4 receptor agonist

0.015 0.013 CID_7515

0.1060.1020.106Sodium channel (voltage-gated) blocker
0.0190.0140.029Inosine monophosphate dehydrogenase 2 inhibitor

0.029 0.008 CID_7515

CID_7515
0.0170.0130.017CXC chemokine 5 receptor antagonist
0.0160.0120.021Carbonic anhydrase VIII inhibitor

0.021 0.007 CID_7515

CID_7515
0.0160.0120.021Carbonic anhydrase X inhibitor

0.021 0.007 CID_7515

CID_7515
0.0210.0170.021Geranylgeranyltransferase inhibitor
0.0310.0270.033Vanilloid 4 antagonist

0.033 0.022 CID_7515

CID_7515
0.0240.020.024Sigma 1 receptor antagonist
0.0210.0180.028Glutamate (mGluR1a) agonist

0.028 0.01 CID_7515

CID_7515
0.0190.0160.019Toll-Like receptor 8 agonist
0.0330.030.0335-Alpha-reductase inhibitor
0.0080.0050.01DNA topoisomerase III inhibitor

0.01 0.004 CID_7515

CID_7515
0.0490.0460.049Leukotriene B4 antagonist
0.040.0370.04Factor Xa inhibitor
0.0150.0120.02Thromboxane A2 agonist

0.02 0.006 CID_7515

CID_7515
0.0360.0340.036AMPA 4 receptor antagonist
0.0480.0470.048Protein kinase C eta inhibitor
0.0240.0230.026Complement factor 1r inhibitor

0.026 0.017 CID_7515

CID_7515
0.0620.060.062MAP kinase kinase 8 inhibitor
0.0480.0460.052Nicotinic alpha7 receptor agonist

0.052 0.04 CID_7515

CID_7515
0.0480.0470.066Nicotinic neuronal receptor agonist

0.066 0.031 CID_7515

CID_7515
0.0160.0150.02Nicotinic acid receptor 1 antagonist

0.02 0.009 CID_7515

CID_7515
0.1760.1750.176Prostaglandin dehydrogenase inhibitor
0.0180.0170.018Progesterone receptor B antagonist
0.0160.0150.016Telomerase stimulant
0.0110.0110.019Carbonic anhydrase XI inhibitor

0.019 0.004 CID_7515

CID_7515
0.010.010.013Imidazoline I2 receptor antagonist

0.013 0.005 CID_7515

CID_7515
0.030.030.033Glutamate (mGluR3) agonist

0.033 0.02 CID_7515

CID_7515
0.0290.030.051Calcium release-activated channel blocker

0.051 0.009 CID_7515

CID_7515
0.0170.0180.019Alpha 2b adrenoreceptor agonist

0.019 0.013 CID_7515

CID_7515
0.0190.0210.021Neuraminidase (Influenza B) inhibitor

0.021 0.015 CID_7515

CID_7515
0.0520.0550.062Phosphodiesterase 1B inhibitor

0.062 0.04 CID_7515

CID_7515
0.0420.0440.047Carbonic anhydrase XIV inhibitor

0.047 0.036 CID_7515

CID_7515
0.0240.0270.026Baculoviral IAP repeat-containing protein 4 inhibitor

0.026 0.024 CID_7515

CID_7515
0.0420.0450.046Adenosine A2b receptor antagonist

0.046 0.038 CID_7515

CID_7515
0.0360.0390.051Carbonic anhydrase IV inhibitor

0.051 0.024 CID_7515

CID_7515
0.0220.0260.025Lysine carboxypeptidase inhibitor

0.025 0.022 CID_7515

CID_7515
0.0430.0470.048HCV NS3/NS4A protease inhibitor

0.048 0.036 CID_7515

CID_7515
0.020.0240.024Fructose-1,6-bisphosphatase 1 inhibitor

0.024 0.015 CID_7515

CID_7515
0.0160.0190.018Complement factor D inhibitor

0.018 0.012 CID_7515

CID_7515
0.0520.0560.055Leukotriene C antagonist

0.055 0.044 CID_7515

CID_7515
0.0520.0560.058Sphingosine kinase inhibitor

0.058 0.043 CID_7515

CID_7515
0.0210.0260.025Glutamate (mGluR1) agonist

0.025 0.016 CID_7515

CID_7515
0.0390.0440.046Potassium channel Kv1.3 blocker

0.046 0.034 CID_7515

CID_7515
0.0330.0380.052Toll-Like receptor 2 agonist

0.052 0.023 CID_7515

CID_7515
0.0130.0180.015Adenosine A2 receptor agonist

0.015 0.013 CID_7515

CID_7515
0.0280.0340.039Arginase inhibitor

0.039 0.023 CID_7515

CID_7515
0.0420.0480.051Beta 2 adrenoreceptor antagonist

0.051 0.034 CID_7515

CID_7515
0.0430.0490.059mTOR inhibitor

0.059 0.029 CID_7515

CID_7515
0.0310.0370.041Glutamate (mGluR3) antagonist

0.041 0.019 CID_7515

CID_7515
0.1820.1880.222Thioredoxin glutathione reductase inhibitor

0.222 0.154 CID_7515

CID_7515
0.0380.0440.041Glycine transporter inhibitor

0.041 0.04 CID_7515

CID_7515
0.0540.0610.099I kappa B kinase 2 inhibitor

0.099 0.013 CID_7515

CID_7515
0.0590.0660.063Prostaglandin-E synthase inhibitor

0.063 0.058 CID_7515

CID_7515
0.0410.0480.068Ribonucleoside-diphosphate reductase inhibitor

0.068 0.03 CID_7515

CID_7515
0.0650.0740.087Fibroblast growth factor 3 antagonist

0.087 0.043 CID_7515

CID_7515
0.0290.0370.038Glutamate (mGluR4) agonist

0.038 0.017 CID_7515

CID_7515
0.2090.2180.226DNA polymerase beta inhibitor

0.226 0.207 CID_7515

CID_7515
0.0280.0370.0435 Hydroxytryptamine 3B antagonist

0.043 0.018 CID_7515

CID_7515
0.0410.050.069Ribonucleotide reductase inhibitor

0.069 0.031 CID_7515

CID_7515
0.0720.0810.076MAP kinase 7 inhibitor

0.076 0.058 CID_7515

CID_7515
0.0690.0790.142I kappa B kinase inhibitor

0.142 0.018 CID_7515

CID_7515
0.0650.0750.111Leucine-rich repeat kinase 2 inhibitor

0.111 0.036 CID_7515

CID_7515
0.0710.0820.093Epidermal growth factor antagonist

0.093 0.05 CID_7515

CID_7515
0.0490.060.067Cyclin A2 inhibitor

0.067 0.041 CID_7515

CID_7515
0.0840.0950.093Granulocyte macrophage colony stimulating factor antagonist

0.093 0.081 CID_7515

CID_7515
0.0350.0460.039Sphingosine kinase 1 inhibitor

0.039 0.033 CID_7515

CID_7515
0.0170.0290.039NMDA receptor glycine site antagonist

0.039 0.009 CID_7515

CID_7515
0.0480.060.061Sphingosine 1-phosphate receptor 3 antagonist

0.061 0.037 CID_7515

CID_7515
0.0450.0570.055EphB4 antagonist

0.055 0.044 CID_7515

CID_7515
0.1030.1160.114Protein kinase C nu inhibitor

0.114 0.1 CID_7515

CID_7515
0.0350.0480.042Carbonic anhydrase VII inhibitor

0.042 0.037 CID_7515

CID_7515
0.0440.0570.0795 Hydroxytryptamine 3 antagonist

0.079 0.025 CID_7515

CID_7515
0.0350.050.059Dihydroorotase inhibitor

0.059 0.017 CID_7515

CID_7515
0.0270.0420.041ATR kinase inhibitor

0.041 0.012 CID_7515

CID_7515
0.0440.0610.052Fibroblast growth factor 4 antagonist

0.052 0.05 CID_7515

CID_7515
0.0260.0420.041Nicotinic acid receptor agonist

0.041 0.02 CID_7515

CID_7515
0.050.0680.068Fibroblast growth factor 2 antagonist

0.068 0.043 CID_7515

CID_7515
0.0520.070.062Beta adrenoreceptor antagonist

0.062 0.051 CID_7515

CID_7515
0.0570.0760.082Rho-associated kinase I inhibitor

0.082 0.045 CID_7515

CID_7515
0.0190.0410.0265 Hydroxytryptamine 4 agonist

0.026 0.013 CID_7515

CID_7515
0.0980.1190.121Lipid peroxidase inhibitor

0.121 0.093 CID_7515

CID_7515
0.030.0520.075Purinergic P2Y antagonist

0.075 0.014 CID_7515

CID_7515
0.0250.0470.032Carnitine palmitoyltransferase inhibitor

0.032 0.027 CID_7515

CID_7515
0.0410.0630.054Beta 1 adrenoreceptor antagonist

0.054 0.041 CID_7515

CID_7515
0.0250.0480.032Carnitine palmitoyltransferase 1 inhibitor

0.032 0.027 CID_7515

CID_7515
0.0420.0660.062Cyclin A inhibitor

0.062 0.042 CID_7515

CID_7515
0.0140.0380.022Alpha 1a adrenoreceptor agonist

0.022 0.016 CID_7515

CID_7515
0.0180.0450.025Thyroid hormone agonist

0.025 0.02 CID_7515

CID_7515
0.1350.1640.198Proto-oncogene tyrosine-protein kinase Fyn inhibitor

0.198 0.075 CID_7515

CID_7515
0.0510.0820.067Vanilloid antagonist

0.067 0.059 CID_7515

CID_7515
0.0490.0810.158CDK1/cyclin B1 inhibitor

0.158 0.014 CID_7515

CID_7515
0.0430.0760.054Cyclin A1 inhibitor

0.054 0.051 CID_7515

CID_7515
0.0350.0680.05CDK4/cyclin D1 inhibitor

0.05 0.049 CID_7515

CID_7515
0.0870.120.175Lck kinase inhibitor

0.175 0.052 CID_7515

CID_7515
0.0540.0890.059Prolactin release inhibitor

0.059 0.055 CID_7515

CID_7515
0.0430.0820.053Sphingosine 1-phosphate receptor 1 antagonist

0.053 0.046 CID_7515

CID_7515
0.1140.1530.124CC chemokine 6 receptor antagonist

0.124 0.097 CID_7515

CID_7515
0.1030.1420.155Ca2+/calmodulin-dependent kinase II gamma inhibitor

0.155 0.086 CID_7515

CID_7515
0.0620.1020.073Sphingosine 1-phosphate receptor antagonist

0.073 0.061 CID_7515

CID_7515
0.0840.1280.143CDK3/cyclin E inhibitor

0.143 0.031 CID_7515

CID_7515
0.0620.1070.103Aurora-A kinase inhibitor

0.103 0.064 CID_7515

CID_7515
0.0870.1330.118Vascular endothelial growth factor 3 antagonist

0.118 0.096 CID_7515

CID_7515
0.0820.130.119CDC-like kinase 3 inhibitor

0.119 0.045 CID_7515

CID_7515
0.0720.1220.102Aurora-B kinase inhibitor

0.102 0.08 CID_7515

CID_7515
0.0360.0890.068Phosphodiesterase 7A inhibitor

0.068 0.013 CID_7515

CID_7515
0.1210.1740.143Death-associated protein kinase 3 inhibitor

0.143 0.134 CID_7515

CID_7515
0.030.0920.133Raf kinase C inhibitor

0.133 0.017 CID_7515

CID_7515
0.0750.1370.109TRKA antagonist

0.109 0.079 CID_7515

CID_7515
0.060.1230.128Mediator release inhibitor

0.128 0.041 CID_7515

CID_7515
0.050.1140.116Platelet activating factor beta antagonist

0.116 0.052 CID_7515

CID_7515
0.1590.2250.361Angiogenesis inhibitor

0.361 0.067 CID_7515

CID_7515
0.0350.1020.044Phosphodiesterase 6C inhibitor

0.044 0.042 CID_7515

CID_7515
0.0770.1440.118Tyrosine-protein kinase receptor antagonist

0.118 0.088 CID_7515

CID_7515
0.1170.1870.166Ca2+/calmodulin-dependent kinase II beta inhibitor

0.166 0.109 CID_7515

CID_7515
0.0070.0770.021Purinergic P2Y1 antagonist

0.021 0.008 CID_7515

CID_7515
0.0560.1270.093CDK2/cyclin A inhibitor

0.093 0.064 CID_7515

CID_7515
0.0390.1120.067Glutamate receptor agonist

0.067 0.066 CID_7515

CID_7515
0.0430.120.08Rho-associated kinase II inhibitor

0.08 0.045 CID_7515

CID_7515
0.0820.160.143Histone deacetylase SIRT1 inhibitor

0.143 0.068 CID_7515

CID_7515
0.0960.1780.124Papain-like protease (SARS coronavirus) inhibitor

0.124 0.071 CID_7515

CID_7515
0.0280.110.085CDK9/cyclin T1 inhibitor

0.085 0.024 CID_7515

CID_7515
0.0160.1020.037DNA gyrase subunit B inhibitor

0.037 0.028 CID_7515

CID_7515
0.1370.2240.191ErbB-1 antagonist

0.191 0.1 CID_7515

CID_7515
0.0470.1340.094Fibroblast growth factor 1 antagonist

0.094 0.063 CID_7515

CID_7515
0.0480.1350.086AXL receptor tyrosine kinase inhibitor

0.086 0.052 CID_7515

CID_7515
0.0370.1250.057CDC25B inhibitor

0.057 0.055 CID_7515

CID_7515
0.0290.1170.087Phosphodiesterase VII inhibitor

0.087 0.02 CID_7515

CID_7515
0.0210.110.037Antibiotic Aminoglycoside-like

0.037 0.024 CID_7515

CID_7515
0.0560.1490.15Vascular endothelial growth factor antagonist

0.15 0.054 CID_7515

CID_7515
0.0720.170.178Tyrosine kinase inhibitor

0.178 0.077 CID_7515

CID_7515
0.1290.2290.198MAP-kinase-activated kinase 5 inhibitor

0.198 0.106 CID_7515

CID_7515
0.0440.1480.066Kallikrein 7 inhibitor

0.066 0.037 CID_7515

CID_7515
0.0430.1540.137Vascular endothelial growth factor 2 antagonist

0.137 0.053 CID_7515

CID_7515
0.0670.1930.163Src kinase inhibitor

0.163 0.075 CID_7515

CID_7515
0.0910.2260.257Interleukin 6 antagonist

0.257 0.022 CID_7515

CID_7515
0.0330.1790.102Cyclin-dependent kinase 1 inhibitor

0.102 0.065 CID_7515

CID_7515
0.0340.180.116Protein kinase (Mos, Mil/Raf, MEKK, RIPK, TESK, LIMK, IRAK, ILK, Activin/TGF-beta) inhibitor

0.116 0.042 CID_7515

CID_7515
0.0350.1850.207Tyrosine-protein kinase receptor FLT3 inhibitor

0.207 0.035 CID_7515

CID_7515
0.0730.2290.135Protein kinase (CK1) gamma 3 inhibitor

0.135 0.107 CID_7515

CID_7515
0.0520.2070.12Interleukin 5 antagonist

0.12 0.023 CID_7515

CID_7515
0.0360.1920.206I kappa B kinase 1 inhibitor

0.206 0.005 CID_7515

CID_7515
0.0390.1990.089Vascular endothelial growth factor 1 antagonist

0.089 0.074 CID_7515

CID_7515
0.0280.2020.157Proto-oncogene tyrosine-protein kinase Kit inhibitor

0.157 0.031 CID_7515

CID_7515
0.0310.2050.071Protein kinase A inhibitor

0.071 0.07 CID_7515

CID_7515
0.020.1960.093Raf kinase inhibitor

0.093 0.037 CID_7515

CID_7515
0.0880.2640.29Ca2+/calmodulin-dependent kinase I alpha inhibitor

0.29 0.043 CID_7515

CID_7515
0.0370.2160.13Protein-tyrosine kinase (PTK, not ETK, WZC) inhibitor

0.13 0.06 CID_7515

CID_7515
0.0360.2180.13Abl kinase inhibitor

0.13 0.06 CID_7515

CID_7515
0.0140.1970.058Raf kinase B inhibitor

0.058 0.043 CID_7515

CID_7515
0.0570.2640.115Protein kinase (CK1) gamma 1 inhibitor

0.115 0.103 CID_7515

CID_7515
0.0280.2580.1c-Src kinase inhibitor

0.1 0.089 CID_7515

CID_7515
0.0970.3310.206Cyclin-dependent kinase 3 inhibitor

0.206 0.03 CID_7515

CID_7515
0.010.2450.266Tyk2 inhibitor

0.266 0.005 CID_7515

CID_7515
0.0250.2920.09Polo-like kinase-2 inhibitor

0.09 0.035 CID_7515

CID_7515
0.0780.3560.169Death-associated protein kinase 1 inhibitor

0.169 0.019 CID_7515

CID_7515
0.1160.4090.214Interleukin 2 agonist

0.214 0.166 CID_7515

CID_7515
0.0280.3230.116TRKB antagonist

0.116 0.078 CID_7515

CID_7515
0.0130.3260.06Check point kinase 1 inhibitor

0.06 0.058 CID_7515

CID_7515
0.0420.4080.088Hematopoietic

0.088 0.052 CID_7515

CID_7515
0.0150.4070.141Protein kinase B gamma inhibitor

0.141 0.019 CID_7515

CID_7515
0.0430.4660.207Polo-like kinase-3 inhibitor

0.207 0.041 CID_7515

CID_7515
0.0060.4610.048Factor VIIa inhibitor

0.048 0.021 CID_7515

CID_7515
0.0050.7260.121DNA gyrase inhibitor

0.121 0.013 CID_7515

CID_7515
0.0290.7690.143NOS3 expression enhancer

0.143 0.08 CID_7515

CID_7515
Ext Pa Pi Pmax Activity Other Results ID Pa_max