| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.938 | 0.001 | 0.939 | Retinoic acid receptor agonist | 0.939 0.001 DBMET01736 | DBMET01736 | |
| 0.905 | 0.005 | 0.907 | Apoptosis agonist | 0.907 0.005 DBMET01736 | DBMET01736 | |
| 0.816 | 0.013 | 0.816 | Antiinflammatory | 0.727 0.026 DBMET01736 | ||
| 0.8 | 0.001 | 0.811 | Retinoic acid receptor gamma antagonist | 0.811 0.001 DBMET01736 | DBMET01736 | |
| 0.798 | 0.001 | 0.798 | Retinoic acid beta receptor agonist | 0.794 0.001 DBMET01736 | ||
| 0.797 | 0.001 | 0.805 | Retinoic acid receptor antagonist | 0.805 0.001 DBMET01736 | DBMET01736 | |
| 0.797 | 0.002 | 0.831 | ABCA1 expression enhancer | 0.831 0.002 DBMET01736 | DBMET01736 | |
| 0.788 | 0.014 | 0.789 | Transcription factor NF kappa B inhibitor | 0.789 0.014 DBMET01736 | DBMET01736 | |
| 0.762 | 0.005 | 0.762 | Antioxidant | 0.707 0.005 DBMET01736 | ||
| 0.746 | 0.001 | 0.762 | Retinoic acid alpha receptor antagonist | 0.762 0.001 DBMET01736 | DBMET01736 | |
| 0.69 | 0.001 | 0.693 | Retinoic acid gamma receptor agonist | 0.693 0.001 DBMET01736 | DBMET01736 | |
| 0.699 | 0.013 | 0.699 | 15-Lipoxygenase inhibitor | 0.378 0.084 DBMET01736 | ||
| 0.666 | 0.001 | 0.666 | Retinoic acid alpha receptor agonist | 0.655 0.001 DBMET01736 | ||
| 0.654 | 0.001 | 0.672 | Retinoic acid beta receptor antagonist | 0.672 0.001 DBMET01736 | DBMET01736 | |
| 0.634 | 0.001 | 0.634 | Keratolytic | 0.48 0.002 DBMET01736 | ||
| 0.617 | 0.009 | 0.617 | Nitric oxide antagonist | 0.587 0.01 DBMET01736 | ||
| 0.596 | 0.01 | 0.777 | Caspase 3 stimulant | 0.777 0.004 DBMET01736 | DBMET01736 | |
| 0.59 | 0.014 | 0.59 | Immunosuppressant | 0.503 0.032 DBMET01736 | ||
| 0.569 | 0.001 | 0.569 | Retinoid X alpha receptor agonist | 0.311 0.002 DBMET01736 | ||
| 0.569 | 0.002 | 0.745 | Ornithine decarboxylase inhibitor | 0.745 0.001 DBMET01736 | DBMET01736 | |
| 0.543 | 0.004 | 0.603 | Aldehyde dehydrogenase inhibitor | 0.603 0.004 DBMET01736 | DBMET01736 | |
| 0.532 | 0.001 | 0.537 | Retinoid X beta receptor agonist | 0.537 0.001 DBMET01736 | DBMET01736 | |
| 0.539 | 0.014 | 0.539 | Lipoxygenase inhibitor | 0.337 0.055 DBMET01736 | ||
| 0.511 | 0.001 | 0.523 | Retinoid X gamma receptor agonist | 0.523 0.001 DBMET01736 | DBMET01736 | |
| 0.524 | 0.013 | 0.524 | Hypoglycemic | 0.511 0.014 DBMET01736 | ||
| 0.508 | 0.001 | 0.508 | Retinoid X receptor agonist | 0.302 0.002 DBMET01736 | ||
| 0.519 | 0.014 | 0.529 | Free radical scavenger | 0.529 0.013 DBMET01736 | DBMET01736 | |
| 0.506 | 0.002 | 0.506 | Transcription factor AP-1 inhibitor | 0.495 0.002 DBMET01736 | ||
| 0.493 | 0.005 | 0.493 | Lipid peroxidase inhibitor | 0.309 0.018 DBMET01736 | ||
| 0.475 | 0 | 0.507 | Retinoid X gamma receptor antagonist | 0.507 0 DBMET01736 | DBMET01736 | |
| 0.472 | 0.033 | 0.472 | Immunostimulant | 0.468 0.033 DBMET01736 | ||
| 0.449 | 0.018 | 0.449 | Hypolipemic | 0.302 0.048 DBMET01736 | ||
| 0.466 | 0.051 | 0.503 | Antibacterial | 0.503 0.04 DBMET01736 | DBMET01736 | |
| 0.383 | 0.012 | 0.383 | Interferon gamma antagonist | 0.261 0.026 DBMET01736 | ||
| 0.373 | 0.006 | 0.373 | Phospholipase A2 inhibitor | 0.301 0.013 DBMET01736 | ||
| 0.426 | 0.077 | 0.426 | Cyclophilin D inhibitor | |||
| 0.347 | 0.002 | 0.347 | Adenylate cyclase stimulant | 0.288 0.003 DBMET01736 | ||
| 0.434 | 0.092 | 0.434 | Caspase 9 stimulant | 0.332 0.161 DBMET01736 | ||
| 0.368 | 0.048 | 0.368 | Apoptosis antagonist | 0.327 0.068 DBMET01736 | ||
| 0.317 | 0.001 | 0.317 | Retinoid X beta receptor antagonist | 0.199 0.001 DBMET01736 | ||
| 0.344 | 0.039 | 0.344 | Tumour necrosis factor alpha release inhibitor | 0.162 0.143 DBMET01736 | ||
| 0.298 | 0.001 | 0.298 | Retinoid X receptor antagonist | 0.146 0.002 DBMET01736 | ||
| 0.299 | 0.01 | 0.299 | Antineoplastic antibiotic | 0.265 0.013 DBMET01736 | ||
| 0.274 | 0.001 | 0.274 | Retinoid X alpha receptor antagonist | 0.133 0.001 DBMET01736 | ||
| 0.341 | 0.078 | 0.341 | Vasodilator, peripheral | |||
| 0.278 | 0.036 | 0.278 | Hepatoprotectant | 0.193 0.069 DBMET01736 | ||
| 0.277 | 0.052 | 0.325 | DNA synthesis inhibitor | 0.325 0.036 DBMET01736 | DBMET01736 | |
| 0.22 | 0.017 | 0.22 | Arachidonic acid antagonist | 0.182 0.052 DBMET01736 | ||
| 0.214 | 0.023 | 0.214 | Alkylator | 0.166 0.039 DBMET01736 | ||
| 0.237 | 0.046 | 0.237 | Neurotrophic factor enhancer | 0.176 0.102 DBMET01736 | ||
| 0.255 | 0.068 | 0.255 | Angiogenesis stimulant | |||
| 0.214 | 0.032 | 0.252 | Bone formation stimulant | 0.252 0.024 DBMET01736 | DBMET01736 | |
| 0.267 | 0.086 | 0.267 | Hypoxia-inducible factor 1 alpha inhibitor | 0.252 0.098 DBMET01736 | ||
| 0.302 | 0.122 | 0.302 | Histamine release inhibitor | |||
| 0.205 | 0.025 | 0.621 | Neurotrophic factor | 0.621 0.003 DBMET01736 | DBMET01736 | |
| 0.209 | 0.042 | 0.209 | Succinate dehydrogenase inhibitor | 0.201 0.048 DBMET01736 | ||
| 0.205 | 0.039 | 0.283 | Melanin inhibitor | 0.283 0.024 DBMET01736 | DBMET01736 | |
| 0.177 | 0.016 | 0.177 | Androgen antagonist | 0.134 0.027 DBMET01736 | ||
| 0.204 | 0.045 | 0.204 | Protein-tyrosine phosphatase inhibitor | |||
| 0.25 | 0.091 | 0.25 | Spasmolytic | |||
| 0.184 | 0.027 | 0.184 | Farnesoid X receptor antagonist | 0.144 0.059 DBMET01736 | ||
| 0.19 | 0.045 | 0.19 | Protein kinase stimulant | |||
| 0.177 | 0.036 | 0.177 | Protein-tyrosine phosphatase 1B inhibitor | |||
| 0.168 | 0.03 | 0.168 | Microtubule formation inhibitor | 0.161 0.032 DBMET01736 | ||
| 0.194 | 0.068 | 0.194 | P-glycoprotein inhibitor | |||
| 0.161 | 0.044 | 0.161 | DNA polymerase I inhibitor | 0.096 0.09 DBMET01736 | ||
| 0.151 | 0.039 | 0.151 | Ca2+-transporting ATPase inhibitor | 0.133 0.104 DBMET01736 | ||
| 0.247 | 0.138 | 0.247 | Vasodilator, coronary | |||
| 0.147 | 0.046 | 0.147 | Cholesterol synthesis inhibitor | 0.132 0.055 DBMET01736 | ||
| 0.118 | 0.018 | 0.118 | Thioredoxin reductase inhibitor | 0.116 0.018 DBMET01736 | ||
| 0.118 | 0.021 | 0.118 | ATPase (Vacuolar H+) inhibitor | 0.103 0.036 DBMET01736 | ||
| 0.211 | 0.12 | 0.211 | Transcription factor STAT3 inhibitor | |||
| 0.128 | 0.038 | 0.128 | Electron transport complex I inhibitor | 0.114 0.055 DBMET01736 | ||
| 0.112 | 0.022 | 0.119 | Na+ K+ transporting ATPase inhibitor | 0.119 0.017 DBMET01736 | DBMET01736 | |
| 0.14 | 0.05 | 0.14 | Vanilloid 1 agonist | |||
| 0.134 | 0.048 | 0.134 | Alpha 2b adrenoreceptor antagonist | |||
| 0.107 | 0.024 | 0.107 | Peroxisome proliferator-activated receptor gamma agonist | |||
| 0.163 | 0.081 | 0.163 | Antipruritic | |||
| 0.085 | 0.006 | 0.085 | Factor III inhibitor | 0.06 0.018 DBMET01736 | ||
| 0.19 | 0.115 | 0.19 | RNA-directed DNA polymerase inhibitor | |||
| 0.256 | 0.182 | 0.266 | Transcription factor inhibitor | 0.266 0.176 DBMET01736 | DBMET01736 | |
| 0.135 | 0.065 | 0.135 | Alpha-N-acetylglucosaminidase inhibitor | 0.127 0.071 DBMET01736 | ||
| 0.077 | 0.008 | 0.077 | Pregnane X receptor antagonist | 0.071 0.013 DBMET01736 | ||
| 0.08 | 0.015 | 0.08 | Heme oxygenase stimulant | 0.079 0.016 DBMET01736 | ||
| 0.122 | 0.056 | 0.24 | TRPA1 agonist | 0.24 0.006 DBMET01736 | DBMET01736 | |
| 0.087 | 0.022 | 0.113 | CDC25B inhibitor | 0.113 0.012 DBMET01736 | DBMET01736 | |
| 0.083 | 0.021 | 0.087 | Exportin-1 inhibitor | 0.087 0.017 DBMET01736 | DBMET01736 | |
| 0.092 | 0.032 | 0.092 | CDC25A inhibitor | |||
| 0.155 | 0.097 | 0.155 | Phospholipase C inhibitor | |||
| 0.107 | 0.053 | 0.107 | Anabolic | 0.095 0.07 DBMET01736 | ||
| 0.069 | 0.017 | 0.069 | Glucose-6-phosphate translocase inhibitor | 0.068 0.017 DBMET01736 | ||
| 0.056 | 0.009 | 0.056 | Kainate receptor agonist | 0.048 0.016 DBMET01736 | ||
| 0.149 | 0.102 | 0.196 | ATPase inhibitor | 0.196 0.041 DBMET01736 | DBMET01736 | |
| 0.113 | 0.067 | 0.113 | Photosensitizer | |||
| 0.058 | 0.014 | 0.058 | Liver X receptor alpha agonist | |||
| 0.112 | 0.071 | 0.112 | Estrogen antagonist | |||
| 0.058 | 0.018 | 0.058 | Collagenase inhibitor | 0.049 0.035 DBMET01736 | ||
| 0.046 | 0.009 | 0.046 | HMG CoA reductase inhibitor | 0.036 0.021 DBMET01736 | ||
| 0.179 | 0.143 | 0.2 | Superoxide dismutase inhibitor | 0.2 0.117 DBMET01736 | DBMET01736 | |
| 0.099 | 0.066 | 0.099 | Estrogen receptor beta antagonist | |||
| 0.087 | 0.055 | 0.087 | Transcription factor NF kappa B stimulant | |||
| 0.038 | 0.009 | 0.038 | Prostaglandin EP2 agonist | |||
| 0.105 | 0.077 | 0.105 | Interleukin 2 antagonist | |||
| 0.032 | 0.006 | 0.032 | Vitamin D receptor antagonist | 0.026 0.009 DBMET01736 | ||
| 0.027 | 0.004 | 0.027 | Vitamin D receptor agonist | 0.015 0.014 DBMET01736 | ||
| 0.199 | 0.179 | 0.199 | Antithrombotic | |||
| 0.168 | 0.151 | 0.168 | Peptidyltransferase inhibitor | |||
| 0.053 | 0.039 | 0.053 | Leukotriene B4 antagonist | |||
| 0.037 | 0.026 | 0.037 | 5-Alpha-reductase inhibitor | |||
| 0.033 | 0.023 | 0.033 | Liver X receptor beta agonist | |||
| 0.045 | 0.035 | 0.045 | Microtubule stabilization | |||
| 0.045 | 0.036 | 0.045 | Peroxisome proliferator-activated receptor alpha agonist | |||
| 0.033 | 0.026 | 0.033 | Tubulin agonist | 0.032 0.029 DBMET01736 | ||
| 0.043 | 0.036 | 0.043 | Parathyroid hormone antagonist | |||
| 0.071 | 0.065 | 0.071 | Estrogen receptor alpha antagonist | |||
| 0.029 | 0.024 | 0.029 | Prostaglandin agonist | |||
| 0.065 | 0.062 | 0.065 | Histone deacetylase SIRT1 stimulant | |||
| 0.065 | 0.062 | 0.065 | Histone deacetylase stimulant | |||
| 0.082 | 0.079 | 0.082 | Uric acid excretion stimulant | |||
| 0.042 | 0.039 | 0.042 | Adenylate cyclase 1 inhibitor | |||
| 0.034 | 0.032 | 0.034 | 2,3-Oxidosqualene-lanosterol cyclase inhibitor | |||
| 0.124 | 0.139 | 0.314 | Platelet adhesion inhibitor | 0.314 0.029 DBMET01736 | DBMET01736 | |
| 0.049 | 0.074 | 0.1 | Lipase inhibitor | 0.1 0.027 DBMET01736 | DBMET01736 | |
| 0.025 | 0.108 | 0.059 | Protein 50S ribosomal subunit inhibitor | 0.059 0.032 DBMET01736 | DBMET01736 | |
| 0.078 | 0.162 | 0.129 | Cathepsin H inhibitor | 0.129 0.064 DBMET01736 | DBMET01736 | |
| 0.05 | 0.305 | 0.12 | 3C-Like protease (SARS coronavirus) inhibitor | 0.12 0.019 DBMET01736 | DBMET01736 | |
| 0.02 | 0.961 | 0.172 | Factor V inhibitor | 0.172 0.011 DBMET01736 | DBMET01736 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |