| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.838 | 0.002 | 0.838 | Proteasome inhibitor | 0.24 0.017 DBMET01061 0.24 0.017 DBMET01062 0.459 0.004 DBMET01081 0.337 0.007 DBMET01122 0.246 0.016 DBMET01124 0.252 0.015 DBMET01063 0.22 0.02 DBMET01065 0.219 0.02 DBMET01082 0.219 0.02 DBMET01084 0.22 0.02 DBMET01066 0.207 0.023 DBMET01067 0.219 0.02 DBMET01085 0.219 0.02 DBMET01086 0.227 0.019 DBMET01064 0.209 0.022 DBMET01068 | ||
| 0.592 | 0.002 | 0.592 | Chymotrypsin inhibitor | 0.099 0.037 DBMET01061 0.099 0.037 DBMET01062 0.152 0.017 DBMET01081 0.095 0.04 DBMET01122 0.1 0.036 DBMET01124 0.11 0.03 DBMET01063 0.095 0.04 DBMET01065 0.091 0.043 DBMET01082 0.091 0.043 DBMET01084 0.095 0.04 DBMET01066 0.091 0.043 DBMET01085 0.091 0.043 DBMET01086 0.122 0.025 DBMET01064 | ||
| 0.593 | 0.011 | 0.593 | Caspase 3 stimulant | 0.212 0.152 DBMET01124 0.192 0.182 DBMET01065 0.192 0.182 DBMET01066 | ||
| 0.572 | 0.003 | 0.572 | Kallikrein inhibitor | 0.055 0.026 DBMET01081 0.083 0.014 DBMET01063 0.092 0.012 DBMET01068 | ||
| 0.554 | 0.037 | 0.554 | Transcription factor NF kappa B inhibitor | 0.219 0.151 DBMET01081 0.185 0.184 DBMET01122 0.223 0.148 DBMET01124 0.206 0.163 DBMET01063 0.27 0.113 DBMET01064 0.244 0.132 DBMET01068 | ||
| 0.532 | 0.025 | 0.532 | Antithrombotic | 0.206 0.17 DBMET01081 0.259 0.119 DBMET01124 0.257 0.121 DBMET01063 0.224 0.149 DBMET01082 0.224 0.149 DBMET01084 0.224 0.149 DBMET01085 0.224 0.149 DBMET01086 0.414 0.046 DBMET01064 0.297 0.089 DBMET01068 | ||
| 0.513 | 0.015 | 0.513 | Antiamyloidogenic | 0.187 0.109 DBMET01061 0.187 0.109 DBMET01062 0.43 0.024 DBMET01081 0.191 0.106 DBMET01122 0.186 0.11 DBMET01124 0.341 0.041 DBMET01063 0.284 0.057 DBMET01082 0.284 0.057 DBMET01084 0.284 0.057 DBMET01085 0.284 0.057 DBMET01086 0.307 0.05 DBMET01064 0.213 0.091 DBMET01068 | ||
| 0.483 | 0.011 | 0.483 | Anticoagulant | 0.139 0.09 DBMET01081 0.149 0.081 DBMET01124 0.22 0.046 DBMET01063 0.249 0.039 DBMET01064 0.128 0.103 DBMET01068 | ||
| 0.476 | 0.005 | 0.476 | Cathepsin G inhibitor | 0.07 0.054 DBMET01061 0.07 0.054 DBMET01062 0.127 0.025 DBMET01081 0.08 0.043 DBMET01124 0.109 0.03 DBMET01063 0.147 0.022 DBMET01064 0.071 0.052 DBMET01068 | ||
| 0.533 | 0.075 | 0.533 | Antiinflammatory | |||
| 0.459 | 0.003 | 0.459 | Carbonic anhydrase III inhibitor | 0.087 0.079 DBMET01081 0.126 0.04 DBMET01063 0.125 0.041 DBMET01064 0.097 0.065 DBMET01068 | ||
| 0.431 | 0.003 | 0.431 | Plasminogen activator inhibitor | |||
| 0.419 | 0.004 | 0.419 | Thrombin inhibitor | 0.069 0.057 DBMET01081 0.085 0.037 DBMET01063 | ||
| 0.463 | 0.052 | 0.463 | Antibacterial | 0.343 0.106 DBMET01122 0.266 0.162 DBMET01124 0.228 0.198 DBMET01065 0.33 0.114 DBMET01082 0.33 0.114 DBMET01084 0.228 0.198 DBMET01066 0.438 0.061 DBMET01067 0.33 0.114 DBMET01085 0.33 0.114 DBMET01086 0.442 0.06 DBMET01068 | ||
| 0.37 | 0.005 | 0.37 | Carbonic anhydrase XV inhibitor | 0.11 0.055 DBMET01063 0.092 0.08 DBMET01064 | ||
| 0.329 | 0.016 | 0.422 | Peptidyltransferase inhibitor | 0.164 0.159 DBMET01061 0.164 0.159 DBMET01062 0.197 0.103 DBMET01124 0.173 0.141 DBMET01063 0.177 0.133 DBMET01065 0.183 0.123 DBMET01082 0.183 0.123 DBMET01084 0.177 0.133 DBMET01066 0.367 0.01 DBMET01067 0.183 0.123 DBMET01085 0.183 0.123 DBMET01086 0.192 0.11 DBMET01064 0.422 0.005 DBMET01068 | DBMET01068 | |
| 0.403 | 0.112 | 0.403 | Apoptosis agonist | 0.304 0.169 DBMET01124 | ||
| 0.299 | 0.017 | 0.299 | Bone formation stimulant | 0.141 0.067 DBMET01081 0.162 0.051 DBMET01122 0.12 0.085 DBMET01124 0.11 0.095 DBMET01063 0.106 0.1 DBMET01082 0.106 0.1 DBMET01084 0.106 0.1 DBMET01085 0.106 0.1 DBMET01086 0.194 0.037 DBMET01064 | ||
| 0.269 | 0.009 | 0.277 | Cathepsin L inhibitor | 0.11 0.019 DBMET01061 0.11 0.019 DBMET01062 0.277 0.008 DBMET01081 0.112 0.018 DBMET01122 0.231 0.01 DBMET01124 0.174 0.013 DBMET01063 0.068 0.031 DBMET01065 0.107 0.019 DBMET01082 0.107 0.019 DBMET01084 0.068 0.031 DBMET01066 0.052 0.047 DBMET01067 0.107 0.019 DBMET01085 0.107 0.019 DBMET01086 0.066 0.033 DBMET01064 0.058 0.041 DBMET01068 | DBMET01081 | |
| 0.246 | 0.004 | 0.246 | Leukocyte elastase inhibitor | 0.041 0.032 DBMET01081 | ||
| 0.323 | 0.101 | 0.397 | Immunosuppressant | 0.356 0.084 DBMET01061 0.356 0.084 DBMET01062 0.31 0.109 DBMET01124 0.397 0.064 DBMET01065 0.369 0.077 DBMET01082 0.369 0.077 DBMET01084 0.397 0.064 DBMET01066 0.328 0.099 DBMET01067 0.369 0.077 DBMET01085 0.369 0.077 DBMET01086 | DBMET01066 | |
| 0.223 | 0.002 | 0.223 | Dipeptidyl peptidase IX inhibitor | |||
| 0.206 | 0.013 | 0.214 | Protease inhibitor | 0.189 0.017 DBMET01061 0.189 0.017 DBMET01062 0.203 0.014 DBMET01081 0.156 0.026 DBMET01122 0.157 0.026 DBMET01124 0.168 0.022 DBMET01063 0.17 0.022 DBMET01065 0.214 0.012 DBMET01082 0.214 0.012 DBMET01084 0.17 0.022 DBMET01066 0.14 0.035 DBMET01067 0.214 0.012 DBMET01085 0.214 0.012 DBMET01086 0.144 0.033 DBMET01064 0.114 0.053 DBMET01068 | DBMET01086 | |
| 0.194 | 0.002 | 0.194 | Dipeptidyl peptidase VIII inhibitor | |||
| 0.192 | 0.006 | 0.192 | Plasmin inhibitor | 0.042 0.037 DBMET01081 0.04 0.038 DBMET01063 | ||
| 0.181 | 0.005 | 0.181 | 3C-Like protease (SARS coronavirus) inhibitor | 0.138 0.013 DBMET01061 0.138 0.013 DBMET01062 0.165 0.007 DBMET01081 0.139 0.012 DBMET01122 0.133 0.014 DBMET01124 0.137 0.013 DBMET01063 0.113 0.023 DBMET01065 0.128 0.016 DBMET01082 0.128 0.016 DBMET01084 0.113 0.023 DBMET01066 0.1 0.033 DBMET01067 0.128 0.016 DBMET01085 0.128 0.016 DBMET01086 0.108 0.026 DBMET01064 0.088 0.049 DBMET01068 | ||
| 0.175 | 0.004 | 0.175 | Dipeptidyl peptidase inhibitor | 0.055 0.033 DBMET01081 0.073 0.016 DBMET01063 | ||
| 0.174 | 0.016 | 0.174 | Carbonic anhydrase VI inhibitor | |||
| 0.225 | 0.089 | 0.458 | Calpain inhibitor | 0.296 0.032 DBMET01061 0.296 0.032 DBMET01062 0.458 0.004 DBMET01081 0.311 0.026 DBMET01122 0.336 0.019 DBMET01124 0.361 0.015 DBMET01063 0.213 0.101 DBMET01065 0.269 0.049 DBMET01082 0.269 0.049 DBMET01084 0.213 0.101 DBMET01066 0.246 0.068 DBMET01067 0.269 0.049 DBMET01085 0.269 0.049 DBMET01086 0.306 0.028 DBMET01064 0.289 0.035 DBMET01068 | DBMET01081 | |
| 0.248 | 0.116 | 0.248 | Immunomodulator | 0.209 0.153 DBMET01064 | ||
| 0.133 | 0.002 | 0.133 | HCV NS3/NS4A protease inhibitor | 0.065 0.018 DBMET01061 0.065 0.018 DBMET01062 0.103 0.004 DBMET01081 0.063 0.019 DBMET01122 0.078 0.012 DBMET01124 0.08 0.011 DBMET01063 0.054 0.027 DBMET01065 0.061 0.02 DBMET01082 0.061 0.02 DBMET01084 0.054 0.027 DBMET01066 0.061 0.02 DBMET01085 0.061 0.02 DBMET01086 0.082 0.01 DBMET01064 0.053 0.029 DBMET01068 | ||
| 0.175 | 0.055 | 0.302 | Neurotensin receptor agonist | 0.245 0.022 DBMET01061 0.245 0.022 DBMET01062 0.302 0.014 DBMET01081 0.25 0.021 DBMET01122 0.23 0.025 DBMET01124 0.278 0.017 DBMET01063 0.167 0.066 DBMET01065 0.184 0.046 DBMET01082 0.184 0.046 DBMET01084 0.167 0.066 DBMET01066 0.184 0.046 DBMET01085 0.184 0.046 DBMET01086 0.297 0.015 DBMET01064 0.17 0.063 DBMET01068 | DBMET01081 | |
| 0.118 | 0.011 | 0.126 | Cathepsin B inhibitor | 0.086 0.021 DBMET01061 0.086 0.021 DBMET01062 0.126 0.01 DBMET01081 0.095 0.018 DBMET01122 0.096 0.018 DBMET01124 0.09 0.02 DBMET01063 0.057 0.038 DBMET01065 0.085 0.022 DBMET01082 0.085 0.022 DBMET01084 0.057 0.038 DBMET01066 0.06 0.035 DBMET01067 0.085 0.022 DBMET01085 0.085 0.022 DBMET01086 0.06 0.035 DBMET01064 0.053 0.044 DBMET01068 | DBMET01081 | |
| 0.118 | 0.013 | 0.118 | Aminopeptidase microsomal inhibitor | 0.049 0.048 DBMET01061 0.049 0.048 DBMET01062 0.084 0.023 DBMET01081 0.057 0.042 DBMET01064 | ||
| 0.116 | 0.012 | 0.116 | Trypsin inhibitor | 0.06 0.048 DBMET01063 0.058 0.052 DBMET01064 | ||
| 0.156 | 0.064 | 0.468 | Thiol protease inhibitor | 0.263 0.024 DBMET01061 0.263 0.024 DBMET01062 0.468 0.011 DBMET01081 0.296 0.02 DBMET01122 0.347 0.015 DBMET01124 0.337 0.016 DBMET01063 0.19 0.043 DBMET01065 0.222 0.033 DBMET01082 0.222 0.033 DBMET01084 0.19 0.043 DBMET01066 0.16 0.061 DBMET01067 0.222 0.033 DBMET01085 0.222 0.033 DBMET01086 0.291 0.02 DBMET01064 0.208 0.036 DBMET01068 | DBMET01081 | |
| 0.097 | 0.005 | 0.097 | Dipeptidyl peptidase IV inhibitor | 0.041 0.039 DBMET01063 | ||
| 0.101 | 0.013 | 0.101 | Aminopeptidase N inhibitor | 0.065 0.022 DBMET01081 | ||
| 0.218 | 0.131 | 0.423 | Insulysin inhibitor | 0.333 0.041 DBMET01061 0.333 0.041 DBMET01062 0.408 0.021 DBMET01081 0.346 0.036 DBMET01122 0.336 0.039 DBMET01124 0.423 0.019 DBMET01063 0.245 0.101 DBMET01065 0.311 0.052 DBMET01082 0.311 0.052 DBMET01084 0.245 0.101 DBMET01066 0.311 0.052 DBMET01085 0.311 0.052 DBMET01086 0.398 0.022 DBMET01064 0.306 0.055 DBMET01068 | DBMET01063 | |
| 0.112 | 0.026 | 0.237 | Hematopoietic | 0.105 0.031 DBMET01061 0.105 0.031 DBMET01062 0.119 0.023 DBMET01081 0.109 0.028 DBMET01122 0.114 0.025 DBMET01124 0.166 0.013 DBMET01063 0.108 0.029 DBMET01065 0.108 0.028 DBMET01082 0.108 0.028 DBMET01084 0.108 0.029 DBMET01066 0.09 0.05 DBMET01067 0.108 0.028 DBMET01085 0.108 0.028 DBMET01086 0.237 0.007 DBMET01064 0.117 0.023 DBMET01068 | DBMET01064 | |
| 0.109 | 0.034 | 0.109 | Carbonic anhydrase XIII inhibitor | |||
| 0.101 | 0.027 | 0.101 | Lipase inhibitor | |||
| 0.091 | 0.018 | 0.091 | Carbonic anhydrase VB inhibitor | |||
| 0.086 | 0.014 | 0.086 | Elastase inhibitor | |||
| 0.153 | 0.085 | 0.363 | Growth hormone agonist | 0.206 0.056 DBMET01061 0.206 0.056 DBMET01062 0.28 0.036 DBMET01081 0.174 0.071 DBMET01122 0.212 0.054 DBMET01124 0.363 0.021 DBMET01063 0.178 0.068 DBMET01065 0.196 0.06 DBMET01082 0.196 0.06 DBMET01084 0.178 0.068 DBMET01066 0.196 0.06 DBMET01085 0.196 0.06 DBMET01086 0.251 0.043 DBMET01064 0.201 0.058 DBMET01068 | DBMET01063 | |
| 0.157 | 0.091 | 0.22 | 3C-like protease (Human coronavirus) inhibitor | 0.195 0.055 DBMET01081 0.141 0.117 DBMET01122 0.22 0.041 DBMET01063 | DBMET01063 | |
| 0.07 | 0.005 | 0.07 | Dipeptidyl peptidase II inhibitor | |||
| 0.078 | 0.014 | 0.078 | Factor X inhibitor | |||
| 0.091 | 0.03 | 0.091 | Carbonic anhydrase V inhibitor | |||
| 0.067 | 0.009 | 0.067 | Trypsin I inhibitor | |||
| 0.08 | 0.023 | 0.263 | Human rhinovirus A protease inhibitor | 0.244 0.005 DBMET01061 0.244 0.005 DBMET01062 0.226 0.005 DBMET01081 0.119 0.012 DBMET01122 0.119 0.012 DBMET01124 0.156 0.008 DBMET01063 0.203 0.005 DBMET01065 0.263 0.004 DBMET01082 0.263 0.004 DBMET01084 0.203 0.005 DBMET01066 0.154 0.008 DBMET01067 0.263 0.004 DBMET01085 0.263 0.004 DBMET01086 0.111 0.014 DBMET01064 0.078 0.025 DBMET01068 | DBMET01086 | |
| 0.068 | 0.014 | 0.068 | CXC chemokine 1 receptor antagonist | |||
| 0.073 | 0.022 | 0.088 | Kallikrein 1 inhibitor | 0.06 0.034 DBMET01081 0.053 0.046 DBMET01122 0.057 0.037 DBMET01124 0.08 0.018 DBMET01063 0.056 0.039 DBMET01067 0.088 0.015 DBMET01068 | DBMET01068 | |
| 0.065 | 0.015 | 0.251 | Cathepsin L2 inhibitor | 0.092 0.009 DBMET01061 0.092 0.009 DBMET01062 0.181 0.005 DBMET01081 0.113 0.006 DBMET01122 0.251 0.004 DBMET01124 0.167 0.005 DBMET01063 0.071 0.013 DBMET01065 0.144 0.005 DBMET01082 0.144 0.005 DBMET01084 0.071 0.013 DBMET01066 0.034 0.033 DBMET01067 0.144 0.005 DBMET01085 0.144 0.005 DBMET01086 0.125 0.006 DBMET01064 0.04 0.028 DBMET01068 | DBMET01124 | |
| 0.081 | 0.031 | 0.161 | Neuropeptide agonist | 0.104 0.026 DBMET01061 0.104 0.026 DBMET01062 0.128 0.02 DBMET01081 0.098 0.027 DBMET01122 0.094 0.028 DBMET01124 0.161 0.01 DBMET01063 0.065 0.036 DBMET01065 0.114 0.024 DBMET01082 0.114 0.024 DBMET01084 0.065 0.036 DBMET01066 0.072 0.034 DBMET01067 0.114 0.024 DBMET01085 0.114 0.024 DBMET01086 0.066 0.036 DBMET01064 0.14 0.016 DBMET01068 | DBMET01063 | |
| 0.073 | 0.029 | 0.159 | Bombesin 1 receptor agonist | 0.082 0.024 DBMET01061 0.082 0.024 DBMET01062 0.111 0.015 DBMET01081 0.094 0.02 DBMET01122 0.091 0.02 DBMET01124 0.159 0.007 DBMET01063 0.069 0.033 DBMET01065 0.075 0.028 DBMET01082 0.075 0.028 DBMET01084 0.069 0.033 DBMET01066 0.075 0.028 DBMET01085 0.075 0.028 DBMET01086 0.058 0.043 DBMET01064 0.081 0.025 DBMET01068 | DBMET01063 | |
| 0.105 | 0.065 | 0.228 | Falcipain 3 inhibitor | 0.178 0.025 DBMET01061 0.178 0.025 DBMET01062 0.228 0.011 DBMET01081 0.189 0.021 DBMET01122 0.187 0.022 DBMET01124 0.187 0.022 DBMET01063 0.118 0.055 DBMET01065 0.141 0.041 DBMET01082 0.141 0.041 DBMET01084 0.118 0.055 DBMET01066 0.141 0.041 DBMET01085 0.141 0.041 DBMET01086 0.185 0.022 DBMET01064 | DBMET01081 | |
| 0.048 | 0.015 | 0.059 | Cathepsin F inhibitor | 0.052 0.01 DBMET01061 0.052 0.01 DBMET01062 0.059 0.005 DBMET01081 0.053 0.01 DBMET01122 0.053 0.009 DBMET01124 0.052 0.01 DBMET01063 0.044 0.022 DBMET01065 0.047 0.016 DBMET01082 0.047 0.016 DBMET01084 0.044 0.022 DBMET01066 0.045 0.021 DBMET01067 0.047 0.016 DBMET01085 0.047 0.016 DBMET01086 0.041 0.032 DBMET01064 0.04 0.033 DBMET01068 | DBMET01081 | |
| 0.103 | 0.071 | 0.202 | Nav1.4 sodium channel blocker | 0.127 0.047 DBMET01061 0.127 0.047 DBMET01062 0.146 0.036 DBMET01081 0.127 0.046 DBMET01122 0.118 0.054 DBMET01124 0.202 0.019 DBMET01063 0.109 0.063 DBMET01065 0.124 0.049 DBMET01082 0.124 0.049 DBMET01084 0.109 0.063 DBMET01066 0.112 0.06 DBMET01067 0.124 0.049 DBMET01085 0.124 0.049 DBMET01086 0.13 0.044 DBMET01064 0.18 0.024 DBMET01068 | DBMET01063 | |
| 0.069 | 0.038 | 0.152 | Protease 3C (Human rhinovirus) inhibitor | 0.095 0.018 DBMET01061 0.095 0.018 DBMET01062 0.152 0.006 DBMET01081 0.107 0.013 DBMET01122 0.098 0.016 DBMET01124 0.127 0.009 DBMET01063 0.075 0.031 DBMET01065 0.078 0.029 DBMET01082 0.078 0.029 DBMET01084 0.075 0.031 DBMET01066 0.078 0.029 DBMET01085 0.078 0.029 DBMET01086 0.077 0.03 DBMET01064 | DBMET01081 | |
| 0.076 | 0.046 | 0.17 | Aminopeptidase I inhibitor | 0.124 0.018 DBMET01061 0.124 0.018 DBMET01062 0.151 0.012 DBMET01081 0.092 0.033 DBMET01122 0.094 0.031 DBMET01124 0.154 0.012 DBMET01063 0.071 0.052 DBMET01065 0.131 0.016 DBMET01082 0.131 0.016 DBMET01084 0.071 0.052 DBMET01066 0.075 0.047 DBMET01067 0.131 0.016 DBMET01085 0.131 0.016 DBMET01086 0.17 0.01 DBMET01064 0.113 0.022 DBMET01068 | DBMET01064 | |
| 0.072 | 0.044 | 0.072 | Carbonic anhydrase VA inhibitor | |||
| 0.097 | 0.071 | 0.225 | Folate antagonist | 0.107 0.053 DBMET01061 0.107 0.053 DBMET01062 0.13 0.031 DBMET01081 0.106 0.054 DBMET01122 0.128 0.033 DBMET01124 0.159 0.019 DBMET01063 0.136 0.028 DBMET01065 0.109 0.051 DBMET01082 0.109 0.051 DBMET01084 0.136 0.028 DBMET01066 0.109 0.051 DBMET01085 0.109 0.051 DBMET01086 0.225 0.007 DBMET01064 0.122 0.038 DBMET01068 | DBMET01064 | |
| 0.148 | 0.124 | 0.314 | Angiogenesis stimulant | 0.231 0.079 DBMET01061 0.231 0.079 DBMET01062 0.275 0.059 DBMET01081 0.219 0.085 DBMET01122 0.268 0.062 DBMET01124 0.314 0.044 DBMET01063 0.22 0.084 DBMET01065 0.215 0.087 DBMET01082 0.215 0.087 DBMET01084 0.22 0.084 DBMET01066 0.215 0.087 DBMET01085 0.215 0.087 DBMET01086 0.313 0.044 DBMET01064 0.234 0.077 DBMET01068 | DBMET01063 | |
| 0.061 | 0.039 | 0.103 | Cathepsin E inhibitor | 0.071 0.029 DBMET01061 0.071 0.029 DBMET01062 0.103 0.013 DBMET01081 0.072 0.028 DBMET01122 0.064 0.036 DBMET01124 0.075 0.025 DBMET01063 0.062 0.037 DBMET01065 0.093 0.016 DBMET01082 0.093 0.016 DBMET01084 0.062 0.037 DBMET01066 0.061 0.04 DBMET01067 0.093 0.016 DBMET01085 0.093 0.016 DBMET01086 0.064 0.035 DBMET01064 0.062 0.037 DBMET01068 | DBMET01081 | |
| 0.054 | 0.034 | 0.054 | Autotaxin inhibitor | |||
| 0.036 | 0.018 | 0.045 | HCV polyprotein inhibitor | 0.041 0.011 DBMET01061 0.041 0.011 DBMET01062 0.045 0.008 DBMET01081 0.04 0.012 DBMET01122 0.041 0.011 DBMET01124 0.041 0.011 DBMET01063 0.037 0.017 DBMET01065 0.038 0.015 DBMET01082 0.038 0.015 DBMET01084 0.037 0.017 DBMET01066 0.037 0.017 DBMET01067 0.038 0.015 DBMET01085 0.038 0.015 DBMET01086 0.045 0.007 DBMET01064 0.036 0.018 DBMET01068 | DBMET01064 | |
| 0.05 | 0.032 | 0.162 | Protease activated receptor 1 antagonist | 0.077 0.02 DBMET01061 0.077 0.02 DBMET01062 0.145 0.006 DBMET01081 0.087 0.017 DBMET01122 0.083 0.018 DBMET01124 0.162 0.005 DBMET01063 0.043 0.035 DBMET01065 0.052 0.031 DBMET01082 0.052 0.031 DBMET01084 0.043 0.035 DBMET01066 0.052 0.031 DBMET01085 0.052 0.031 DBMET01086 0.093 0.015 DBMET01068 | DBMET01063 | |
| 0.049 | 0.032 | 0.072 | Bombesin antagonist | 0.053 0.025 DBMET01061 0.053 0.025 DBMET01062 0.068 0.013 DBMET01081 0.053 0.026 DBMET01122 0.055 0.023 DBMET01124 0.072 0.012 DBMET01063 0.043 0.042 DBMET01065 0.05 0.029 DBMET01082 0.05 0.029 DBMET01084 0.043 0.042 DBMET01066 0.05 0.029 DBMET01085 0.05 0.029 DBMET01086 0.047 0.035 DBMET01068 | DBMET01063 | |
| 0.042 | 0.028 | 0.067 | Neurokinin 2 agonist | 0.046 0.023 DBMET01061 0.046 0.023 DBMET01062 0.06 0.013 DBMET01081 0.044 0.025 DBMET01122 0.046 0.023 DBMET01124 0.067 0.009 DBMET01063 0.04 0.031 DBMET01082 0.04 0.031 DBMET01084 0.04 0.031 DBMET01085 0.04 0.031 DBMET01086 0.037 0.035 DBMET01068 | DBMET01063 | |
| 0.034 | 0.021 | 0.047 | Calpain 1 inhibitor | 0.038 0.014 DBMET01061 0.038 0.014 DBMET01062 0.047 0.005 DBMET01081 0.037 0.014 DBMET01122 0.036 0.016 DBMET01124 0.04 0.01 DBMET01063 0.034 0.021 DBMET01082 0.034 0.021 DBMET01084 0.033 0.025 DBMET01067 0.034 0.021 DBMET01085 0.034 0.021 DBMET01086 0.034 0.022 DBMET01064 0.032 0.027 DBMET01068 | DBMET01081 | |
| 0.06 | 0.047 | 0.084 | Caspase 9 inhibitor | 0.072 0.03 DBMET01061 0.072 0.03 DBMET01062 0.083 0.021 DBMET01081 0.068 0.034 DBMET01122 0.062 0.044 DBMET01124 0.066 0.037 DBMET01063 0.058 0.051 DBMET01065 0.084 0.021 DBMET01082 0.084 0.021 DBMET01084 0.058 0.051 DBMET01066 0.059 0.049 DBMET01067 0.084 0.021 DBMET01085 0.084 0.021 DBMET01086 0.077 0.025 DBMET01064 | DBMET01086 | |
| 0.053 | 0.041 | 0.11 | Bombesin 3 receptor antagonist | 0.066 0.027 DBMET01061 0.066 0.027 DBMET01062 0.093 0.014 DBMET01081 0.069 0.025 DBMET01122 0.064 0.029 DBMET01124 0.11 0.009 DBMET01063 0.058 0.035 DBMET01065 0.057 0.036 DBMET01082 0.057 0.036 DBMET01084 0.058 0.035 DBMET01066 0.057 0.036 DBMET01085 0.057 0.036 DBMET01086 0.061 0.032 DBMET01064 0.051 0.045 DBMET01068 | DBMET01063 | |
| 0.031 | 0.02 | 0.06 | Plasmepsin I inhibitor | 0.042 0.012 DBMET01061 0.042 0.012 DBMET01062 0.06 0.005 DBMET01081 0.04 0.013 DBMET01122 0.037 0.014 DBMET01124 0.06 0.005 DBMET01063 0.029 0.022 DBMET01065 0.05 0.008 DBMET01082 0.05 0.008 DBMET01084 0.029 0.022 DBMET01066 0.029 0.023 DBMET01067 0.05 0.008 DBMET01085 0.05 0.008 DBMET01086 0.032 0.019 DBMET01064 0.044 0.01 DBMET01068 | DBMET01063 | |
| 0.059 | 0.049 | 0.126 | Glucagon-like peptide 1 agonist | 0.115 0.015 DBMET01061 0.115 0.015 DBMET01062 0.095 0.025 DBMET01081 0.076 0.037 DBMET01122 0.083 0.033 DBMET01124 0.109 0.017 DBMET01063 0.107 0.018 DBMET01065 0.095 0.024 DBMET01082 0.095 0.024 DBMET01084 0.107 0.018 DBMET01066 0.094 0.025 DBMET01067 0.095 0.024 DBMET01085 0.095 0.024 DBMET01086 0.126 0.013 DBMET01064 0.083 0.033 DBMET01068 | DBMET01064 | |
| 0.051 | 0.041 | 0.051 | Heparanase inhibitor | |||
| 0.059 | 0.052 | 0.171 | Histone deacetylase SIRT3 inhibitor | 0.071 0.026 DBMET01061 0.071 0.026 DBMET01062 0.12 0.007 DBMET01081 0.085 0.015 DBMET01122 0.103 0.009 DBMET01124 0.171 0.004 DBMET01063 0.065 0.035 DBMET01065 0.063 0.042 DBMET01082 0.063 0.042 DBMET01084 0.065 0.035 DBMET01066 0.063 0.042 DBMET01085 0.063 0.042 DBMET01086 0.074 0.023 DBMET01064 0.078 0.019 DBMET01068 | DBMET01063 | |
| 0.053 | 0.046 | 0.1 | Immunoglobulin Fc receptor antagonist | 0.068 0.013 DBMET01061 0.068 0.013 DBMET01062 0.1 0.004 DBMET01081 0.063 0.019 DBMET01122 0.054 0.043 DBMET01124 0.096 0.004 DBMET01063 0.069 0.012 DBMET01082 0.069 0.012 DBMET01084 0.069 0.012 DBMET01085 0.069 0.012 DBMET01086 0.052 0.048 DBMET01064 0.053 0.045 DBMET01068 | DBMET01081 | |
| 0.028 | 0.021 | 0.097 | Thrombin receptor antagonist | 0.041 0.011 DBMET01061 0.041 0.011 DBMET01062 0.097 0.004 DBMET01081 0.054 0.008 DBMET01122 0.07 0.006 DBMET01124 0.096 0.004 DBMET01063 0.026 0.023 DBMET01082 0.026 0.023 DBMET01084 0.026 0.023 DBMET01085 0.026 0.023 DBMET01086 0.031 0.017 DBMET01064 0.054 0.008 DBMET01068 | DBMET01081 | |
| 0.032 | 0.029 | 0.17 | Renin inhibitor | 0.17 0.004 DBMET01061 0.17 0.004 DBMET01062 0.143 0.005 DBMET01081 0.036 0.025 DBMET01122 0.032 0.029 DBMET01124 0.044 0.021 DBMET01063 0.091 0.007 DBMET01065 0.144 0.005 DBMET01082 0.144 0.005 DBMET01084 0.091 0.007 DBMET01066 0.109 0.005 DBMET01067 0.144 0.005 DBMET01085 0.144 0.005 DBMET01086 | DBMET01062 | |
| 0.044 | 0.041 | 0.044 | Carbonic anhydrase XIV inhibitor | |||
| 0.04 | 0.037 | 0.067 | Neurotensin receptor antagonist | 0.049 0.029 DBMET01061 0.049 0.029 DBMET01062 0.067 0.021 DBMET01081 0.053 0.026 DBMET01122 0.045 0.031 DBMET01063 0.051 0.027 DBMET01064 | DBMET01081 | |
| 0.069 | 0.066 | 0.149 | Somatostatin 1 agonist | 0.085 0.046 DBMET01061 0.085 0.046 DBMET01062 0.095 0.038 DBMET01081 0.085 0.046 DBMET01122 0.092 0.039 DBMET01124 0.149 0.014 DBMET01063 0.076 0.056 DBMET01065 0.096 0.037 DBMET01082 0.096 0.037 DBMET01084 0.076 0.056 DBMET01066 0.078 0.053 DBMET01067 0.096 0.037 DBMET01085 0.096 0.037 DBMET01086 0.073 0.06 DBMET01064 0.139 0.017 DBMET01068 | DBMET01063 | |
| 0.046 | 0.044 | 0.138 | Ribonucleoside-diphosphate reductase inhibitor | 0.093 0.021 DBMET01061 0.093 0.021 DBMET01062 0.138 0.013 DBMET01081 0.068 0.03 DBMET01122 0.073 0.028 DBMET01124 0.094 0.02 DBMET01063 0.046 0.044 DBMET01065 0.09 0.022 DBMET01082 0.09 0.022 DBMET01084 0.046 0.044 DBMET01066 0.09 0.022 DBMET01085 0.09 0.022 DBMET01086 0.122 0.016 DBMET01064 0.048 0.042 DBMET01068 | DBMET01081 | |
| 0.08 | 0.079 | 0.108 | Aminoacyl-tRNA synthetase inhibitor | 0.09 0.059 DBMET01063 0.09 0.059 DBMET01064 0.108 0.038 DBMET01068 | DBMET01068 | |
| 0.032 | 0.033 | 0.05 | Bombesin 1 receptor antagonist | 0.036 0.027 DBMET01061 0.036 0.027 DBMET01062 0.045 0.018 DBMET01081 0.037 0.025 DBMET01122 0.04 0.022 DBMET01124 0.05 0.013 DBMET01063 | DBMET01063 | |
| 0.043 | 0.046 | 0.142 | Bombesin 2 receptor antagonist | 0.064 0.022 DBMET01061 0.064 0.022 DBMET01062 0.142 0.01 DBMET01081 0.06 0.024 DBMET01122 0.092 0.015 DBMET01124 0.115 0.013 DBMET01063 0.069 0.02 DBMET01082 0.069 0.02 DBMET01084 0.069 0.02 DBMET01085 0.069 0.02 DBMET01086 0.081 0.017 DBMET01064 0.051 0.032 DBMET01068 | DBMET01081 | |
| 0.044 | 0.047 | 0.132 | Ribonucleotide reductase inhibitor | 0.092 0.023 DBMET01061 0.092 0.023 DBMET01062 0.132 0.015 DBMET01081 0.068 0.032 DBMET01122 0.072 0.03 DBMET01124 0.092 0.023 DBMET01063 0.089 0.023 DBMET01082 0.089 0.023 DBMET01084 0.089 0.023 DBMET01085 0.089 0.023 DBMET01086 0.116 0.017 DBMET01064 0.046 0.045 DBMET01068 | DBMET01081 | |
| 0.01 | 0.013 | 0.014 | 3C-Like protease (MERS coronavirus) inhibitor | 0.012 0.009 DBMET01061 0.012 0.009 DBMET01062 0.014 0.005 DBMET01081 0.011 0.009 DBMET01122 | DBMET01081 | |
| 0.044 | 0.051 | 0.184 | Cathepsin D inhibitor | 0.149 0.008 DBMET01061 0.149 0.008 DBMET01062 0.131 0.01 DBMET01081 0.058 0.035 DBMET01122 0.054 0.038 DBMET01124 0.076 0.026 DBMET01063 0.129 0.01 DBMET01065 0.184 0.005 DBMET01082 0.184 0.005 DBMET01084 0.129 0.01 DBMET01066 0.113 0.014 DBMET01067 0.184 0.005 DBMET01085 0.184 0.005 DBMET01086 0.052 0.04 DBMET01064 | DBMET01086 | |
| 0.015 | 0.024 | 0.029 | Human T-cell leukemia virus type I protease inhibitor | 0.019 0.017 DBMET01061 0.019 0.017 DBMET01062 0.026 0.01 DBMET01081 0.019 0.017 DBMET01122 0.019 0.018 DBMET01124 0.029 0.009 DBMET01063 0.023 0.012 DBMET01082 0.023 0.012 DBMET01084 0.023 0.012 DBMET01085 0.023 0.012 DBMET01086 | DBMET01063 | |
| 0.042 | 0.053 | 0.056 | Prolyl endopeptidase inhibitor | 0.056 0.028 DBMET01081 | DBMET01081 | |
| 0.01 | 0.021 | 0.033 | Protease activated receptor agonist | 0.028 0.008 DBMET01081 0.033 0.007 DBMET01063 | DBMET01063 | |
| 0.052 | 0.064 | 0.078 | Gonadotropin-releasing hormone receptor agonist | 0.059 0.042 DBMET01061 0.059 0.042 DBMET01062 0.073 0.023 DBMET01081 0.058 0.044 DBMET01122 0.062 0.036 DBMET01124 0.078 0.019 DBMET01063 0.055 0.053 DBMET01068 | DBMET01063 | |
| 0.006 | 0.02 | 0.016 | Protease activated receptor 1 agonist | 0.013 0.007 DBMET01081 0.016 0.005 DBMET01063 | DBMET01063 | |
| 0.016 | 0.031 | 0.041 | Aminopeptidase P inhibitor | 0.022 0.017 DBMET01081 0.041 0.005 DBMET01063 0.022 0.017 DBMET01082 0.022 0.017 DBMET01084 0.022 0.017 DBMET01085 0.022 0.017 DBMET01086 0.023 0.016 DBMET01064 0.031 0.009 DBMET01068 | DBMET01063 | |
| 0.071 | 0.087 | 0.182 | Falcipain inhibitor | 0.101 0.054 DBMET01061 0.101 0.054 DBMET01062 0.182 0.019 DBMET01081 0.112 0.048 DBMET01122 0.176 0.021 DBMET01124 0.125 0.042 DBMET01063 | DBMET01081 | |
| 0.029 | 0.046 | 0.152 | Erythropoietin receptor agonist | 0.038 0.031 DBMET01061 0.038 0.031 DBMET01062 0.043 0.026 DBMET01081 0.035 0.034 DBMET01124 0.067 0.015 DBMET01063 0.152 0.008 DBMET01064 0.045 0.024 DBMET01068 | DBMET01064 | |
| 0.014 | 0.031 | 0.023 | Tryptophan hydroxylase 1 inhibitor | 0.023 0.005 DBMET01064 | DBMET01064 | |
| 0.023 | 0.04 | 0.055 | Calcitonin receptor agonist | 0.034 0.023 DBMET01061 0.034 0.023 DBMET01062 0.055 0.016 DBMET01081 0.029 0.028 DBMET01122 0.03 0.027 DBMET01124 0.053 0.016 DBMET01063 0.038 0.021 DBMET01082 0.038 0.021 DBMET01084 0.038 0.021 DBMET01085 0.038 0.021 DBMET01086 0.05 0.017 DBMET01064 0.035 0.023 DBMET01068 | DBMET01081 | |
| 0.01 | 0.027 | 0.018 | KiSS-1 receptor antagonist | 0.018 0.011 DBMET01063 | DBMET01063 | |
| 0.028 | 0.046 | 0.062 | Cholecystokinin B agonist | 0.043 0.021 DBMET01081 0.034 0.031 DBMET01124 0.062 0.011 DBMET01063 0.035 0.03 DBMET01064 0.034 0.032 DBMET01068 | DBMET01063 | |
| 0.033 | 0.051 | 0.127 | Plasmepsin II inhibitor | 0.094 0.005 DBMET01061 0.094 0.005 DBMET01062 0.127 0.004 DBMET01081 0.054 0.015 DBMET01122 0.058 0.013 DBMET01124 0.101 0.004 DBMET01063 0.064 0.01 DBMET01065 0.112 0.004 DBMET01082 0.112 0.004 DBMET01084 0.064 0.01 DBMET01066 0.047 0.02 DBMET01067 0.112 0.004 DBMET01085 0.112 0.004 DBMET01086 0.049 0.019 DBMET01064 0.053 0.016 DBMET01068 | DBMET01081 | |
| 0.03 | 0.049 | 0.128 | Endothelin-converting enzyme inhibitor | 0.045 0.034 DBMET01061 0.045 0.034 DBMET01062 0.088 0.016 DBMET01081 0.046 0.034 DBMET01063 0.05 0.03 DBMET01082 0.05 0.03 DBMET01084 0.05 0.03 DBMET01085 0.05 0.03 DBMET01086 0.128 0.011 DBMET01064 | DBMET01064 | |
| 0.032 | 0.051 | 0.068 | HIV-1 protease inhibitor | 0.053 0.018 DBMET01061 0.053 0.018 DBMET01062 0.068 0.008 DBMET01081 0.042 0.031 DBMET01122 0.039 0.037 DBMET01124 0.049 0.023 DBMET01063 0.049 0.022 DBMET01065 0.066 0.009 DBMET01082 0.066 0.009 DBMET01084 0.049 0.022 DBMET01066 0.045 0.027 DBMET01067 0.066 0.009 DBMET01085 0.066 0.009 DBMET01086 0.045 0.027 DBMET01064 0.041 0.033 DBMET01068 | DBMET01081 | |
| 0.133 | 0.153 | 0.24 | Catenin beta inhibitor | 0.179 0.053 DBMET01061 0.179 0.053 DBMET01062 0.197 0.035 DBMET01081 0.201 0.031 DBMET01122 0.195 0.036 DBMET01124 0.24 0.013 DBMET01063 0.184 0.047 DBMET01065 0.178 0.055 DBMET01082 0.178 0.055 DBMET01084 0.184 0.047 DBMET01066 0.178 0.055 DBMET01085 0.178 0.055 DBMET01086 0.209 0.026 DBMET01064 | DBMET01063 | |
| 0.068 | 0.088 | 0.177 | Falcipain 2 inhibitor | 0.097 0.054 DBMET01061 0.097 0.054 DBMET01062 0.177 0.019 DBMET01081 0.108 0.048 DBMET01122 0.172 0.021 DBMET01124 0.121 0.042 DBMET01063 | DBMET01081 | |
| 0.053 | 0.076 | 0.105 | Elastase 1 inhibitor | 0.071 0.045 DBMET01061 0.071 0.045 DBMET01062 0.093 0.024 DBMET01081 0.089 0.028 DBMET01122 0.064 0.055 DBMET01124 0.074 0.042 DBMET01063 0.066 0.052 DBMET01065 0.088 0.029 DBMET01082 0.088 0.029 DBMET01084 0.066 0.052 DBMET01066 0.088 0.029 DBMET01085 0.088 0.029 DBMET01086 0.105 0.018 DBMET01064 | DBMET01064 | |
| 0.011 | 0.034 | 0.025 | Angiotensin-converting enzyme 2 inhibitor | 0.025 0.005 DBMET01064 | DBMET01064 | |
| 0.019 | 0.043 | 0.039 | Cathepsin K inhibitor | 0.039 0.01 DBMET01081 0.025 0.022 DBMET01122 0.027 0.018 DBMET01082 0.027 0.018 DBMET01084 0.027 0.018 DBMET01085 0.027 0.018 DBMET01086 | DBMET01081 | |
| 0.019 | 0.045 | 0.076 | Plasma kallikrein inhibitor | 0.041 0.017 DBMET01081 0.031 0.026 DBMET01124 0.063 0.008 DBMET01063 0.03 0.027 DBMET01067 0.076 0.006 DBMET01068 | DBMET01068 | |
| 0.038 | 0.064 | 0.064 | Collagenase inhibitor | 0.046 0.042 DBMET01061 0.046 0.042 DBMET01062 0.064 0.013 DBMET01081 | DBMET01081 | |
| 0.025 | 0.051 | 0.178 | Cathepsin L1 inhibitor | 0.051 0.019 DBMET01061 0.051 0.019 DBMET01062 0.178 0.006 DBMET01081 0.077 0.012 DBMET01122 0.159 0.006 DBMET01124 0.132 0.007 DBMET01063 0.045 0.023 DBMET01082 0.045 0.023 DBMET01084 0.045 0.023 DBMET01085 0.045 0.023 DBMET01086 | DBMET01081 | |
| 0.026 | 0.052 | 0.038 | Growth factor receptor-bound protein 2 antagonist | 0.032 0.031 DBMET01081 0.038 0.017 DBMET01063 | DBMET01063 | |
| 0.011 | 0.039 | 0.028 | Growth hormone releasing factor antagonist | 0.028 0.014 DBMET01063 | DBMET01063 | |
| 0.01 | 0.04 | 0.021 | Neurokinin 1 agonist | 0.021 0.014 DBMET01081 0.021 0.014 DBMET01063 | DBMET01063 | |
| 0.018 | 0.049 | 0.084 | Dipeptidyl peptidase I inhibitor | 0.041 0.012 DBMET01081 0.038 0.014 DBMET01122 0.037 0.015 DBMET01124 0.084 0.005 DBMET01063 0.035 0.016 DBMET01064 | DBMET01063 | |
| 0.009 | 0.042 | 0.15 | Integrin beta7 antagonist | 0.018 0.015 DBMET01081 0.038 0.008 DBMET01063 0.019 0.014 DBMET01067 0.15 0.003 DBMET01064 0.069 0.005 DBMET01068 | DBMET01064 | |
| 0.023 | 0.06 | 0.053 | GHS receptor antagonist | 0.051 0.007 DBMET01081 0.031 0.025 DBMET01122 0.031 0.026 DBMET01124 0.053 0.006 DBMET01063 | DBMET01063 | |
| 0.026 | 0.063 | 0.058 | Growth hormone release inhibitor | 0.037 0.036 DBMET01081 0.058 0.017 DBMET01063 0.046 0.025 DBMET01068 | DBMET01063 | |
| 0.007 | 0.046 | 0.26 | Integrin alpha4beta7 antagonist | 0.021 0.014 DBMET01081 0.033 0.008 DBMET01063 0.26 0.003 DBMET01064 | DBMET01064 | |
| 0.004 | 0.043 | 0.048 | Melanocortin 5 agonist | 0.048 0.012 DBMET01063 | DBMET01063 | |
| 0.042 | 0.081 | 0.075 | Angiotensin-converting enzyme inhibitor | 0.058 0.033 DBMET01081 0.075 0.016 DBMET01064 | DBMET01064 | |
| 0.019 | 0.059 | 0.076 | Complement C3a chemotactic receptor antagonist | 0.041 0.032 DBMET01081 0.046 0.029 DBMET01063 0.076 0.015 DBMET01064 | DBMET01064 | |
| 0.005 | 0.044 | 0.05 | Melanocortin 3 agonist | 0.05 0.012 DBMET01063 | DBMET01063 | |
| 0.026 | 0.067 | 0.073 | Tryptophan 5 hydroxylase inhibitor | 0.04 0.015 DBMET01063 0.073 0.003 DBMET01064 0.036 0.023 DBMET01068 | DBMET01064 | |
| 0.083 | 0.125 | 0.117 | Factor V inhibitor | 0.094 0.085 DBMET01061 0.094 0.085 DBMET01062 0.109 0.052 DBMET01081 0.117 0.042 DBMET01124 0.108 0.054 DBMET01063 0.112 0.047 DBMET01065 0.095 0.083 DBMET01082 0.095 0.083 DBMET01084 0.112 0.047 DBMET01066 0.095 0.083 DBMET01085 0.095 0.083 DBMET01086 0.095 0.083 DBMET01064 | DBMET01124 | |
| 0.005 | 0.047 | 0.054 | Melanocortin 1 agonist | 0.054 0.013 DBMET01063 | DBMET01063 | |
| 0.063 | 0.106 | 0.208 | Aminopeptidase B inhibitor | 0.148 0.039 DBMET01061 0.148 0.039 DBMET01062 0.193 0.023 DBMET01081 0.086 0.076 DBMET01122 0.084 0.078 DBMET01124 0.129 0.048 DBMET01063 0.143 0.041 DBMET01082 0.143 0.041 DBMET01084 0.143 0.041 DBMET01085 0.143 0.041 DBMET01086 0.208 0.019 DBMET01064 | DBMET01064 | |
| 0.007 | 0.051 | 0.044 | Neutral endopeptidase inhibitor | 0.023 0.014 DBMET01081 0.044 0.008 DBMET01064 | DBMET01064 | |
| 0.004 | 0.051 | 0.015 | Glucagon agonist | 0.015 0.01 DBMET01064 | DBMET01064 | |
| 0.039 | 0.086 | 0.168 | Carbonic anhydrase stimulant | 0.07 0.032 DBMET01061 0.07 0.032 DBMET01062 0.12 0.014 DBMET01081 0.059 0.042 DBMET01122 0.076 0.028 DBMET01124 0.111 0.016 DBMET01063 0.052 0.051 DBMET01065 0.054 0.047 DBMET01082 0.054 0.047 DBMET01084 0.052 0.051 DBMET01066 0.06 0.04 DBMET01067 0.054 0.047 DBMET01085 0.054 0.047 DBMET01086 0.168 0.009 DBMET01064 0.104 0.018 DBMET01068 | DBMET01064 | |
| 0.02 | 0.068 | 0.081 | Melanocortin 1 antagonist | 0.064 0.016 DBMET01081 0.036 0.029 DBMET01122 0.053 0.019 DBMET01124 0.081 0.013 DBMET01063 0.034 0.03 DBMET01068 | DBMET01063 | |
| 0.019 | 0.068 | 0.029 | Baculoviral IAP repeat-containing protein 4 inhibitor | 0.028 0.017 DBMET01081 0.029 0.016 DBMET01063 0.027 0.019 DBMET01064 | DBMET01063 | |
| 0.02 | 0.07 | 0.08 | Carbonic anhydrase I stimulant | 0.044 0.02 DBMET01081 0.033 0.032 DBMET01124 0.036 0.028 DBMET01063 0.08 0.007 DBMET01064 | DBMET01064 | |
| 0.02 | 0.072 | 0.06 | Melanocortin 4 antagonist | 0.046 0.026 DBMET01081 0.06 0.019 DBMET01063 | DBMET01063 | |
| 0.005 | 0.059 | 0.037 | Melanocortin 3 antagonist | 0.037 0.017 DBMET01063 | DBMET01063 | |
| 0.012 | 0.066 | 0.028 | Bombesin agonist | 0.022 0.015 DBMET01081 0.028 0.009 DBMET01063 | DBMET01063 | |
| 0.007 | 0.062 | 0.021 | Cathepsin S inhibitor | 0.021 0.012 DBMET01081 0.018 0.014 DBMET01082 0.018 0.014 DBMET01084 0.018 0.014 DBMET01085 0.018 0.014 DBMET01086 | DBMET01081 | |
| 0.086 | 0.141 | 0.204 | Cathepsin H inhibitor | 0.144 0.05 DBMET01061 0.144 0.05 DBMET01062 0.192 0.025 DBMET01081 0.171 0.033 DBMET01122 0.134 0.059 DBMET01124 0.204 0.021 DBMET01063 0.169 0.034 DBMET01082 0.169 0.034 DBMET01084 0.169 0.034 DBMET01085 0.169 0.034 DBMET01086 0.167 0.035 DBMET01064 0.107 0.095 DBMET01068 | DBMET01063 | |
| 0.026 | 0.083 | 0.098 | Metalloproteinase-3 inhibitor | 0.048 0.035 DBMET01061 0.048 0.035 DBMET01062 0.098 0.011 DBMET01081 0.051 0.032 DBMET01122 0.051 0.031 DBMET01063 0.045 0.039 DBMET01082 0.045 0.039 DBMET01084 0.045 0.039 DBMET01085 0.045 0.039 DBMET01086 0.069 0.019 DBMET01064 | DBMET01081 | |
| 0.025 | 0.082 | 0.063 | Melanocortin antagonist | 0.051 0.028 DBMET01081 0.063 0.019 DBMET01063 | DBMET01063 | |
| 0.033 | 0.091 | 0.048 | Baculoviral IAP repeat-containing protein inhibitor | 0.048 0.025 DBMET01081 0.044 0.038 DBMET01063 | DBMET01081 | |
| 0.006 | 0.064 | 0.019 | Carbonic anhydrase IV stimulant | 0.019 0.007 DBMET01064 | DBMET01064 | |
| 0.007 | 0.066 | 0.045 | Melanocortin agonist | 0.045 0.014 DBMET01063 | DBMET01063 | |
| 0.035 | 0.096 | 0.073 | Carbonic anhydrase II stimulant | 0.055 0.03 DBMET01081 0.048 0.044 DBMET01063 0.073 0.012 DBMET01064 | DBMET01064 | |
| 0.006 | 0.067 | 0.016 | Aminopeptidase A inhibitor | 0.016 0.015 DBMET01064 | DBMET01064 | |
| 0.009 | 0.07 | 0.063 | Somatostatin 2 antagonist | 0.063 0.011 DBMET01063 0.048 0.016 DBMET01068 | DBMET01063 | |
| 0.011 | 0.074 | 0.034 | Somatostatin 4 antagonist | 0.034 0.01 DBMET01063 0.028 0.013 DBMET01068 | DBMET01063 | |
| 0.029 | 0.093 | 0.063 | Integrin alpha1beta1 antagonist | 0.042 0.016 DBMET01081 0.063 0.004 DBMET01064 | DBMET01064 | |
| 0.006 | 0.07 | 0.283 | VLA-4 antagonist | 0.043 0.014 DBMET01063 0.283 0.003 DBMET01064 | DBMET01064 | |
| 0.006 | 0.071 | 0.034 | Melanocortin 4 agonist | 0.034 0.014 DBMET01063 | DBMET01063 | |
| 0.009 | 0.075 | 0.02 | Bombesin 3 receptor agonist | 0.02 0.012 DBMET01063 | DBMET01063 | |
| 0.01 | 0.076 | 0.106 | Integrin alphaVbeta1 antagonist | 0.018 0.016 DBMET01063 0.106 0.004 DBMET01064 | DBMET01064 | |
| 0.022 | 0.089 | 0.109 | Integrin alpha5beta1 antagonist | 0.049 0.018 DBMET01063 0.109 0.005 DBMET01064 | DBMET01064 | |
| 0.033 | 0.102 | 0.129 | Protease activated receptor antagonist | 0.057 0.052 DBMET01061 0.057 0.052 DBMET01062 0.108 0.012 DBMET01081 0.064 0.041 DBMET01122 0.065 0.041 DBMET01124 0.129 0.007 DBMET01063 0.07 0.034 DBMET01068 | DBMET01063 | |
| 0.015 | 0.084 | 0.044 | Peptide deformylase inhibitor | 0.044 0.013 DBMET01081 | DBMET01081 | |
| 0.017 | 0.087 | 0.069 | Somatostatin 1 antagonist | 0.069 0.012 DBMET01063 0.061 0.015 DBMET01068 | DBMET01063 | |
| 0.005 | 0.076 | 0.405 | Integrin alpha4 antagonist | 0.027 0.017 DBMET01081 0.032 0.015 DBMET01063 0.405 0.003 DBMET01064 | DBMET01064 | |
| 0.032 | 0.104 | 0.075 | Factor IXa inhibitor | 0.058 0.028 DBMET01064 0.075 0.018 DBMET01068 | DBMET01068 | |
| 0.009 | 0.081 | 0.043 | Geranylgeranyltransferase I inhibitor | 0.043 0.005 DBMET01124 0.022 0.014 DBMET01064 | DBMET01124 | |
| 0.011 | 0.084 | 0.022 | Caspase 8 inhibitor | 0.022 0.01 DBMET01081 0.022 0.01 DBMET01064 | DBMET01064 | |
| 0.038 | 0.111 | 0.171 | Catalase inhibitor | 0.065 0.059 DBMET01081 0.069 0.055 DBMET01063 0.171 0.021 DBMET01064 0.098 0.039 DBMET01068 | DBMET01064 | |
| 0.003 | 0.076 | 0.007 | Phosphoribosylglycinamide formyltransferase inhibitor | 0.007 0.005 DBMET01064 | DBMET01064 | |
| 0.018 | 0.097 | 0.054 | Oxytocin agonist | 0.053 0.022 DBMET01081 0.054 0.021 DBMET01063 | DBMET01063 | |
| 0.156 | 0.236 | 0.628 | Calpain 2 inhibitor | 0.338 0.093 DBMET01061 0.338 0.093 DBMET01062 0.628 0.005 DBMET01081 0.414 0.054 DBMET01122 0.482 0.029 DBMET01124 0.419 0.051 DBMET01063 0.209 0.179 DBMET01082 0.209 0.179 DBMET01084 0.281 0.127 DBMET01067 0.209 0.179 DBMET01085 0.209 0.179 DBMET01086 0.378 0.073 DBMET01064 0.333 0.095 DBMET01068 | DBMET01081 | |
| 0.016 | 0.097 | 0.029 | Motilin receptor antagonist | 0.029 0.016 DBMET01063 | DBMET01063 | |
| 0.019 | 0.105 | 0.103 | Antimetabolite | 0.056 0.028 DBMET01124 0.043 0.037 DBMET01063 0.103 0.016 DBMET01064 | DBMET01064 | |
| 0.038 | 0.131 | 0.076 | Sirtuin 1 inhibitor | 0.068 0.048 DBMET01081 0.076 0.039 DBMET01124 0.075 0.04 DBMET01063 0.062 0.056 DBMET01064 | DBMET01124 | |
| 0.027 | 0.121 | 0.205 | VCAM antagonist | 0.039 0.027 DBMET01124 0.043 0.017 DBMET01063 0.205 0.004 DBMET01064 | DBMET01064 | |
| 0.027 | 0.121 | 0.204 | VCAM-1 antagonist | 0.039 0.027 DBMET01124 0.044 0.017 DBMET01063 0.204 0.004 DBMET01064 | DBMET01064 | |
| 0.01 | 0.107 | 0.069 | Growth hormone releasing factor agonist | 0.067 0.008 DBMET01061 0.067 0.008 DBMET01062 0.055 0.011 DBMET01063 0.069 0.007 DBMET01065 0.068 0.007 DBMET01082 0.068 0.007 DBMET01084 0.069 0.007 DBMET01066 0.068 0.007 DBMET01085 0.068 0.007 DBMET01086 | DBMET01066 | |
| 0.108 | 0.205 | 0.368 | Immunostimulant | 0.308 0.076 DBMET01061 0.308 0.076 DBMET01062 0.318 0.074 DBMET01081 0.199 0.121 DBMET01124 0.221 0.109 DBMET01063 0.34 0.067 DBMET01065 0.368 0.059 DBMET01082 0.368 0.059 DBMET01084 0.34 0.067 DBMET01066 0.309 0.076 DBMET01067 0.368 0.059 DBMET01085 0.368 0.059 DBMET01086 0.248 0.097 DBMET01064 0.259 0.093 DBMET01068 | DBMET01086 | |
| 0.052 | 0.152 | 0.102 | Vanilloid 4 agonist | 0.07 0.065 DBMET01061 0.07 0.065 DBMET01062 0.102 0.015 DBMET01081 0.07 0.066 DBMET01122 0.069 0.066 DBMET01124 | DBMET01081 | |
| 0.026 | 0.127 | 0.103 | Farnesyltransferase inhibitor | 0.056 0.022 DBMET01081 0.103 0.007 DBMET01124 0.069 0.016 DBMET01063 0.074 0.014 DBMET01064 | DBMET01124 | |
| 0.006 | 0.108 | 0.026 | Cholecystokinin agonist | 0.026 0.01 DBMET01063 | DBMET01063 | |
| 0.167 | 0.269 | 0.292 | Ca(v)3.3 blocker | 0.249 0.102 DBMET01081 0.218 0.155 DBMET01122 0.243 0.111 DBMET01124 0.292 0.05 DBMET01063 0.223 0.147 DBMET01064 | DBMET01063 | |
| 0.018 | 0.12 | 0.041 | Carboxypeptidase B inhibitor | 0.03 0.029 DBMET01081 0.032 0.025 DBMET01063 0.041 0.012 DBMET01064 | DBMET01064 | |
| 0.162 | 0.266 | 0.343 | Interleukin 2 agonist | 0.225 0.149 DBMET01061 0.225 0.149 DBMET01062 0.222 0.154 DBMET01081 0.211 0.171 DBMET01122 0.247 0.121 DBMET01082 0.247 0.121 DBMET01084 0.235 0.136 DBMET01067 0.247 0.121 DBMET01085 0.247 0.121 DBMET01086 0.343 0.049 DBMET01064 0.241 0.129 DBMET01068 | DBMET01064 | |
| 0.042 | 0.146 | 0.178 | Secretase beta inhibitor | 0.117 0.011 DBMET01061 0.117 0.011 DBMET01062 0.176 0.004 DBMET01081 0.095 0.021 DBMET01122 0.178 0.004 DBMET01124 0.164 0.005 DBMET01063 0.095 0.021 DBMET01065 0.172 0.004 DBMET01082 0.172 0.004 DBMET01084 0.095 0.021 DBMET01066 0.083 0.033 DBMET01067 0.172 0.004 DBMET01085 0.172 0.004 DBMET01086 0.146 0.005 DBMET01064 0.12 0.01 DBMET01068 | DBMET01124 | |
| 0.005 | 0.109 | 0.053 | Growth hormone release promoting | 0.048 0.006 DBMET01061 0.048 0.006 DBMET01062 0.031 0.01 DBMET01063 0.053 0.005 DBMET01065 0.05 0.005 DBMET01082 0.05 0.005 DBMET01084 0.053 0.005 DBMET01066 0.05 0.005 DBMET01085 0.05 0.005 DBMET01086 | DBMET01066 | |
| 0.023 | 0.127 | 0.063 | GHS receptor agonist | 0.063 0.012 DBMET01063 | DBMET01063 | |
| 0.022 | 0.13 | 0.118 | Opioid delta receptor antagonist | 0.06 0.046 DBMET01081 0.064 0.043 DBMET01124 0.118 0.026 DBMET01063 | DBMET01063 | |
| 0.075 | 0.185 | 0.237 | Histone deacetylase SIRT1 inhibitor | 0.113 0.1 DBMET01061 0.113 0.1 DBMET01062 0.167 0.048 DBMET01081 0.113 0.1 DBMET01122 0.172 0.045 DBMET01124 0.237 0.02 DBMET01063 0.141 0.069 DBMET01064 0.156 0.057 DBMET01068 | DBMET01063 | |
| 0.007 | 0.119 | 0.022 | Somatostatin 3 antagonist | 0.022 0.012 DBMET01063 | DBMET01063 | |
| 0.006 | 0.12 | 0.096 | Cholecystokinin A antagonist | 0.043 0.022 DBMET01081 0.046 0.021 DBMET01124 0.096 0.009 DBMET01063 | DBMET01063 | |
| 0.198 | 0.311 | 0.532 | 5 Hydroxytryptamine release inhibitor | 0.344 0.121 DBMET01061 0.344 0.121 DBMET01062 0.415 0.069 DBMET01081 0.294 0.172 DBMET01122 0.258 0.217 DBMET01124 0.437 0.058 DBMET01063 0.255 0.221 DBMET01065 0.347 0.118 DBMET01082 0.347 0.118 DBMET01084 0.255 0.221 DBMET01066 0.304 0.161 DBMET01067 0.347 0.118 DBMET01085 0.347 0.118 DBMET01086 0.532 0.023 DBMET01064 0.426 0.063 DBMET01068 | DBMET01064 | |
| 0.06 | 0.174 | 0.124 | Vanilloid agonist | 0.124 0.017 DBMET01122 | DBMET01122 | |
| 0.023 | 0.138 | 0.066 | Histamine H1 receptor agonist | 0.056 0.012 DBMET01081 0.04 0.039 DBMET01122 0.044 0.031 DBMET01124 0.066 0.006 DBMET01063 0.042 0.036 DBMET01064 | DBMET01063 | |
| 0.058 | 0.174 | 0.203 | Interleukin 1 beta converting enzyme inhibitor | 0.125 0.031 DBMET01061 0.125 0.031 DBMET01062 0.203 0.005 DBMET01081 0.127 0.03 DBMET01122 0.115 0.04 DBMET01124 0.122 0.034 DBMET01063 0.111 0.044 DBMET01082 0.111 0.044 DBMET01084 0.111 0.044 DBMET01085 0.111 0.044 DBMET01086 0.182 0.009 DBMET01064 | DBMET01081 | |
| 0.09 | 0.208 | 0.513 | Interleukin antagonist | 0.19 0.09 DBMET01061 0.19 0.09 DBMET01062 0.349 0.039 DBMET01081 0.216 0.076 DBMET01122 0.378 0.034 DBMET01124 0.513 0.019 DBMET01063 0.191 0.089 DBMET01065 0.225 0.072 DBMET01082 0.225 0.072 DBMET01084 0.191 0.089 DBMET01066 0.225 0.072 DBMET01085 0.225 0.072 DBMET01086 0.255 0.06 DBMET01064 0.357 0.038 DBMET01068 | DBMET01063 | |
| 0.065 | 0.187 | 0.335 | Thrombolytic | 0.149 0.082 DBMET01061 0.149 0.082 DBMET01062 0.208 0.048 DBMET01081 0.142 0.088 DBMET01122 0.214 0.045 DBMET01124 0.179 0.062 DBMET01063 0.122 0.108 DBMET01065 0.142 0.088 DBMET01082 0.142 0.088 DBMET01084 0.122 0.108 DBMET01066 0.142 0.088 DBMET01085 0.142 0.088 DBMET01086 0.335 0.019 DBMET01064 0.125 0.104 DBMET01068 | DBMET01064 | |
| 0.05 | 0.184 | 0.103 | Factor XII inhibitor | 0.079 0.068 DBMET01081 0.095 0.043 DBMET01063 0.103 0.034 DBMET01064 | DBMET01064 | |
| 0.011 | 0.146 | 0.021 | Follicle-stimulating hormone antagonist | 0.021 0.011 DBMET01063 0.02 0.011 DBMET01064 | DBMET01063 | |
| 0.016 | 0.151 | 0.058 | Opioid agonist | 0.058 0.031 DBMET01063 | DBMET01063 | |
| 0.01 | 0.146 | 0.543 | Integrin antagonist | 0.042 0.03 DBMET01081 0.051 0.027 DBMET01063 0.543 0.004 DBMET01064 | DBMET01064 | |
| 0.006 | 0.141 | 0.016 | Cholecystokinin A agonist | 0.016 0.011 DBMET01063 | DBMET01063 | |
| 0.054 | 0.195 | 0.243 | Histone deacetylase class III inhibitor | 0.101 0.089 DBMET01061 0.101 0.089 DBMET01062 0.171 0.03 DBMET01081 0.159 0.038 DBMET01124 0.243 0.01 DBMET01063 0.152 0.042 DBMET01064 0.143 0.049 DBMET01068 | DBMET01063 | |
| 0.013 | 0.155 | 0.054 | Growth hormone secretagogue receptor antagonist | 0.041 0.021 DBMET01081 0.054 0.016 DBMET01063 | DBMET01063 | |
| 0.015 | 0.161 | 0.05 | Somatostatin 5 agonist | 0.05 0.012 DBMET01063 0.037 0.022 DBMET01068 | DBMET01063 | |
| 0.021 | 0.17 | 0.069 | Selectin antagonist | 0.069 0.043 DBMET01063 0.068 0.044 DBMET01064 0.056 0.053 DBMET01068 | DBMET01063 | |
| 0.014 | 0.163 | 0.039 | Macrophage elastase inhibitor | 0.039 0.035 DBMET01081 | DBMET01081 | |
| 0.01 | 0.16 | 0.037 | Opioid delta receptor agonist | 0.037 0.022 DBMET01063 | DBMET01063 | |
| 0.005 | 0.155 | 0.038 | Cholecystokinin B antagonist | 0.028 0.024 DBMET01081 0.038 0.015 DBMET01063 | DBMET01063 | |
| 0.006 | 0.162 | 0.075 | Cholecystokinin antagonist | 0.053 0.023 DBMET01081 0.04 0.03 DBMET01124 0.075 0.013 DBMET01063 0.04 0.029 DBMET01065 0.04 0.029 DBMET01066 | DBMET01063 | |
| 0.013 | 0.169 | 0.082 | Matrix metalloproteinase 1 inhibitor | 0.082 0.02 DBMET01081 0.046 0.041 DBMET01063 | DBMET01081 | |
| 0.008 | 0.167 | 0.064 | Geranylgeranyltransferase inhibitor | 0.024 0.013 DBMET01081 0.064 0.004 DBMET01124 0.03 0.009 DBMET01063 0.038 0.006 DBMET01064 | DBMET01124 | |
| 0.009 | 0.17 | 0.049 | Gonadotropin-releasing hormone receptor antagonist | 0.049 0.017 DBMET01063 | DBMET01063 | |
| 0.015 | 0.18 | 0.08 | Histamine H2 receptor agonist | 0.058 0.016 DBMET01081 0.042 0.03 DBMET01122 0.061 0.014 DBMET01124 0.08 0.007 DBMET01063 0.04 0.034 DBMET01068 | DBMET01063 | |
| 0.012 | 0.177 | 0.035 | Toll-Like receptor 2 agonist | 0.035 0.034 DBMET01063 | DBMET01063 | |
| 0.017 | 0.183 | 0.106 | Opioid mu receptor antagonist | 0.106 0.03 DBMET01063 0.058 0.056 DBMET01082 0.058 0.056 DBMET01084 0.058 0.056 DBMET01085 0.058 0.056 DBMET01086 | DBMET01063 | |
| 0.049 | 0.221 | 0.16 | Lanosterol 14 alpha demethylase inhibitor | 0.113 0.038 DBMET01061 0.113 0.038 DBMET01062 0.129 0.023 DBMET01081 0.113 0.038 DBMET01122 0.091 0.07 DBMET01124 0.14 0.016 DBMET01063 0.116 0.035 DBMET01065 0.107 0.045 DBMET01082 0.107 0.045 DBMET01084 0.116 0.035 DBMET01066 0.102 0.053 DBMET01067 0.107 0.045 DBMET01085 0.107 0.045 DBMET01086 0.16 0.009 DBMET01064 0.135 0.018 DBMET01068 | DBMET01064 | |
| 0.01 | 0.187 | 0.06 | Opioid mu receptor agonist | 0.06 0.024 DBMET01063 | DBMET01063 | |
| 0.057 | 0.239 | 0.203 | Cyclooxygenase 3 inhibitor | 0.16 0.04 DBMET01081 0.119 0.079 DBMET01122 0.148 0.05 DBMET01124 0.138 0.059 DBMET01063 0.108 0.092 DBMET01082 0.108 0.092 DBMET01084 0.108 0.092 DBMET01085 0.108 0.092 DBMET01086 0.203 0.018 DBMET01064 0.125 0.072 DBMET01068 | DBMET01064 | |
| 0.018 | 0.204 | 0.096 | AICAR transformylase inhibitor | 0.044 0.03 DBMET01081 0.05 0.022 DBMET01063 0.096 0.005 DBMET01064 | DBMET01064 | |
| 0.013 | 0.199 | 0.096 | Neutrophil collagenase inhibitor | 0.096 0.024 DBMET01081 0.072 0.037 DBMET01063 0.058 0.053 DBMET01064 | DBMET01081 | |
| 0.009 | 0.197 | 0.017 | Potassium channel (Inward rectifier) 11 blocker | 0.017 0.016 DBMET01065 0.017 0.016 DBMET01066 | DBMET01066 | |
| 0.013 | 0.202 | 0.071 | Factor XIIIa inhibitor | 0.046 0.018 DBMET01081 0.034 0.03 DBMET01122 0.048 0.017 DBMET01124 0.071 0.009 DBMET01063 0.04 0.023 DBMET01064 | DBMET01063 | |
| 0.018 | 0.209 | 0.037 | Aggrecanase 1 inhibitor | 0.037 0.032 DBMET01064 | DBMET01064 | |
| 0.01 | 0.202 | 0.078 | Ornithine carbamoyltransferase inhibitor | 0.046 0.043 DBMET01063 0.078 0.022 DBMET01064 0.052 0.038 DBMET01068 | DBMET01064 | |
| 0.002 | 0.196 | 0.08 | Integrin alpha4beta1 antagonist | 0.08 0.004 DBMET01064 | DBMET01064 | |
| 0.034 | 0.229 | 0.129 | Opioid antagonist | 0.086 0.062 DBMET01081 0.081 0.067 DBMET01124 0.129 0.032 DBMET01063 0.093 0.053 DBMET01082 0.093 0.053 DBMET01084 0.093 0.053 DBMET01085 0.093 0.053 DBMET01086 | DBMET01063 | |
| 0.016 | 0.212 | 0.082 | Lysophosphatidic acid 3 receptor antagonist | 0.048 0.039 DBMET01081 0.082 0.009 DBMET01064 | DBMET01064 | |
| 0.014 | 0.211 | 0.041 | Membrane dipeptidase inhibitor | 0.038 0.03 DBMET01081 0.041 0.025 DBMET01064 | DBMET01064 | |
| 0.014 | 0.221 | 0.029 | Glucosylceramidase stimulant | 0.029 0.013 DBMET01081 0.028 0.018 DBMET01063 | DBMET01081 | |
| 0.022 | 0.23 | 0.112 | Histone deacetylase inhibitor | 0.072 0.038 DBMET01081 0.088 0.025 DBMET01124 0.112 0.014 DBMET01063 | DBMET01063 | |
| 0.018 | 0.23 | 0.134 | Matrix metalloproteinase inhibitor | 0.134 0.016 DBMET01081 0.062 0.052 DBMET01063 | DBMET01081 | |
| 0.126 | 0.34 | 0.352 | Tyrosine 3 hydroxylase inhibitor | 0.185 0.165 DBMET01061 0.185 0.165 DBMET01062 0.214 0.112 DBMET01081 0.198 0.139 DBMET01122 0.214 0.112 DBMET01124 0.254 0.064 DBMET01063 0.187 0.16 DBMET01065 0.187 0.16 DBMET01066 0.352 0.016 DBMET01064 | DBMET01064 | |
| 0.026 | 0.244 | 0.145 | Metalloproteinase-9 inhibitor | 0.145 0.016 DBMET01081 0.072 0.051 DBMET01063 0.067 0.063 DBMET01064 | DBMET01081 | |
| 0.016 | 0.24 | 0.082 | Matrix metalloproteinase (membrane-type) inhibitor | 0.082 0.019 DBMET01081 | DBMET01081 | |
| 0.004 | 0.229 | 0.079 | GP IIb/IIIa receptor antagonist | 0.079 0.022 DBMET01064 | DBMET01064 | |
| 0.01 | 0.244 | 0.04 | Histone deacetylase 7 inhibitor | 0.035 0.028 DBMET01081 0.04 0.023 DBMET01124 0.039 0.024 DBMET01063 0.034 0.029 DBMET01064 | DBMET01124 | |
| 0.014 | 0.248 | 0.064 | Nicotinic receptor alpha3 subunit antagonist | 0.044 0.031 DBMET01081 0.064 0.018 DBMET01063 | DBMET01063 | |
| 0.027 | 0.262 | 0.115 | Histone deacetylase SIRT1 stimulant | 0.102 0.026 DBMET01124 0.115 0.02 DBMET01063 0.114 0.02 DBMET01064 0.078 0.046 DBMET01068 | DBMET01063 | |
| 0.027 | 0.262 | 0.115 | Histone deacetylase stimulant | 0.102 0.026 DBMET01124 0.115 0.02 DBMET01063 0.114 0.02 DBMET01064 0.078 0.046 DBMET01068 | DBMET01063 | |
| 0.004 | 0.241 | 0.047 | Somatostatin 5 antagonist | 0.047 0.014 DBMET01063 0.038 0.019 DBMET01068 | DBMET01063 | |
| 0.007 | 0.244 | 0.041 | AMPA 2 receptor antagonist | 0.041 0.014 DBMET01064 | DBMET01064 | |
| 0.024 | 0.263 | 0.112 | Metalloproteinase-2 inhibitor | 0.112 0.033 DBMET01081 0.079 0.054 DBMET01064 | DBMET01081 | |
| 0.006 | 0.246 | 0.035 | Integrin alphaVbeta3 antagonist | 0.035 0.006 DBMET01064 | DBMET01064 | |
| 0.05 | 0.291 | 0.497 | Cell adhesion inhibitor | 0.163 0.039 DBMET01081 0.121 0.064 DBMET01124 0.156 0.043 DBMET01063 0.497 0.004 DBMET01064 | DBMET01064 | |
| 0.024 | 0.266 | 0.06 | Parathyroid hormone antagonist | 0.06 0.011 DBMET01065 0.06 0.011 DBMET01066 | DBMET01066 | |
| 0.003 | 0.247 | 0.016 | Integrin alphaVbeta6 antagonist | 0.016 0.008 DBMET01064 | DBMET01064 | |
| 0.054 | 0.302 | 0.178 | Cell wall synthesis inhibitor | 0.12 0.1 DBMET01064 0.178 0.042 DBMET01068 | DBMET01068 | |
| 0.099 | 0.354 | 0.289 | Neuropeptide Y2 antagonist | 0.193 0.133 DBMET01061 0.193 0.133 DBMET01062 0.289 0.025 DBMET01081 0.199 0.121 DBMET01122 0.227 0.08 DBMET01124 0.277 0.033 DBMET01063 0.189 0.14 DBMET01082 0.189 0.14 DBMET01084 0.189 0.14 DBMET01085 0.189 0.14 DBMET01086 0.229 0.078 DBMET01064 0.246 0.06 DBMET01068 | DBMET01081 | |
| 0.019 | 0.277 | 0.113 | Nav1.8 sodium channel blocker | 0.113 0.023 DBMET01063 | DBMET01063 | |
| 0.005 | 0.265 | 0.116 | Prostacyclin antagonist | 0.116 0.004 DBMET01064 | DBMET01064 | |
| 0.047 | 0.311 | 0.082 | Ca(v)3.1 blocker | 0.082 0.053 DBMET01124 | DBMET01124 | |
| 0.005 | 0.273 | 0.041 | Lysine carboxypeptidase inhibitor | 0.041 0.01 DBMET01064 | DBMET01064 | |
| 0.025 | 0.294 | 0.085 | Corticotropin releasing factor 2 receptor antagonist | 0.067 0.033 DBMET01081 0.085 0.013 DBMET01063 | DBMET01063 | |
| 0.005 | 0.275 | 0.064 | AMPA 3 receptor antagonist | 0.039 0.014 DBMET01063 0.064 0.005 DBMET01064 | DBMET01064 | |
| 0.003 | 0.276 | 0.081 | AMPA 1 receptor antagonist | 0.042 0.014 DBMET01063 0.081 0.007 DBMET01064 | DBMET01064 | |
| 0.037 | 0.311 | 0.161 | Caspase 3 inhibitor | 0.103 0.087 DBMET01061 0.103 0.087 DBMET01062 0.161 0.021 DBMET01081 0.103 0.086 DBMET01122 0.1 0.092 DBMET01082 0.1 0.092 DBMET01084 0.1 0.092 DBMET01085 0.1 0.092 DBMET01086 0.142 0.034 DBMET01064 | DBMET01081 | |
| 0.007 | 0.289 | 0.197 | Oxytocin antagonist | 0.197 0.005 DBMET01082 0.197 0.005 DBMET01084 0.197 0.005 DBMET01085 0.197 0.005 DBMET01086 | DBMET01086 | |
| 0.014 | 0.299 | 0.041 | Somatostatin 4 agonist | 0.041 0.021 DBMET01063 | DBMET01063 | |
| 0.004 | 0.289 | 0.021 | Follicle-stimulating hormone agonist | 0.021 0.017 DBMET01063 | DBMET01063 | |
| 0.009 | 0.295 | 0.04 | Factor XIa inhibitor | 0.04 0.029 DBMET01063 | DBMET01063 | |
| 0.043 | 0.333 | 0.25 | Calcium channel N-type blocker | 0.196 0.017 DBMET01081 0.134 0.048 DBMET01122 0.25 0.008 DBMET01124 0.104 0.089 DBMET01063 | DBMET01124 | |
| 0.015 | 0.309 | 0.441 | Histidine decarboxylase inhibitor | 0.066 0.055 DBMET01124 0.158 0.018 DBMET01063 0.441 0.003 DBMET01064 0.105 0.03 DBMET01068 | DBMET01064 | |
| 0.004 | 0.307 | 0.032 | Vitronectin receptor antagonist | 0.032 0.01 DBMET01064 | DBMET01064 | |
| 0.013 | 0.319 | 0.143 | Histone deacetylase SIRT2 inhibitor | 0.143 0.009 DBMET01063 0.065 0.061 DBMET01064 0.067 0.058 DBMET01068 | DBMET01063 | |
| 0.018 | 0.325 | 0.064 | Protein kinase C iota inhibitor | 0.064 0.037 DBMET01063 | DBMET01063 | |
| 0.011 | 0.323 | 0.046 | Ceramide glucosyltransferase inhibitor | 0.046 0.01 DBMET01068 | DBMET01068 | |
| 0.005 | 0.317 | 0.046 | Geranyltranstransferase inhibitor | 0.046 0.027 DBMET01124 0.045 0.028 DBMET01064 | DBMET01124 | |
| 0.005 | 0.32 | 0.055 | Protocollagen prolyl hydroxylase inhibitor | 0.055 0.005 DBMET01064 | DBMET01064 | |
| 0.008 | 0.327 | 0.03 | Somatostatin agonist | 0.03 0.023 DBMET01063 | DBMET01063 | |
| 0.004 | 0.325 | 0.075 | Kainate receptor 2 antagonist | 0.075 0.008 DBMET01064 | DBMET01064 | |
| 0.029 | 0.35 | 0.126 | Chelator | 0.091 0.09 DBMET01124 0.126 0.048 DBMET01064 | DBMET01064 | |
| 0.018 | 0.339 | 0.062 | Botulinum neurotoxin type A inhibitor | 0.054 0.047 DBMET01063 0.062 0.035 DBMET01064 | DBMET01064 | |
| 0.028 | 0.351 | 0.391 | Cell adhesion molecule inhibitor | 0.087 0.045 DBMET01081 0.074 0.062 DBMET01063 0.391 0.005 DBMET01064 | DBMET01064 | |
| 0.039 | 0.365 | 0.201 | DOPA decarboxylase inhibitor | 0.121 0.044 DBMET01063 0.201 0.006 DBMET01064 | DBMET01064 | |
| 0.01 | 0.339 | 0.08 | Argininosuccinate synthase inhibitor | 0.08 0.025 DBMET01064 | DBMET01064 | |
| 0.099 | 0.429 | 0.292 | Apoptosis antagonist | 0.267 0.111 DBMET01081 0.238 0.14 DBMET01124 0.21 0.166 DBMET01063 0.228 0.149 DBMET01082 0.228 0.149 DBMET01084 0.228 0.149 DBMET01085 0.228 0.149 DBMET01086 0.292 0.091 DBMET01064 | DBMET01064 | |
| 0.011 | 0.341 | 0.065 | Cyclin A1 inhibitor | 0.065 0.029 DBMET01063 | DBMET01063 | |
| 0.004 | 0.335 | 0.032 | Glucagon receptor antagonist | 0.032 0.019 DBMET01064 | DBMET01064 | |
| 0.015 | 0.349 | 0.065 | CXC chemokine 4 receptor antagonist | 0.058 0.044 DBMET01124 0.065 0.039 DBMET01063 | DBMET01063 | |
| 0.008 | 0.344 | 0.057 | ICAM 1 antagonist | 0.022 0.019 DBMET01124 0.026 0.011 DBMET01063 0.057 0.004 DBMET01064 | DBMET01064 | |
| 0.035 | 0.377 | 0.091 | Granulocyte macrophage colony stimulating factor agonist | 0.091 0.05 DBMET01064 | DBMET01064 | |
| 0.015 | 0.357 | 0.053 | Kainate receptor agonist | 0.053 0.011 DBMET01064 | DBMET01064 | |
| 0.088 | 0.434 | 0.488 | Histamine release inhibitor | 0.213 0.188 DBMET01061 0.213 0.188 DBMET01062 0.364 0.093 DBMET01081 0.249 0.156 DBMET01122 0.215 0.185 DBMET01124 0.276 0.138 DBMET01063 0.247 0.157 DBMET01082 0.247 0.157 DBMET01084 0.38 0.086 DBMET01067 0.247 0.157 DBMET01085 0.247 0.157 DBMET01086 0.488 0.033 DBMET01064 0.473 0.039 DBMET01068 | DBMET01064 | |
| 0.026 | 0.372 | 0.081 | Keratolytic | 0.081 0.047 DBMET01064 | DBMET01064 | |
| 0.005 | 0.353 | 0.052 | Diacylglycerol O-acyltransferase 1 inhibitor | 0.052 0.009 DBMET01064 | DBMET01064 | |
| 0.024 | 0.373 | 0.114 | Glutamate dehydrogenase inhibitor | 0.07 0.056 DBMET01063 0.114 0.025 DBMET01064 0.079 0.045 DBMET01068 | DBMET01064 | |
| 0.009 | 0.373 | 0.048 | AMPA 4 receptor antagonist | 0.048 0.016 DBMET01064 | DBMET01064 | |
| 0.015 | 0.38 | 0.069 | Analgesic, opioid | 0.069 0.063 DBMET01063 | DBMET01063 | |
| 0.02 | 0.392 | 0.072 | Potassium channel (Tandem pore domain) blocker | 0.072 0.057 DBMET01081 0.071 0.059 DBMET01063 0.07 0.064 DBMET01064 | DBMET01081 | |
| 0.062 | 0.442 | 0.477 | Superoxide dismutase inhibitor | 0.172 0.153 DBMET01081 0.245 0.078 DBMET01124 0.384 0.029 DBMET01063 0.477 0.015 DBMET01064 0.274 0.061 DBMET01068 | DBMET01064 | |
| 0.076 | 0.459 | 0.232 | 5 Hydroxytryptamine release stimulant | 0.169 0.154 DBMET01081 0.232 0.098 DBMET01063 0.212 0.112 DBMET01064 | DBMET01063 | |
| 0.004 | 0.388 | 0.019 | Integrin alphaLbeta2 antagonist | 0.019 0.005 DBMET01064 | DBMET01064 | |
| 0.068 | 0.453 | 0.147 | Papain-like protease (SARS coronavirus) inhibitor | 0.139 0.046 DBMET01124 0.147 0.037 DBMET01065 0.147 0.037 DBMET01066 | DBMET01066 | |
| 0.012 | 0.397 | 0.066 | Aconitate hydratase inhibitor | 0.066 0.021 DBMET01064 | DBMET01064 | |
| 0.007 | 0.395 | 0.077 | Glycine transporter 2 inhibitor | 0.077 0.018 DBMET01064 | DBMET01064 | |
| 0.02 | 0.413 | 0.107 | Nitric-oxide synthase inhibitor | 0.107 0.05 DBMET01063 0.096 0.067 DBMET01064 | DBMET01063 | |
| 0.035 | 0.442 | 0.295 | Nav1.2 sodium channel blocker | 0.142 0.062 DBMET01081 0.135 0.068 DBMET01124 0.295 0.015 DBMET01063 0.152 0.056 DBMET01064 0.157 0.053 DBMET01068 | DBMET01063 | |
| 0.006 | 0.413 | 0.02 | Toll-Like receptor 8 agonist | 0.02 0.016 DBMET01068 | DBMET01068 | |
| 0.009 | 0.418 | 0.067 | Collagenase 3 inhibitor | 0.067 0.034 DBMET01081 0.053 0.051 DBMET01063 0.066 0.035 DBMET01064 | DBMET01081 | |
| 0.023 | 0.435 | 0.121 | Neurotrophic factor | 0.121 0.093 DBMET01081 0.115 0.103 DBMET01063 | DBMET01081 | |
| 0.021 | 0.442 | 0.26 | GABA C receptor agonist | 0.131 0.043 DBMET01063 0.26 0.012 DBMET01064 0.11 0.057 DBMET01068 | DBMET01064 | |
| 0.063 | 0.486 | 0.311 | Gastrin inhibitor | 0.256 0.072 DBMET01081 0.255 0.074 DBMET01124 0.257 0.071 DBMET01063 0.311 0.026 DBMET01064 | DBMET01064 | |
| 0.03 | 0.457 | 0.124 | DNA polymerase I inhibitor | 0.124 0.065 DBMET01124 | DBMET01124 | |
| 0.021 | 0.45 | 0.098 | Prolactin inhibitor | 0.098 0.057 DBMET01064 | DBMET01064 | |
| 0.025 | 0.455 | 0.232 | Alpha-N-acetylglucosaminidase inhibitor | 0.232 0.026 DBMET01064 0.13 0.068 DBMET01068 | DBMET01064 | |
| 0.005 | 0.442 | 0.031 | RNA-directed RNA polymerase inhibitor | 0.031 0.028 DBMET01064 | DBMET01064 | |
| 0.034 | 0.472 | 0.207 | Peroxidase inhibitor | 0.207 0.057 DBMET01064 0.192 0.061 DBMET01068 | DBMET01064 | |
| 0.002 | 0.44 | 0.028 | Integrin beta2 antagonist | 0.028 0.004 DBMET01064 | DBMET01064 | |
| 0.027 | 0.467 | 0.119 | Toll-Like receptor 2 antagonist | 0.119 0.079 DBMET01064 | DBMET01064 | |
| 0.005 | 0.445 | 0.066 | LFA antagonist | 0.026 0.023 DBMET01063 0.066 0.005 DBMET01064 | DBMET01064 | |
| 0.042 | 0.485 | 0.125 | Melanin inhibitor | 0.125 0.124 DBMET01064 | DBMET01064 | |
| 0.017 | 0.461 | 0.434 | Psychostimulant | 0.145 0.121 DBMET01081 0.145 0.12 DBMET01124 0.348 0.032 DBMET01063 0.174 0.097 DBMET01065 0.174 0.097 DBMET01066 0.434 0.018 DBMET01064 0.383 0.025 DBMET01068 | DBMET01064 | |
| 0.011 | 0.457 | 0.062 | Sphingosine 1-phosphate receptor 3 antagonist | 0.062 0.036 DBMET01064 | DBMET01064 | |
| 0.085 | 0.533 | 0.227 | Nitric-oxide synthase stimulant | 0.205 0.081 DBMET01063 0.22 0.06 DBMET01064 0.227 0.052 DBMET01068 | DBMET01068 | |
| 0.004 | 0.452 | 0.167 | Secretase gamma inhibitor | 0.167 0.004 DBMET01061 0.167 0.004 DBMET01062 0.083 0.008 DBMET01065 0.036 0.035 DBMET01082 0.036 0.035 DBMET01084 0.083 0.008 DBMET01066 0.148 0.004 DBMET01067 0.036 0.035 DBMET01085 0.036 0.035 DBMET01086 | DBMET01062 | |
| 0.003 | 0.451 | 0.058 | Kainate receptor antagonist | 0.058 0.017 DBMET01064 | DBMET01064 | |
| 0.046 | 0.494 | 0.36 | Transcription factor STAT3 inhibitor | 0.174 0.173 DBMET01061 0.174 0.173 DBMET01062 0.351 0.032 DBMET01081 0.237 0.094 DBMET01122 0.256 0.078 DBMET01124 0.36 0.03 DBMET01063 0.223 0.108 DBMET01064 | DBMET01063 | |
| 0.004 | 0.453 | 0.135 | Phosphorylase inhibitor | 0.056 0.027 DBMET01063 0.135 0.008 DBMET01064 0.051 0.03 DBMET01068 | DBMET01064 | |
| 0.008 | 0.458 | 0.06 | Glutamate (mGluR1a) antagonist | 0.06 0.015 DBMET01063 0.058 0.016 DBMET01064 0.054 0.018 DBMET01068 | DBMET01063 | |
| 0.03 | 0.489 | 0.168 | Amyloid beta aggregation inhibitor | 0.168 0.096 DBMET01122 | DBMET01122 | |
| 0.009 | 0.469 | 0.054 | Adenosine deaminase inhibitor | 0.046 0.034 DBMET01063 0.054 0.026 DBMET01064 | DBMET01064 | |
| 0.009 | 0.47 | 0.194 | Phenylalanine 4-hydroxylase inhibitor | 0.077 0.04 DBMET01063 0.194 0.007 DBMET01064 0.117 0.019 DBMET01068 | DBMET01064 | |
| 0.001 | 0.462 | 0.02 | Integrin alphaVbeta5 antagonist | 0.02 0.004 DBMET01064 | DBMET01064 | |
| 0.003 | 0.465 | 0.036 | Squalene synthetase inhibitor | 0.036 0.02 DBMET01124 | DBMET01124 | |
| 0.003 | 0.466 | 0.148 | Vasopressin 1B antagonist | 0.148 0.004 DBMET01061 0.148 0.004 DBMET01062 0.146 0.004 DBMET01065 0.024 0.023 DBMET01082 0.024 0.023 DBMET01084 0.146 0.004 DBMET01066 0.112 0.004 DBMET01067 0.024 0.023 DBMET01085 0.024 0.023 DBMET01086 | DBMET01062 | |
| 0.03 | 0.493 | 0.104 | Photosensitizer | 0.104 0.081 DBMET01064 | DBMET01064 | |
| 0.013 | 0.476 | 0.035 | Glutamate (mGluR8) antagonist | 0.035 0.026 DBMET01064 | DBMET01064 | |
| 0.009 | 0.473 | 0.131 | Porphobilinogen synthase inhibitor | 0.083 0.045 DBMET01063 0.131 0.025 DBMET01064 0.069 0.056 DBMET01068 | DBMET01064 | |
| 0.005 | 0.469 | 0.037 | Angiotensin II receptor antagonist | 0.037 0.019 DBMET01064 | DBMET01064 | |
| 0.02 | 0.486 | 0.094 | Sphingomyelinase inhibitor | 0.094 0.066 DBMET01068 | DBMET01068 | |
| 0.023 | 0.489 | 0.156 | Beta amyloid protein antagonist | 0.099 0.09 DBMET01081 0.155 0.037 DBMET01063 0.156 0.036 DBMET01064 | DBMET01064 | |
| 0.007 | 0.473 | 0.034 | Glutamate (mGluR1) agonist | 0.034 0.007 DBMET01064 | DBMET01064 | |
| 0.009 | 0.486 | 0.021 | Vitamin D receptor antagonist | 0.021 0.019 DBMET01065 0.021 0.019 DBMET01066 | DBMET01066 | |
| 0.012 | 0.489 | 0.119 | Alkylator | 0.119 0.069 DBMET01064 0.111 0.077 DBMET01068 | DBMET01064 | |
| 0.094 | 0.572 | 0.282 | 5 Hydroxytryptamine uptake stimulant | 0.261 0.07 DBMET01063 0.282 0.055 DBMET01064 | DBMET01064 | |
| 0.038 | 0.518 | 0.147 | Adenylate cyclase stimulant | 0.126 0.111 DBMET01124 0.128 0.106 DBMET01063 0.147 0.069 DBMET01064 0.138 0.086 DBMET01068 | DBMET01064 | |
| 0.009 | 0.495 | 0.113 | Glutamate decarboxylase inhibitor | 0.071 0.054 DBMET01063 0.105 0.027 DBMET01064 0.113 0.023 DBMET01068 | DBMET01068 | |
| 0.034 | 0.522 | 0.219 | DNA synthesis inhibitor | 0.219 0.095 DBMET01064 | DBMET01064 | |
| 0.024 | 0.515 | 0.256 | Insulin sensitizer | 0.147 0.138 DBMET01081 0.165 0.113 DBMET01063 0.256 0.031 DBMET01064 0.158 0.122 DBMET01068 | DBMET01064 | |
| 0.042 | 0.537 | 0.163 | NOS3 expression enhancer | 0.163 0.061 DBMET01122 0.127 0.102 DBMET01064 | DBMET01122 | |
| 0.004 | 0.5 | 0.089 | Glutamate (mGluR group I) agonist | 0.056 0.026 DBMET01063 0.089 0.01 DBMET01064 | DBMET01064 | |
| 0.01 | 0.507 | 0.082 | Epithelial sodium channel blocker | 0.082 0.012 DBMET01063 0.051 0.048 DBMET01068 | DBMET01063 | |
| 0.1 | 0.601 | 0.217 | MAP kinase kinase 3 inhibitor | 0.217 0.08 DBMET01124 0.211 0.093 DBMET01063 0.203 0.113 DBMET01068 | DBMET01124 | |
| 0.006 | 0.509 | 0.055 | Integrin alpha2beta1 antagonist | 0.055 0.004 DBMET01064 | DBMET01064 | |
| 0.03 | 0.537 | 0.161 | Succinate dehydrogenase inhibitor | 0.161 0.093 DBMET01064 | DBMET01064 | |
| 0.01 | 0.518 | 0.041 | Glutamate (mGluR8) agonist | 0.041 0.021 DBMET01064 | DBMET01064 | |
| 0.101 | 0.612 | 0.484 | Calcium channel L-type activator | 0.385 0.091 DBMET01067 0.275 0.18 DBMET01064 0.484 0.034 DBMET01068 | DBMET01068 | |
| 0.004 | 0.515 | 0.097 | Cannabinoid CB1 receptor agonist | 0.055 0.047 DBMET01081 0.097 0.021 DBMET01063 | DBMET01063 | |
| 0.008 | 0.521 | 0.053 | Beta 2 adrenoreceptor antagonist | 0.053 0.033 DBMET01068 | DBMET01068 | |
| 0.005 | 0.518 | 0.052 | Glutamate (mGluR3) antagonist | 0.052 0.011 DBMET01064 | DBMET01064 | |
| 0.02 | 0.535 | 0.07 | Glutamate (mGluR6) antagonist | 0.07 0.039 DBMET01064 | DBMET01064 | |
| 0.025 | 0.541 | 0.141 | Electron transport complex I inhibitor | 0.141 0.026 DBMET01122 | DBMET01122 | |
| 0.012 | 0.53 | 0.089 | Phospholipase D inhibitor | 0.068 0.057 DBMET01124 0.089 0.023 DBMET01064 | DBMET01064 | |
| 0.058 | 0.578 | 0.229 | Sodium/bile acid cotransporter inhibitor | 0.2 0.188 DBMET01081 0.229 0.151 DBMET01064 | DBMET01064 | |
| 0.004 | 0.525 | 0.045 | Angiotensin AT1 receptor antagonist | 0.045 0.025 DBMET01064 | DBMET01064 | |
| 0.004 | 0.525 | 0.064 | NMDA 2A receptor antagonist | 0.064 0.027 DBMET01064 0.055 0.033 DBMET01068 | DBMET01064 | |
| 0.009 | 0.531 | 0.059 | Aryl hydrocarbon receptor antagonist | 0.059 0.056 DBMET01063 | DBMET01063 | |
| 0.01 | 0.533 | 0.049 | Dopamine beta hydroxylase inhibitor | 0.049 0.032 DBMET01063 0.046 0.04 DBMET01064 | DBMET01063 | |
| 0.004 | 0.529 | 0.053 | Glutamate (mGluR5) agonist | 0.053 0.023 DBMET01064 | DBMET01064 | |
| 0.002 | 0.531 | 0.028 | Glutamate (mGluR1a) agonist | 0.028 0.01 DBMET01064 | DBMET01064 | |
| 0.004 | 0.535 | 0.083 | Thymidylate synthase inhibitor | 0.083 0.006 DBMET01064 | DBMET01064 | |
| 0.004 | 0.542 | 0.111 | Antineoplastic antibiotic | 0.111 0.041 DBMET01067 | DBMET01067 | |
| 0.005 | 0.545 | 0.07 | Phosphofructokinase-1 inhibitor | 0.07 0.048 DBMET01064 | DBMET01064 | |
| 0.034 | 0.574 | 0.18 | Transcription factor STAT6 inhibitor | 0.18 0.01 DBMET01063 0.138 0.034 DBMET01068 | DBMET01063 | |
| 0.004 | 0.543 | 0.083 | Vasopressin 1 antagonist | 0.083 0.011 DBMET01061 0.083 0.011 DBMET01062 0.078 0.011 DBMET01065 0.078 0.011 DBMET01066 0.039 0.018 DBMET01067 | DBMET01062 | |
| 0.007 | 0.547 | 0.073 | Integrin alpha2 antagonist | 0.073 0.005 DBMET01064 | DBMET01064 | |
| 0.018 | 0.561 | 0.164 | Calcium channel (voltage-sensitive) blocker | 0.12 0.056 DBMET01081 0.164 0.027 DBMET01124 | DBMET01124 | |
| 0.006 | 0.55 | 0.048 | Glutamate (mGluR4) agonist | 0.048 0.012 DBMET01064 | DBMET01064 | |
| 0.022 | 0.568 | 0.128 | Acetylcholine release stimulant | 0.128 0.037 DBMET01063 0.119 0.05 DBMET01064 0.103 0.081 DBMET01068 | DBMET01063 | |
| 0.021 | 0.571 | 0.118 | UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor | 0.118 0.04 DBMET01064 | DBMET01064 | |
| 0.011 | 0.564 | 0.033 | Antibiotic Aminoglycoside-like | 0.033 0.031 DBMET01082 0.033 0.031 DBMET01084 0.033 0.031 DBMET01085 0.033 0.031 DBMET01086 | DBMET01086 | |
| 0.017 | 0.572 | 0.063 | Exportin-1 inhibitor | 0.063 0.062 DBMET01063 0.063 0.062 DBMET01068 | DBMET01068 | |
| 0.016 | 0.575 | 0.119 | GABA C receptor rho-1 antagonist | 0.099 0.064 DBMET01063 0.119 0.041 DBMET01064 | DBMET01064 | |
| 0.039 | 0.602 | 0.397 | Cholesterol antagonist | 0.397 0.05 DBMET01064 | DBMET01064 | |
| 0.009 | 0.572 | 0.085 | NMDA receptor agonist | 0.085 0.026 DBMET01064 | DBMET01064 | |
| 0.007 | 0.573 | 0.102 | Diacylglycerol O-acyltransferase inhibitor | 0.102 0.007 DBMET01064 | DBMET01064 | |
| 0.011 | 0.578 | 0.079 | Caspase 7 inhibitor | 0.079 0.065 DBMET01081 | DBMET01081 | |
| 0.001 | 0.571 | 0.025 | Egl nine homolog 1 inhibitor | 0.025 0.005 DBMET01064 | DBMET01064 | |
| 0.006 | 0.577 | 0.069 | Thromboxane synthase inhibitor | 0.069 0.018 DBMET01064 | DBMET01064 | |
| 0.003 | 0.579 | 0.094 | AMPA receptor antagonist | 0.042 0.041 DBMET01063 0.094 0.013 DBMET01064 | DBMET01064 | |
| 0.003 | 0.579 | 0.116 | Glutamate (mGluR1) antagonist | 0.086 0.021 DBMET01063 0.051 0.047 DBMET01065 0.051 0.047 DBMET01066 0.116 0.012 DBMET01064 | DBMET01064 | |
| 0.036 | 0.612 | 0.392 | Transcription factor STAT inhibitor | 0.348 0.035 DBMET01081 0.249 0.087 DBMET01122 0.244 0.091 DBMET01124 0.392 0.021 DBMET01063 0.217 0.115 DBMET01064 0.199 0.14 DBMET01068 | DBMET01063 | |
| 0.004 | 0.582 | 0.073 | Antidiuretic hormone antagonist | 0.073 0.017 DBMET01061 0.073 0.017 DBMET01062 0.065 0.018 DBMET01065 0.065 0.018 DBMET01066 0.036 0.03 DBMET01067 | DBMET01062 | |
| 0.045 | 0.628 | 0.392 | Nootropic | 0.207 0.148 DBMET01061 0.207 0.148 DBMET01062 0.331 0.06 DBMET01081 0.392 0.041 DBMET01063 0.316 0.067 DBMET01082 0.316 0.067 DBMET01084 0.316 0.067 DBMET01085 0.316 0.067 DBMET01086 0.347 0.055 DBMET01064 0.25 0.108 DBMET01068 | DBMET01063 | |
| 0.011 | 0.595 | 0.074 | Glutamate (mGluR4) antagonist | 0.074 0.009 DBMET01064 | DBMET01064 | |
| 0.072 | 0.657 | 0.139 | Heat shock protein 70 antagonist | 0.139 0.079 DBMET01064 | DBMET01064 | |
| 0.027 | 0.613 | 0.144 | GABA C receptor rho-2 antagonist | 0.144 0.082 DBMET01064 | DBMET01064 | |
| 0.016 | 0.606 | 0.181 | Free radical scavenger | 0.181 0.114 DBMET01124 | DBMET01124 | |
| 0.011 | 0.604 | 0.089 | Mediator release inhibitor | 0.089 0.083 DBMET01064 | DBMET01064 | |
| 0.03 | 0.624 | 0.27 | Interleukin agonist | 0.205 0.116 DBMET01063 0.27 0.065 DBMET01064 0.26 0.072 DBMET01068 | DBMET01064 | |
| 0.003 | 0.603 | 0.034 | Glutamate (mGluR group II) antagonist | 0.034 0.033 DBMET01064 | DBMET01064 | |
| 0.045 | 0.652 | 0.201 | Growth factor agonist | 0.201 0.062 DBMET01124 | DBMET01124 | |
| 0.012 | 0.621 | 0.138 | Ferrochelatase inhibitor | 0.108 0.063 DBMET01064 0.138 0.043 DBMET01068 | DBMET01068 | |
| 0.01 | 0.62 | 0.112 | Mucolytic | 0.112 0.062 DBMET01064 | DBMET01064 | |
| 0.004 | 0.615 | 0.061 | Cannabinoid receptor agonist | 0.061 0.048 DBMET01063 | DBMET01063 | |
| 0.021 | 0.634 | 0.126 | Cytokine production inhibitor | 0.126 0.084 DBMET01063 0.125 0.085 DBMET01064 | DBMET01063 | |
| 0.009 | 0.624 | 0.067 | Glutamate (mGluR7) antagonist | 0.067 0.048 DBMET01064 | DBMET01064 | |
| 0.005 | 0.621 | 0.068 | Beta 1 adrenoreceptor antagonist | 0.068 0.028 DBMET01068 | DBMET01068 | |
| 0.017 | 0.639 | 0.121 | Adenylate cyclase inhibitor | 0.093 0.091 DBMET01124 0.093 0.091 DBMET01063 0.104 0.081 DBMET01064 0.121 0.067 DBMET01068 | DBMET01068 | |
| 0.017 | 0.641 | 0.053 | DNA helicase inhibitor | 0.053 0.041 DBMET01064 | DBMET01064 | |
| 0.019 | 0.643 | 0.138 | Neuropeptide Y1 antagonist | 0.138 0.085 DBMET01063 | DBMET01063 | |
| 0.005 | 0.63 | 0.071 | Carbamoyl phosphate synthetase inhibitor | 0.071 0.034 DBMET01064 | DBMET01064 | |
| 0.017 | 0.643 | 0.235 | Antibacterial (Helicobacter pylori) | 0.235 0.014 DBMET01124 0.125 0.074 DBMET01064 | DBMET01124 | |
| 0.006 | 0.635 | 0.066 | Beta 2 adrenoreceptor agonist | 0.066 0.029 DBMET01068 | DBMET01068 | |
| 0.004 | 0.642 | 0.058 | Neuronal nicotinic receptor antagonist | 0.058 0.057 DBMET01063 | DBMET01063 | |
| 0.005 | 0.644 | 0.05 | Beta adrenoreceptor agonist | 0.05 0.017 DBMET01068 | DBMET01068 | |
| 0.007 | 0.649 | 0.069 | S-adenosyl-L-methionine decarboxylase inhibitor | 0.069 0.063 DBMET01063 | DBMET01063 | |
| 0.006 | 0.649 | 0.069 | Beta adrenoreceptor antagonist | 0.069 0.04 DBMET01068 | DBMET01068 | |
| 0.002 | 0.647 | 0.065 | Diamine oxidase inhibitor | 0.034 0.032 DBMET01063 0.065 0.008 DBMET01068 | DBMET01068 | |
| 0.034 | 0.679 | 0.269 | Vasodilator, coronary | 0.269 0.115 DBMET01064 0.254 0.13 DBMET01068 | DBMET01064 | |
| 0.007 | 0.655 | 0.092 | Glutamate (mGluR group III) agonist | 0.092 0.011 DBMET01064 | DBMET01064 | |
| 0.018 | 0.672 | 0.235 | Hemostatic | 0.187 0.038 DBMET01081 0.132 0.092 DBMET01124 0.235 0.024 DBMET01063 0.167 0.051 DBMET01064 0.119 0.116 DBMET01068 | DBMET01063 | |
| 0.023 | 0.678 | 0.1 | Glutamate (mGluR7) agonist | 0.1 0.06 DBMET01064 0.092 0.079 DBMET01068 | DBMET01064 | |
| 0.042 | 0.7 | 0.22 | GABA C receptor rho-3 antagonist | 0.22 0.184 DBMET01064 | DBMET01064 | |
| 0.009 | 0.672 | 0.099 | GABA C receptor antagonist | 0.099 0.079 DBMET01064 | DBMET01064 | |
| 0.025 | 0.69 | 0.107 | Adenylate kinase inhibitor | 0.107 0.057 DBMET01064 | DBMET01064 | |
| 0.012 | 0.681 | 0.376 | Platelet antagonist | 0.196 0.104 DBMET01081 0.165 0.13 DBMET01063 0.376 0.032 DBMET01064 0.151 0.143 DBMET01068 | DBMET01064 | |
| 0.025 | 0.695 | 0.093 | Toll-Like receptor 3 antagonist | 0.093 0.062 DBMET01068 | DBMET01068 | |
| 0.075 | 0.754 | 0.35 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.35 0.15 DBMET01063 0.266 0.261 DBMET01064 0.295 0.22 DBMET01068 | DBMET01063 | |
| 0.007 | 0.688 | 0.101 | Urease inhibitor | 0.101 0.065 DBMET01068 | DBMET01068 | |
| 0.011 | 0.697 | 0.152 | Calcium channel blocker | 0.152 0.057 DBMET01124 | DBMET01124 | |
| 0.008 | 0.695 | 0.104 | Polo-like kinase-1 inhibitor | 0.104 0.041 DBMET01063 | DBMET01063 | |
| 0.005 | 0.698 | 0.067 | Protein kinase B gamma inhibitor | 0.067 0.061 DBMET01063 | DBMET01063 | |
| 0.011 | 0.706 | 0.195 | ATPase (Vacuolar H+) inhibitor | 0.195 0.003 DBMET01122 | DBMET01122 | |
| 0.07 | 0.767 | 0.171 | 5 Hydroxytryptamine 3E antagonist | 0.171 0.134 DBMET01063 | DBMET01063 | |
| 0.013 | 0.71 | 0.128 | Interleukin 8 antagonist | 0.128 0.052 DBMET01064 | DBMET01064 | |
| 0.005 | 0.703 | 0.103 | Alcohol dehydrogenase inhibitor | 0.103 0.05 DBMET01064 | DBMET01064 | |
| 0.009 | 0.708 | 0.084 | Uric acid excretion stimulant | 0.084 0.075 DBMET01064 | DBMET01064 | |
| 0.008 | 0.711 | 0.119 | Cystathionine beta-synthase inhibitor | 0.119 0.059 DBMET01064 | DBMET01064 | |
| 0.021 | 0.728 | 0.138 | Phospholipase C inhibitor | 0.138 0.133 DBMET01064 | DBMET01064 | |
| 0.028 | 0.736 | 0.301 | Vasodilator, peripheral | 0.301 0.096 DBMET01064 0.255 0.123 DBMET01068 | DBMET01064 | |
| 0.027 | 0.746 | 0.375 | Cyclophilin D inhibitor | 0.375 0.106 DBMET01064 0.347 0.125 DBMET01068 | DBMET01064 | |
| 0.006 | 0.725 | 0.051 | Glutamate (mGluR group III) antagonist | 0.051 0.019 DBMET01064 | DBMET01064 | |
| 0.01 | 0.73 | 0.138 | Nav1.6 sodium channel blocker | 0.138 0.069 DBMET01063 | DBMET01063 | |
| 0.009 | 0.735 | 0.198 | Spasmolytic | 0.198 0.121 DBMET01068 | DBMET01068 | |
| 0.005 | 0.743 | 0.075 | Peroxisome proliferator-activated receptor gamma antagonist | 0.075 0.041 DBMET01064 | DBMET01064 | |
| 0.017 | 0.759 | 0.208 | Platelet adhesion inhibitor | 0.148 0.108 DBMET01081 0.208 0.067 DBMET01064 | DBMET01064 | |
| 0.014 | 0.757 | 0.188 | DNA damaging | 0.188 0.126 DBMET01064 | DBMET01064 | |
| 0.005 | 0.749 | 0.138 | CDK2/cyclin A inhibitor | 0.138 0.031 DBMET01061 0.138 0.031 DBMET01062 0.116 0.045 DBMET01067 | DBMET01062 | |
| 0.021 | 0.768 | 0.11 | Interleukin 4 antagonist | 0.11 0.101 DBMET01068 | DBMET01068 | |
| 0.004 | 0.753 | 0.224 | Diuretic | 0.171 0.06 DBMET01124 0.183 0.052 DBMET01063 0.224 0.036 DBMET01064 0.134 0.09 DBMET01068 | DBMET01064 | |
| 0.012 | 0.767 | 0.186 | Insulin secretagoues | 0.186 0.044 DBMET01064 | DBMET01064 | |
| 0.004 | 0.76 | 0.101 | Inducible nitric-oxide synthase inhibitor | 0.101 0.036 DBMET01064 | DBMET01064 | |
| 0.003 | 0.766 | 0.074 | TRPA1 antagonist | 0.074 0.029 DBMET01124 | DBMET01124 | |
| 0.045 | 0.808 | 0.16 | MAP kinase kinase 5 inhibitor | 0.16 0.115 DBMET01065 0.16 0.115 DBMET01066 | DBMET01066 | |
| 0.005 | 0.776 | 0.069 | HIV-1 integrase inhibitor | 0.069 0.05 DBMET01064 | DBMET01064 | |
| 0.003 | 0.777 | 0.137 | Glutamate receptor agonist | 0.137 0.021 DBMET01064 | DBMET01064 | |
| 0.004 | 0.783 | 0.156 | Cyclin B inhibitor | 0.156 0.005 DBMET01061 0.156 0.005 DBMET01062 0.056 0.036 DBMET01065 0.056 0.036 DBMET01066 0.125 0.007 DBMET01067 | DBMET01062 | |
| 0.002 | 0.784 | 0.096 | NMDA 2 receptor antagonist | 0.096 0.034 DBMET01068 | DBMET01068 | |
| 0.004 | 0.787 | 0.133 | Adrenaline agonist | 0.133 0.02 DBMET01068 | DBMET01068 | |
| 0.005 | 0.789 | 0.111 | Gastric antisecretory | 0.111 0.052 DBMET01124 | DBMET01124 | |
| 0.004 | 0.813 | 0.184 | Sodium channel blocker | 0.184 0.039 DBMET01063 | DBMET01063 | |
| 0.004 | 0.83 | 0.146 | Sodium channel (voltage-gated) blocker | 0.146 0.057 DBMET01063 | DBMET01063 | |
| 0.004 | 0.842 | 0.382 | Cyclin-dependent kinase 5 inhibitor | 0.382 0.005 DBMET01061 0.382 0.005 DBMET01062 0.105 0.071 DBMET01065 0.105 0.071 DBMET01066 0.34 0.007 DBMET01067 | DBMET01062 | |
| 0.007 | 0.853 | 0.086 | Telomerase inhibitor | 0.068 0.055 DBMET01061 0.068 0.055 DBMET01062 0.086 0.041 DBMET01065 0.086 0.041 DBMET01066 | DBMET01066 | |
| 0.009 | 0.855 | 0.413 | Toll-Like receptor agonist | 0.413 0.055 DBMET01064 0.227 0.172 DBMET01068 | DBMET01064 | |
| 0.009 | 0.857 | 0.406 | Toll-Like receptor 7 agonist | 0.406 0.057 DBMET01064 0.215 0.183 DBMET01068 | DBMET01064 | |
| 0.005 | 0.879 | 0.148 | Platelet aggregation inhibitor | 0.148 0.13 DBMET01064 | DBMET01064 | |
| 0.004 | 0.897 | 0.219 | Anticonvulsant | 0.219 0.07 DBMET01063 0.17 0.107 DBMET01068 | DBMET01063 | |
| 0.004 | 0.904 | 0.221 | Bronchodilator | 0.095 0.07 DBMET01067 0.221 0.015 DBMET01068 | DBMET01068 | |
| 0.005 | 0.912 | 0.173 | Vasodilator | 0.173 0.129 DBMET01068 | DBMET01068 | |
| 0.005 | 0.914 | 0.302 | Antiobesity | 0.302 0.115 DBMET01068 | DBMET01068 | |
| 0.004 | 0.914 | 0.107 | Glutamate receptor antagonist | 0.107 0.088 DBMET01064 | DBMET01064 | |
| 0.004 | 0.915 | 0.512 | Dyrk kinase inhibitor | 0.512 0.013 DBMET01061 0.512 0.013 DBMET01062 0.415 0.024 DBMET01067 | DBMET01062 | |
| 0.004 | 0.917 | 0.533 | Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor | 0.533 0.009 DBMET01061 0.533 0.009 DBMET01062 0.45 0.018 DBMET01067 | DBMET01062 | |
| 0.007 | 0.93 | 0.199 | Hypoglycemic | 0.189 0.124 DBMET01124 0.199 0.113 DBMET01064 | DBMET01064 | |
| 0.005 | 0.944 | 0.195 | Cardiotonic | 0.185 0.135 DBMET01124 0.195 0.124 DBMET01064 0.19 0.128 DBMET01068 | DBMET01064 | |
| 0.004 | 0.971 | 0.148 | Antimitotic | 0.148 0.123 DBMET01122 | DBMET01122 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |