Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.9930.0010.993Alpha 2b adrenoreceptor antagonist

0.737 0.003 DBMET00757

0.9810.0020.981Alpha 2a adrenoreceptor antagonist

0.559 0.004 DBMET00757

0.9570.0010.957Alpha 2c adrenoreceptor antagonist

0.626 0.003 DBMET00757

0.9560.0020.956Alpha 2 adrenoreceptor antagonist

0.492 0.004 DBMET00757

0.910.0020.915 Hydroxytryptamine 2B antagonist

0.548 0.005 DBMET00757

0.9020.0020.902Dopamine D2 agonist

0.614 0.003 DBMET00757

0.8950.0020.8955 Hydroxytryptamine 2C antagonist

0.393 0.005 DBMET00757

0.8640.0030.864Dopamine agonist

0.707 0.004 DBMET00757

0.82200.822Prolactin inhibitor

0.58 0.001 DBMET00757

0.7680.0030.768Dopamine D2 antagonist

0.329 0.009 DBMET00757

0.7680.0040.7685 Hydroxytryptamine antagonist

0.38 0.012 DBMET00757

0.7620.0020.762Dopamine D1 antagonist

0.518 0.003 DBMET00757

0.7410.0030.7415 Hydroxytryptamine 1 antagonist

0.25 0.013 DBMET00757

0.7290.0040.729Dopamine antagonist

0.351 0.009 DBMET00757

0.7250.0040.725Alpha adrenoreceptor antagonist

0.331 0.013 DBMET00757

0.7190.0040.7195 Hydroxytryptamine 2 antagonist

0.39 0.01 DBMET00757

0.690.0030.695 Hydroxytryptamine 1A antagonist

0.247 0.011 DBMET00757

0.6720.0090.8275 Hydroxytryptamine release stimulant

0.827 0.003 DBMET00757

DBMET00757
0.6280.0040.6285 Hydroxytryptamine 2A antagonist

0.333 0.01 DBMET00757

0.6070.0030.6075 Hydroxytryptamine 5A antagonist

0.211 0.005 DBMET00757

0.5890.0030.5895 Hydroxytryptamine 1D antagonist

0.137 0.014 DBMET00757

0.5740.0010.574Prolactin release inhibitor

0.364 0.001 DBMET00757

0.5630.0030.563Alpha 1d adrenoreceptor antagonist

0.149 0.014 DBMET00757

0.5530.0030.5535 Hydroxytryptamine 5 antagonist

0.181 0.005 DBMET00757

0.5140.0040.514Dopamine D3 antagonist

0.155 0.014 DBMET00757

0.5060.0040.5165 Hydroxytryptamine 1F antagonist

0.516 0.004 DBMET00757

DBMET00757
0.5130.0210.513Spasmolytic

0.441 0.033 DBMET00757

0.50.0090.536Sigma receptor agonist

0.536 0.007 DBMET00757

DBMET00757
0.4870.0050.487Alpha 1a adrenoreceptor antagonist

0.165 0.021 DBMET00757

0.490.0120.49Psychostimulant

0.435 0.018 DBMET00757

0.4440.0050.444Alpha 1 adrenoreceptor antagonist

0.17 0.026 DBMET00757

0.3850.0080.385Cholinergic antagonist

0.321 0.013 DBMET00757

0.3740.0090.374Acetylcholine antagonist

0.312 0.013 DBMET00757

0.3650.0070.3655 Hydroxytryptamine 1E antagonist

0.349 0.01 DBMET00757

0.3530.0060.3535 Hydroxytryptamine agonist

0.251 0.01 DBMET00757

0.3290.0020.3295 Hydroxytryptamine 2B agonist

0.164 0.003 DBMET00757

0.3160.0050.3165 Hydroxytryptamine 1B antagonist

0.137 0.014 DBMET00757

0.2940.0140.294Antiadrenergic

0.217 0.021 DBMET00757

0.3730.0960.587Analgesic

0.587 0.029 DBMET00757

DBMET00757
0.2880.0140.288Adrenaline antagonist

0.213 0.021 DBMET00757

0.2630.0080.2635 Hydroxytryptamine 1 agonist

0.189 0.012 DBMET00757

0.2520.0250.296Acetylcholine M1 receptor antagonist

0.296 0.015 DBMET00757

DBMET00757
0.2190.0030.2195 Hydroxytryptamine 1D agonist

0.059 0.008 DBMET00757

0.210.0090.317Opioid kappa receptor antagonist

0.317 0.005 DBMET00757

DBMET00757
0.1920.0070.192Dopamine D4 agonist

0.087 0.017 DBMET00757

0.1970.0130.307Acetylcholine nicotinic antagonist

0.307 0.007 DBMET00757

DBMET00757
0.1960.0150.248Opioid antagonist

0.248 0.008 DBMET00757

DBMET00757
0.1850.0040.1855 Hydroxytryptamine 2 agonist

0.081 0.015 DBMET00757

0.1770.0040.177Alpha 2d adrenoreceptor antagonist

0.149 0.009 DBMET00757

0.1790.0170.179Alpha 1b adrenoreceptor antagonist

0.111 0.032 DBMET00757

0.1610.0060.275Dopamine D5 antagonist

0.275 0.004 DBMET00757

DBMET00757
0.1620.0150.21Opioid mu receptor antagonist

0.21 0.008 DBMET00757

DBMET00757
0.1550.0150.172Alpha adrenoreceptor agonist

0.172 0.012 DBMET00757

DBMET00757
0.1480.0180.162Dopamine D4 antagonist

0.162 0.016 DBMET00757

DBMET00757
0.1450.0160.164Analgesic, opioid

0.164 0.013 DBMET00757

DBMET00757
0.1470.020.184Opioid delta receptor antagonist

0.184 0.014 DBMET00757

DBMET00757
0.150.0440.15Acetylcholine muscarinic antagonist

0.116 0.072 DBMET00757

0.1230.0170.188Neuronal nicotinic receptor antagonist

0.188 0.009 DBMET00757

DBMET00757
0.1150.0110.143Alpha 2 adrenoreceptor agonist

0.143 0.007 DBMET00757

DBMET00757
0.1080.0060.108Dopamine D3 agonist

0.07 0.011 DBMET00757

0.1660.0650.166Cholinergic
0.1950.0970.308Cyclic AMP phosphodiesterase inhibitor

0.308 0.039 DBMET00757

DBMET00757
0.1340.040.142Nav1.1 sodium channel blocker

0.142 0.036 DBMET00757

DBMET00757
0.0980.0040.129Dopamine autoreceptor agonist

0.129 0.004 DBMET00757

DBMET00757
0.1960.1040.196Peptidyltransferase inhibitor
0.1940.1090.212Vasodilator

0.212 0.095 DBMET00757

DBMET00757
0.0860.0060.1075 Hydroxytryptamine 3B antagonist

0.107 0.004 DBMET00757

DBMET00757
0.1010.0260.1085 Hydroxytryptamine uptake inhibitor

0.108 0.024 DBMET00757

DBMET00757
0.0920.0180.1265 Hydroxytryptamine 2A agonist

0.126 0.008 DBMET00757

DBMET00757
0.0980.0260.0985 Hydroxytryptamine 7 antagonist

0.091 0.027 DBMET00757

0.0760.0140.0765 Hydroxytryptamine 1B agonist

0.059 0.028 DBMET00757

0.0850.0230.14Dopamine uptake inhibitor

0.14 0.011 DBMET00757

DBMET00757
0.0850.0240.085Adrenaline uptake inhibitor

0.081 0.026 DBMET00757

0.1020.0540.102Antihistaminic
0.0660.0180.09Nicotinic receptor alpha4 subunit antagonist

0.09 0.01 DBMET00757

DBMET00757
0.0690.0220.1155 Hydroxytryptamine 1A agonist

0.115 0.013 DBMET00757

DBMET00757
0.050.0050.077Dopamine D1 agonist

0.077 0.004 DBMET00757

DBMET00757
0.0890.0490.09Histamine H1 receptor antagonist

0.09 0.048 DBMET00757

DBMET00757
0.1190.0790.119Acetylcholinesterase inhibitor
0.0920.0530.092Acetylcholine agonist
0.0920.0530.092Histamine antagonist
0.0640.0260.096Sigma receptor antagonist

0.096 0.017 DBMET00757

DBMET00757
0.0620.0240.083Dopamine transporter inhibitor

0.083 0.016 DBMET00757

DBMET00757
0.0620.0280.079Opioid agonist

0.079 0.019 DBMET00757

DBMET00757
0.0570.0270.0865 Hydroxytryptamine 4 antagonist

0.086 0.011 DBMET00757

DBMET00757
0.0720.0470.072CXC chemokine receptor antagonist
0.0810.0560.098Acetylcholine nicotinic agonist

0.098 0.039 DBMET00757

DBMET00757
0.0370.0160.049CXC chemokine 3 receptor antagonist

0.049 0.01 DBMET00757

DBMET00757
0.0580.0370.0725 Hydroxytryptamine 3 antagonist

0.072 0.028 DBMET00757

DBMET00757
0.150.1290.533Anticonvulsant

0.533 0.01 DBMET00757

DBMET00757
0.0630.0420.063Acetylcholine M2 receptor antagonist
0.1250.1060.246NOS3 expression enhancer

0.246 0.027 DBMET00757

DBMET00757
0.0390.0210.064p53 inhibitor

0.064 0.007 DBMET00757

DBMET00757
0.0390.020.039Opioid delta receptor agonist

0.039 0.02 DBMET00757

0.1660.1490.166DNA damaging
0.0470.0310.078Opioid mu receptor agonist

0.078 0.018 DBMET00757

DBMET00757
0.0530.0380.094Nicotinic receptor alpha7 subunit antagonist

0.094 0.013 DBMET00757

DBMET00757
0.0520.0420.101Protein kinase C eta inhibitor

0.101 0.017 DBMET00757

DBMET00757
0.0420.0340.0765 Hydroxytryptamine 2C agonist

0.076 0.012 DBMET00757

DBMET00757
0.0350.030.058Somatostatin 1 antagonist

0.058 0.016 DBMET00757

DBMET00757
0.0260.0210.034Somatostatin 2 antagonist

0.034 0.019 DBMET00757

DBMET00757
0.0760.0740.076Ca(v)3.1 blocker
0.0380.0370.079Opioid kappa receptor agonist

0.079 0.013 DBMET00757

DBMET00757
0.070.0810.116Antineoplastic alkaloid

0.116 0.039 DBMET00757

DBMET00757
0.0290.0410.035Protein kinase C beta I inhibitor

0.035 0.018 DBMET00757

DBMET00757
0.0850.10.148Toll-Like receptor 4 antagonist

0.148 0.022 DBMET00757

DBMET00757
0.0090.0290.015NMDA receptor phencyclidine site antagonist

0.015 0.012 DBMET00757

DBMET00757
0.0250.0490.046Nicotinic receptor beta4 subunit antagonist

0.046 0.018 DBMET00757

DBMET00757
0.0390.0740.071Alpha 1 adrenoreceptor agonist

0.071 0.027 DBMET00757

DBMET00757
0.070.1270.162Adenylate cyclase inhibitor

0.162 0.037 DBMET00757

DBMET00757
0.1640.2220.415Vasodilator, peripheral

0.415 0.051 DBMET00757

DBMET00757
0.0480.1060.153Nicotinic alpha4beta2 receptor antagonist

0.153 0.007 DBMET00757

DBMET00757
0.0680.1320.079CC chemokine 5 receptor agonist

0.079 0.068 DBMET00757

DBMET00757
0.110.1790.185Antipruritic

0.185 0.06 DBMET00757

DBMET00757
0.0080.0870.039Somatostatin 5 antagonist

0.039 0.019 DBMET00757

DBMET00757
0.0560.1350.084Protein kinase C delta inhibitor

0.084 0.071 DBMET00757

DBMET00757
0.0190.0990.04511-Beta-hydroxysteroid dehydrogenase 1 inhibitor

0.045 0.034 DBMET00757

DBMET00757
0.0920.180.153MAP3K9 inhibitor

0.153 0.055 DBMET00757

DBMET00757
0.030.1290.0595 Hydroxytryptamine 3A antagonist

0.059 0.058 DBMET00757

DBMET00757
0.0150.1330.112NMDA 2A receptor antagonist

0.112 0.011 DBMET00757

DBMET00757
0.0310.150.088Nicotinic alpha3beta2 receptor antagonist

0.088 0.01 DBMET00757

DBMET00757
0.020.140.07Nicotinic receptor alpha3 subunit antagonist

0.07 0.015 DBMET00757

DBMET00757
0.0640.2330.123Neurotrophic factor

0.123 0.091 DBMET00757

DBMET00757
0.0460.230.112GABA C receptor antagonist

0.112 0.061 DBMET00757

DBMET00757
0.0240.2430.171NMDA receptor antagonist

0.171 0.019 DBMET00757

DBMET00757
0.1030.3310.339Immunosuppressant

0.339 0.093 DBMET00757

DBMET00757
0.0680.3010.14GABA C receptor rho-2 antagonist

0.14 0.088 DBMET00757

DBMET00757
0.0080.3150.08NMDA 2C receptor antagonist

0.08 0.025 DBMET00757

DBMET00757
0.0320.3440.108GABA C receptor rho-1 antagonist

0.108 0.052 DBMET00757

DBMET00757
0.0050.3250.115NMDA 2 receptor antagonist

0.115 0.025 DBMET00757

DBMET00757
0.0640.4220.171DNA synthesis inhibitor

0.171 0.166 DBMET00757

DBMET00757
0.120.5110.279Calcium channel L-type activator

0.279 0.175 DBMET00757

DBMET00757
0.0160.4390.123Glutamate receptor antagonist

0.123 0.071 DBMET00757

DBMET00757
0.0610.5090.219Antibacterial

0.219 0.208 DBMET00757

DBMET00757
0.0710.5360.229GABA C receptor rho-3 antagonist

0.229 0.174 DBMET00757

DBMET00757
0.0760.5790.184Tyrosine 3 hydroxylase inhibitor

0.184 0.168 DBMET00757

DBMET00757
0.0370.5540.224Transcription factor NF kappa B inhibitor

0.224 0.147 DBMET00757

DBMET00757
0.0310.6070.2Hypoxia-inducible factor 1 alpha inhibitor

0.2 0.152 DBMET00757

DBMET00757
0.0580.6530.339Antiinflammatory

0.339 0.181 DBMET00757

DBMET00757
0.0510.7090.136Ca2+-transporting ATPase inhibitor

0.136 0.088 DBMET00757

DBMET00757
0.0030.6680.041GABA uptake inhibitor

0.041 0.025 DBMET00757

DBMET00757
0.010.7590.038Glutamate (mGluR8) antagonist

0.038 0.019 DBMET00757

DBMET00757
0.0050.8220.099GABA C receptor agonist

0.099 0.068 DBMET00757

DBMET00757
Ext Pa Pi Pmax Activity Other Results ID Pa_max