Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.5930.0120.5935 Hydroxytryptamine release inhibitor

0.482 0.039 DBMET00415

0.5480.0040.548Protein kinase (CK1) inhibitor

0.352 0.012 DBMET00415

0.5280.0130.528MAP kinase kinase 6 inhibitor

0.44 0.038 DBMET00415

0.530.0160.53Nootropic

0.474 0.024 DBMET00415

0.5290.0190.529GABA C receptor rho-3 antagonist

0.513 0.022 DBMET00415

0.5020.0280.502Histamine release inhibitor

0.306 0.121 DBMET00415

0.5020.0330.502Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.464 0.052 DBMET00415

0.4590.0040.459GABA C receptor agonist

0.313 0.009 DBMET00415

0.4480.0020.448MAP kinase kinase 3 inhibitor

0.385 0.003 DBMET00415

0.4480.0040.448Histone deacetylase stimulant

0.132 0.013 DBMET00415

0.4480.0040.448Histone deacetylase SIRT1 stimulant

0.132 0.013 DBMET00415

0.4450.0040.445Glutamate (mGluR) agonist

0.215 0.008 DBMET00415

0.4040.0040.404Glutamate (mGluR) antagonist

0.209 0.009 DBMET00415

0.3970.0030.397Glutamate (mGluR group II) agonist

0.148 0.005 DBMET00415

0.3910.0030.391Glutamate (mGluR2) agonist

0.141 0.005 DBMET00415

0.3670.0060.367Glutamate receptor antagonist

0.224 0.02 DBMET00415

0.3730.0250.373Peroxidase inhibitor

0.311 0.035 DBMET00415

0.360.0150.36TRKC antagonist

0.156 0.096 DBMET00415

0.3480.0050.379Polo-like kinase-3 inhibitor

0.379 0.004 DBMET00415

DBMET00415
0.3440.0040.344Macrophage colony-stimulating factor 1 receptor antagonist

0.228 0.006 DBMET00415

0.3660.0330.366Superoxide dismutase inhibitor

0.258 0.069 DBMET00415

0.3550.0240.355Ca2+/calmodulin-dependent kinase I alpha inhibitor

0.295 0.041 DBMET00415

0.3160.0060.316Protein kinase (CaMK, MLCK, PhK, SNF, KIN, NIM1, MAPKAP, POLO, CHK, ULK, RSK-2nd domain) inhibitor

0.214 0.012 DBMET00415

0.3140.0060.314Histidine decarboxylase inhibitor

0.206 0.012 DBMET00415

0.3170.0140.317Protein kinase (CK1) gamma 3 inhibitor
0.3380.0390.338Insulysin inhibitor

0.312 0.052 DBMET00415

0.3030.0050.303Porphobilinogen synthase inhibitor

0.177 0.015 DBMET00415

0.3250.0270.325RNA-directed DNA polymerase inhibitor

0.276 0.038 DBMET00415

0.3160.0210.316Protein kinase C nu inhibitor

0.12 0.093 DBMET00415

0.2940.0040.388Nav1.8 sodium channel blocker

0.388 0.004 DBMET00415

DBMET00415
0.3120.0240.312MAP-kinase-activated kinase 5 inhibitor

0.286 0.038 DBMET00415

0.290.0140.29Nitric-oxide synthase stimulant

0.258 0.027 DBMET00415

0.2810.0070.281Check point kinase 2 inhibitor

0.206 0.015 DBMET00415

0.270.0060.27Protein kinase C mu inhibitor

0.201 0.012 DBMET00415

0.3020.040.302Anticonvulsant

0.177 0.102 DBMET00415

0.2670.0060.267Glutamate receptor agonist

0.097 0.039 DBMET00415

0.3010.0430.301DNA synthesis inhibitor

0.267 0.057 DBMET00415

0.2860.0310.286Dual specificity tyrosine-phosphorylation regulated kinase 3 inhibitor

0.163 0.107 DBMET00415

0.3240.070.324Calcium channel activator

0.252 0.145 DBMET00415

0.310.0570.31Ca2+/calmodulin-dependent kinase II alpha inhibitor

0.245 0.111 DBMET00415

0.2540.0090.254Histone deacetylase class III inhibitor

0.141 0.051 DBMET00415

0.2670.0250.267Protein kinase (CK1) gamma inhibitor
0.2580.0240.258Heat shock protein 90 alpha antagonist

0.138 0.1 DBMET00415

0.2440.0140.247Ferrochelatase inhibitor

0.247 0.014 DBMET00415

DBMET00415
0.2450.0210.245Protein kinase (CK1) gamma 2 inhibitor
0.2410.020.332Sodium channel blocker

0.332 0.008 DBMET00415

DBMET00415
0.2220.0090.253GABA C receptor antagonist

0.253 0.006 DBMET00415

DBMET00415
0.2180.0060.249GABA C receptor rho-1 antagonist

0.249 0.004 DBMET00415

DBMET00415
0.2150.0050.215Histone deacetylase SIRT2 inhibitor

0.104 0.026 DBMET00415

0.2480.0390.248LIM domain kinase 1 inhibitor

0.168 0.082 DBMET00415

0.2610.0540.261Ca2+/calmodulin-dependent protein kinase inhibitor

0.179 0.089 DBMET00415

0.2760.0690.289Aryl hydrocarbon receptor agonist

0.289 0.064 DBMET00415

DBMET00415
0.2990.0930.299Angiogenesis inhibitor
0.2270.0220.227Cyclin-dependent kinase 8 inhibitor

0.15 0.079 DBMET00415

0.2170.0120.217Beta amyloid protein antagonist

0.159 0.035 DBMET00415

0.2560.0510.288MAP kinase kinase 2 inhibitor

0.288 0.039 DBMET00415

DBMET00415
0.210.0060.21Alcohol oxidase inhibitor

0.093 0.02 DBMET00415

0.2260.0230.226Histone deacetylase SIRT1 inhibitor

0.142 0.068 DBMET00415

0.2290.0260.229Nav1.2 sodium channel blocker
0.2230.0220.231Sodium channel (voltage-gated) blocker

0.231 0.02 DBMET00415

DBMET00415
0.2330.0330.233Protein kinase (CK1) gamma 1 inhibitor
0.2660.0660.2665 Hydroxytryptamine uptake stimulant

0.225 0.11 DBMET00415

0.240.0440.24Neurotrophic factor enhancer

0.165 0.117 DBMET00415

0.2110.0160.211CF transmembrane conductance regulator agonist

0.17 0.047 DBMET00415

0.2560.0630.256Tyrosine 3 hydroxylase inhibitor

0.228 0.093 DBMET00415

0.2210.0290.221Heat shock protein 90 antagonist

0.137 0.089 DBMET00415

0.2050.0160.205Ca2+/calmodulin-dependent protein kinase kinase B inhibitor

0.187 0.027 DBMET00415

0.2180.0290.218Alpha-N-acetylglucosaminidase inhibitor

0.152 0.054 DBMET00415

0.210.0240.21GABA C receptor rho-2 antagonist

0.209 0.024 DBMET00415

0.220.0360.225 Hydroxytryptamine 3E antagonist

0.203 0.057 DBMET00415

0.1920.010.192Check point kinase 1 inhibitor

0.136 0.017 DBMET00415

0.2330.0540.233Interleukin-1 receptor-associated protein kinase 1 inhibitor
0.1860.0090.186I kappa B kinase inhibitor

0.112 0.031 DBMET00415

0.180.0050.18Lanosterol 14 alpha demethylase inhibitor

0.088 0.075 DBMET00415

0.180.0060.18I kappa B kinase 1 inhibitor
0.210.0370.21NOS3 expression enhancer
0.2410.070.241HERG channel blocker
0.2240.0540.224Ca2+/calmodulin-dependent kinase II gamma inhibitor

0.216 0.057 DBMET00415

0.180.0120.18Glutamate dehydrogenase inhibitor

0.175 0.012 DBMET00415

0.2570.090.257Ca(v)3.3 blocker
0.2180.0570.218I kappa B kinase epsilon inhibitor

0.217 0.058 DBMET00415

0.1730.0120.173Pim-3 kinase inhibitor

0.122 0.03 DBMET00415

0.1920.0330.192Cell wall synthesis inhibitor

0.138 0.077 DBMET00415

0.1910.0330.22TRKA antagonist

0.22 0.025 DBMET00415

DBMET00415
0.1770.0190.177Pim-1 kinase inhibitor

0.14 0.031 DBMET00415

0.1720.0160.172Alcohol dehydrogenase inhibitor

0.083 0.075 DBMET00415

0.1740.0190.174Adenylate kinase inhibitor

0.124 0.04 DBMET00415

0.1680.0140.168DOPA decarboxylase inhibitor

0.121 0.044 DBMET00415

0.1640.0120.164MAP kinase kinase 1 inhibitor

0.142 0.02 DBMET00415

0.2220.070.222Pyruvate kinase inhibitor
0.1850.0340.185Protein kinase (CK1) delta inhibitor
0.2190.0680.219Clk dual-specificity kinase inhibitor

0.215 0.071 DBMET00415

0.210.0610.21CDC-like kinase 2 inhibitor
0.1970.0510.197Succinate dehydrogenase inhibitor

0.165 0.087 DBMET00415

0.2260.0790.226Potassium channel (Voltage-sensitive) blocker
0.1810.0360.181MAP kinase kinase inhibitor

0.139 0.058 DBMET00415

0.2080.0640.22CDC-like kinase 4 inhibitor

0.22 0.058 DBMET00415

DBMET00415
0.1470.0050.147Polo-like kinase-2 inhibitor

0.103 0.023 DBMET00415

0.1470.0040.147Diacylglycerol O-acyltransferase 1 inhibitor

0.11 0.005 DBMET00415

0.1570.0140.157Polo-like kinase-1 inhibitor

0.115 0.033 DBMET00415

0.1510.0090.151Biliverdin reductase inhibitor

0.138 0.011 DBMET00415

0.1870.0460.201Tyrosine-protein kinase receptor antagonist

0.201 0.04 DBMET00415

DBMET00415
0.1950.0550.195Anticoagulant

0.131 0.099 DBMET00415

0.1590.0210.159Creatine kinase inhibitor

0.102 0.057 DBMET00415

0.140.0040.14Glutamate (mGluR1a) antagonist

0.061 0.014 DBMET00415

0.140.0040.14S-adenosyl-L-methionine decarboxylase inhibitor

0.118 0.006 DBMET00415

0.1520.0160.152CYP2A6 inhibitor
0.2290.0930.229DNA damaging
0.1640.0320.164Granulocyte macrophage colony stimulating factor antagonist

0.114 0.058 DBMET00415

0.1490.0170.149Acetylcholine release stimulant
0.2080.0760.208Psychostimulant
0.1720.0410.172MAP kinase 3 inhibitor

0.158 0.056 DBMET00415

0.2560.1280.256Vasodilator, coronary
0.130.0040.13Glutamate (mGluR group II) antagonist

0.043 0.021 DBMET00415

0.1410.0150.141Tyk2 inhibitor

0.073 0.04 DBMET00415

0.2510.1250.251Antithrombotic
0.1970.0720.197Focal adhesion kinase 2 inhibitor

0.171 0.099 DBMET00415

0.1980.0760.198Death-associated protein kinase 3 inhibitor

0.146 0.129 DBMET00415

0.1290.0070.129I kappa B kinase 2 inhibitor

0.084 0.02 DBMET00415

0.2480.1270.248Cholesterol antagonist
0.2050.0840.205EphB2 antagonist
0.1510.0310.151Protein kinase C gamma inhibitor

0.125 0.048 DBMET00415

0.1250.0060.125Histone deacetylase SIRT3 inhibitor

0.086 0.014 DBMET00415

0.1380.020.145Rho-associated kinase II inhibitor

0.145 0.018 DBMET00415

DBMET00415
0.1520.0340.152MAP kinase kinase kinase inhibitor

0.094 0.072 DBMET00415

0.190.0720.267Tyrosine kinase inhibitor

0.267 0.05 DBMET00415

DBMET00415
0.1260.0090.126Secretase beta inhibitor

0.121 0.01 DBMET00415

0.1510.0350.151GABA receptor agonist

0.119 0.057 DBMET00415

0.1250.010.125Glutamate (mGluR1) antagonist
0.2210.1060.2215 Hydroxytryptamine release stimulant

0.179 0.142 DBMET00415

0.1250.0110.125Transforming growth factor antagonist
0.2080.0940.208Antiamyloidogenic
0.1720.0590.172Neurotensin receptor agonist

0.15 0.101 DBMET00415

0.1180.0050.118Exportin-1 inhibitor

0.064 0.06 DBMET00415

0.1330.020.151MAP-kinase-activated kinase inhibitor

0.151 0.014 DBMET00415

DBMET00415
0.1150.0040.115Glutamate (mGluR2) antagonist

0.032 0.018 DBMET00415

0.1410.030.141CDK2/cyclin A inhibitor

0.134 0.033 DBMET00415

0.1440.0330.144Carbonic anhydrase XV inhibitor
0.1250.0150.134Janus tyrosine kinase 1 inhibitor

0.134 0.012 DBMET00415

DBMET00415
0.2040.0940.204Peptidyltransferase inhibitor

0.172 0.142 DBMET00415

0.1680.060.168Dual specificity tyrosine-phosphorylation regulated kinase 1B inhibitor
0.1710.0640.171Dual specificity tyrosine-phosphorylation-regulated kinase 4 inhibitor
0.2170.1120.2175 Hydroxytryptamine 1E antagonist
0.1410.0370.141CC chemokine 6 receptor antagonist

0.132 0.064 DBMET00415

0.1440.040.144Cyclin-dependent kinase 2 inhibitor

0.114 0.057 DBMET00415

0.1160.0130.116Human rhinovirus A protease inhibitor

0.062 0.033 DBMET00415

0.1180.0160.118Carbamoyl phosphate synthetase inhibitor

0.095 0.022 DBMET00415

0.1750.0740.175MAP kinase kinase 5 inhibitor

0.163 0.105 DBMET00415

0.1730.0720.1733C-like protease (Human coronavirus) inhibitor
0.1410.040.141DNA repair enzyme inhibitor

0.122 0.069 DBMET00415

0.1410.0410.1415 Hydroxytryptamine 3A agonist

0.132 0.047 DBMET00415

0.1870.0890.187Histone acetyltransferase inhibitor
0.130.0320.13Folate antagonist
0.1280.0310.128Interleukin-1 receptor-associated protein kinase 4 inhibitor

0.092 0.054 DBMET00415

0.1130.0160.113MAP3K7 inhibitor

0.085 0.034 DBMET00415

0.1020.0060.102Corticotropin releasing factor 2 receptor antagonist

0.078 0.019 DBMET00415

0.1070.0110.107Protein kinase C beta inhibitor

0.078 0.033 DBMET00415

0.0980.0040.098Dopamine beta hydroxylase inhibitor

0.066 0.01 DBMET00415

0.10.0080.1Aconitate hydratase inhibitor

0.065 0.022 DBMET00415

0.130.0380.13MAP kinase 8 inhibitor
0.110.0190.121CDC7 inhibitor

0.121 0.015 DBMET00415

DBMET00415
0.0960.0040.096Protein kinase (CK1) epsilon inhibitor

0.052 0.011 DBMET00415

0.1130.0220.113Glutamate (mGluR group I) antagonist
0.1290.0380.129Carbonic anhydrase III inhibitor
0.1170.0260.117Phosphofructokinase-1 inhibitor

0.079 0.042 DBMET00415

0.1320.0420.132Transcription factor STAT6 inhibitor

0.105 0.094 DBMET00415

0.1380.0490.138Protein kinase (CK2) alpha inhibitor
0.0980.010.098Glutamate (mGluR group III) agonist
0.0930.0050.093Histamine H2 receptor agonist

0.088 0.005 DBMET00415

0.1520.0640.152Ca2+/calmodulin-dependent kinase II delta inhibitor

0.12 0.084 DBMET00415

0.1520.0650.152Activin receptor-like kinase 2 inhibitor

0.131 0.083 DBMET00415

0.1050.0190.105Transforming growth factor beta 3 antagonist
0.1090.0240.132MAP-kinase-activated kinase 2 inhibitor

0.132 0.016 DBMET00415

DBMET00415
0.0970.0120.097Glutamate (mGluR6) antagonist

0.072 0.036 DBMET00415

0.0980.0130.098Protein kinase C epsilon inhibitor

0.059 0.032 DBMET00415

0.1160.0320.116Histamine N-methyltransferase inhibitor

0.106 0.04 DBMET00415

0.1510.0670.199Hemostatic

0.199 0.033 DBMET00415

DBMET00415
0.0920.0090.092Stearoyl-CoA desaturase inhibitor

0.044 0.03 DBMET00415

0.0930.0090.093Glutamate (mGluR group I) agonist

0.042 0.04 DBMET00415

0.1070.0240.107Aminopeptidase I inhibitor

0.08 0.042 DBMET00415

0.1430.0620.143Ca2+-transporting ATPase inhibitor

0.132 0.108 DBMET00415

0.2130.1320.214Ca2+/calmodulin-dependent kinase IV inhibitor

0.214 0.13 DBMET00415

DBMET00415
0.1130.0330.113NADH dehydrogenase inhibitor

0.102 0.042 DBMET00415

0.090.010.096Diacylglycerol O-acyltransferase inhibitor

0.096 0.008 DBMET00415

DBMET00415
0.1860.1070.186Dyrk kinase inhibitor
0.1350.0560.135Alkylator
0.0950.0160.095Pim-2 kinase inhibitor

0.069 0.024 DBMET00415

0.1080.0310.108Inducible nitric-oxide synthase inhibitor
0.120.0430.12UDP-glucose 4-epimerase inhibitor

0.114 0.048 DBMET00415

0.1050.0280.105Granulocyte macrophage colony stimulating factor agonist

0.089 0.053 DBMET00415

0.1130.0370.113Triose-phosphate isomerase inhibitor

0.091 0.058 DBMET00415

0.2520.1750.252Antibacterial

0.231 0.195 DBMET00415

0.2060.130.206Transcription factor STAT inhibitor
0.1360.060.136Antibacterial (Helicobacter pylori)
0.0990.0230.099Nav1.7 sodium channel blocker

0.074 0.039 DBMET00415

0.1060.0320.112Rho-associated kinase inhibitor

0.112 0.029 DBMET00415

DBMET00415
0.0920.0180.092Aryl hydrocarbon receptor antagonist
0.1610.0870.161Phospholipase C inhibitor
0.0880.0150.088AMPA receptor antagonist

0.044 0.038 DBMET00415

0.0910.0180.091Ornithine carbamoyltransferase inhibitor

0.048 0.041 DBMET00415

0.0930.020.093MAP kinase kinase 7 inhibitor

0.09 0.025 DBMET00415

0.1020.0290.102Glutamate decarboxylase inhibitor
0.0810.0090.081Adenosine deaminase inhibitor

0.07 0.013 DBMET00415

0.0890.0180.089Bruton tyrosine kinase inhibitor

0.054 0.042 DBMET00415

0.1390.0680.139Cyclin-dependent kinase 7 inhibitor
0.1340.0630.134Cyclooxygenase 3 inhibitor
0.0870.0170.087Mannitol-1-phosphate 5-dehydrogenase inhibitor

0.073 0.024 DBMET00415

0.1220.0520.122Nav1.5 sodium channel blocker
0.0970.0270.097Phenylalanine 4-hydroxylase inhibitor

0.081 0.037 DBMET00415

0.1040.0340.104GABA A receptor agonist

0.086 0.053 DBMET00415

0.140.070.14Cytokine production inhibitor
0.0880.0190.088Glutamate (mGluR7) antagonist

0.065 0.053 DBMET00415

0.0850.0160.085Fatty acid synthase inhibitor
0.1940.1260.194Interleukin agonist

0.187 0.133 DBMET00415

0.0720.0040.072Histamine H1 receptor agonist

0.061 0.008 DBMET00415

0.1120.0440.112Nitric-oxide synthase inhibitor
0.120.0520.12Aminopeptidase B inhibitor

0.084 0.078 DBMET00415

0.090.0220.09Protein kinase C iota inhibitor
0.110.0420.11Glutamate (mGluR7) agonist
0.0890.0220.089Carbonic anhydrase stimulant

0.059 0.041 DBMET00415

0.0850.020.085Acyl-CoA dehydrogenase inhibitor

0.06 0.033 DBMET00415

0.0990.0350.099mTOR complex 2 inhibitor
0.0970.0330.097Nicotinic alpha4beta2 receptor antagonist
0.0980.0340.098Phosphodiesterase XI inhibitor
0.0980.0340.098Phosphodiesterase 11A inhibitor
0.0920.0290.092Phosphodiesterase 4B inhibitor
0.0780.0150.078Transforming growth factor beta 1 antagonist
0.1410.0780.148Adenylate cyclase stimulant

0.148 0.067 DBMET00415

DBMET00415
0.2170.1540.217Transcription factor NF kappa B inhibitor
0.0930.030.093Protein kinase B beta inhibitor

0.069 0.059 DBMET00415

0.1270.0650.127TRKB antagonist
0.1180.0550.118Activin receptor-like kinase 4 inhibitor
0.1020.040.102Bcr-Abl kinase inhibitor
0.1440.0820.144Diuretic
0.1240.0620.124Proteasome inhibitor
0.0880.0280.088MAP kinase kinase 8 inhibitor
0.0910.0310.091Benzodiazepine agonist
0.1380.0790.138CDC-like kinase 1 inhibitor
0.0830.0240.092Argininosuccinate synthase inhibitor

0.092 0.021 DBMET00415

DBMET00415
0.0660.0070.066Nerve growth factor antagonist
0.1350.0770.148Ribosomal protein S6 kinase inhibitor

0.148 0.066 DBMET00415

DBMET00415
0.1060.0480.106UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor

0.098 0.056 DBMET00415

0.1540.0960.154Tumour necrosis factor antagonist
0.1360.0790.136Vascular endothelial growth factor 3 antagonist
0.1110.0540.111Protein kinase (CK2) inhibitor
0.1680.1110.168Angiogenesis stimulant
0.0960.040.096Hematopoietic
0.1180.0630.118Glycogen synthase kinase-3 beta inhibitor
0.110.0550.11Urease inhibitor
0.0730.0180.073Histamine agonist

0.065 0.023 DBMET00415

0.0930.0390.093D-Ala-D-Ala ligase inhibitor

0.081 0.066 DBMET00415

0.0680.0140.068Glutamate (mGluR5) agonist
0.0610.0080.061Glutamate (mGluR4) agonist

0.031 0.029 DBMET00415

0.0580.0050.058Transforming growth factor beta 2 antagonist
0.0710.0180.071Epithelial sodium channel blocker
0.0820.0290.082Potassium channel (Tandem pore domain) blocker
0.0650.0120.068AICAR transformylase inhibitor

0.068 0.01 DBMET00415

DBMET00415
0.0820.0290.0825 Hydroxytryptamine 3A antagonist

0.059 0.057 DBMET00415

0.1370.0850.137Heat shock protein 70 antagonist
0.1390.0870.139MAP kinase kinase 4 inhibitor
0.110.0580.11Mediator release inhibitor
0.0620.0110.062Kainate receptor 2 antagonist

0.033 0.027 DBMET00415

0.0930.0430.093Histamine H2 receptor antagonist

0.083 0.06 DBMET00415

0.0620.0120.062Geranyltranstransferase inhibitor
0.0720.0230.072Bombesin 3 receptor antagonist
0.0830.0350.083GABA B receptor agonist
0.1080.0610.108AMP-activated protein kinase stimulant

0.096 0.076 DBMET00415

0.0650.0180.065Farnesyltransferase inhibitor
0.1690.1230.169Cyclic AMP phosphodiesterase inhibitor
0.0840.0380.084Syk tyrosine kinase inhibitor

0.076 0.043 DBMET00415

0.0870.0410.087Keratolytic
0.0670.0210.067Chemokine receptor agonist
0.1110.0660.111Cystathionine beta-synthase inhibitor
0.130.0860.13Mannose-6-phosphate isomerase inhibitor
0.0660.0230.072Antimetabolite

0.072 0.021 DBMET00415

DBMET00415
0.1530.1110.153Anesthetic general
0.0620.0190.062HCV NS3/NS4A protease inhibitor
0.1090.0660.109Mucolytic
0.1110.0690.111Glycogen synthase kinase-3 inhibitor
0.1620.1220.162Glyceraldehyde-3-phosphate dehydrogenase inhibitor
0.0560.0150.056Glutamate (mGluR group III) antagonist
0.0540.0140.054Alpha 1d adrenoreceptor agonist
0.0670.0270.067Cyclin A1 inhibitor

0.067 0.026 DBMET00415

0.0530.0140.053Factor XIIIa inhibitor
0.1220.0830.122Glycogen synthase kinase-3 alpha inhibitor
0.1860.1470.186Neuropeptide Y2 antagonist
0.0430.0050.043Purinergic P2Y15 antagonist

0.035 0.01 DBMET00415

0.0780.0410.078Protein kinase B alpha inhibitor

0.061 0.06 DBMET00415

0.1170.0810.168RET inhibitor

0.168 0.053 DBMET00415

DBMET00415
0.1250.0890.125Nav1.6 sodium channel blocker
0.0720.0370.072Cyclin A2 inhibitor
0.0940.060.094HIV-1 integrase (Overall Integration) inhibitor
0.0450.0110.045AMPA 3 receptor antagonist
0.0750.0410.075Carbonic anhydrase VA inhibitor
0.130.0970.13Thiol protease inhibitor
0.0960.0630.096Electrolyte absorption antagonist
0.1750.1420.175Calpain inhibitor
0.0380.0050.038Glucosylceramidase stimulant
0.070.0370.07Cyclin A inhibitor
0.0740.0420.074Neuronal nicotinic receptor antagonist

0.066 0.048 DBMET00415

0.1360.1050.136Arachidonic acid antagonist
0.0690.0380.069Protease 3C (Human rhinovirus) inhibitor

0.058 0.057 DBMET00415

0.0470.0170.047Diamine oxidase inhibitor

0.033 0.032 DBMET00415

0.0440.0130.044ATM kinase inhibitor
0.0790.0480.141Janus tyrosine kinase 2 inhibitor

0.141 0.023 DBMET00415

DBMET00415
0.050.0210.05Glutamate (mGluR4) antagonist
0.0410.0120.041ATR kinase inhibitor

0.036 0.016 DBMET00415

0.0450.0160.045Glutamate (mGluR8) agonist
0.0370.0080.037MAP3K8 inhibitor
0.0650.0360.065Neuropeptide agonist
0.0460.0180.046Vascular adhesion protein 1 inhibitor
0.0380.0090.038Nicotinic alpha4beta2 receptor agonist
0.0740.0460.074Glycine receptor agonist
0.0440.0160.044Glutamate (mGluR3) antagonist
0.0320.0040.032Complement factor D inhibitor

0.02 0.009 DBMET00415

0.1590.1310.159Aldehyde oxidase inhibitor
0.070.0430.07Acetylcholine M5 receptor agonist
0.0380.0110.038Nicotinic alpha3beta4 receptor agonist
0.0810.0550.081Acetylcholine nicotinic agonist
0.0710.0440.071Sirtuin 1 inhibitor

0.069 0.045 DBMET00415

0.0410.0140.041Tryptophan 5 hydroxylase inhibitor

0.035 0.026 DBMET00415

0.0340.0080.034Glutamate (mGluR1) agonist

0.024 0.019 DBMET00415

0.0340.0070.034Glutamate (mGluR1a) agonist
0.0540.0280.054Bombesin 2 receptor antagonist
0.0630.0370.063Potassium channel intermediate-conductance Ca-activated blocker
0.130.1040.13Hexokinase inhibitor
0.1010.0750.101Nav1.4 sodium channel blocker
0.1080.0830.108Cyclin-dependent kinase inhibitor
0.0380.0130.091Poly(ADP-ribose) polymerase 2 inhibitor

0.091 0.005 DBMET00415

DBMET00415
0.0310.0060.031ICAM 1 antagonist
0.0810.0560.081Histamine H1 receptor antagonist
0.0610.0380.061Heat shock protein 90 beta antagonist
0.0440.0210.044Membrane dipeptidase inhibitor

0.039 0.027 DBMET00415

0.0710.0480.071Amidase inhibitor
0.0650.0420.0655 Hydroxytryptamine 3 agonist
0.050.0270.05CC chemokine 4 receptor antagonist
0.0560.0340.056Lysine-specific demethylase 1A inhibitor
0.0440.0220.044Kainate receptor agonist

0.042 0.027 DBMET00415

0.0320.010.032Hedgehog signaling activator
0.1280.1060.128Pregnane X receptor agonist
0.1160.0940.116Interleukin 1 antagonist
0.0350.0130.035CDK4/cyclin D3 inhibitor
0.0470.0250.047Dipeptidyl peptidase IV inhibitor
0.0550.0330.055Dipeptidyl peptidase inhibitor
0.0420.020.042DNA gyrase subunit B inhibitor

0.034 0.033 DBMET00415

0.0830.0620.0963C-Like protease (SARS coronavirus) inhibitor

0.096 0.037 DBMET00415

DBMET00415
0.0570.0360.057Ribonucleoside-diphosphate reductase inhibitor
0.0670.0460.067Potassium channel (ATP-sensitive) blocker
0.0360.0160.036Methionyl aminopeptidase 1 inhibitor
0.0370.0170.037HCV polyprotein inhibitor
0.0660.0460.066Carbonic anhydrase V inhibitor
0.0480.0290.048Benzodiazepine inverse agonist
0.0570.0380.057Ribonucleotide reductase inhibitor
0.0810.0610.081Phosphodiesterase IV inhibitor
0.0380.0190.038CXC chemokine receptor agonist
0.0420.0230.042MAP3K5 inhibitor
0.0360.0170.036AMPA 1 receptor antagonist
0.1270.1080.127Sphingosine 1-phosphate receptor 5 antagonist
0.0490.0310.049Glucose-6-phosphate isomerase inhibitor
0.0850.0670.085Aminoacyl-tRNA synthetase inhibitor
0.060.0430.06Purinergic P2X1 antagonist
0.0430.0260.043Kainate receptor antagonist
0.0350.0190.035Protein kinase (CK2) beta inhibitor

0.031 0.03 DBMET00415

0.0490.0330.049Cytokine production stimulant
0.0210.0050.021CDK2/cyclin A3 inhibitor

0.017 0.01 DBMET00415

0.0870.0710.087Protein kinase C zeta inhibitor
0.0580.0430.058Bombesin 1 receptor agonist

0.055 0.047 DBMET00415

0.0310.0170.085Histamine H3 receptor agonist

0.085 0.007 DBMET00415

DBMET00415
0.0580.0430.058Cyclin-dependent kinase 6 inhibitor
0.0370.0220.037Calcitonin receptor agonist
0.0330.0190.033Acetylcholine M4 receptor agonist
0.0360.0220.036Fumarate hydratase inhibitor
0.0810.0670.081Ornithine decarboxylase inhibitor
0.0270.0130.027Complement factor 1s inhibitor
0.0590.0440.059Alpha 2 adrenoreceptor agonist
0.0550.0420.055Xanthine dehydrogenase inhibitor
0.0230.0090.023Toll-Like receptor 8 agonist
0.0580.0450.058Cyclin D1 inhibitor
0.1040.0910.104Aldehyde dehydrogenase inhibitor

0.1 0.098 DBMET00415

0.0750.0630.075Leucine-rich repeat kinase 2 inhibitor
0.0230.010.023Factor XIII inhibitor
0.0440.0320.118Poly(ADP-ribose) polymerase inhibitor

0.118 0.006 DBMET00415

DBMET00415
0.0620.050.062Histone deacetylase inhibitor
0.0680.0570.068Phospholipase D inhibitor
0.0410.030.0413-Hydroxyanthranilate 3,4-dioxygenase inhibitor
0.0390.0290.039VCAM-1 antagonist
0.0440.0340.044Factor Xa inhibitor
0.0540.0440.054Immunoglobulin Fc receptor antagonist
0.0390.0290.039VCAM antagonist
0.030.020.03AMPA 2 receptor antagonist
0.0220.0120.022Hexokinase stimulant
0.1450.1350.145Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor
0.0730.0640.073Acetylcholine nicotinic antagonist
0.1830.1740.228Gastrin inhibitor

0.228 0.108 DBMET00415

DBMET00415
0.020.0110.02Cyclin T1 inhibitor
0.0520.0430.052Thromboxane synthase inhibitor
0.0180.0090.018Nicotinic alpha4 receptor agonist
0.050.0410.05Toll-Like receptor 8 antagonist
0.0310.0220.031Potassium channel small-conductance Ca-activated activator
0.1830.1750.187Hypoxia-inducible factor 1 alpha inhibitor

0.187 0.168 DBMET00415

DBMET00415
0.0680.060.068Rho-associated kinase I inhibitor
0.0520.0450.052MAP kinase kinase 9 inhibitor
0.0180.010.018CC chemokine 9 receptor antagonist
0.0320.0250.032Plasma kallikrein inhibitor
0.0260.0190.026Thymidine phosphorylase inhibitor
0.0460.0390.046Potassium channel (Inward rectifier) blocker
0.0430.0370.043Thymidylate synthase inhibitor
0.010.0030.01CC chemokine 6 receptor agonist

0.006 0.005 DBMET00415

0.0770.070.077Acetylcholine agonist
0.0880.0810.088Gastric antisecretory
0.0270.020.02711-Beta-hydroxysteroid dehydrogenase 2 inhibitor
0.0350.0290.035Melanocortin 1 antagonist
0.0270.0210.027Thrombin receptor antagonist
0.1760.170.176Transcription factor STAT3 inhibitor
0.0850.080.085Interleukin 1 beta converting enzyme inhibitor
0.1040.0990.104Cathepsin H inhibitor
0.0260.0210.028Hypoxanthine phosphoribosyltransferase inhibitor

0.028 0.019 DBMET00415

DBMET00415
0.0340.0290.034Inosine monophosphate dehydrogenase inhibitor
0.0450.040.045Adenosine A2b receptor antagonist
0.070.0650.071Fibroblast growth factor 3 antagonist

0.071 0.064 DBMET00415

DBMET00415
0.0780.0740.281Protein kinase (Mos, Mil/Raf, MEKK, RIPK, TESK, LIMK, IRAK, ILK, Activin/TGF-beta) inhibitor

0.281 0.01 DBMET00415

DBMET00415
0.020.0160.02Geranylgeranyltransferase I inhibitor
0.0880.0840.088Falcipain 3 inhibitor
0.0950.090.095Protein-tyrosine kinase (PTK, not ETK, WZC) inhibitor
0.0690.0650.069Phosphodiesterase VI inhibitor
0.0210.0170.021Geranylgeranyltransferase inhibitor
0.0940.090.094Abl kinase inhibitor
0.0290.0250.029Endothelial nitric-oxide synthase inhibitor
0.1450.1410.145Potassium channel blocker
0.0260.0220.026Protocollagen prolyl hydroxylase inhibitor
0.0490.0460.049Carbonic anhydrase VB inhibitor
0.0580.0550.058Phosphodiesterase 1C inhibitor
0.0550.0520.055Gonadotropin-releasing hormone receptor agonist
0.0130.010.0131-Deoxy-D-xylulose-5-phosphate reductoisomerase inhibitor
0.0140.0120.014Egl nine homolog 1 inhibitor
0.0170.0150.017Histamine H4 receptor agonist
0.1040.1020.104Phosphodiesterase inhibitor
0.2010.20.539Toll-Like receptor agonist

0.539 0.025 DBMET00415

DBMET00415
0.0250.0240.025Myristoyl transferase inhibitor
0.10.0980.1Nav1.3 sodium channel blocker
0.0480.0470.048Alpha-mannosidase inhibitor
0.0930.0920.093Aurora-B kinase inhibitor
0.0480.0470.048Nicotinic neuronal receptor agonist
0.0140.0130.014Dipeptidyl peptidase IX inhibitor
0.0710.070.071Protein kinase A inhibitor
0.0240.0230.024Lysine carboxypeptidase inhibitor
0.0810.080.081Prolactin inhibitor
0.0330.0340.083Poly(ADP-ribose) polymerase 1 inhibitor

0.083 0.009 DBMET00415

DBMET00415
0.010.0110.011Purine nucleoside phosphorylase inhibitor

0.011 0.009 DBMET00415

DBMET00415
0.0770.0990.088Insulin receptor antagonist

0.088 0.08 DBMET00415

DBMET00415
0.190.2140.532Toll-Like receptor 7 agonist

0.532 0.026 DBMET00415

DBMET00415
0.0250.050.047Carbonic anhydrase I stimulant

0.047 0.018 DBMET00415

DBMET00415
0.1490.1770.208Cardiotonic

0.208 0.111 DBMET00415

DBMET00415
0.040.0730.053Carbonic anhydrase II stimulant

0.053 0.034 DBMET00415

DBMET00415
0.0490.0830.248Raf kinase inhibitor

0.248 0.009 DBMET00415

DBMET00415
0.1080.1740.411Interleukin antagonist

0.411 0.029 DBMET00415

DBMET00415
0.1570.2310.24Vasodilator, peripheral

0.24 0.135 DBMET00415

DBMET00415
0.0480.1250.077ALK inhibitor

0.077 0.063 DBMET00415

DBMET00415
0.0210.1080.037Somatostatin 4 agonist

0.037 0.026 DBMET00415

DBMET00415
0.0630.1620.343MAP kinase 12 inhibitor

0.343 0.005 DBMET00415

DBMET00415
0.0360.1370.069CXC chemokine receptor antagonist

0.069 0.051 DBMET00415

DBMET00415
0.0230.1260.208Raf kinase B inhibitor

0.208 0.009 DBMET00415

DBMET00415
0.1860.2980.292Calcium channel L-type activator

0.292 0.164 DBMET00415

DBMET00415
0.0410.1620.121Tyrosine-protein kinase receptor FLT3 inhibitor

0.121 0.067 DBMET00415

DBMET00415
0.0350.160.233Proto-oncogene tyrosine-protein kinase c-hck inhibitor

0.233 0.004 DBMET00415

DBMET00415
0.0610.2120.15Src kinase inhibitor

0.15 0.083 DBMET00415

DBMET00415
0.0580.2220.158Alpha 2d adrenoreceptor antagonist

0.158 0.007 DBMET00415

DBMET00415
0.150.3590.315Cyclophilin D inhibitor

0.315 0.149 DBMET00415

DBMET00415
0.0060.2840.03Alpha 2d adrenoreceptor agonist

0.03 0.009 DBMET00415

DBMET00415
0.0210.3160.123c-Src kinase inhibitor

0.123 0.073 DBMET00415

DBMET00415
0.0390.4710.162Vasodilator

0.162 0.14 DBMET00415

DBMET00415
0.0250.580.659Interleukin 5 antagonist

0.659 0.002 DBMET00415

DBMET00415
0.0020.8350.02Thyroid hormone alpha agonist

0.02 0.007 DBMET00415

DBMET00415
0.0020.920.02Thyroid hormone alpha antagonist

0.02 0.008 DBMET00415

DBMET00415
Ext Pa Pi Pmax Activity Other Results ID Pa_max