Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.6880.0020.688NMDA 2B receptor antagonist

0.065 0.028 DBMET00327

0.6890.0040.689Glutamate receptor antagonist

0.472 0.005 DBMET00327

0.6410.020.641Analgesic
0.620.0040.62NMDA receptor antagonist

0.412 0.004 DBMET00327

0.5750.0150.5755 Hydroxytryptamine release inhibitor

0.488 0.036 DBMET00327

0.4730.0040.473NMDA 2 receptor antagonist
0.4810.0310.481GABA C receptor rho-3 antagonist

0.462 0.037 DBMET00327

0.4060.0040.406ATPase inhibitor

0.172 0.068 DBMET00327

0.4020.0090.402Amylase inhibitor

0.225 0.036 DBMET00327

0.3810.0040.381Autotaxin inhibitor
0.4710.10.471Antiinflammatory
0.3680.0040.368Dopamine D2 agonist
0.420.0650.42Histamine release inhibitor

0.394 0.079 DBMET00327

0.3960.0480.424Aldehyde oxidase inhibitor

0.424 0.044 DBMET00327

DBMET00327
0.3770.0430.417Lipoxygenase inhibitor

0.417 0.033 DBMET00327

DBMET00327
0.3270.0090.336Alkaline phosphatase inhibitor

0.336 0.008 DBMET00327

DBMET00327
0.320.0040.32NMDA 2C receptor antagonist

0.061 0.043 DBMET00327

0.3240.0270.324RNA-directed DNA polymerase inhibitor

0.254 0.047 DBMET00327

0.3040.0170.304Cyclooxygenase inhibitor

0.273 0.022 DBMET00327

0.360.0810.36Calpain 2 inhibitor
0.2840.0070.284Nav1.6 sodium channel blocker
0.2710.0040.271Mineralocorticoid receptor antagonist
0.2830.0250.283Diuretic
0.2950.0420.295Anticonvulsant
0.2550.0020.283Kynurenine 3 monooxygenase inhibitor

0.283 0.002 DBMET00327

DBMET00327
0.2970.0460.3145 Hydroxytryptamine uptake stimulant

0.314 0.038 DBMET00327

DBMET00327
0.2580.0070.258HIV-1 reverse transcriptase inhibitor
0.2570.0130.2575 Hydroxytryptamine 3E antagonist
0.2620.020.262Hemostatic
0.2460.0050.246Macrophage migration inhibitory factor inhibitor

0.229 0.006 DBMET00327

0.3060.0680.3065 Hydroxytryptamine release stimulant
0.2390.0070.239Dopamine agonist
0.2720.0440.272Ca2+/calmodulin-dependent kinase II beta inhibitor
0.2490.0250.249Antipruritic
0.2410.0210.241Insulin secretagoues
0.2920.0730.292Spasmolytic
0.2240.010.224Potassium channel (Ca-activated) activator

0.079 0.077 DBMET00327

0.2140.0070.214Inducible nitric-oxide synthase inhibitor

0.154 0.015 DBMET00327

0.2490.0450.249Ca2+/calmodulin-dependent kinase II gamma inhibitor
0.2040.0060.204Potassium channel large-conductance Ca-activated activator
0.3140.1250.314Antibacterial

0.232 0.194 DBMET00327

0.2220.0340.254Succinate dehydrogenase inhibitor

0.254 0.021 DBMET00327

DBMET00327
0.2590.0760.259Cardiotonic
0.2340.0530.234Dual specificity tyrosine-phosphorylation regulated kinase 3 inhibitor
0.1820.0050.352NMDA receptor subunit 3B antagonist

0.352 0.003 DBMET00327

DBMET00327
0.2260.0540.226Neurotrophic factor enhancer

0.196 0.08 DBMET00327

0.2780.1070.278Vasodilator, coronary
0.2110.0460.2113C-like protease (Human coronavirus) inhibitor
0.1750.0120.175Electrolyte absorption antagonist

0.132 0.028 DBMET00327

0.1690.0160.169Nitric-oxide synthase inhibitor

0.144 0.025 DBMET00327

0.1680.0160.168Phosphodiesterase 7B inhibitor
0.3260.1790.326Ca2+/calmodulin-dependent protein kinase kinase A inhibitor
0.1490.0050.1495 Hydroxytryptamine 2A agonist
0.2280.0850.228DNA synthesis inhibitor

0.227 0.086 DBMET00327

0.1570.0160.157Acetylcholine M3 receptor agonist
0.1790.0380.179Sodium channel (voltage-gated) blocker
0.1480.0070.148NMDA 2A receptor antagonist
0.2110.0720.225Nitric-oxide synthase stimulant

0.225 0.054 DBMET00327

DBMET00327
0.1440.0070.144Kallikrein 1 inhibitor
0.1620.030.162GABA receptor agonist
0.250.1180.25Thyroid hormone beta antagonist
0.1320.0040.132Factor XIa inhibitor
0.1610.0340.161Alpha 2b adrenoreceptor antagonist

0.156 0.036 DBMET00327

0.1430.0170.143MAP-kinase-activated kinase inhibitor
0.2480.1250.248Thyroid hormone antagonist
0.1360.0150.136MAP-kinase-activated kinase 2 inhibitor
0.1480.0270.148UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor

0.083 0.075 DBMET00327

0.1690.0520.169GABA C receptor rho-2 antagonist

0.152 0.072 DBMET00327

0.1430.0260.143DNA directed RNA polymerase inhibitor
0.1230.0060.251NMDA receptor subunit 3A antagonist

0.251 0.004 DBMET00327

DBMET00327
0.220.1040.224Tyrosine 3 hydroxylase inhibitor

0.224 0.097 DBMET00327

DBMET00327
0.1240.0090.124Acetylcholine M5 receptor agonist
0.1310.0170.131Bromodomain-containing protein 2 inhibitor
0.1220.0080.122NMDA receptor glycine site agonist
0.2550.1410.255Calcium channel activator
0.1220.010.122Alpha 2 adrenoreceptor agonist
0.1180.0070.118Phospholipase D inhibitor
0.1320.0250.1325 Hydroxytryptamine agonist
0.1290.0220.129Protein kinase B gamma inhibitor
0.1440.0390.1445 Hydroxytryptamine 3A agonist
0.1280.0250.167NADH dehydrogenase inhibitor

0.167 0.014 DBMET00327

DBMET00327
0.1670.0690.193Arachidonic acid antagonist

0.193 0.04 DBMET00327

DBMET00327
0.1110.0160.111NMDA receptor agonist
0.210.1190.215 Hydroxytryptamine 1E antagonist
0.0950.0040.095Factor XI inhibitor
0.1320.0420.132GABA C receptor agonist

0.118 0.051 DBMET00327

0.120.0320.12Potassium channel activator
0.1020.0150.102GABA receptor antagonist
0.0960.010.0965 Hydroxytryptamine 2 agonist
0.1180.0320.135Dopamine antagonist

0.135 0.029 DBMET00327

DBMET00327
0.1680.0820.168Interleukin-1 receptor-associated protein kinase 1 inhibitor
0.1910.1070.191Aryl hydrocarbon receptor agonist
0.0890.0050.089Fructose-1,6-bisphosphatase inhibitor

0.088 0.005 DBMET00327

0.120.0370.12Acetylcholine agonist
0.1480.0660.148Adenylate cyclase stimulant

0.141 0.079 DBMET00327

0.1030.0210.326Phosphodiesterase III inhibitor

0.326 0.004 DBMET00327

DBMET00327
0.1050.0240.12D-Ala-D-Ala ligase inhibitor

0.12 0.014 DBMET00327

DBMET00327
0.0930.0130.391Phosphodiesterase 3B inhibitor

0.391 0.003 DBMET00327

DBMET00327
0.1430.0640.145Ca2+-transporting ATPase inhibitor

0.145 0.055 DBMET00327

DBMET00327
0.1040.0260.104Alpha adrenoreceptor agonist
0.0810.0030.081Elastase 2A inhibitor
0.0810.0030.081Elastase 2 inhibitor
0.0940.0160.0945 Hydroxytryptamine 1A agonist
0.1410.0640.141Sodium channel blocker
0.0850.010.085Progesterone antagonist
0.1120.0380.112Androgen antagonist
0.1050.0310.112Dopamine D2 antagonist

0.112 0.029 DBMET00327

DBMET00327
0.1420.070.142Pregnane X receptor agonist
0.0930.0220.0935 Hydroxytryptamine 1 agonist
0.0960.0250.096Nav1.7 sodium channel blocker
0.2830.2130.283Caspase 9 stimulant

0.282 0.214 DBMET00327

0.170.10.17Psychostimulant
0.0790.0080.079Factor VII inhibitor
0.1250.0560.1255 Hydroxytryptamine 2B antagonist

0.102 0.081 DBMET00327

0.1010.0320.1015 Hydroxytryptamine 1A antagonist
0.0730.0040.073ATP citrate lysase inhibitor

0.068 0.004 DBMET00327

0.1110.0440.111MAP kinase kinase 1 inhibitor
0.0710.0050.071Endothelial nitric-oxide synthase inhibitor
0.1220.0570.281Cystathionine beta-synthase inhibitor

0.281 0.011 DBMET00327

DBMET00327
0.0950.0310.095CDC25A inhibitor
0.1130.050.113Alpha adrenoreceptor antagonist
0.0680.0040.068Calcitonin gene-related peptide antagonist
0.0840.020.084GABA A receptor antagonist
0.0730.010.073Potassium channel (Inward rectifier) activator
0.0790.0170.079AMPA receptor antagonist
0.0770.0160.077Kallikrein inhibitor
0.0740.0130.074Aldosterone antagonist
0.0810.020.081Thromboxane antagonist
0.0770.0160.077Thromboxane A2 antagonist
0.070.010.07Potassium channel (ATP-sensitive) activator
0.1280.070.133Alpha-N-acetylglucosaminidase inhibitor

0.133 0.066 DBMET00327

DBMET00327
0.0950.0370.095Glycine receptor antagonist
0.1150.0570.115Ferrochelatase inhibitor
0.0780.0210.078Enoyl-[acyl-carrier-protein] reductase inhibitor

0.077 0.021 DBMET00327

0.1010.0470.101Alpha 2 adrenoreceptor antagonist

0.076 0.071 DBMET00327

0.0770.0240.077MDM2 inhibitor
0.1750.1240.175ErbB-1 antagonist
0.1170.0660.1175 Hydroxytryptamine antagonist
0.1060.0550.138UDP-glucose 4-epimerase inhibitor

0.138 0.034 DBMET00327

DBMET00327
0.0780.0280.078Aryl hydrocarbon receptor antagonist
0.090.0410.095 Hydroxytryptamine 1 antagonist
0.0550.0060.055Carnitine palmitoyltransferase 1 inhibitor
0.0550.0060.055Carnitine palmitoyltransferase inhibitor
0.1820.1330.182Calpain inhibitor
0.0920.0430.092Glutamate receptor agonist
0.1380.0910.138Anticoagulant
0.0610.0140.061Purinergic P2X4 antagonist
0.0910.0450.091Acetylcholine nicotinic agonist
0.1630.1170.163HERG channel blocker
0.060.0140.06Dopamine D3 agonist
0.1240.0780.133NADPH oxidase inhibitor

0.133 0.068 DBMET00327

DBMET00327
0.0940.0490.094Interleukin 5 antagonist

0.09 0.055 DBMET00327

0.1070.0620.128DOPA decarboxylase inhibitor

0.128 0.036 DBMET00327

DBMET00327
0.0650.020.065Acetylcholine M1 receptor agonist
0.120.0750.12Cathepsin H inhibitor
0.0690.0240.069Prostaglandin E2 antagonist
0.0710.0270.071Acetylcholine muscarinic agonist
0.0610.0170.061Adenylate cyclase 1 inhibitor
0.0820.0380.082GABA B receptor agonist

0.07 0.068 DBMET00327

0.0770.0350.259Dopamine D1 antagonist

0.259 0.007 DBMET00327

DBMET00327
0.0740.0320.074Glutamate (mGluR6) antagonist
0.0890.0490.089GABA A receptor agonist
0.0670.0270.067Neuropeptide Y5 antagonist
0.0980.0580.098Lanosterol 14 alpha demethylase inhibitor
0.1490.1090.149Phospholipase C inhibitor

0.14 0.127 DBMET00327

0.080.0410.08Vanilloid 4 agonist
0.0920.0540.092Ca(v)2.2 blocker
0.0540.0160.054GABA B receptor antagonist

0.047 0.023 DBMET00327

0.0660.0280.066CC chemokine 2 receptor antagonist
0.0420.0040.042Acid ceramidase inhibitor
0.0710.0340.0715 Hydroxytryptamine 3 agonist

0.06 0.049 DBMET00327

0.1290.0920.494Peroxidase inhibitor

0.494 0.01 DBMET00327

DBMET00327
0.0390.0050.039Fructose-1,6-bisphosphatase 1 inhibitor

0.022 0.02 DBMET00327

0.1240.090.124Lipid peroxidase inhibitor
0.0750.0420.075Peroxisome proliferator-activated receptor gamma antagonist

0.074 0.044 DBMET00327

0.0710.0380.0715 Hydroxytryptamine uptake inhibitor
0.1070.0730.107Nav1.5 sodium channel blocker
0.0460.0130.046Acetylcholine M4 receptor agonist
0.0660.0350.066Plasminogen activator inhibitor
0.0840.0530.084Adrenaline agonist
0.0630.0330.063Nicotinic neuronal receptor agonist
0.0640.0340.064Beta 2 adrenoreceptor agonist
0.1070.0770.11TRPA1 agonist

0.11 0.071 DBMET00327

DBMET00327
0.0490.020.049Factor VIIa inhibitor
0.0960.0670.096Glutamate (mGluR7) agonist
0.0520.0230.052Benzodiazepine antagonist
0.0420.0140.042Potassium channel small-conductance Ca-activated activator
0.0940.0660.106Sphingomyelinase inhibitor

0.106 0.053 DBMET00327

DBMET00327
0.1210.0950.121Sphingosine 1-phosphate receptor 2 antagonist

0.116 0.106 DBMET00327

0.1270.1020.127Thiol protease inhibitor
0.0530.0280.053Glutamate (mGluR group I) agonist
0.0470.0220.047Alpha 1L adrenoreceptor agonist
0.060.0360.06Alpha 1 adrenoreceptor agonist
0.20.1770.2Antithrombotic
0.0370.0150.037Cholesterol ester transfer protein antagonist
0.0710.050.071Benzodiazepine agonist
0.1120.0910.112Glycogen synthase kinase-3 alpha inhibitor
0.0280.0080.028Imidazoline I1 receptor antagonist
0.050.0290.05Glutamate (mGluR5) antagonist
0.0880.0670.088Glutamate release inhibitor

0.088 0.066 DBMET00327

0.0930.0730.093GABA C receptor rho-1 antagonist
0.0720.0520.113Lipase inhibitor

0.113 0.021 DBMET00327

DBMET00327
0.1510.1320.151Insulin sensitizer
0.0610.0420.073Purinergic P2X1 antagonist

0.073 0.029 DBMET00327

DBMET00327
0.0990.080.106GABA C receptor antagonist

0.106 0.07 DBMET00327

DBMET00327
0.0690.050.069Prostaglandin-E synthase inhibitor
0.0820.0640.082Histamine N-methyltransferase inhibitor
0.0330.0140.033Carnitine palmitoyltransferase 1A inhibitor
0.0380.020.038Plasma kallikrein inhibitor
0.0540.0370.054Nicotinic alpha7 receptor agonist
0.060.0430.07Carbamoyl phosphate synthetase inhibitor

0.07 0.035 DBMET00327

DBMET00327
0.0470.030.047Glutamate (mGluR5) agonist
0.0890.0730.151Creatine kinase inhibitor

0.151 0.024 DBMET00327

DBMET00327
0.0940.0770.094Mediator release inhibitor
0.0980.0810.098Protein kinase C gamma inhibitor
0.0340.0180.034Prostaglandin EP3 antagonist
0.0690.0540.069Epoxide hydrolase inhibitor
0.0490.0340.049Bromodomain-containing protein 3 inhibitor
0.0580.0430.058Androgen agonist

0.054 0.05 DBMET00327

0.0710.0560.088Alpha 2a adrenoreceptor antagonist

0.088 0.043 DBMET00327

DBMET00327
0.0560.0420.056Dopamine uptake inhibitor
0.1020.0880.102Microtubule formation inhibitor
0.1090.0960.109Sphingosine 1-phosphate receptor 4 antagonist
0.0550.0420.0555 Hydroxytryptamine 7 agonist
0.1070.0940.107Cyclooxygenase 3 inhibitor
0.0550.0430.064Pregnane X receptor antagonist

0.064 0.023 DBMET00327

DBMET00327
0.0410.0290.0573-Hydroxyanthranilate 3,4-dioxygenase inhibitor

0.057 0.009 DBMET00327

DBMET00327
0.0660.0540.066Glutamate (mGluR group I) antagonist
0.0190.0090.019Calcitonin gene-related peptide 1 receptor antagonist
0.0390.0290.047CF transmembrane conductance regulator antagonist

0.047 0.011 DBMET00327

DBMET00327
0.020.0110.02Progesterone agonist
0.0380.030.038Dopamine D5 agonist

0.038 0.031 DBMET00327

0.1340.1260.134Platelet adhesion inhibitor
0.0650.0570.065Exportin-1 inhibitor
0.0890.0810.0895 Hydroxytryptamine 2 antagonist
0.0450.0380.045Carnitine palmitoyltransferase 1B inhibitor
0.0360.0290.036TRPM8 blocker
0.0820.0750.082HIV-1 integrase (Overall Integration) inhibitor

0.082 0.075 DBMET00327

0.0420.0350.042Histamine H1 receptor agonist
0.050.0430.05Acetylcholine M2 receptor agonist
0.0810.0740.084Triose-phosphate isomerase inhibitor

0.084 0.069 DBMET00327

DBMET00327
0.0250.0190.025Sodium/glucose cotransporter inhibitor
0.0260.020.026Integrin alpha2beta1 antagonist
0.0520.0460.052Dihydroorotate oxidase inhibitor
0.0610.0570.061Alpha 1a adrenoreceptor antagonist
0.0140.010.014Glucagon agonist
0.0510.0480.119Dopamine D4 antagonist

0.119 0.022 DBMET00327

DBMET00327
0.0340.0310.034Integrin alpha2 antagonist
0.0350.0330.035Vascular adhesion protein 1 inhibitor
0.0650.0630.065Alpha 1 adrenoreceptor antagonist
0.1440.1420.144Potassium channel (Voltage-sensitive) blocker
0.0680.0660.068GABA aminotransferase inhibitor
0.0640.0630.064Vanilloid antagonist
0.10.1180.188Interleukin 4 antagonist

0.188 0.026 DBMET00327

DBMET00327
0.0380.0570.045Glucose-6-phosphate isomerase inhibitor

0.045 0.038 DBMET00327

DBMET00327
0.0240.0440.048Phosphoglycerate kinase inhibitor

0.048 0.015 DBMET00327

DBMET00327
0.0430.0660.068Dopamine D3 antagonist

0.068 0.039 DBMET00327

DBMET00327
0.1060.1290.158Mannose-6-phosphate isomerase inhibitor

0.158 0.058 DBMET00327

DBMET00327
0.0270.050.055Urate transporter 1 inhibitor

0.055 0.016 DBMET00327

DBMET00327
0.0640.0880.122Chymotrypsin inhibitor

0.122 0.025 DBMET00327

DBMET00327
0.0640.0880.103Estrogen receptor alpha antagonist

0.103 0.025 DBMET00327

DBMET00327
0.1170.1420.145Interferon gamma antagonist

0.145 0.085 DBMET00327

DBMET00327
0.0480.0830.094Histidine decarboxylase inhibitor

0.094 0.034 DBMET00327

DBMET00327
0.1510.1860.167Superoxide dismutase inhibitor

0.167 0.159 DBMET00327

DBMET00327
0.0670.1060.097Urease inhibitor

0.097 0.071 DBMET00327

DBMET00327
0.0180.0620.035Estradiol 17 beta-dehydrogenase 3 inhibitor

0.035 0.019 DBMET00327

DBMET00327
0.1120.1560.344Amyloid beta precursor protein antagonist

0.344 0.01 DBMET00327

DBMET00327
0.0360.0950.057Protease activated receptor antagonist

0.057 0.051 DBMET00327

DBMET00327
0.0370.0970.055Fatty acid synthase inhibitor

0.055 0.042 DBMET00327

DBMET00327
0.1040.1960.407P-glycoprotein inhibitor

0.407 0.015 DBMET00327

DBMET00327
0.1620.2560.2115-Lipoxygenase inhibitor

0.21 0.202 DBMET00327

DBMET00327
0.1270.2210.157Glyceraldehyde-3-phosphate dehydrogenase inhibitor

0.157 0.134 DBMET00327

DBMET00327
0.0630.170.277Cyclooxygenase 1 inhibitor

0.277 0.017 DBMET00327

DBMET00327
0.1320.2390.20112-Lipoxygenase inhibitor

0.201 0.15 DBMET00327

DBMET00327
0.1220.2330.556Prostaglandin dehydrogenase inhibitor

0.556 0.031 DBMET00327

DBMET00327
0.0120.1330.031Melatonin 2 agonist

0.031 0.026 DBMET00327

DBMET00327
0.0340.1550.059Heat shock protein 90 beta antagonist

0.059 0.041 DBMET00327

DBMET00327
0.0520.1740.121Alpha 2c adrenoreceptor antagonist

0.121 0.049 DBMET00327

DBMET00327
0.0250.1520.0553(or 17)beta-hydroxysteroid dehydrogenase inhibitor

0.055 0.035 DBMET00327

DBMET00327
0.0560.1860.204Cyclooxygenase 2 inhibitor

0.204 0.029 DBMET00327

DBMET00327
0.1350.2810.383Alpha-glucosidase inhibitor

0.383 0.122 DBMET00327

DBMET00327
0.0490.2090.21Estrogen receptor beta antagonist

0.21 0.009 DBMET00327

DBMET00327
0.0420.2230.098Uric acid excretion stimulant

0.098 0.055 DBMET00327

DBMET00327
0.0650.2770.179Heat shock protein 90 alpha antagonist

0.179 0.063 DBMET00327

DBMET00327
0.0050.230.08Leukotriene A4 hydrolase inhibitor

0.08 0.009 DBMET00327

DBMET00327
0.0150.2470.08Elastase inhibitor

0.08 0.016 DBMET00327

DBMET00327
0.0560.3020.155Heat shock protein 90 antagonist

0.155 0.07 DBMET00327

DBMET00327
0.0130.2710.039Estrogen-related receptor beta antagonist

0.039 0.012 DBMET00327

DBMET00327
0.0240.2870.1795-Lipoxygenase inhibitor

0.179 0.029 DBMET00327

DBMET00327
0.0410.3540.182Estrogen antagonist

0.182 0.015 DBMET00327

DBMET00327
0.0050.3340.611Dopamine D5 antagonist

0.611 0.003 DBMET00327

DBMET00327
0.0520.410.168Antioxidant

0.168 0.144 DBMET00327

DBMET00327
0.0360.40.137Dual specificity phosphatase inhibitor

0.137 0.11 DBMET00327

DBMET00327
0.0030.3830.042Estrogen receptor alpha agonist

0.042 0.02 DBMET00327

DBMET00327
0.0030.4130.096Estrogen receptor beta agonist

0.096 0.012 DBMET00327

DBMET00327
0.0040.4920.022Integrin alphaVbeta3 antagonist

0.022 0.015 DBMET00327

DBMET00327
0.0040.6390.057Estrogen agonist

0.057 0.031 DBMET00327

DBMET00327
0.0030.7490.036Estradiol 17 beta-dehydrogenase 2 inhibitor

0.036 0.024 DBMET00327

DBMET00327
0.0030.7940.033Sphingosine 1-phosphate receptor 3 agonist

0.033 0.025 DBMET00327

DBMET00327
Ext Pa Pi Pmax Activity Other Results ID Pa_max