Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.9420.0020.942Alpha adrenoreceptor agonist

0.662 0.003 DBMET00464

0.715 0.003 DBMET00465

0.9350.0010.935Alpha 2 adrenoreceptor agonist

0.635 0.002 DBMET00464

0.671 0.002 DBMET00465

0.8530.0010.853Alpha 2b adrenoreceptor agonist

0.326 0.002 DBMET00464

0.243 0.002 DBMET00465

0.7660.0010.766Alpha 2c adrenoreceptor agonist

0.205 0.002 DBMET00464

0.134 0.002 DBMET00465

0.7380.0010.738Alpha 2a adrenoreceptor agonist

0.391 0.001 DBMET00464

0.404 0.001 DBMET00465

0.7330.0040.733Antiadrenergic

0.569 0.005 DBMET00464

0.544 0.005 DBMET00465

0.7310.0040.731Adrenaline antagonist

0.566 0.005 DBMET00464

0.542 0.005 DBMET00465

0.6820.0030.682Alpha 2a adrenoreceptor antagonist

0.366 0.005 DBMET00464

0.333 0.005 DBMET00465

0.6520.0030.652Alpha 2b adrenoreceptor antagonist

0.403 0.005 DBMET00464

0.357 0.006 DBMET00465

0.6280.0020.628Prostacyclin antagonist

0.403 0.003 DBMET00464

0.417 0.003 DBMET00465

0.6060.0040.606Alpha 2 adrenoreceptor antagonist

0.301 0.008 DBMET00464

0.267 0.01 DBMET00465

0.550.0030.55Alpha 2c adrenoreceptor antagonist

0.313 0.006 DBMET00464

0.292 0.007 DBMET00465

0.5090.0010.509Alpha 2d adrenoreceptor agonist

0.424 0.001 DBMET00464

0.407 0.001 DBMET00465

0.5050.0310.505Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.47 0.049 DBMET00464

0.326 0.179 DBMET00465

0.4610.0010.461Alpha 1b adrenoreceptor agonist

0.346 0.001 DBMET00464

0.339 0.001 DBMET00465

0.4220.0040.422Alpha 1 adrenoreceptor agonist

0.18 0.007 DBMET00464

0.161 0.009 DBMET00465

0.3440.0120.344Alpha adrenoreceptor antagonist

0.236 0.022 DBMET00464

0.154 0.037 DBMET00465

0.3850.0580.385Angiogenesis inhibitor

0.308 0.089 DBMET00464

0.194 0.177 DBMET00465

0.3140.0030.314Vitronectin receptor antagonist

0.178 0.004 DBMET00464

0.286 0.003 DBMET00465

0.3170.0220.317MAP-kinase-activated kinase 5 inhibitor

0.276 0.044 DBMET00464

0.285 0.038 DBMET00465

0.2740.0040.274Adrenaline agonist

0.234 0.005 DBMET00464

0.265 0.004 DBMET00465

0.2860.0280.305Src kinase inhibitor

0.305 0.025 DBMET00464

0.145 0.087 DBMET00465

DBMET00464
0.2770.020.277Lck kinase inhibitor

0.181 0.049 DBMET00464

0.142 0.071 DBMET00465

0.2530.0020.253Alpha 1a adrenoreceptor agonist

0.206 0.002 DBMET00464

0.196 0.002 DBMET00465

0.2990.0510.299Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor

0.252 0.067 DBMET00464

0.187 0.101 DBMET00465

0.2960.0540.296Dyrk kinase inhibitor

0.249 0.072 DBMET00464

0.173 0.116 DBMET00465

0.2620.0230.262Bone formation stimulant

0.191 0.038 DBMET00464

0.228 0.029 DBMET00465

0.2510.0290.251Protein-tyrosine kinase Lyn inhibitor

0.156 0.063 DBMET00464

0.106 0.097 DBMET00465

0.2240.0120.224Alpha 1b adrenoreceptor antagonist

0.175 0.018 DBMET00464

0.124 0.028 DBMET00465

0.1920.010.192Alpha 1d adrenoreceptor antagonist

0.134 0.017 DBMET00464

0.086 0.028 DBMET00465

0.220.0550.22I kappa B kinase epsilon inhibitor

0.207 0.065 DBMET00464

0.2010.0420.201Dual specificity tyrosine-phosphorylation regulated kinase 1B inhibitor

0.155 0.07 DBMET00464

0.190.0350.19Protein kinase (CK1) gamma 2 inhibitor

0.115 0.069 DBMET00464

0.1770.0240.177Alpha 1 adrenoreceptor antagonist

0.123 0.036 DBMET00464

0.068 0.06 DBMET00465

0.1750.0290.177Aurora-C kinase inhibitor

0.177 0.028 DBMET00464

0.175 0.029 DBMET00465

DBMET00464
0.1620.0190.162Insulin growth factor antagonist

0.109 0.041 DBMET00464

0.1890.0480.189Protein kinase (CK1) gamma inhibitor

0.124 0.086 DBMET00464

0.1410.0030.141Integrin alphaVbeta1 antagonist

0.072 0.004 DBMET00464

0.067 0.004 DBMET00465

0.1390.0020.139Alpha 1L adrenoreceptor agonist

0.115 0.002 DBMET00464

0.135 0.002 DBMET00465

0.1550.0190.155Insulin like growth factor 1 antagonist

0.103 0.04 DBMET00464

0.1770.0450.177Cyclin-dependent kinase inhibitor

0.154 0.054 DBMET00464

0.109 0.082 DBMET00465

0.1360.0040.136Integrin alphaVbeta3 antagonist

0.071 0.004 DBMET00464

0.123 0.004 DBMET00465

0.1350.0140.135Alpha 2d adrenoreceptor antagonist

0.107 0.038 DBMET00464

0.09 0.072 DBMET00465

0.120.0010.12Integrin beta6 antagonist

0.066 0.002 DBMET00464

0.084 0.002 DBMET00465

0.2980.1820.298MAP kinase 1 inhibitor
0.1290.0140.133CXC chemokine receptor antagonist

0.133 0.014 DBMET00464

0.1 0.024 DBMET00465

DBMET00464
0.1310.020.1315 Hydroxytryptamine 7 antagonist

0.083 0.03 DBMET00464

0.1690.0620.185Cyclin-dependent kinase 3 inhibitor

0.185 0.044 DBMET00464

DBMET00464
0.110.0020.11Imidazoline I1 receptor antagonist

0.037 0.005 DBMET00464

0.036 0.005 DBMET00465

0.1170.0120.117NMDA 2B receptor antagonist

0.076 0.022 DBMET00464

0.270.1670.27MAP kinase kinase 6 inhibitor

0.249 0.191 DBMET00464

0.235 0.21 DBMET00465

0.1550.0520.228c-Src kinase inhibitor

0.228 0.029 DBMET00464

DBMET00464
0.1640.0610.164Growth factor antagonist

0.123 0.089 DBMET00464

0.1330.0470.133Interleukin 8 antagonist
0.110.0240.11Nicotinic alpha4beta2 receptor antagonist
0.1240.0390.124CDK2/cyclin A inhibitor

0.118 0.044 DBMET00464

0.1870.1050.208ErbB-1 antagonist

0.208 0.081 DBMET00464

DBMET00464
0.1640.0830.164Tyrosine kinase inhibitor

0.155 0.087 DBMET00464

0.0910.0120.124Potassium channel (Ca-activated) blocker

0.063 0.036 DBMET00464

0.124 0.006 DBMET00465

DBMET00465
0.1740.0950.174Focal adhesion kinase 2 inhibitor

0.152 0.128 DBMET00464

0.120.0410.12CDK/cyclin complex inhibitor

0.1 0.052 DBMET00464

0.1470.070.147Protein kinase (CK1) inhibitor

0.107 0.102 DBMET00464

0.0920.0140.092Cyclin B1 inhibitor

0.077 0.025 DBMET00464

0.1310.0550.131Protein kinase (CK2) alpha inhibitor
0.0770.0050.077Dopamine beta hydroxylase inhibitor

0.046 0.04 DBMET00465

0.1050.0340.105Alpha 1a adrenoreceptor antagonist

0.074 0.048 DBMET00464

0.1590.0890.159Phospholipase C inhibitor

0.153 0.1 DBMET00465

0.0810.0140.081Cyclin B2 inhibitor

0.07 0.021 DBMET00464

0.051 0.045 DBMET00465

0.1130.0470.113Protein kinase C mu inhibitor
0.0930.0270.093CDC7 inhibitor

0.075 0.039 DBMET00464

0.1160.0510.116Protein kinase (CK2) inhibitor

0.083 0.079 DBMET00464

0.1640.10.164Anesthetic general
0.2320.1690.232Calcium channel activator
0.1070.0480.256Protein kinase (Mos, Mil/Raf, MEKK, RIPK, TESK, LIMK, IRAK, ILK, Activin/TGF-beta) inhibitor

0.256 0.012 DBMET00464

DBMET00464
0.0940.0350.094Focal adhesion kinase 1 inhibitor

0.08 0.049 DBMET00464

0.0710.0120.071Potassium channel small-conductance Ca-activated blocker
0.0880.030.088Neuronal nicotinic receptor antagonist

0.074 0.042 DBMET00464

0.0750.0180.075Cyclin B inhibitor

0.064 0.027 DBMET00464

0.1140.0580.114Cyclin-dependent kinase 1 inhibitor

0.107 0.062 DBMET00464

0.086 0.077 DBMET00465

0.0840.0290.084ZAP-70 protein tyrosine kinase inhibitor
0.0920.0370.259Raf kinase inhibitor

0.259 0.009 DBMET00464

DBMET00464
0.1130.0620.113Activin receptor-like kinase 4 inhibitor
0.1120.0630.1125 Hydroxytryptamine 3A agonist
0.1310.0820.131Protein kinase C nu inhibitor
0.1090.0610.109CDC-like kinase 3 inhibitor

0.102 0.075 DBMET00464

0.0970.0490.097Histamine N-methyltransferase inhibitor
0.0790.0320.0795 Hydroxytryptamine 3A antagonist
0.0680.0220.068Nicotinic receptor alpha7 subunit antagonist
0.1350.0890.156Dual specificity tyrosine-phosphorylation-regulated kinase 4 inhibitor

0.156 0.073 DBMET00464

DBMET00464
0.0770.0310.077Potassium channel (ATP-sensitive) blocker
0.0490.0050.132Integrin beta5 antagonist

0.034 0.008 DBMET00464

0.132 0.004 DBMET00465

DBMET00465
0.2710.2270.271Caspase 9 stimulant
0.1070.0630.107Cyclin-dependent kinase 2 inhibitor

0.093 0.078 DBMET00464

0.0470.0030.047Complement factor 1r inhibitor

0.042 0.004 DBMET00464

0.041 0.004 DBMET00465

0.0630.020.063Nicotinic receptor alpha4 subunit antagonist

0.063 0.02 DBMET00464

0.0910.0480.091Dual specificity tyrosine-phosphorylation regulated kinase 2 inhibitor

0.091 0.048 DBMET00464

0.1290.0880.129Protein kinase (CK1) gamma 1 inhibitor
0.1160.0770.116Epidermal growth factor receptor kinase inhibitor
0.0880.050.088ALK inhibitor
0.1350.0970.135Cyclin-dependent kinase 8 inhibitor
0.1070.070.107Glycogen synthase kinase-3 beta inhibitor
0.0920.0550.092Pim-3 kinase inhibitor

0.079 0.078 DBMET00464

0.1010.0650.101Gastric antisecretory
0.0880.0520.088TIE antagonist
0.0860.0510.086TIE-2 antagonist
0.1050.070.105EphA2 antagonist
0.1190.0850.119Glycogen synthase kinase-3 alpha inhibitor

0.108 0.096 DBMET00464

0.1070.0730.107Glycogen synthase kinase-3 inhibitor
0.0490.0190.054Integrin alpha5beta1 antagonist

0.038 0.032 DBMET00464

0.054 0.015 DBMET00465

DBMET00465
0.150.120.15Dual specificity tyrosine-phosphorylation regulated kinase 3 inhibitor
0.0660.0380.093Raf kinase C inhibitor

0.093 0.027 DBMET00464

DBMET00464
0.0560.0280.056CXC chemokine 1 receptor antagonist

0.052 0.033 DBMET00465

0.0620.0340.062Cyclin A1 inhibitor

0.057 0.046 DBMET00464

0.0810.0530.081Acetylcholine nicotinic antagonist
0.0920.0650.107Pim-1 kinase inhibitor

0.107 0.051 DBMET00464

DBMET00464
0.0930.0660.093MAP kinase kinase 1 inhibitor
0.0340.0080.049Integrin beta3 antagonist

0.018 0.016 DBMET00464

0.049 0.006 DBMET00465

DBMET00465
0.1320.1070.24Polo-like kinase-3 inhibitor

0.24 0.028 DBMET00464

DBMET00464
0.1720.1470.18Nitric-oxide synthase stimulant

0.18 0.127 DBMET00464

DBMET00464
0.0290.0040.029Complement factor 1 inhibitor

0.022 0.006 DBMET00464

0.022 0.006 DBMET00465

0.0280.0030.028Imidazoline I2 receptor antagonist
0.0620.0390.062Cyclin D1 inhibitor
0.0330.0090.033Thymidine phosphorylase inhibitor

0.026 0.019 DBMET00464

0.026 0.018 DBMET00465

0.080.0580.08Leucine-rich repeat kinase 2 inhibitor
0.0680.0470.084Cyclin B3 inhibitor

0.084 0.036 DBMET00464

DBMET00464
0.0370.0160.037Protein kinase (CK2) beta inhibitor

0.031 0.03 DBMET00464

0.033 0.023 DBMET00465

0.1170.10.117Activin receptor-like kinase 2 inhibitor
0.0520.0340.052H+/K+-transporting ATPase inhibitor
0.0450.0280.045Histamine H1 receptor agonist
0.060.0460.06Cyclin A2 inhibitor
0.0750.0620.084Platelet growth factor antagonist

0.084 0.053 DBMET00464

DBMET00464
0.0880.0760.088Aurora-A kinase inhibitor
0.030.0180.03MAP3K8 inhibitor
0.1740.1630.174DNA synthesis inhibitor
0.0660.0550.066NMDA 2 receptor antagonist
0.0290.0190.029Nicotinic alpha4beta2 receptor agonist
0.0850.0750.085Platelet activating factor beta antagonist
0.0150.0060.015Cyclin D2 inhibitor

0.014 0.008 DBMET00464

0.0940.0850.0945 Hydroxytryptamine antagonist
0.0860.0770.086Check point kinase 2 inhibitor

0.086 0.078 DBMET00464

0.1460.1390.146Proto-oncogene tyrosine-protein kinase Fyn inhibitor
0.0540.0470.054CDK4/cyclin D inhibitor
0.0590.0530.059Cyclin-dependent kinase 4 inhibitor
0.0560.050.056CDK1/cyclin B inhibitor
0.2060.2010.206GABA C receptor rho-3 antagonist
0.0360.0310.036Potassium channel Kv1.1 blocker
0.0830.080.111DNA directed RNA polymerase inhibitor

0.111 0.045 DBMET00464

DBMET00464
0.0160.0130.016Nicotinic alpha4 receptor agonist
0.0370.0350.037Thymidine kinase inhibitor
0.0350.0330.035Alpha 1d adrenoreceptor agonist
0.0840.0830.084MAP kinase 8 inhibitor
0.0130.0120.013Integrin alphaVbeta6 antagonist

0.013 0.011 DBMET00465

0.0340.0340.049Integrin antagonist

0.049 0.028 DBMET00465

DBMET00465
0.0260.0270.029DNA polymerase III inhibitor

0.029 0.018 DBMET00465

DBMET00465
0.0240.0260.025Thymidine kinase (Herpes simplex virus 1) inhibitor

0.025 0.023 DBMET00464

DBMET00464
0.0990.1010.289MAP kinase 12 inhibitor

0.289 0.008 DBMET00464

DBMET00464
0.0710.0760.086MAP-kinase-activated kinase inhibitor

0.086 0.054 DBMET00464

DBMET00464
0.0180.0230.02Thymidine kinase (Herpes simplex virus 2) inhibitor

0.02 0.016 DBMET00464

DBMET00464
0.1890.2020.203Ca2+/calmodulin-dependent kinase IV inhibitor

0.203 0.158 DBMET00464

0.196 0.176 DBMET00465

DBMET00464
0.060.0770.075MAP-kinase-activated kinase 2 inhibitor

0.075 0.05 DBMET00464

DBMET00464
0.1730.1930.217Ca2+/calmodulin-dependent kinase II alpha inhibitor

0.217 0.138 DBMET00464

DBMET00464
0.0390.0690.162Raf kinase B inhibitor

0.162 0.012 DBMET00464

DBMET00464
0.0620.0970.139NMDA receptor antagonist

0.139 0.028 DBMET00465

DBMET00465
0.1040.1650.137Clk dual-specificity kinase inhibitor

0.137 0.127 DBMET00464

DBMET00464
0.0090.0840.06Kainate receptor 4 antagonist

0.06 0.005 DBMET00465

DBMET00465
0.090.1720.129CDC-like kinase 4 inhibitor

0.129 0.119 DBMET00464

DBMET00464
0.0570.1460.095Polo-like kinase-4 inhibitor

0.095 0.082 DBMET00464

DBMET00464
0.10.2060.122Death-associated protein kinase 1 inhibitor

0.122 0.107 DBMET00464

DBMET00464
0.0070.1140.026Kainate receptor 3 antagonist

0.026 0.006 DBMET00465

DBMET00465
0.0060.1230.038Kainate receptor 5 antagonist

0.038 0.007 DBMET00465

DBMET00465
0.0550.1840.145Glutamate receptor antagonist

0.109 0.086 DBMET00464

0.145 0.054 DBMET00465

DBMET00465
0.0950.230.162Platelet aggregation inhibitor

0.162 0.115 DBMET00464

DBMET00464
0.1060.2530.177Death-associated protein kinase 2 inhibitor

0.177 0.058 DBMET00464

0.153 0.099 DBMET00465

DBMET00464
0.0250.2040.147Proto-oncogene tyrosine-protein kinase c-hck inhibitor

0.147 0.015 DBMET00464

DBMET00464
0.0070.2090.051AMPA 2 receptor antagonist

0.051 0.011 DBMET00465

DBMET00465
0.0250.5290.188Interleukin antagonist

0.188 0.091 DBMET00464

DBMET00464
0.0140.8580.317Interleukin 5 antagonist

0.317 0.004 DBMET00464

DBMET00464
Ext Pa Pi Pmax Activity Other Results ID Pa_max