Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.570.010.57Calpain 2 inhibitor
0.5030.0740.503Transcription factor inhibitor
0.4440.0540.444Calcium channel L-type activator

0.395 0.085 DBMET00249

0.360.0050.416Androgen antagonist

0.416 0.004 DBMET00249

DBMET00249
0.430.0760.43Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.338 0.164 DBMET00249

0.4170.0670.417Histamine release inhibitor
0.3270.0410.327Transcription factor STAT3 inhibitor
0.2750.0050.275Potassium channel activator

0.215 0.007 DBMET00249

0.2970.0310.297Calpain inhibitor
0.3090.0510.309Transcription factor STAT inhibitor
0.2850.0270.285Neuropeptide Y2 antagonist
0.3840.1260.384DNA polymerase beta inhibitor
0.3810.1230.468Caspase 9 stimulant

0.468 0.074 DBMET00249

DBMET00249
0.2550.0080.255Catalase inhibitor

0.087 0.044 DBMET00249

0.3070.0690.307Interleukin 2 agonist
0.3030.0780.30312-Lipoxygenase inhibitor

0.185 0.168 DBMET00249

0.2260.0050.226Prostaglandin-E synthase inhibitor

0.151 0.011 DBMET00249

0.2230.0040.223NMDA receptor agonist

0.095 0.021 DBMET00249

0.2510.0320.251Amyloid beta precursor protein antagonist
0.3350.1290.3355 Hydroxytryptamine release inhibitor
0.3440.1390.344Alpha-glucosidase inhibitor
0.3440.140.344DNA directed DNA polymerase inhibitor
0.2320.0350.2323C-like protease (Human coronavirus) inhibitor
0.1980.0030.198NMDA receptor glycine site agonist

0.117 0.01 DBMET00249

0.2970.1040.297Thioredoxin glutathione reductase inhibitor
0.3140.1290.314Beta lactamase inhibitor
0.1960.0130.196Sphingosine 1-phosphate receptor 5 antagonist

0.137 0.085 DBMET00249

0.2280.0510.228Nitric-oxide synthase stimulant

0.198 0.092 DBMET00249

0.2140.0390.214Succinate dehydrogenase inhibitor

0.193 0.054 DBMET00249

0.1790.0050.238Androgen agonist

0.238 0.004 DBMET00249

DBMET00249
0.2650.0940.265Streptokinase A inhibitor
0.2720.1040.272Thyroid hormone beta antagonist
0.2790.1130.33Calcium channel activator

0.33 0.064 DBMET00249

DBMET00249
0.2730.1090.273Thyroid hormone antagonist
0.2370.0820.237Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase inhibitor

0.163 0.127 DBMET00249

0.1860.0380.186M17 leucyl aminopeptidase inhibitor
0.1890.0440.189Thiol protease inhibitor
0.1450.0030.145Dihydroorotate oxidase inhibitor

0.073 0.015 DBMET00249

0.1790.0370.202CF transmembrane conductance regulator agonist

0.202 0.02 DBMET00249

DBMET00249
0.1390.0050.139Glutamate (mGluR group III) agonist
0.2250.0930.225Superoxide dismutase inhibitor

0.212 0.105 DBMET00249

0.160.0290.16Sphingosine 1-phosphate receptor 2 antagonist
0.1560.0260.156Potassium channel (Ca-activated) activator

0.112 0.046 DBMET00249

0.2310.1030.231Gastrin inhibitor

0.184 0.173 DBMET00249

0.1560.0280.156Sphingosine 1-phosphate receptor 4 antagonist

0.125 0.064 DBMET00249

0.1510.0230.151Urease inhibitor

0.148 0.024 DBMET00249

0.1410.0160.141Potassium channel (Voltage-sensitive) activator
0.150.0270.15CDK3/cyclin E inhibitor
0.2120.0960.212Aryl hydrocarbon receptor agonist
0.1560.0420.156Cathepsin H inhibitor
0.1410.0350.141Caspase 3 inhibitor
0.1710.0660.171Death-associated protein kinase 2 inhibitor
0.1360.0340.168UDP-glucose 4-epimerase inhibitor

0.168 0.024 DBMET00249

DBMET00249
0.2090.1130.209Interleukin agonist

0.164 0.154 DBMET00249

0.1840.0890.184Dual specificity tyrosine-phosphorylation regulated kinase 3 inhibitor
0.0970.0040.097NMDA receptor glycine site antagonist

0.038 0.009 DBMET00249

0.1370.0440.137Aminopeptidase B inhibitor
0.1420.0520.142Death-associated protein kinase 1 inhibitor
0.1010.0110.101Dihydroorotate dehydrogenase inhibitor

0.049 0.038 DBMET00249

0.1150.0260.115Glutathione S-transferase inhibitor

0.081 0.059 DBMET00249

0.1270.0410.127Falcipain inhibitor
0.1250.040.125Falcipain 2 inhibitor
0.1180.0330.211Triose-phosphate isomerase inhibitor

0.211 0.01 DBMET00249

DBMET00249
0.0960.0110.096Exportin-1 inhibitor

0.077 0.029 DBMET00249

0.1650.0840.165LIM domain kinase 1 inhibitor
0.0850.0050.085Glutamate (mGluR4) agonist
0.0860.0060.086Potassium channel (Inward rectifier) activator

0.077 0.009 DBMET00249

0.0880.0090.088Kainate receptor antagonist

0.045 0.024 DBMET00249

0.0830.0060.083Potassium channel (ATP-sensitive) activator

0.074 0.008 DBMET00249

0.1420.0680.142Pregnane X receptor agonist

0.137 0.08 DBMET00249

0.0860.0130.086Sphingosine 1-phosphate receptor 3 antagonist
0.1070.0350.107Bcr-Abl kinase inhibitor
0.0960.0240.096Sphingosine 1-phosphate receptor antagonist
0.0960.0250.096Potassium channel large-conductance Ca-activated activator

0.08 0.035 DBMET00249

0.1130.0430.113UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor

0.111 0.045 DBMET00249

0.0740.0040.074Glutamate (mGluR8) agonist

0.073 0.005 DBMET00249

0.1030.0340.103Vanilloid antagonist
0.1380.070.138Calcium channel blocker
0.2150.1470.215Prostaglandin dehydrogenase inhibitor
0.1150.0480.154Adenylate kinase inhibitor

0.154 0.025 DBMET00249

DBMET00249
0.1560.0910.156ATPase inhibitor
0.090.0310.09Vanilloid 1 antagonist
0.1170.060.117Calcium channel (voltage-sensitive) blocker
0.0670.0110.067Collagenase inhibitor
0.080.0250.08NMDA 2C receptor antagonist

0.057 0.049 DBMET00249

0.1370.0860.137Neuropeptide Y1 antagonist
0.0980.0490.098Calcium antagonist
0.0590.0110.059Delayed rectifier potassium channel activator
0.0590.0110.059Potassium channel KCNQ activator
0.090.0450.09D-Ala-D-Ala ligase inhibitor
0.1490.1050.149Neurotensin receptor agonist
0.0880.0440.094Thioredoxin reductase inhibitor

0.094 0.035 DBMET00249

DBMET00249
0.0580.0150.058Glutamate (mGluR4) antagonist

0.043 0.031 DBMET00249

0.1010.0590.149Creatine kinase inhibitor

0.149 0.024 DBMET00249

DBMET00249
0.0980.0570.098Interleukin 12 antagonist
0.0520.0120.052Potassium channel Kv1.1 blocker
0.0630.0240.063Glycine transporter 2 inhibitor
0.070.0320.101Biliverdin reductase inhibitor

0.101 0.018 DBMET00249

DBMET00249
0.0530.0150.06Nerve growth factor antagonist

0.06 0.01 DBMET00249

DBMET00249
0.0990.0630.133Anabolic

0.133 0.029 DBMET00249

DBMET00249
0.0780.0420.078Calcium channel L-type blocker
0.2020.1670.202Transcription factor NF kappa B inhibitor
0.0780.0440.078Epoxide hydrolase inhibitor
0.0480.0150.048Glucagon-like peptide 1 receptor antagonist
0.0390.0070.039Kainate receptor 1 antagonist
0.0480.0170.048Kainate receptor 2 antagonist
0.0330.0040.077Progesterone receptor B antagonist

0.077 0.002 DBMET00249

DBMET00249
0.0410.0130.045Catechol O-methyltransferase inhibitor

0.045 0.011 DBMET00249

DBMET00249
0.0490.0210.058CDK5/p25 inhibitor

0.058 0.016 DBMET00249

DBMET00249
0.0550.0270.055Plasminogen activator inhibitor antagonist
0.0620.0350.107Argininosuccinate synthase inhibitor

0.107 0.017 DBMET00249

DBMET00249
0.0760.050.076Vanilloid 4 agonist
0.1950.1690.238Cholesterol antagonist

0.238 0.134 DBMET00249

DBMET00249
0.1220.0970.197Mannose-6-phosphate isomerase inhibitor

0.197 0.032 DBMET00249

DBMET00249
0.0740.0490.074Metalloproteinase-9 inhibitor
0.0660.0420.066Neuraminidase (influenza) inhibitor
0.0970.0740.097Ferrochelatase inhibitor
0.1320.1080.132Heat shock protein 90 alpha antagonist
0.1040.0810.104TRPA1 agonist

0.096 0.095 DBMET00249

0.0620.0390.062Enoyl-[acyl-carrier-protein] reductase inhibitor
0.110.0880.11Alpha-N-acetylglucosaminidase inhibitor

0.103 0.097 DBMET00249

0.0830.0610.0833C-Like protease (SARS coronavirus) inhibitor
0.1160.0960.116Vanilloid 1 agonist
0.0640.0440.083Transcription factor RelA inhibitor

0.083 0.015 DBMET00249

DBMET00249
0.120.10.12Cytidine deaminase inhibitor
0.0280.0090.028Protease (Human cytomegalovirus) inhibitor
0.0260.0070.026Factor XIII inhibitor
0.0720.0530.072Nav1.8 sodium channel blocker
0.1860.1680.186MAP kinase kinase 3 inhibitor
0.0920.0740.092Nitric-oxide synthase inhibitor
0.0350.0170.035AMPA 1 receptor antagonist
0.0980.0810.109DOPA decarboxylase inhibitor

0.109 0.06 DBMET00249

DBMET00249
0.0590.0420.059Ca(v)3.2 blocker
0.0230.0060.025Potassium channel (Inward rectifier) 11 blocker

0.025 0.005 DBMET00249

DBMET00249
0.0750.0580.075Metalloproteinase-2 inhibitor
0.0580.0410.058Cathepsin L inhibitor
0.0440.0290.044Carbonic anhydrase IV inhibitor
0.0260.0110.026Kainate receptor 5 antagonist

0.02 0.015 DBMET00249

0.0590.0440.059Neuraminidase inhibitor
0.080.0650.08CC chemokine 5 receptor agonist
0.0850.0710.085HIV-1 integrase (Overall Integration) inhibitor
0.1010.0870.101Interleukin 2 antagonist
0.0440.0310.044Dihydroorotase inhibitor
0.0270.0150.027Kainate receptor 4 antagonist

0.023 0.019 DBMET00249

0.0320.0220.032Methionyl aminopeptidase 1 inhibitor
0.060.0510.06Neutrophil collagenase inhibitor
0.0550.0460.055Botulinum neurotoxin type A inhibitor
0.0370.0280.037TRPM8 blocker
0.0680.0590.09Glutamate dehydrogenase inhibitor

0.09 0.037 DBMET00249

DBMET00249
0.0780.0690.078NMDA receptor antagonist

0.075 0.072 DBMET00249

0.0450.0360.045AMPA receptor antagonist
0.0150.0060.015Human herpes virus 5 capsid protein P40 inhibitor
0.110.1010.11Interleukin 4 antagonist
0.1150.1070.146Cell wall synthesis inhibitor

0.146 0.07 DBMET00249

DBMET00249
0.020.0130.025-Alpha-reductase 2 inhibitor
0.0340.0270.034Nicotinic acid receptor agonist
0.0590.0520.059Histone deacetylase SIRT3 inhibitor
0.0470.0410.047Lysophosphatidic acid 3 receptor antagonist
0.040.0350.04NMDA receptor subunit 3B antagonist
0.0290.0240.029Cyclophilin A inhibitor
0.0690.0640.069GABA aminotransferase inhibitor
0.0410.0370.041Glutamate (mGluR group III) antagonist
0.0250.0220.027NMDA 2D receptor antagonist

0.027 0.019 DBMET00249

DBMET00249
0.0470.0440.047CD45 antagonist
0.180.1770.181Tyrosine 3 hydroxylase inhibitor

0.181 0.175 DBMET00249

DBMET00249
0.0280.0260.028Epoxide hydrolase 1 inhibitor
0.0480.0460.048Acetyl-CoA transferase inhibitor
0.0990.0970.099Calcium channel N-type blocker
0.0110.010.013Glutamate (mGluR6) agonist

0.013 0.007 DBMET00249

DBMET00249
0.0460.0450.046Neuropeptide agonist
0.0150.0140.015Kainate receptor 3 antagonist
0.1450.1460.149Neurotrophic factor enhancer

0.149 0.14 DBMET00249

DBMET00249
0.0460.050.083Alcohol oxidase inhibitor

0.083 0.023 DBMET00249

DBMET00249
0.0590.0690.111Porphobilinogen synthase inhibitor

0.111 0.031 DBMET00249

DBMET00249
0.0670.0810.074GABA B receptor agonist

0.074 0.057 DBMET00249

DBMET00249
0.0490.0660.066Purinergic P2X1 antagonist

0.066 0.036 DBMET00249

DBMET00249
0.0230.040.032Progesterone antagonist

0.032 0.027 DBMET00249

DBMET00249
0.120.150.158Anesthetic general

0.158 0.106 DBMET00249

DBMET00249
0.1240.1580.14Ca2+-transporting ATPase inhibitor

0.14 0.075 DBMET00249

DBMET00249
0.0440.0790.098Phosphofructokinase-1 inhibitor

0.098 0.032 DBMET00249

DBMET00249
0.0450.0910.071Histidine decarboxylase inhibitor

0.071 0.05 DBMET00249

DBMET00249
0.0780.1560.101Factor V inhibitor

0.101 0.067 DBMET00249

DBMET00249
0.1780.2580.332Antibacterial

0.332 0.113 DBMET00249

DBMET00249
0.0130.0970.031Fumarate hydratase inhibitor

0.031 0.027 DBMET00249

DBMET00249
0.1330.2310.183MAP kinase kinase 5 inhibitor

0.183 0.058 DBMET00249

DBMET00249
0.0580.1620.098Lanosterol 14 alpha demethylase inhibitor

0.098 0.058 DBMET00249

DBMET00249
0.060.1740.121AMP-activated protein kinase stimulant

0.121 0.048 DBMET00249

DBMET00249
0.0460.1720.061Calcium channel P-type blocker

0.061 0.056 DBMET00249

DBMET00249
0.0260.2710.113Epidermal growth factor antagonist

0.113 0.036 DBMET00249

DBMET00249
Ext Pa Pi Pmax Activity Other Results ID Pa_max