| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.716 | 0.002 | 0.716 | HIV-1 protease inhibitor | 0.5 0.003 DBMET01182 0.686 0.002 DBMET01183 0.293 0.003 DBMET00084 0.57 0.003 DBMET00385 | ||
| 0.6 | 0.003 | 0.6 | Protease inhibitor | 0.442 0.004 DBMET01182 0.592 0.003 DBMET01183 0.315 0.005 DBMET00084 0.522 0.004 DBMET00385 | ||
| 0.256 | 0.06 | 0.343 | Calpain inhibitor | 0.223 0.091 DBMET01182 0.343 0.018 DBMET01183 0.199 0.114 DBMET00385 | DBMET01183 | |
| 0.204 | 0.024 | 0.263 | Proteasome inhibitor | 0.202 0.024 DBMET01182 0.263 0.014 DBMET01183 0.196 0.026 DBMET00385 | DBMET01183 | |
| 0.129 | 0.017 | 0.145 | Alpha 2d adrenoreceptor antagonist | 0.145 0.01 DBMET01182 0.138 0.013 DBMET00084 0.088 0.075 DBMET00385 | DBMET01182 | |
| 0.119 | 0.013 | 0.161 | Cathepsin D inhibitor | 0.118 0.013 DBMET01182 0.161 0.007 DBMET01183 0.058 0.035 DBMET00084 0.116 0.014 DBMET00385 | DBMET01183 | |
| 0.24 | 0.138 | 0.348 | Apoptosis antagonist | 0.325 0.069 DBMET01183 0.348 0.057 DBMET00084 0.239 0.139 DBMET00385 | DBMET00084 | |
| 0.086 | 0.008 | 0.176 | Renin inhibitor | 0.08 0.009 DBMET01182 0.176 0.004 DBMET01183 0.034 0.027 DBMET00084 0.086 0.008 DBMET00385 | DBMET01183 | |
| 0.124 | 0.049 | 0.15 | Nav1.4 sodium channel blocker | 0.125 0.048 DBMET01182 0.15 0.034 DBMET01183 0.106 0.067 DBMET00084 0.109 0.063 DBMET00385 | DBMET01183 | |
| 0.085 | 0.019 | 0.109 | Cathepsin E inhibitor | 0.088 0.018 DBMET01182 0.109 0.011 DBMET01183 0.062 0.038 DBMET00084 0.081 0.021 DBMET00385 | DBMET01183 | |
| 0.086 | 0.021 | 0.116 | Human rhinovirus A protease inhibitor | 0.083 0.022 DBMET01182 0.116 0.013 DBMET01183 0.081 0.023 DBMET00385 | DBMET01183 | |
| 0.16 | 0.102 | 0.16 | P-glycoprotein inhibitor | 0.158 0.105 DBMET01182 | ||
| 0.07 | 0.021 | 0.084 | Endothelin-converting enzyme inhibitor | 0.07 0.021 DBMET01182 0.084 0.017 DBMET01183 0.064 0.023 DBMET00385 | DBMET01183 | |
| 0.091 | 0.045 | 0.106 | 3C-Like protease (SARS coronavirus) inhibitor | 0.087 0.052 DBMET01182 0.106 0.028 DBMET01183 0.087 0.052 DBMET00385 | DBMET01183 | |
| 0.103 | 0.062 | 0.129 | Factor V inhibitor | 0.104 0.061 DBMET01182 0.129 0.031 DBMET01183 0.105 0.059 DBMET00385 | DBMET01183 | |
| 0.199 | 0.16 | 0.24 | Nootropic | 0.24 0.117 DBMET01183 | DBMET01183 | |
| 0.07 | 0.031 | 0.093 | Caspase 9 inhibitor | 0.061 0.046 DBMET01182 0.093 0.016 DBMET01183 0.065 0.038 DBMET00385 | DBMET01183 | |
| 0.067 | 0.03 | 0.106 | Cathepsin B inhibitor | 0.052 0.046 DBMET01182 0.106 0.014 DBMET01183 0.063 0.033 DBMET00385 | DBMET01183 | |
| 0.045 | 0.014 | 0.081 | Caspase 2 inhibitor | 0.081 0.006 DBMET01183 0.041 0.015 DBMET00084 0.044 0.014 DBMET00385 | DBMET01183 | |
| 0.074 | 0.044 | 0.13 | Secretase beta inhibitor | 0.095 0.021 DBMET01182 0.13 0.008 DBMET01183 | DBMET01183 | |
| 0.039 | 0.013 | 0.058 | Plasmepsin I inhibitor | 0.04 0.012 DBMET01182 0.058 0.005 DBMET01183 0.028 0.024 DBMET00084 0.037 0.014 DBMET00385 | DBMET01183 | |
| 0.078 | 0.054 | 0.117 | Somatostatin 1 agonist | 0.117 0.024 DBMET01182 0.085 0.046 DBMET01183 0.076 0.056 DBMET00385 | DBMET01182 | |
| 0.051 | 0.028 | 0.059 | Bombesin antagonist | 0.059 0.019 DBMET01182 0.059 0.02 DBMET01183 0.048 0.032 DBMET00385 | DBMET01183 | |
| 0.078 | 0.056 | 0.116 | Chymotrypsin inhibitor | 0.076 0.06 DBMET01182 0.116 0.027 DBMET01183 0.073 0.065 DBMET00385 | DBMET01183 | |
| 0.203 | 0.184 | 0.315 | Interleukin 2 agonist | 0.315 0.064 DBMET01182 0.235 0.136 DBMET01183 | DBMET01182 | |
| 0.064 | 0.046 | 0.088 | Glucagon-like peptide 1 agonist | 0.054 0.053 DBMET01182 0.088 0.029 DBMET01183 0.067 0.044 DBMET00084 0.056 0.051 DBMET00385 | DBMET01183 | |
| 0.035 | 0.018 | 0.04 | Calpain 1 inhibitor | 0.031 0.03 DBMET01182 0.04 0.01 DBMET01183 0.035 0.02 DBMET00385 | DBMET01183 | |
| 0.057 | 0.045 | 0.086 | Bombesin 1 receptor agonist | 0.086 0.023 DBMET01182 0.069 0.032 DBMET01183 | DBMET01182 | |
| 0.037 | 0.026 | 0.046 | Bombesin 1 receptor antagonist | 0.034 0.029 DBMET01182 0.046 0.017 DBMET01183 | DBMET01183 | |
| 0.026 | 0.025 | 0.033 | HCV NS5A inhibitor | 0.033 0.011 DBMET01183 | DBMET01183 | |
| 0.051 | 0.051 | 0.058 | Kallikrein 1 inhibitor | 0.058 0.037 DBMET01183 | DBMET01183 | |
| 0.016 | 0.019 | 0.041 | Neutral endopeptidase inhibitor | 0.041 0.009 DBMET01182 0.033 0.011 DBMET01183 | DBMET01182 | |
| 0.022 | 0.029 | 0.031 | Cathepsin K inhibitor | 0.031 0.014 DBMET01183 | DBMET01183 | |
| 0.015 | 0.023 | 0.023 | Human T-cell leukemia virus type I protease inhibitor | 0.023 0.013 DBMET01183 | DBMET01183 | |
| 0.027 | 0.041 | 0.074 | Cathepsin L2 inhibitor | 0.074 0.012 DBMET01183 | DBMET01183 | |
| 0.045 | 0.06 | 0.061 | Bombesin 3 receptor antagonist | 0.061 0.032 DBMET01182 0.06 0.032 DBMET01183 | DBMET01182 | |
| 0.029 | 0.045 | 0.036 | HCV polyprotein inhibitor | 0.036 0.019 DBMET01183 | DBMET01183 | |
| 0.032 | 0.05 | 0.039 | Acetyl-CoA carboxylase inhibitor | 0.039 0.032 DBMET01183 | DBMET01183 | |
| 0.07 | 0.089 | 0.129 | Falcipain inhibitor | 0.129 0.04 DBMET01183 | DBMET01183 | |
| 0.046 | 0.07 | 0.058 | Protease activated receptor antagonist | 0.058 0.05 DBMET01182 | DBMET01182 | |
| 0.026 | 0.052 | 0.033 | Tubulin agonist | 0.033 0.027 DBMET01182 | DBMET01182 | |
| 0.043 | 0.07 | 0.05 | Angiotensin-converting enzyme inhibitor | 0.05 0.046 DBMET01182 0.05 0.048 DBMET01183 | DBMET01183 | |
| 0.036 | 0.07 | 0.11 | Aminopeptidase microsomal inhibitor | 0.11 0.015 DBMET01182 0.079 0.026 DBMET01183 | DBMET01182 | |
| 0.062 | 0.101 | 0.112 | Falcipain 2 inhibitor | 0.112 0.045 DBMET01183 | DBMET01183 | |
| 0.046 | 0.089 | 0.058 | Gonadotropin-releasing hormone receptor agonist | 0.058 0.044 DBMET01182 | DBMET01182 | |
| 0.025 | 0.068 | 0.092 | Aminopeptidase N inhibitor | 0.092 0.015 DBMET01182 0.059 0.025 DBMET01183 | DBMET01182 | |
| 0.032 | 0.076 | 0.039 | Cathepsin F inhibitor | 0.039 0.037 DBMET01182 | DBMET01182 | |
| 0.038 | 0.082 | 0.052 | Carbonic anhydrase II stimulant | 0.052 0.035 DBMET01182 | DBMET01182 | |
| 0.034 | 0.085 | 0.05 | Elastase inhibitor | 0.05 0.042 DBMET01183 | DBMET01183 | |
| 0.02 | 0.071 | 0.037 | Carbonic anhydrase I stimulant | 0.037 0.027 DBMET01182 | DBMET01182 | |
| 0.04 | 0.092 | 0.057 | Acetyl-CoA transferase 2 inhibitor | 0.057 0.039 DBMET01182 | DBMET01182 | |
| 0.033 | 0.094 | 0.047 | HCV NS3/NS4A protease inhibitor | 0.047 0.039 DBMET01183 | DBMET01183 | |
| 0.007 | 0.094 | 0.052 | Aminopeptidase P inhibitor | 0.052 0.004 DBMET01182 | DBMET01182 | |
| 0.077 | 0.164 | 0.106 | Cell adhesion inhibitor | 0.106 0.079 DBMET01182 | DBMET01182 | |
| 0.092 | 0.188 | 0.17 | Growth hormone agonist | 0.17 0.073 DBMET01182 0.149 0.088 DBMET01183 | DBMET01182 | |
| 0.057 | 0.184 | 0.116 | Histone deacetylase class III inhibitor | 0.116 0.073 DBMET01183 | DBMET01183 | |
| 0.071 | 0.205 | 0.139 | Angiogenesis stimulant | 0.136 0.131 DBMET01182 0.139 0.129 DBMET01183 | DBMET01183 | |
| 0.082 | 0.216 | 0.221 | Thiol protease inhibitor | 0.221 0.033 DBMET01183 | DBMET01183 | |
| 0.121 | 0.277 | 0.405 | Calpain 2 inhibitor | 0.405 0.059 DBMET01183 | DBMET01183 | |
| 0.055 | 0.225 | 0.103 | Microtubule formation inhibitor | 0.103 0.085 DBMET01182 | DBMET01182 | |
| 0.031 | 0.211 | 0.075 | Protease 3C (Human rhinovirus) inhibitor | 0.075 0.031 DBMET01183 | DBMET01183 | |
| 0.035 | 0.221 | 0.086 | Opioid antagonist | 0.086 0.062 DBMET01182 | DBMET01182 | |
| 0.07 | 0.274 | 0.134 | Interleukin antagonist | 0.134 0.132 DBMET01182 | DBMET01182 | |
| 0.045 | 0.258 | 0.122 | Thrombolytic | 0.122 0.108 DBMET01183 | DBMET01183 | |
| 0.011 | 0.242 | 0.069 | Cathepsin L inhibitor | 0.069 0.03 DBMET01183 | DBMET01183 | |
| 0.014 | 0.259 | 0.04 | Plasmepsin II inhibitor | 0.04 0.031 DBMET01183 | DBMET01183 | |
| 0.005 | 0.263 | 0.041 | Cathepsin L1 inhibitor | 0.041 0.025 DBMET01183 | DBMET01183 | |
| 0.006 | 0.273 | 0.059 | Ribonucleoside-diphosphate reductase inhibitor | 0.056 0.036 DBMET01182 0.059 0.035 DBMET01183 | DBMET01183 | |
| 0.005 | 0.277 | 0.076 | Ribonucleotide reductase inhibitor | 0.056 0.039 DBMET01182 0.076 0.028 DBMET01183 | DBMET01183 | |
| 0.101 | 0.418 | 0.163 | Peptidyltransferase inhibitor | 0.163 0.162 DBMET01182 | DBMET01182 | |
| 0.031 | 0.4 | 0.182 | Cathepsin H inhibitor | 0.114 0.084 DBMET01182 0.182 0.028 DBMET01183 | DBMET01183 | |
| 0.07 | 0.48 | 0.298 | Toll-Like receptor agonist | 0.298 0.112 DBMET00385 | DBMET00385 | |
| 0.06 | 0.472 | 0.242 | Antithrombotic | 0.242 0.133 DBMET01183 | DBMET01183 | |
| 0.07 | 0.484 | 0.295 | Toll-Like receptor 7 agonist | 0.295 0.113 DBMET00385 | DBMET00385 | |
| 0.009 | 0.425 | 0.071 | Catalase inhibitor | 0.071 0.054 DBMET01183 | DBMET01183 | |
| 0.019 | 0.487 | 0.086 | Interleukin 1 beta converting enzyme inhibitor | 0.086 0.079 DBMET01183 | DBMET01183 | |
| 0.011 | 0.484 | 0.067 | Carbonic anhydrase stimulant | 0.067 0.034 DBMET01182 | DBMET01182 | |
| 0.015 | 0.601 | 0.152 | Aminopeptidase B inhibitor | 0.152 0.037 DBMET01182 | DBMET01182 | |
| 0.013 | 0.647 | 0.176 | Immunostimulant | 0.176 0.135 DBMET01182 | DBMET01182 | |
| 0.017 | 0.659 | 0.054 | Immunoglobulin Fc receptor antagonist | 0.054 0.043 DBMET01182 | DBMET01182 | |
| 0.007 | 0.662 | 0.081 | Aminopeptidase I inhibitor | 0.081 0.041 DBMET01182 | DBMET01182 | |
| 0.014 | 0.85 | 0.191 | Insulysin inhibitor | 0.191 0.171 DBMET01182 | DBMET01182 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |