Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.8470.0020.8475 Hydroxytryptamine 2C agonist

0.149 0.005 DBMET00949

0.8250.0030.8255 Hydroxytryptamine agonist

0.165 0.019 DBMET00949

0.7480.0050.7485 Hydroxytryptamine release stimulant

0.686 0.008 DBMET00949

0.21 0.113 DBMET00950

0.690.0020.69GABA C receptor agonist

0.656 0.002 DBMET00949

0.231 0.016 DBMET00950

0.6490.0040.649GABA C receptor rho-3 antagonist

0.439 0.046 DBMET00949

0.301 0.115 DBMET00950

0.6360.0040.636Alpha-N-acetylglucosaminidase inhibitor

0.386 0.01 DBMET00949

0.561 0.004 DBMET00950

0.6170.0060.617Superoxide dismutase inhibitor

0.272 0.062 DBMET00949

0.186 0.134 DBMET00950

0.5860.0040.5865 Hydroxytryptamine 1F antagonist
0.5980.0190.598Aldehyde oxidase inhibitor

0.167 0.125 DBMET00950

0.5950.0210.595Antiobesity
0.6030.0360.603Caspase 9 stimulant

0.431 0.093 DBMET00949

0.307 0.186 DBMET00950

0.5720.0110.572Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.467 0.051 DBMET00949

0.297 0.217 DBMET00950

0.540.0050.54Antiadrenergic
0.5390.0050.539Adrenaline antagonist
0.5150.0040.5155 Hydroxytryptamine uptake stimulant

0.475 0.005 DBMET00949

0.26 0.072 DBMET00950

0.5050.0040.5055 Hydroxytryptamine uptake inhibitor

0.096 0.028 DBMET00949

0.4880.0040.4885 Hydroxytryptamine 7 antagonist
0.4910.010.491Peroxidase inhibitor

0.112 0.108 DBMET00949

0.4790.0070.479Calcium channel activator

0.334 0.061 DBMET00949

0.251 0.146 DBMET00950

0.4990.0330.4995 Hydroxytryptamine release inhibitor

0.289 0.178 DBMET00949

0.4940.0290.494Vasodilator, peripheral

0.339 0.078 DBMET00949

0.232 0.142 DBMET00950

0.4730.010.473Ca2+/calmodulin-dependent kinase II alpha inhibitor
0.4560.0050.456Tyrosine 3 hydroxylase inhibitor

0.375 0.011 DBMET00949

0.294 0.036 DBMET00950

0.4460.0050.446Protein kinase (CaMK, MLCK, PhK, SNF, KIN, NIM1, MAPKAP, POLO, CHK, ULK, RSK-2nd domain) inhibitor

0.07 0.06 DBMET00949

0.4550.020.455HERG channel blocker
0.4290.0030.429GABA C receptor antagonist

0.36 0.004 DBMET00949

0.117 0.055 DBMET00950

0.4640.0430.464Calcium channel L-type activator

0.361 0.109 DBMET00949

0.420.0030.42Protein kinase C mu inhibitor

0.116 0.044 DBMET00949

0.410.0040.41Ferrochelatase inhibitor

0.14 0.042 DBMET00949

0.116 0.057 DBMET00950

0.3760.0050.376Check point kinase 1 inhibitor

0.065 0.051 DBMET00949

0.4110.0520.411MAP kinase kinase 6 inhibitor
0.3860.0290.386Potassium channel (Voltage-sensitive) blocker
0.3630.0090.363Ca2+/calmodulin-dependent kinase IV inhibitor

0.278 0.038 DBMET00949

0.3780.0250.378DNA synthesis inhibitor

0.287 0.048 DBMET00949

0.325 0.036 DBMET00950

0.4160.0670.416Histamine release inhibitor
0.3720.0270.372Psychostimulant

0.18 0.093 DBMET00949

0.3610.0230.361Cyclic AMP phosphodiesterase inhibitor

0.183 0.108 DBMET00950

0.3640.0250.364Interleukin agonist

0.266 0.068 DBMET00949

0.176 0.144 DBMET00950

0.3370.0040.337MAP-kinase-activated kinase inhibitor

0.117 0.027 DBMET00949

0.3480.0150.348Cyclin-dependent kinase inhibitor

0.146 0.058 DBMET00949

0.3470.0140.347Phospholipase C inhibitor

0.16 0.087 DBMET00949

0.154 0.099 DBMET00950

0.3320.0040.332Adrenaline uptake inhibitor

0.123 0.014 DBMET00949

0.330.0030.33GABA C receptor rho-1 antagonist

0.28 0.004 DBMET00949

0.094 0.071 DBMET00950

0.3720.0450.372Vasodilator, coronary

0.257 0.128 DBMET00949

0.263 0.122 DBMET00950

0.330.0040.33Cyclin-dependent kinase 4 inhibitor

0.07 0.041 DBMET00949

0.3270.0040.327CXC chemokine 4 receptor antagonist

0.084 0.029 DBMET00949

0.3250.0050.325Activin receptor-like kinase 4 inhibitor
0.3220.0050.322GABA C receptor rho-2 antagonist

0.202 0.028 DBMET00949

0.3270.0170.327MAP-kinase-activated kinase 5 inhibitor
0.3260.0170.3265 Hydroxytryptamine 1E antagonist

0.256 0.068 DBMET00949

0.3150.0080.315Nitric-oxide synthase stimulant

0.233 0.045 DBMET00949

0.213 0.07 DBMET00950

0.310.0040.315 Hydroxytryptamine 3E antagonist

0.23 0.027 DBMET00949

0.3050.0040.305MAP-kinase-activated kinase 2 inhibitor

0.111 0.023 DBMET00949

0.3040.0050.304ALK inhibitor
0.3010.0040.3015 Hydroxytryptamine 3A agonist

0.182 0.021 DBMET00949

0.3040.010.304UDP-glucose 4-epimerase inhibitor

0.159 0.026 DBMET00949

0.2 0.018 DBMET00950

0.2940.0050.294Pim-1 kinase inhibitor
0.3140.0290.314RNA-directed DNA polymerase inhibitor

0.212 0.083 DBMET00949

0.191 0.114 DBMET00950

0.310.0320.31MAP kinase kinase 2 inhibitor
0.3080.0310.308Anesthetic general

0.144 0.12 DBMET00949

0.134 0.132 DBMET00950

0.3210.0470.321Insulysin inhibitor

0.234 0.112 DBMET00949

0.2790.0040.279Protein kinase C delta inhibitor
0.2980.0340.298Gastrin inhibitor

0.225 0.112 DBMET00949

0.2670.0030.267Nicotinic receptor alpha4 subunit antagonist

0.094 0.009 DBMET00949

0.2830.0210.283Tyrosine-protein kinase receptor FLT3 inhibitor
0.2640.0080.2645 Hydroxytryptamine 1 agonist
0.2720.0160.272Succinate dehydrogenase inhibitor

0.167 0.084 DBMET00949

0.176 0.073 DBMET00950

0.2580.0050.258Alcohol oxidase inhibitor

0.06 0.035 DBMET00949

0.137 0.012 DBMET00950

0.2560.0070.256Porphobilinogen synthase inhibitor

0.069 0.056 DBMET00949

0.2740.0260.274I kappa B kinase epsilon inhibitor

0.142 0.129 DBMET00949

0.2530.010.253Adenylate kinase inhibitor

0.112 0.051 DBMET00949

0.165 0.022 DBMET00950

0.2590.0190.259Cyclin-dependent kinase 7 inhibitor
0.2430.0040.243Toll-Like receptor 7 antagonist

0.067 0.049 DBMET00949

0.2430.0040.243CDK4/cyclin D1 inhibitor
0.2640.0270.264Tumour necrosis factor antagonist
0.2410.0040.241Protein kinase C alpha inhibitor
0.2590.0240.2593C-like protease (Human coronavirus) inhibitor

0.163 0.082 DBMET00949

0.2430.0080.243NADH dehydrogenase inhibitor

0.097 0.047 DBMET00949

0.136 0.021 DBMET00950

0.30.0660.3Hypoxia-inducible factor 1 alpha inhibitor
0.2420.010.242UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor

0.131 0.033 DBMET00949

0.156 0.025 DBMET00950

0.2360.0080.236Triose-phosphate isomerase inhibitor

0.104 0.044 DBMET00949

0.157 0.018 DBMET00950

0.2320.0050.232Cyclin B3 inhibitor

0.088 0.034 DBMET00949

0.2880.0620.288DNA damaging
0.3050.0850.305Antithrombotic

0.241 0.133 DBMET00950

0.2580.0390.258Glyceraldehyde-3-phosphate dehydrogenase inhibitor

0.218 0.059 DBMET00949

0.248 0.044 DBMET00950

0.3060.0870.306Cholesterol antagonist

0.188 0.176 DBMET00950

0.2220.0050.933Poly(ADP-ribose) polymerase inhibitor

0.933 0.001 DBMET00949

DBMET00949
0.2270.0110.227Polo-like kinase-4 inhibitor
0.2230.0070.223Adenylate cyclase stimulant

0.17 0.035 DBMET00949

0.166 0.04 DBMET00950

0.2570.0440.257DNA methyltransferase I inhibitor

0.182 0.079 DBMET00949

0.2340.0240.234Toll-Like receptor 9 antagonist

0.163 0.055 DBMET00949

0.2150.0090.215Creatine kinase inhibitor

0.104 0.055 DBMET00949

0.171 0.017 DBMET00950

0.2240.0190.224Alpha 2b adrenoreceptor antagonist

0.103 0.072 DBMET00949

0.2160.0110.216Histidine decarboxylase inhibitor

0.077 0.045 DBMET00949

0.063 0.058 DBMET00950

0.2380.0370.238Protein kinase C nu inhibitor
0.2060.0050.206I kappa B kinase 1 inhibitor
0.2480.0490.248DNA methylase inhibitor

0.187 0.088 DBMET00949

0.2030.0050.203Protein kinase C iota inhibitor

0.103 0.018 DBMET00949

0.2030.0050.203CDK4/cyclin D inhibitor
0.240.0430.24Focal adhesion kinase 2 inhibitor
0.2190.0230.219Cyclin-dependent kinase 1 inhibitor

0.168 0.034 DBMET00949

0.1980.0030.198Alpha 1b adrenoreceptor agonist
0.2270.0320.227Acetylcholine M1 receptor antagonist

0.223 0.033 DBMET00949

0.128 0.098 DBMET00950

0.2010.0090.2015 Hydroxytryptamine 1A agonist
0.1960.0040.196Alpha 2 adrenoreceptor agonist

0.112 0.012 DBMET00949

0.20.0090.2Prolactin inhibitor

0.145 0.024 DBMET00949

0.2360.0470.236Neurotrophic factor enhancer
0.1910.0030.191Motilin receptor agonist

0.029 0.01 DBMET00949

0.1910.0050.925Poly(ADP-ribose) polymerase 1 inhibitor

0.925 0.001 DBMET00949

DBMET00949
0.1930.0060.193Biliverdin reductase inhibitor

0.065 0.036 DBMET00949

0.095 0.02 DBMET00950

0.2160.030.216Activin receptor-like kinase 2 inhibitor
0.20.0140.2Protein kinase C gamma inhibitor

0.101 0.075 DBMET00949

0.1950.0090.195Alpha adrenoreceptor agonist

0.08 0.038 DBMET00949

0.2120.0270.212Toll-Like receptor antagonist

0.119 0.086 DBMET00949

0.2150.030.215NADPH oxidase inhibitor
0.1930.0080.193Carbamoyl phosphate synthetase inhibitor

0.104 0.019 DBMET00949

0.133 0.013 DBMET00950

0.1970.0120.197HIV-1 integrase (Overall Integration) inhibitor

0.085 0.071 DBMET00949

0.1840.0050.184Nicotinic alpha4beta2 receptor antagonist

0.132 0.012 DBMET00949

0.1890.0090.189CDK1/cyclin B1 inhibitor

0.154 0.015 DBMET00949

0.2150.0360.215Vascular endothelial growth factor 3 antagonist
0.20.0210.2CF transmembrane conductance regulator agonist

0.138 0.099 DBMET00949

0.146 0.083 DBMET00950

0.1880.010.188Electrolyte absorption antagonist
0.1970.0190.197CDK/cyclin complex inhibitor

0.081 0.067 DBMET00949

0.1850.0080.185Phenylalanine 4-hydroxylase inhibitor
0.2050.0280.205Catenin beta inhibitor
0.1820.0060.182Ca2+-transporting ATPase inhibitor

0.153 0.035 DBMET00949

0.168 0.014 DBMET00950

0.1770.0010.177Alpha 1L adrenoreceptor agonist

0.042 0.032 DBMET00949

0.190.0150.19Protein kinase A inhibitor
0.2350.0610.235Ca2+/calmodulin-dependent protein kinase inhibitor
0.190.0160.19Acetylcholine agonist

0.156 0.024 DBMET00949

0.2020.0290.202Cell wall synthesis inhibitor

0.159 0.057 DBMET00949

0.116 0.106 DBMET00950

0.2140.0410.214Cytidine deaminase inhibitor
0.2040.0320.581Death-associated protein kinase 2 inhibitor

0.581 0.002 DBMET00949

DBMET00949
0.1760.0040.1765 Hydroxytryptamine 3 agonist

0.095 0.017 DBMET00949

0.1890.0190.189Alpha 2 adrenoreceptor antagonist

0.098 0.05 DBMET00949

0.180.010.18Acetylcholine nicotinic agonist

0.137 0.021 DBMET00949

0.1850.0160.185Alpha 2a adrenoreceptor antagonist

0.08 0.049 DBMET00949

0.1810.0130.362Death-associated protein kinase 1 inhibitor

0.362 0.003 DBMET00949

DBMET00949
0.2370.0690.237Neuropeptide Y2 antagonist

0.208 0.105 DBMET00949

0.2560.0890.256Spasmolytic
0.2080.0410.208Amylase inhibitor

0.109 0.088 DBMET00950

0.20.0330.2Arachidonic acid antagonist

0.192 0.041 DBMET00950

0.1870.020.187Check point kinase 2 inhibitor
0.1740.0080.174Histamine N-methyltransferase inhibitor

0.078 0.069 DBMET00949

0.170.0040.175 Hydroxytryptamine 1B agonist
0.180.0150.18Acetylcholine nicotinic antagonist

0.115 0.032 DBMET00949

0.1830.0180.183Interleukin 8 antagonist

0.119 0.062 DBMET00949

0.1920.0270.192Toll-Like receptor 2 antagonist

0.109 0.091 DBMET00949

0.1990.0360.199Cyclin-dependent kinase 8 inhibitor

0.133 0.099 DBMET00949

0.1690.0060.169Protein kinase C eta inhibitor
0.1990.0350.199Neurotensin receptor agonist

0.164 0.072 DBMET00949

0.1870.0240.187Nav1.6 sodium channel blocker
0.1830.0210.183Sphingosine 1-phosphate receptor 5 antagonist

0.138 0.084 DBMET00949

0.1660.0040.166Somatostatin 4 agonist

0.085 0.008 DBMET00949

0.1660.0050.166Glycine receptor antagonist

0.104 0.029 DBMET00949

0.092 0.041 DBMET00950

0.1660.0050.166Alpha 2d adrenoreceptor antagonist
0.1710.010.171Acetylcholine M3 receptor agonist

0.126 0.032 DBMET00949

0.1740.0140.174Phosphofructokinase-1 inhibitor

0.079 0.041 DBMET00949

0.149 0.018 DBMET00950

0.2970.1380.324Antibacterial

0.324 0.118 DBMET00950

DBMET00950
0.1670.0080.167Acyl-CoA dehydrogenase inhibitor

0.047 0.046 DBMET00949

0.087 0.02 DBMET00950

0.1620.0050.1625 Hydroxytryptamine 2A agonist

0.089 0.02 DBMET00949

0.2020.0450.202Ca2+/calmodulin-dependent kinase II delta inhibitor
0.1570.0030.157Dopamine D5 agonist

0.117 0.004 DBMET00949

0.04 0.027 DBMET00950

0.170.0160.17Nitric-oxide synthase inhibitor

0.126 0.034 DBMET00949

0.1760.0230.176Alpha 2c adrenoreceptor antagonist

0.112 0.055 DBMET00949

0.1560.0040.156Cyclin D3 inhibitor
0.1630.0140.163Glutamate dehydrogenase inhibitor

0.082 0.043 DBMET00949

0.102 0.029 DBMET00950

0.1660.0170.166Protein kinase C zeta inhibitor

0.095 0.057 DBMET00949

0.1670.0190.167Calcium antagonist
0.1590.0110.159Neuronal nicotinic receptor antagonist

0.103 0.023 DBMET00949

0.1570.0110.157Argininosuccinate synthase inhibitor

0.071 0.03 DBMET00949

0.087 0.023 DBMET00950

0.1760.030.176Cyclooxygenase 3 inhibitor

0.14 0.058 DBMET00950

0.1830.0370.183Cholinergic antagonist

0.156 0.049 DBMET00949

0.2060.0610.206Histone acetyltransferase inhibitor
0.2280.0830.416Vasodilator

0.156 0.149 DBMET00949

0.416 0.02 DBMET00950

DBMET00950
0.1590.0140.159Inducible nitric-oxide synthase inhibitor

0.107 0.031 DBMET00949

0.1760.0310.176Cystathionine beta-synthase inhibitor

0.092 0.087 DBMET00950

0.1490.0050.1495 Hydroxytryptamine 2 agonist

0.056 0.032 DBMET00949

0.1470.0030.147Phospholipase D inhibitor

0.086 0.026 DBMET00949

0.1730.0290.173Aminopeptidase B inhibitor

0.116 0.055 DBMET00949

0.160.0170.16Transcription factor STAT6 inhibitor

0.11 0.08 DBMET00949

0.180.0370.18Acetylcholine antagonist

0.153 0.049 DBMET00949

0.1590.0170.159DOPA decarboxylase inhibitor

0.124 0.041 DBMET00949

0.1 0.076 DBMET00950

0.1640.0210.164DNA repair enzyme inhibitor

0.114 0.085 DBMET00949

0.1660.0240.166Sphingosine 1-phosphate receptor 2 antagonist
0.2380.0960.238Transcription factor STAT inhibitor
0.1720.0310.277Aurora-C kinase inhibitor

0.277 0.006 DBMET00949

DBMET00949
0.1460.0050.146Acetylcholine M5 receptor agonist

0.084 0.031 DBMET00949

0.1850.0440.185Ribosomal protein S6 kinase inhibitor
0.1470.0060.147Protein kinase C epsilon inhibitor
0.1440.0040.144Myc inhibitor

0.094 0.009 DBMET00949

0.150.010.15CXC chemokine receptor antagonist
0.1480.0080.148Viral attachment inhibitor

0.088 0.036 DBMET00949

0.1520.0130.152Glutamate decarboxylase inhibitor

0.073 0.052 DBMET00949

0.078 0.046 DBMET00950

0.160.0210.16Sphingosine 1-phosphate receptor 2 agonist
0.1530.0150.153Acetylcholine release stimulant

0.107 0.071 DBMET00949

0.136 0.028 DBMET00950

0.1870.0490.187ATPase inhibitor
0.1480.010.148Acetylcholine muscarinic agonist

0.114 0.015 DBMET00949

0.1710.0340.171MAP3K9 inhibitor
0.1650.030.165Falcipain 3 inhibitor
0.1370.0030.137Alpha 1a adrenoreceptor agonist
0.1610.0270.161Heat shock protein 70 antagonist

0.133 0.107 DBMET00949

0.190.0560.19Antipruritic
0.1650.0310.165Pregnane X receptor agonist

0.143 0.067 DBMET00949

0.2160.0830.216Potassium channel blocker
0.1650.0320.165Cyclin-dependent kinase 2 inhibitor
0.140.0080.14Glycine receptor agonist

0.099 0.022 DBMET00949

0.083 0.035 DBMET00950

0.2030.0710.203Proto-oncogene tyrosine-protein kinase Fyn inhibitor
0.1510.0190.151Rho-associated kinase inhibitor
0.1350.0040.135Mannosidase inhibitor

0.08 0.009 DBMET00949

0.081 0.008 DBMET00950

0.1340.0030.1345 Hydroxytryptamine 2B agonist

0.052 0.012 DBMET00949

0.1440.0140.144Lanosterol 14 alpha demethylase inhibitor

0.09 0.073 DBMET00949

0.111 0.04 DBMET00950

0.2440.1140.244Nootropic
0.1750.0460.175Hemostatic
0.1650.0370.165Cathepsin H inhibitor

0.118 0.078 DBMET00949

0.111 0.088 DBMET00950

0.1330.0050.133Protein kinase C beta inhibitor

0.077 0.034 DBMET00949

0.1360.0090.136Acetylcholine M1 receptor agonist

0.105 0.012 DBMET00949

0.1370.0090.137Mannitol-1-phosphate 5-dehydrogenase inhibitor

0.079 0.021 DBMET00950

0.1510.0240.151Beta glucuronidase inhibitor
0.1550.030.155Chemokine receptor antagonist
0.1730.0470.173Mannose-6-phosphate isomerase inhibitor
0.130.0050.13GABA B receptor agonist

0.081 0.04 DBMET00949

0.081 0.04 DBMET00950

0.1280.0030.128Alpha 1d adrenoreceptor agonist

0.038 0.028 DBMET00949

0.1380.0130.138Glutamate release inhibitor
0.1360.0130.136Interferon agonist
0.160.0370.165 Hydroxytryptamine 2B antagonist
0.1320.010.132Granulocyte macrophage colony stimulating factor agonist

0.083 0.067 DBMET00949

0.1750.0530.175Hexokinase inhibitor
0.170.0470.17Nav1.2 sodium channel blocker
0.160.0380.16Acetylcholine muscarinic antagonist

0.142 0.049 DBMET00949

0.1520.030.152Photosensitizer
0.1280.0060.128Cyclin B1 inhibitor
0.1370.0150.137Aminopeptidase I inhibitor

0.074 0.049 DBMET00949

0.092 0.033 DBMET00950

0.1780.0570.178Cholinergic

0.161 0.069 DBMET00950

0.1650.0440.165Neuropeptide Y1 antagonist

0.153 0.061 DBMET00949

0.1270.0060.127Histamine agonist

0.066 0.022 DBMET00949

0.1240.0040.124MAP kinase kinase 7 inhibitor

0.099 0.013 DBMET00949

0.095 0.018 DBMET00950

0.1590.0390.159Adenylate cyclase inhibitor
0.2450.1250.245Interleukin 2 agonist

0.242 0.128 DBMET00950

0.1250.0050.125Protein kinase C theta inhibitor
0.1390.0190.139CYP2A6 inhibitor
0.1730.0540.173Protein kinase stimulant

0.112 0.102 DBMET00949

0.126 0.087 DBMET00950

0.1270.0080.127Nicotinic receptor alpha7 subunit antagonist

0.08 0.017 DBMET00949

0.1260.0080.1265 Hydroxytryptamine 3A antagonist

0.067 0.046 DBMET00949

0.1390.0220.139Pim-3 kinase inhibitor

0.097 0.049 DBMET00949

0.1360.0180.136Glutamate (mGluR7) agonist

0.09 0.083 DBMET00949

0.1360.0190.136Adrenaline agonist
0.1250.0080.125Dopamine transporter inhibitor

0.07 0.021 DBMET00949

0.1190.0020.119Phenylethanolamine N methyltransferase inhibitor

0.082 0.004 DBMET00949

0.1440.0280.144Catalase inhibitor
0.2230.1080.223Transcription factor STAT3 inhibitor
0.1380.0220.138MAP kinase kinase 1 inhibitor
0.1310.0170.131Bromodomain-containing protein 2 inhibitor

0.088 0.058 DBMET00949

0.1190.0050.119Exportin-1 inhibitor
0.1180.0050.118Alpha-mannosidase inhibitor

0.078 0.012 DBMET00949

0.094 0.007 DBMET00950

0.1840.0710.184LIM domain kinase 1 inhibitor
0.1180.0050.118Poly(ADP-ribose) polymerase 2 inhibitor
0.1270.0130.127Carbonic anhydrase stimulant
0.1680.0550.168Protein kinase (CK1) inhibitor
0.1210.0080.121CC chemokine 5 receptor agonist

0.115 0.01 DBMET00949

0.2570.1450.257Calpain 2 inhibitor
0.1550.0430.1555 Hydroxytryptamine 2 antagonist
0.220.1090.22Immunostimulant
0.1960.0850.196Anticonvulsant
0.1170.0060.117Cyclin-dependent kinase 6 inhibitor

0.087 0.017 DBMET00949

0.1440.0330.144Carbonic anhydrase XV inhibitor
0.1240.0130.124Caspase 7 inhibitor
0.1150.0050.115Nicotinic alpha3beta2 receptor antagonist

0.104 0.007 DBMET00949

0.1460.0370.146Sphingosine 1-phosphate receptor 4 antagonist
0.1680.0590.168Interferon gamma antagonist

0.151 0.076 DBMET00950

0.2110.1030.211Calpain inhibitor
0.1890.0810.285Death-associated protein kinase 3 inhibitor

0.285 0.042 DBMET00949

DBMET00949
0.1570.0490.157Sodium channel (voltage-gated) blocker
0.1180.0110.118NMDA 2C receptor antagonist

0.111 0.013 DBMET00949

0.1160.0090.116Nicotinic neuronal receptor agonist

0.086 0.018 DBMET00949

0.1110.0040.111Ryanodine receptor antagonist

0.066 0.023 DBMET00949

0.058 0.044 DBMET00950

0.1360.030.1365 Hydroxytryptamine 2C antagonist
0.1420.0370.142Mucolytic

0.102 0.075 DBMET00950

0.1130.0080.129Cyclin B inhibitor

0.129 0.006 DBMET00949

DBMET00949
0.1170.0130.117Alpha 1 adrenoreceptor agonist
0.1060.0030.106Nicotinic alpha4 receptor agonist

0.047 0.004 DBMET00949

0.1210.0170.121Acetylcholine M4 receptor antagonist

0.09 0.037 DBMET00949

0.1120.0090.112Interferon inducer
0.1620.0590.162Thiol protease inhibitor
0.1080.0060.108Cyclin D1 inhibitor
0.1130.0120.1135 Hydroxytryptamine 6 antagonist

0.057 0.039 DBMET00949

0.1080.0070.108Glucosylceramidase inhibitor

0.058 0.034 DBMET00949

0.054 0.04 DBMET00950

0.150.0490.155 Hydroxytryptamine antagonist
0.2370.1370.237Transcription factor NF kappa B inhibitor
0.130.030.13Phosphodiesterase 7B inhibitor
0.130.0310.13Anabolic

0.088 0.081 DBMET00949

0.123 0.037 DBMET00950

0.110.0110.11Vanilloid 4 agonist

0.095 0.02 DBMET00949

0.07 0.063 DBMET00950

0.1220.0230.122Phosphodiesterase 6D inhibitor
0.1360.0370.136Nav1.5 sodium channel blocker
0.1570.0580.157Proto-oncogene tyrosine-protein kinase Yes inhibitor
0.1060.0070.106Ca(v)3.2 blocker
0.1080.0090.108S-adenosyl-L-methionine decarboxylase inhibitor

0.08 0.037 DBMET00949

0.075 0.047 DBMET00950

0.1170.0190.117mTOR complex 2 inhibitor

0.079 0.072 DBMET00949

0.1470.0490.147Nav1.3 sodium channel blocker
0.1560.0590.156MAP kinase 3 inhibitor

0.133 0.099 DBMET00949

0.1040.0070.104Sphingosine kinase 2 inhibitor

0.075 0.018 DBMET00949

0.077 0.017 DBMET00950

0.1090.0140.1095 Hydroxytryptamine 5A antagonist

0.06 0.045 DBMET00949

0.1030.0080.103Toll-Like receptor 8 antagonist

0.052 0.039 DBMET00949

0.1020.0080.102Aconitate hydratase inhibitor

0.047 0.044 DBMET00950

0.1310.0370.131Carbonic anhydrase III inhibitor
0.1010.0070.101Cyclin H inhibitor

0.07 0.028 DBMET00949

0.1030.0090.103Glutamate (mGluR6) antagonist

0.074 0.032 DBMET00949

0.069 0.041 DBMET00950

0.0960.0030.096Imidazoline I1 receptor antagonist

0.032 0.006 DBMET00949

0.1460.0530.146MAP kinase kinase inhibitor
0.1150.0220.115Myeloperoxidase inhibitor
0.1830.0910.183Ca2+/calmodulin-dependent kinase II beta inhibitor
0.1090.0160.109Estrogen-related receptor beta agonist

0.077 0.076 DBMET00950

0.0970.0050.097Purinergic P2X4 antagonist
0.1060.0140.106NMDA receptor glycine site agonist

0.087 0.023 DBMET00949

0.1240.0320.124Interleukin 1 beta converting enzyme inhibitor
0.1130.0210.113Na+ K+ transporting ATPase inhibitor

0.096 0.035 DBMET00949

0.103 0.029 DBMET00950

0.1060.0150.106Ornithine carbamoyltransferase inhibitor

0.052 0.037 DBMET00949

0.061 0.031 DBMET00950

0.110.0190.11D-Ala-D-Ala ligase inhibitor
0.0960.0050.096Histamine H4 receptor antagonist

0.074 0.01 DBMET00949

0.1340.0440.134TRPA1 agonist
0.1070.0170.107NMDA receptor agonist

0.098 0.02 DBMET00949

0.1040.0140.1045 Hydroxytryptamine 5 antagonist

0.052 0.051 DBMET00949

0.1360.0460.136Microtubule formation inhibitor
0.0930.0040.093Dopamine beta hydroxylase inhibitor
0.140.0510.14Vanilloid 1 agonist
0.140.0520.14Alkylator

0.097 0.091 DBMET00949

0.123 0.066 DBMET00950

0.0960.0080.096Epithelial sodium channel blocker

0.059 0.03 DBMET00949

0.1130.0250.113Histamine H2 receptor antagonist

0.079 0.067 DBMET00949

0.1310.0430.131Alpha adrenoreceptor antagonist
0.0910.0030.091Alpha 2a adrenoreceptor agonist
0.1160.0280.116I kappa B kinase inhibitor
0.1410.0530.141Aldehyde dehydrogenase inhibitor
0.1370.050.137Beta amyloid protein antagonist
0.0960.0090.096Cyclin B2 inhibitor

0.093 0.01 DBMET00949

0.0950.0080.095Corticotropin releasing factor 2 receptor antagonist

0.058 0.051 DBMET00949

0.1060.020.1065 Hydroxytryptamine 1D antagonist

0.058 0.051 DBMET00949

0.0940.0080.0945 Hydroxytryptamine 7 agonist

0.078 0.014 DBMET00949

0.1030.0170.1035 Hydroxytryptamine 3 antagonist

0.053 0.044 DBMET00949

0.0940.0090.094MDM2 inhibitor
0.1060.0210.1065 Hydroxytryptamine 1B antagonist
0.0940.0090.094Sphingosine kinase inhibitor

0.083 0.014 DBMET00949

0.071 0.023 DBMET00950

0.1590.0740.159Polo-like kinase-3 inhibitor
0.090.0050.09Adenylate cyclase 1 inhibitor

0.043 0.038 DBMET00950

0.0950.010.095Topoisomerase II beta inhibitor

0.047 0.038 DBMET00949

0.0890.0050.089Histamine H2 receptor agonist
0.1480.0640.148Cytokine production inhibitor
0.1230.040.123CDK2/cyclin A inhibitor

0.087 0.071 DBMET00949

0.1480.0650.148MAP kinase kinase 4 inhibitor
0.1150.0330.115Polo-like kinase-1 inhibitor
0.1220.040.122Sphingomyelinase inhibitor
0.0890.0070.089Glucose-6-phosphate isomerase inhibitor

0.047 0.035 DBMET00949

0.078 0.009 DBMET00950

0.1390.0570.139Antibacterial (Helicobacter pylori)
0.0880.0070.088Sodium/calcium exchanger inhibitor
0.0990.0180.099GP IIb/IIIa receptor antagonist
0.1190.0380.1195 Hydroxytryptamine 2A antagonist
0.0840.0030.084Nicotinic alpha4beta2 receptor agonist

0.065 0.004 DBMET00949

0.190.1090.19Platelet antagonist
0.1560.0750.156Anticoagulant
0.0890.0090.093Lysine-specific demethylase 1A inhibitor

0.093 0.008 DBMET00949

DBMET00949
0.0940.0140.094Glutamate (mGluR7) antagonist
0.0970.0170.097Purinergic P2X1 antagonist

0.057 0.048 DBMET00950

0.0920.0140.092Heat shock protein 90 beta antagonist
0.1540.0760.154Melanin inhibitor

0.127 0.12 DBMET00950

0.0960.0180.096Acetylcholine M5 receptor antagonist

0.058 0.045 DBMET00949

0.0820.0050.082Vascular adhesion protein 1 inhibitor
0.0820.0050.082Acetylcholine M4 receptor agonist

0.04 0.015 DBMET00949

0.1520.0760.152Diuretic
0.1270.0510.127GABA receptor agonist
0.1020.0260.102GABA aminotransferase inhibitor
0.0910.0160.091I kappa B kinase 2 inhibitor

0.059 0.049 DBMET00949

0.0780.0030.078Nicotinic alpha3beta4 receptor agonist

0.067 0.004 DBMET00949

0.0850.0110.085Acetylcholine M2 receptor agonist

0.059 0.03 DBMET00949

0.0930.0190.093Beta adrenoreceptor antagonist

0.062 0.051 DBMET00949

0.1750.1010.175Insulin sensitizer
0.10.0280.1Histone deacetylase SIRT1 stimulant
0.10.0280.1Histone deacetylase stimulant
0.1120.0390.112NMDA receptor antagonist

0.086 0.058 DBMET00949

0.0930.020.093Dopamine uptake inhibitor

0.065 0.034 DBMET00949

0.1380.0660.138Sodium channel blocker
0.0860.0150.086Histone deacetylase SIRT3 inhibitor
0.1180.0470.118Cyclin-dependent kinase 9 inhibitor

0.096 0.067 DBMET00949

0.0740.0040.074Alpha 2d adrenoreceptor agonist
0.0850.0150.085Beta 1 adrenoreceptor antagonist
0.0960.0260.096CDC7 inhibitor
0.0740.0040.074Protein kinase C beta II inhibitor
0.0970.0280.097Polo-like kinase-2 inhibitor
0.0740.0040.074Histamine H1 receptor agonist

0.053 0.015 DBMET00949

0.0920.0230.092Secretase beta inhibitor
0.1290.060.129Anesthetic local
0.0760.0070.076Histamine H3 receptor agonist
0.0740.0060.074Potassium channel small-conductance Ca-activated activator
0.1020.0340.102Alpha 1b adrenoreceptor antagonist
0.1410.0730.141Glycogen synthase kinase-3 alpha inhibitor
0.0880.020.088Potassium channel (Tandem pore domain) blocker
0.0990.0320.099NMDA 2 receptor antagonist

0.074 0.048 DBMET00949

0.1390.0720.139Histone deacetylase SIRT1 inhibitor
0.080.0140.08Cyclin A1 inhibitor

0.057 0.044 DBMET00949

0.0890.0220.089Acetylcholine M3 receptor antagonist

0.061 0.04 DBMET00949

0.1270.0610.127MAP kinase 12 inhibitor
0.0710.0040.071Protein kinase (CK2) beta inhibitor

0.043 0.01 DBMET00949

0.0810.0150.081Phosphodiesterase 1A inhibitor
0.0830.0170.083Phosphodiesterase 1C inhibitor
0.0720.0070.072Geranyltranstransferase inhibitor
0.1560.090.156Interleukin-1 receptor-associated protein kinase 1 inhibitor
0.0770.0120.077Dihydroorotate oxidase inhibitor
0.070.0040.07Kainate receptor agonist

0.056 0.009 DBMET00949

0.046 0.019 DBMET00950

0.0870.0220.087Protease 3C (Human rhinovirus) inhibitor

0.059 0.054 DBMET00949

0.0710.0060.071Acid-sensing ion channel blocker
0.1160.0520.116AMP-activated protein kinase stimulant
0.0720.0080.072Kainate receptor 2 antagonist

0.031 0.029 DBMET00949

0.0740.010.074CC chemokine receptor 2B antagonist
0.0740.010.074Pregnane X receptor antagonist
0.1160.0530.116Expectorant
0.070.0070.07GABA uptake inhibitor

0.055 0.012 DBMET00949

0.0810.0190.081NMDA 2A receptor antagonist
0.070.0080.07GABA B receptor antagonist

0.049 0.021 DBMET00949

0.0710.010.071Immunoglobulin Fc receptor antagonist

0.052 0.049 DBMET00949

0.1180.0570.118MAP kinase 13 inhibitor
0.1030.0410.103Phosphodiesterase I inhibitor
0.0950.0350.095Rho-associated kinase I inhibitor
0.0710.0110.071Potassium channel (Inward rectifier) activator
0.0740.0140.074Nicotinic receptor alpha3 subunit antagonist

0.056 0.021 DBMET00949

0.0720.0120.072Kainate receptor antagonist
0.0690.0090.069GHS receptor agonist

0.043 0.029 DBMET00949

0.1030.0430.103Bile acid receptor antagonist

0.091 0.07 DBMET00949

0.080.020.08Pim-2 kinase inhibitor
0.0730.0130.073Growth hormone secretagogue receptor agonist
0.0640.0050.064Methionyl aminopeptidase 1 inhibitor
0.0680.0090.068Fumarate hydratase inhibitor

0.047 0.015 DBMET00950

0.0740.0150.074NMDA receptor subunit 3B antagonist

0.048 0.026 DBMET00949

0.0660.0070.066Sphingosine kinase 1 inhibitor

0.057 0.011 DBMET00949

0.047 0.019 DBMET00950

0.1220.0640.122Proteasome inhibitor
0.0660.0080.066Arginase inhibitor

0.053 0.013 DBMET00949

0.0650.0080.065Guanylate cyclase inhibitor

0.044 0.028 DBMET00950

0.0680.010.068Potassium channel (ATP-sensitive) activator
0.0980.040.098Carbonic anhydrase VI inhibitor
0.0640.0060.064Hypoxanthine phosphoribosyltransferase inhibitor

0.027 0.02 DBMET00949

0.024 0.023 DBMET00950

0.0910.0340.091Protein kinase B alpha inhibitor
0.1010.0440.101Interleukin-1 receptor-associated protein kinase 4 inhibitor

0.079 0.072 DBMET00949

0.0730.0160.0735 Hydroxytryptamine 4 antagonist

0.05 0.039 DBMET00949

0.080.0230.08Beta 3 adrenoreceptor antagonist

0.065 0.044 DBMET00949

0.0630.0070.063Protein kinase (CK1) epsilon inhibitor
0.0920.0360.092Keratolytic
0.0710.0160.071Beta 2 adrenoreceptor antagonist

0.048 0.04 DBMET00949

0.0650.010.0655 Hydroxytryptamine 3B antagonist

0.032 0.03 DBMET00949

0.110.0550.11Urease inhibitor
0.0850.030.085Nav1.7 sodium channel blocker
0.0850.030.085Cyclin A2 inhibitor

0.074 0.036 DBMET00949

0.0610.0070.0613-Hydroxyanthranilate 3,4-dioxygenase inhibitor
0.0660.0120.066Glutamate (mGluR4) antagonist

0.054 0.018 DBMET00949

0.0590.0050.059CDK6/cyclin D3 inhibitor
0.0710.0170.071Dipeptidyl peptidase inhibitor

0.053 0.035 DBMET00949

0.0980.0440.098Alpha 1 adrenoreceptor antagonist
0.0740.0210.074Nicotinic alpha7 receptor agonist

0.049 0.044 DBMET00949

0.0660.0120.066CC chemokine 4 receptor antagonist
0.0570.0040.057Myristoyl transferase inhibitor

0.029 0.014 DBMET00949

0.0750.0230.075Enoyl-[acyl-carrier-protein] reductase inhibitor
0.0990.0460.099Aminoacyl-tRNA synthetase inhibitor
0.070.0180.07Chemokine receptor agonist
0.0610.0090.061Nerve growth factor antagonist
0.0560.0040.056Histamine H4 receptor agonist

0.021 0.01 DBMET00949

0.0610.010.061AMPA 4 receptor antagonist

0.05 0.015 DBMET00949

0.0810.030.081Alpha 1d adrenoreceptor antagonist
0.0560.0050.058Epoxide hydrolase 1 inhibitor

0.058 0.005 DBMET00949

DBMET00949
0.1070.0560.107Gastric antisecretory
0.0660.0160.066Adenosine deaminase inhibitor

0.041 0.039 DBMET00950

0.0760.0260.097Androgen agonist

0.097 0.016 DBMET00950

DBMET00950
0.1710.120.171Aryl hydrocarbon receptor agonist
0.060.010.06Diamine oxidase inhibitor
0.080.030.08Acetylcholine M2 receptor antagonist

0.065 0.041 DBMET00949

0.070.020.07Neurokinin antagonist
0.0580.0080.058Glutamate (mGluR8) agonist

0.04 0.022 DBMET00949

0.039 0.023 DBMET00950

0.1070.0580.107Protein kinase (CK2) inhibitor
0.0540.0050.054Bombesin agonist
0.0570.0080.057Endothelial nitric-oxide synthase inhibitor

0.052 0.009 DBMET00949

0.10.0520.1Alcohol dehydrogenase inhibitor
0.0530.0040.0535 Hydroxytryptamine 6 agonist

0.031 0.015 DBMET00949

0.080.0320.117Cyclin E inhibitor

0.117 0.019 DBMET00949

DBMET00949
0.0520.0030.052Alpha 2c adrenoreceptor agonist

0.017 0.016 DBMET00949

0.080.0320.08Cyclin A inhibitor

0.066 0.04 DBMET00949

0.0560.0080.056Integrin alpha2 antagonist

0.042 0.018 DBMET00949

0.0670.0190.067Potassium channel (Inward rectifier) blocker
0.0580.0110.058Membrane dipeptidase inhibitor
0.0510.0030.051Alpha 2b adrenoreceptor agonist
0.080.0330.08Dopamine D1 antagonist
0.0720.0250.072Calcium channel P-type blocker

0.065 0.04 DBMET00950

0.0830.0360.083Phosphodiesterase VI inhibitor
0.1070.060.107MAP kinase kinase kinase inhibitor
0.1170.070.117TRKA antagonist
0.0820.0350.082Sphingosine 1-phosphate receptor 4 agonist
0.0880.0410.088Alpha 1a adrenoreceptor antagonist
0.0860.040.086Rho-associated kinase II inhibitor
0.0880.0420.0885 Hydroxytryptamine 1 antagonist
0.0760.030.076Aryl hydrocarbon receptor antagonist
0.0610.0150.061Glutamate (mGluR1a) antagonist
0.0610.0160.061Oxytocin agonist

0.039 0.033 DBMET00949

0.0620.0160.062NMDA receptor subunit 3A antagonist

0.035 0.029 DBMET00949

0.0580.0120.058Dihydropteroate synthase inhibitor

0.037 0.03 DBMET00949

0.0620.0160.062Thymidylate synthase inhibitor
0.060.0140.06Neurokinin 1 antagonist
0.1410.0960.141Heat shock protein 90 alpha antagonist
0.0870.0420.087Focal adhesion kinase 1 inhibitor
0.0520.0070.052Lysine carboxypeptidase inhibitor

0.031 0.015 DBMET00949

0.0880.0430.088Transforming growth factor beta 3 antagonist
0.0510.0070.051CDK4/cyclin D3 inhibitor

0.033 0.014 DBMET00949

0.0650.0210.065Bombesin 2 receptor antagonist
0.0530.0090.0535 Hydroxytryptamine 1D agonist

0.038 0.015 DBMET00949

0.0490.0050.049Bombesin 3 receptor agonist
0.110.0650.11EphA2 antagonist
0.1670.1230.167Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase inhibitor
0.0480.0040.048Estrogen-related receptor gamma antagonist
0.150.1060.15Platelet adhesion inhibitor
0.0720.0280.072Phosphodiesterase 1B inhibitor
0.1140.0710.114Cholesterol synthesis inhibitor

0.108 0.077 DBMET00950

0.050.0070.05Ceramide glucosyltransferase inhibitor

0.037 0.021 DBMET00949

0.04 0.017 DBMET00950

0.0560.0120.056DNA gyrase subunit A inhibitor

0.04 0.035 DBMET00949

0.070.0270.07Potassium channel intermediate-conductance Ca-activated blocker
0.060.0170.06Potassium channel small-conductance Ca-activated blocker
0.1130.070.113Caspase 3 inhibitor
0.0580.0150.058Thymidine kinase inhibitor

0.043 0.026 DBMET00950

0.0580.0150.058Cytokine production stimulant
0.0940.0510.094Ornithine decarboxylase inhibitor
0.0580.0150.058AICAR transformylase inhibitor

0.048 0.025 DBMET00950

0.0570.0140.057Dipeptidyl peptidase IV inhibitor

0.044 0.032 DBMET00949

0.0470.0050.047Thymidine phosphorylase inhibitor

0.024 0.023 DBMET00949

0.0820.040.082Epoxide hydrolase inhibitor

0.066 0.059 DBMET00949

0.090.0480.09GABA A receptor agonist
0.0560.0140.056Parathyroid hormone antagonist
0.050.0080.05Uridine phosphorylase inhibitor
0.1340.0920.134Heat shock protein 90 antagonist
0.0460.0050.046Protein kinase C beta I inhibitor
0.0870.0460.087NAD(P)H dehydrogenase (quinone) inhibitor
0.0810.040.0815 Hydroxytryptamine 1A antagonist
0.0690.0280.069Carbonic anhydrase VB inhibitor
0.0480.0070.048Transforming growth factor beta 2 antagonist
0.0440.0040.044Acid ceramidase inhibitor

0.026 0.016 DBMET00949

0.1380.0970.138Ca2+/calmodulin-dependent protein kinase kinase B inhibitor
0.0580.0170.058CDK7/cyclin H inhibitor
0.0430.0030.043Imidazoline I2 receptor antagonist
0.0740.0340.074Potassium channel (ATP-sensitive) blocker
0.0440.0050.044Glutamate (mGluR1a) agonist
0.0440.0050.044Purinergic P2Y15 antagonist

0.028 0.021 DBMET00949

0.034 0.011 DBMET00950

0.0610.0230.061Prolyl endopeptidase inhibitor
0.0890.050.089Leucine-rich repeat kinase 2 inhibitor
0.1120.0740.112Calcium channel N-type blocker
0.0430.0050.043MAP3K8 inhibitor
0.0660.0280.066Beta 2 adrenoreceptor agonist
0.0650.0280.065CC chemokine 2 receptor antagonist
0.0450.0080.045Tryptophan 5 hydroxylase inhibitor
0.0450.0090.045Purinergic P2Y14 antagonist
0.080.0440.08Cathepsin G inhibitor
0.1940.1580.19412-Lipoxygenase inhibitor
0.050.0130.05Prostacyclin antagonist
0.2340.1980.234Analgesic
0.1010.0650.101Nav1.1 sodium channel blocker
0.0490.0130.049Potassium channel Kv1.1 blocker
0.0590.0230.059Lysophosphatidic acid 3 receptor antagonist
0.0650.030.116Cyclin E1 inhibitor

0.116 0.015 DBMET00949

DBMET00949
0.1210.0860.121Tyrosine-protein kinase receptor antagonist
0.0940.0590.094Antihistaminic
0.0590.0240.059Carbonic anhydrase II stimulant
0.090.0550.09Insulin growth factor antagonist
0.0570.0220.057Aldosterone antagonist
0.0530.0180.053Glutamate (mGluR group III) antagonist

0.047 0.025 DBMET00949

0.0670.0330.067Glutamate (mGluR1) antagonist
0.0650.0310.065Botulinum neurotoxin type A inhibitor
0.0430.0090.043Estrogen-related receptor beta antagonist
0.040.0070.04Kainate receptor 1 antagonist
0.0760.0430.076Benzodiazepine agonist
0.0440.0110.044Cyclin E2 inhibitor
0.0570.0240.057Squalene epoxidase inhibitor
0.0610.0280.0613(or 17)beta-hydroxysteroid dehydrogenase inhibitor
0.0690.0360.069Phosphodiesterase VII inhibitor
0.1050.0720.105Monophenol monooxygenase inhibitor
0.0430.0110.043Lysophosphatidic acid 2 receptor antagonist
0.0360.0040.036Complement factor 1s inhibitor
0.0930.0610.093Potassium channel (Ca-activated) activator
0.0410.0090.041NMDA 2D receptor antagonist
0.0620.030.062GABA receptor antagonist
0.0850.0540.085Insulin like growth factor 1 antagonist
0.0360.0040.036Cyclin T1 inhibitor

0.03 0.005 DBMET00949

0.0660.0350.066Plasminogen activator inhibitor
0.0370.0060.037Nicotinic acid receptor 2 antagonist
0.0450.0150.045Somatostatin 5 agonist
0.0530.0220.053Dihydroorotase inhibitor
0.0360.0050.036Glutaminyl-peptide cyclotransferase inhibitor
0.0730.0420.073Dopamine agonist
0.0490.0180.049Renin inhibitor
0.0550.0250.055HCV NS3/NS4A protease inhibitor
0.0960.0670.096Insulin receptor antagonist
0.1130.0830.113TRKB antagonist
0.10.0710.1Granulocyte macrophage colony stimulating factor antagonist
0.0470.0180.047Heme oxygenase inhibitor
0.0780.0490.078MAP kinase 11 inhibitor
0.0450.0160.045Phosphoglycerate kinase inhibitor
0.0570.0280.057Heparanase inhibitor
0.0360.0070.036Glutamate (mGluR1) agonist

0.027 0.013 DBMET00949

0.0920.0640.092Fibroblast growth factor 1 antagonist
0.0740.0450.074Orexin receptor 1 antagonist
0.0720.0440.072Carbonic anhydrase VA inhibitor
0.0440.0150.044Somatostatin agonist
0.080.0510.08Fibroblast growth factor 3 antagonist
0.1170.0880.117Bone formation stimulant
0.0390.0110.039Glutamate (mGluR3) agonist

0.031 0.027 DBMET00949

0.0620.0330.062Fatty acid synthase inhibitor
0.0730.0450.073CDK2/cyclin E2 inhibitor

0.068 0.05 DBMET00949

0.0470.0190.047Substance P antagonist
0.0620.0350.062Sphingosine 1-phosphate receptor 3 antagonist
0.0790.0520.08Somatostatin 1 agonist

0.08 0.051 DBMET00949

DBMET00949
0.0790.0520.079CC chemokine receptor antagonist
0.040.0130.04Melatonin receptor 1A agonist
0.0340.0070.034Glucosylceramidase stimulant
0.0310.0040.031Carbonic anhydrase X inhibitor
0.0310.0040.031Carbonic anhydrase VIII inhibitor
0.0410.0140.041CXC chemokine receptor agonist
0.0660.0390.066Transcription factor RelA inhibitor
0.1170.0910.117Calcium channel blocker
0.0850.0590.085Histamine antagonist
0.0430.0170.043Glutamate (mGluR3) antagonist

0.036 0.026 DBMET00950

0.0620.0360.062Cathepsin L inhibitor
0.1050.0790.105CDK3/cyclin E inhibitor
0.0340.0080.034Thymidine kinase (Herpes simplex virus 1) inhibitor

0.028 0.015 DBMET00950

0.1090.0830.109Protein kinase (CK1) delta inhibitor
0.0580.0320.058GABA A receptor antagonist
0.0390.0140.039ATR kinase inhibitor

0.031 0.026 DBMET00949

0.030.0050.03Factor XIII inhibitor
0.0390.0140.039AMPA 3 receptor antagonist

0.031 0.019 DBMET00949

0.0510.0260.051Purinergic P2Y antagonist
0.1880.1630.188MAP kinase kinase 3 inhibitor
0.0730.0480.073Calcium channel L-type blocker
0.0350.0110.035Methionyl aminopeptidase 2 inhibitor
0.0340.010.034Calcium-sensing receptor agonist
0.0550.030.055Phosphodiesterase 7A inhibitor
0.0330.0090.033Hedgehog signaling activator

0.027 0.021 DBMET00950

0.0290.0050.029Thymidine kinase (Herpes simplex virus 2) inhibitor

0.021 0.013 DBMET00950

0.0440.020.044Nicotinic receptor beta4 subunit antagonist
0.1550.1310.155MAP kinase kinase 5 inhibitor
0.0750.0510.075Adenosine A3 receptor antagonist
0.0670.0430.067Neutrophil collagenase inhibitor
0.1270.1040.127Tyrosine kinase inhibitor
0.0440.020.044Carbonic anhydrase I stimulant
0.0320.0090.032Lysophosphatidic acid receptor 1 agonist
0.0380.0150.038Dipeptidyl peptidase II inhibitor

0.036 0.018 DBMET00949

0.0260.0030.026Cyclin D2 inhibitor

0.014 0.008 DBMET00949

0.0330.010.033Integrin alpha2beta1 antagonist
0.0310.0080.031Vanilloid 2 agonist

0.024 0.022 DBMET00950

0.0840.0610.084Hematopoietic
0.1450.1220.145Non-steroidal antiinflammatory agent
0.0380.0150.038Adenosine uptake inhibitor
0.0750.0530.075Carbonic anhydrase XIII inhibitor
0.0830.0610.083Bcr-Abl kinase inhibitor
0.0410.020.041Delayed rectifier potassium channel blocker
0.0520.030.052Antimetabolite
0.0990.0770.099Protein kinase (CK2) alpha inhibitor
0.0340.0130.034DNA topoisomerase IV inhibitor
0.0260.0050.026Histone-lysine N-methyltransferase EZH2 inhibitor
0.0910.070.091MAO A inhibitor
0.0370.0160.037Peptide deformylase inhibitor
0.0360.0150.036Vanilloid 4 antagonist
0.050.0290.05Cholesterol esterase inhibitor
0.0730.0530.073Janus tyrosine kinase 2 inhibitor
0.0420.0220.042MAP3K5 inhibitor
0.0380.0180.038Carnitine palmitoyltransferase 1 inhibitor
0.0720.0520.072Metalloproteinase-9 inhibitor
0.0860.0660.086Potassium channel activator
0.0660.0460.066Carbonic anhydrase V inhibitor
0.0760.0560.076Estrogen receptor alpha antagonist
0.0380.0180.038Carnitine palmitoyltransferase inhibitor
0.0280.0090.0285 Hydroxytryptamine 4 agonist

0.027 0.01 DBMET00949

0.0430.0240.043Cathepsin L1 inhibitor
0.0710.0520.071Macrophage colony-stimulating factor 1 receptor antagonist
0.0320.0130.032CXC chemokine 2 receptor antagonist
0.0410.0220.041CF transmembrane conductance regulator antagonist

0.039 0.029 DBMET00950

0.0530.0350.053mTOR inhibitor
0.0220.0050.022CXC chemokine 4 receptor agonist

0.015 0.011 DBMET00949

0.0440.0270.044Toll-Like receptor 2 agonist
0.0310.0140.031LFA antagonist
0.0340.0180.034AMPA 1 receptor antagonist
0.0260.010.026ICAM 1 antagonist
0.0250.0080.025Neuraminidase (Influenza B) inhibitor
0.0480.0320.048Glutamate (mGluR group I) agonist
0.050.0340.05Transforming growth factor beta 1 antagonist
0.0880.0720.088Potassium channel (Voltage-sensitive) activator
0.0210.0050.021CDK2/cyclin A3 inhibitor
0.0350.0190.035Carboxypeptidase B inhibitor

0.031 0.027 DBMET00949

0.0220.0060.022Methylmalonyl-CoA mutase inhibitor

0.018 0.014 DBMET00950

0.0680.0530.068Phosphodiesterase V inhibitor
0.0390.0240.039Factor XIIIa inhibitor
0.0580.0430.058Collagenase 3 inhibitor
0.0550.040.055MAP kinase kinase 9 inhibitor
0.0390.0240.039Vanilloid 3 antagonist
0.0460.0310.046Glutamate (mGluR5) agonist
0.0390.0250.039DNA gyrase subunit B inhibitor
0.0760.0620.076Histamine H1 receptor antagonist
0.0360.0220.036Calcitonin receptor agonist
0.0250.0110.025Protease (Human cytomegalovirus) inhibitor
0.0210.0070.021Complement factor D inhibitor
0.2130.1990.21315-Lipoxygenase inhibitor
0.0390.0250.039Melanocortin 1 antagonist
0.0360.0230.036Opioid delta receptor agonist
0.020.0070.02NMDA receptor phencyclidine site antagonist
0.0180.0050.018Carbonic anhydrase XI inhibitor
0.020.0070.02Telomerase stimulant

0.019 0.009 DBMET00950

0.0450.0320.045Fructose-1,6-bisphosphatase inhibitor
0.0210.0090.021Estrogen-related receptor gamma agonist
0.0750.0630.075MAP kinase 7 inhibitor
0.0690.0570.069Nav1.8 sodium channel blocker
0.0660.0540.066Transforming growth factor antagonist
0.0790.0670.079Androgen antagonist
0.0520.040.052Ribonucleoside-diphosphate reductase inhibitor
0.0210.0090.021Antibiotic Anthracycline-like

0.018 0.014 DBMET00950

0.0530.0410.053Ribonucleotide reductase inhibitor
0.0770.0660.077Glutathione S-transferase inhibitor
0.0790.0680.079T cell inhibitor
0.0560.0440.056Calcium channel T-type blocker
0.0220.0110.022Toll-Like receptor 8 agonist
0.0610.0510.061Fibroblast growth factor 2 antagonist
0.0580.0470.058Dopamine D3 antagonist
0.0720.0620.072Metalloproteinase-2 inhibitor
0.0180.0080.018Thromboxane A2 agonist

0.016 0.01 DBMET00950

0.060.050.068Prolactin release inhibitor

0.068 0.026 DBMET00950

DBMET00950
0.0240.0140.024Isoleucine-tRNA ligase inhibitor
0.0650.0550.065Syk tyrosine kinase inhibitor

0.062 0.058 DBMET00949

0.0280.0190.02811-Beta-hydroxysteroid dehydrogenase 2 inhibitor
0.0960.0870.096Aurora-B kinase inhibitor
0.0160.0070.016Lysophosphatidic acid receptor 3 agonist
0.0150.0060.0151-Deoxy-D-xylulose-5-phosphate reductoisomerase inhibitor
0.0450.0370.045AMPA receptor antagonist
0.0420.0340.042Stearoyl-CoA desaturase inhibitor
0.0620.0540.062Orexin receptor antagonist
0.0350.0270.035Nicotinic acid receptor agonist
0.0110.0030.011DNA topoisomerase III inhibitor
0.0170.0090.017Purinergic P2Y1 agonist
0.0640.0570.064Phosphodiesterase 5A inhibitor
0.0370.030.037Histone deacetylase 9 inhibitor
0.0990.0920.099MAO inhibitor
0.0220.0150.022Adenosine kinase inhibitor
0.0460.0390.046Adenosine A2b receptor antagonist
0.0750.0680.075AXL receptor tyrosine kinase inhibitor
0.0450.0390.045Benzodiazepine antagonist
0.0130.0070.013Glutamate (mGluR6) agonist
0.0270.0210.027Thrombin receptor antagonist
0.0640.0590.064Dopamine antagonist
0.1370.1320.137Dual specificity tyrosine-phosphorylation regulated kinase 3 inhibitor
0.0120.0070.012Purine nucleoside phosphorylase inhibitor
0.1350.130.135Pyruvate kinase inhibitor
0.0290.0240.029Dipeptidyl peptidase I inhibitor
0.0220.0180.022Dopamine autoreceptor agonist
0.0390.0340.039Sphingosine 1-phosphate receptor 1 agonist
0.0390.0340.039Plasmepsin II inhibitor
0.0130.0080.013Integrin beta2 antagonist
0.0290.0250.029Cholesterol ester transfer protein antagonist
0.1270.1230.127TRKC antagonist
0.120.1160.12Ca2+/calmodulin-dependent kinase II gamma inhibitor
0.0080.0040.008Integrin alpha5beta6 antagonist
0.0070.0040.007CC chemokine 6 receptor agonist

0.006 0.005 DBMET00949

0.0110.0080.011Melatonin 5 antagonist
0.0530.050.053Leukotriene C antagonist
0.0660.0630.066Protein kinase B gamma inhibitor
0.0160.0140.016Nicotinic acid receptor 1 antagonist
0.0220.020.022Fructose-1,6-bisphosphatase 1 inhibitor
0.0620.060.062Janus tyrosine kinase 3 inhibitor
0.0520.0490.052Sphingosine 1-phosphate receptor 1 antagonist
0.0330.030.033Histone deacetylase 7 inhibitor
0.0240.0220.024Sodium/glucose cotransporter inhibitor
0.0370.0350.037CDK5/p25 inhibitor
0.0540.0520.056CDK1/cyclin B inhibitor

0.056 0.05 DBMET00949

DBMET00949
0.0490.0480.049Matrix metalloproteinase (membrane-type) inhibitor
0.0140.0120.014Adenosine A2a receptor agonist
0.0430.0410.043Beta adrenoreceptor agonist
0.0220.020.022NMDA receptor glycine site antagonist
0.0150.0140.015Adenosine A2 receptor agonist
0.0370.0360.037Histamine H3 receptor antagonist
0.0110.010.011Egl nine homolog 3 inhibitor
0.010.0090.01Purinergic P2Y2 agonist
0.0110.010.011Melatonin 2 antagonist
0.0090.0080.009Progesterone receptor A antagonist
0.0040.0030.004Reverse transcriptase (HBV) inhibitor
0.0130.0120.013Integrin alphaVbeta6 antagonist
0.0350.040.04Integrin alpha1beta1 antagonist

0.04 0.021 DBMET00949

DBMET00949
0.0620.1080.155Dual specificity tyrosine-phosphorylation regulated kinase 2 inhibitor

0.155 0.013 DBMET00949

DBMET00949
0.0120.0680.045AMPA 2 receptor antagonist

0.045 0.012 DBMET00949

DBMET00949
0.1440.2110.196Peptidyltransferase inhibitor

0.196 0.105 DBMET00950

DBMET00950
0.050.160.179MAP kinase 9 inhibitor

0.179 0.028 DBMET00949

DBMET00949
0.0120.1290.041,3-Beta-glucan synthase inhibitor

0.04 0.004 DBMET00950

DBMET00950
0.0480.1680.159Cyclin-dependent kinase 5 inhibitor

0.159 0.036 DBMET00949

DBMET00949
0.0810.2130.145Sigma receptor agonist

0.145 0.088 DBMET00950

DBMET00950
0.0330.1730.182MAP kinase 10 inhibitor

0.182 0.011 DBMET00949

DBMET00949
0.0180.1950.039Antibiotic Aminoglycoside-like

0.039 0.021 DBMET00950

DBMET00950
0.0540.2570.0783C-Like protease (SARS coronavirus) inhibitor

0.078 0.077 DBMET00949

DBMET00949
0.0090.2590.072Opioid kappa receptor agonist

0.072 0.014 DBMET00950

DBMET00950
0.020.3090.08MAP kinase kinase 10 inhibitor

0.08 0.029 DBMET00949

DBMET00949
0.0550.390.152Hepatoprotectant

0.152 0.108 DBMET00950

DBMET00950
0.0760.4790.204Sodium/bile acid cotransporter inhibitor

0.204 0.183 DBMET00950

DBMET00950
0.0120.4960.399Nitric oxide donor

0.065 0.04 DBMET00949

0.399 0.001 DBMET00950

DBMET00950
0.0190.5860.273Angiogenesis stimulant

0.273 0.06 DBMET00950

DBMET00950
0.0030.7390.046Adenosine A1 receptor agonist

0.046 0.006 DBMET00950

DBMET00950
Ext Pa Pi Pmax Activity Other Results ID Pa_max