Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.7910.0030.791Protein kinase (Mos, Mil/Raf, MEKK, RIPK, TESK, LIMK, IRAK, ILK, Activin/TGF-beta) inhibitor
0.7770.0030.777Raf kinase inhibitor
0.7480.0010.748Raf kinase C inhibitor

0.401 0.004 DBMET00675

0.7340.0030.734Raf kinase B inhibitor
0.5960.0060.596Calcium channel L-type activator

0.565 0.01 DBMET00675

0.4360.0050.436TIE antagonist
0.440.0180.44Antimitotic

0.283 0.049 DBMET00675

0.4230.0050.423TIE-2 antagonist
0.3880.0290.444Calcium channel activator

0.444 0.012 DBMET00675

DBMET00675
0.4060.0520.406Angiogenesis inhibitor
0.3740.020.374EphB2 antagonist
0.3440.0040.44Potassium channel (Ca-activated) blocker

0.44 0.003 DBMET00675

DBMET00675
0.3280.0160.328Tubulin antagonist

0.169 0.05 DBMET00675

0.3420.0480.342Hypoxia-inducible factor 1 alpha inhibitor

0.242 0.108 DBMET00675

0.2760.0050.276Hedgehog signaling inhibitor
0.2610.0080.261Catalase inhibitor

0.087 0.044 DBMET00675

0.2490.0090.249Microtubule formation inhibitor

0.119 0.061 DBMET00675

0.2770.0420.277Platelet aggregation inhibitor

0.154 0.124 DBMET00675

0.2410.0070.241Gastric antisecretory

0.092 0.075 DBMET00675

0.2290.0120.311Check point kinase 2 inhibitor

0.311 0.006 DBMET00675

DBMET00675
0.2780.0730.372Insulysin inhibitor

0.372 0.027 DBMET00675

DBMET00675
0.3470.1480.347Caspase 9 stimulant

0.332 0.161 DBMET00675

0.2890.0970.315Vasodilator, coronary

0.315 0.076 DBMET00675

DBMET00675
0.2170.0260.217ATPase inhibitor

0.162 0.082 DBMET00675

0.2140.0230.214Platelet activating factor antagonist
0.290.10.29Transcription factor NF kappa B inhibitor
0.20.0160.2Platelet activating factor alpha antagonist
0.1890.0140.267HIV-1 integrase (Overall Integration) inhibitor

0.267 0.004 DBMET00675

DBMET00675
0.2110.0370.211Dual specificity tyrosine-phosphorylation regulated kinase 1B inhibitor

0.203 0.041 DBMET00675

0.1440.0060.144Granulocyte macrophage colony stimulating factor agonist

0.137 0.008 DBMET00675

0.1330.0060.133Potassium channel (ATP-sensitive) blocker

0.109 0.012 DBMET00675

0.1560.0360.156Interleukin 1b antagonist

0.15 0.04 DBMET00675

0.1730.0540.173NOS3 expression enhancer
0.1860.0720.186Interleukin-1 receptor-associated protein kinase 1 inhibitor
0.1310.0190.131mTOR complex 1 inhibitor
0.120.0130.12DNA gyrase inhibitor
0.1660.0590.166Protein kinase (CK1) gamma inhibitor

0.112 0.099 DBMET00675

0.1220.0190.122Prostaglandin-E synthase inhibitor

0.07 0.049 DBMET00675

0.2370.1350.237Cholesterol antagonist

0.217 0.15 DBMET00675

0.160.060.16Lck kinase inhibitor
0.1540.0540.187MAP kinase kinase 4 inhibitor

0.187 0.019 DBMET00675

DBMET00675
0.1020.0050.102Factor XIa inhibitor
0.1180.0230.118Glutamate release inhibitor

0.101 0.041 DBMET00675

0.1490.0580.149Interleukin 1 antagonist

0.129 0.077 DBMET00675

0.1480.0580.148Pregnane X receptor agonist

0.147 0.059 DBMET00675

0.2040.1150.204Cardiotonic
0.1770.090.177Growth factor agonist
0.1410.0540.141Antibacterial (Helicobacter pylori)

0.109 0.1 DBMET00675

0.1330.050.133DNA repair enzyme inhibitor
0.1290.0460.161Protein kinase C gamma inhibitor

0.161 0.026 DBMET00675

DBMET00675
0.1410.0580.141Protein kinase (CK1) delta inhibitor
0.1070.0280.107Histamine H2 receptor antagonist

0.094 0.041 DBMET00675

0.090.0130.124Factor IXa inhibitor

0.124 0.005 DBMET00675

DBMET00675
0.1130.0370.119Potassium channel activator

0.119 0.033 DBMET00675

DBMET00675
0.1360.060.136Vascular endothelial growth factor antagonist
0.1850.1110.26Aryl hydrocarbon receptor agonist

0.26 0.075 DBMET00675

DBMET00675
0.0920.0180.092CDK4/cyclin D1 inhibitor
0.1590.0890.159LIM domain kinase 1 inhibitor
0.1230.0530.135Photosensitizer

0.135 0.042 DBMET00675

DBMET00675
0.1730.1030.173Insulin sensitizer

0.173 0.104 DBMET00675

0.1250.0580.125Vascular endothelial growth factor 2 antagonist
0.1090.0460.109CDK/cyclin complex inhibitor
0.0670.0050.067Factor XI inhibitor
0.0770.0230.077CDK4/cyclin D inhibitor
0.0960.0440.096Platelet growth factor antagonist

0.077 0.06 DBMET00675

0.1810.1310.232RNA-directed DNA polymerase inhibitor

0.232 0.063 DBMET00675

DBMET00675
0.0530.0040.053HCV NS5A inhibitor
0.1140.0660.114Protein kinase (CK2) alpha inhibitor
0.2830.2360.397Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.397 0.103 DBMET00675

DBMET00675
0.0730.0270.073Transcription factor AP-1 inhibitor
0.0690.0240.069Alpha tubulin antagonist
0.1470.1040.147Tumour necrosis factor antagonist
0.070.0280.086Cyclin D1 inhibitor

0.086 0.014 DBMET00675

DBMET00675
0.0980.0570.098Proto-oncogene tyrosine-protein kinase Kit inhibitor
0.10.0630.1Cyclin-dependent kinase 9 inhibitor
0.1240.0880.124Protein kinase (CK1) inhibitor
0.1090.0750.109Protein kinase (CK1) gamma 2 inhibitor

0.098 0.086 DBMET00675

0.0360.0050.036Acid ceramidase inhibitor

0.031 0.008 DBMET00675

0.1480.1170.245Pyruvate kinase inhibitor

0.245 0.062 DBMET00675

DBMET00675
0.1350.1070.135Protein kinase (CK1) gamma 3 inhibitor
0.1080.080.108Interleukin 8 antagonist

0.1 0.096 DBMET00675

0.030.0030.031Granulocyte colony stimulating factor receptor agonist

0.031 0.003 DBMET00675

DBMET00675
0.120.0950.12CDC-like kinase 1 inhibitor
0.1570.1330.56Aldehyde oxidase inhibitor

0.56 0.024 DBMET00675

DBMET00675
0.0620.0390.062Beta tubulin antagonist
0.2270.2040.227Transcription factor inhibitor
0.0480.0260.087Potassium channel small-conductance Ca-activated blocker

0.087 0.008 DBMET00675

DBMET00675
0.1150.0930.115Interleukin 4 antagonist
0.0330.0150.04Elastase 2B inhibitor

0.04 0.008 DBMET00675

DBMET00675
0.0330.0150.04Elastase 3A inhibitor

0.04 0.008 DBMET00675

DBMET00675
0.0330.0150.04Elastase 3B inhibitor

0.04 0.008 DBMET00675

DBMET00675
0.060.0440.06Cyclin B1 inhibitor
0.0990.0830.099CDC-like kinase 3 inhibitor
0.1060.090.115MAP kinase 12 inhibitor

0.115 0.076 DBMET00675

DBMET00675
0.050.0350.093Potassium channel (Inward rectifier) activator

0.093 0.005 DBMET00675

DBMET00675
0.1430.1280.143P-glycoprotein inhibitor
0.0540.040.054Cyclin B2 inhibitor

0.052 0.044 DBMET00675

0.0480.0340.09Potassium channel (ATP-sensitive) activator

0.09 0.005 DBMET00675

DBMET00675
0.1120.0980.112Cytokine production inhibitor
0.0830.0710.083ATPase (Vacuolar H+) inhibitor
0.1410.130.155I kappa B kinase epsilon inhibitor

0.155 0.115 DBMET00675

DBMET00675
0.0790.0670.079Stem cell growth factor agonist
0.0750.0640.08MAP kinase kinase 7 inhibitor

0.08 0.045 DBMET00675

DBMET00675
0.0320.0210.032Cholesterol ester transfer protein antagonist
0.0920.0830.092Folate antagonist
0.0620.0530.062Alpha adrenoreceptor agonist
0.0560.0480.056Alpha 2 adrenoreceptor agonist
0.0480.0410.048H+/K+-transporting ATPase inhibitor
0.0510.0440.056Heparanase inhibitor

0.056 0.031 DBMET00675

DBMET00675
0.0160.0090.0224-Hydroxyphenylpyruvate dioxygenase inhibitor

0.022 0.004 DBMET00675

DBMET00675
0.0590.0530.059Fibroblast growth factor 2 antagonist
0.0290.0240.029Lysophosphatidic acid 2 receptor antagonist
0.0750.0720.075Dual specificity tyrosine-phosphorylation regulated kinase 2 inhibitor
0.0540.0530.054CDK1/cyclin B inhibitor
0.0860.0850.086Insulin receptor antagonist
0.2130.2140.318Antibacterial

0.318 0.122 DBMET00675

DBMET00675
0.0470.0490.075Protein kinase C eta inhibitor

0.075 0.026 DBMET00675

DBMET00675
0.0160.0230.018Potassium channel (Inward rectifier) 11 blocker

0.018 0.014 DBMET00675

DBMET00675
0.1390.1470.167Dyrk kinase inhibitor

0.167 0.12 DBMET00675

DBMET00675
0.1760.1850.244Gastrin inhibitor

0.244 0.086 DBMET00675

DBMET00675
0.030.0390.036Protein kinase C beta I inhibitor

0.036 0.016 DBMET00675

DBMET00675
0.0070.0220.017Imidazoline I2 receptor antagonist

0.017 0.004 DBMET00675

DBMET00675
0.0750.0910.086Hematopoietic

0.086 0.058 DBMET00675

DBMET00675
0.0270.0440.037Diamine oxidase inhibitor

0.037 0.027 DBMET00675

DBMET00675
0.070.0890.078MAP kinase 7 inhibitor

0.078 0.052 DBMET00675

DBMET00675
0.0860.110.124DOPA decarboxylase inhibitor

0.124 0.04 DBMET00675

DBMET00675
0.1490.1750.197DNA damaging

0.197 0.118 DBMET00675

DBMET00675
0.0620.0890.076Ornithine decarboxylase inhibitor

0.076 0.072 DBMET00675

DBMET00675
0.2290.2590.3395 Hydroxytryptamine release inhibitor

0.339 0.125 DBMET00675

DBMET00675
0.0260.0580.04Urokinase inhibitor

0.04 0.039 DBMET00675

DBMET00675
0.0240.0570.032Protein kinase C beta II inhibitor

0.032 0.024 DBMET00675

DBMET00675
0.1120.1460.154GABA C receptor rho-2 antagonist

0.154 0.069 DBMET00675

DBMET00675
0.0480.0820.077Cyclin B3 inhibitor

0.077 0.04 DBMET00675

DBMET00675
0.0160.0510.037Nicotinic alpha4beta2 receptor agonist

0.037 0.01 DBMET00675

DBMET00675
0.060.0960.091Carbonic anhydrase VI inhibitor

0.091 0.046 DBMET00675

DBMET00675
0.1250.1620.157Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor

0.157 0.124 DBMET00675

DBMET00675
0.1560.1960.301Prostaglandin dehydrogenase inhibitor

0.301 0.101 DBMET00675

DBMET00675
0.1850.2290.29515-Lipoxygenase inhibitor

0.295 0.135 DBMET00675

DBMET00675
0.0440.1020.079Protein kinase C beta inhibitor

0.079 0.031 DBMET00675

DBMET00675
0.0180.0770.035Factor VIIa inhibitor

0.035 0.03 DBMET00675

DBMET00675
0.1310.1910.196Cyclic AMP phosphodiesterase inhibitor

0.196 0.097 DBMET00675

DBMET00675
0.070.130.674Nav1.1 sodium channel blocker

0.674 0.003 DBMET00675

DBMET00675
0.0530.1140.085S-adenosyl-L-methionine decarboxylase inhibitor

0.085 0.028 DBMET00675

DBMET00675
0.0720.1370.172Amylase inhibitor

0.172 0.054 DBMET00675

DBMET00675
0.0720.1390.269Nav1.4 sodium channel blocker

0.269 0.005 DBMET00675

DBMET00675
0.1440.2160.221DNA synthesis inhibitor

0.221 0.093 DBMET00675

DBMET00675
0.0960.1680.168Arachidonic acid antagonist

0.168 0.068 DBMET00675

DBMET00675
0.0650.1410.098Adenylate cyclase inhibitor

0.098 0.086 DBMET00675

DBMET00675
0.0250.1010.044Dihydrofolate reductase inhibitor

0.044 0.029 DBMET00675

DBMET00675
0.0820.1640.182Peroxidase inhibitor

0.182 0.065 DBMET00675

DBMET00675
0.070.1580.125Adenylate kinase inhibitor

0.125 0.039 DBMET00675

DBMET00675
0.0120.1050.039Potassium channel small-conductance Ca-activated activator

0.039 0.016 DBMET00675

DBMET00675
0.1460.240.2015 Hydroxytryptamine 3E antagonist

0.201 0.061 DBMET00675

DBMET00675
0.0570.1550.092NADH dehydrogenase inhibitor

0.092 0.053 DBMET00675

DBMET00675
0.020.1180.039Histamine H2 receptor agonist

0.039 0.036 DBMET00675

DBMET00675
0.1480.2460.195Vasodilator, peripheral

0.195 0.182 DBMET00675

DBMET00675
0.1410.2440.195Nitric-oxide synthase stimulant

0.195 0.097 DBMET00675

DBMET00675
0.0190.1250.047Thymidylate synthase inhibitor

0.047 0.032 DBMET00675

DBMET00675
0.1030.2140.1383C-like protease (Human coronavirus) inhibitor

0.138 0.125 DBMET00675

DBMET00675
0.1130.2260.241Streptokinase A inhibitor

0.241 0.108 DBMET00675

DBMET00675
0.0080.1220.023Integrin beta5 antagonist

0.023 0.012 DBMET00675

DBMET00675
0.040.1560.103Potassium channel (Ca-activated) activator

0.103 0.053 DBMET00675

DBMET00675
0.1570.2750.382GABA C receptor rho-3 antagonist

0.382 0.07 DBMET00675

DBMET00675
0.0260.1440.077Aldosterone antagonist

0.077 0.012 DBMET00675

DBMET00675
0.0590.1790.083MAP kinase kinase 1 inhibitor

0.083 0.082 DBMET00675

DBMET00675
0.1350.2580.197Calpain 2 inhibitor

0.197 0.19 DBMET00675

DBMET00675
0.0580.1860.082D-Ala-D-Ala ligase inhibitor

0.082 0.062 DBMET00675

DBMET00675
0.1550.2850.327Interleukin 2 agonist

0.327 0.057 DBMET00675

DBMET00675
0.1190.250.277Superoxide dismutase inhibitor

0.277 0.06 DBMET00675

DBMET00675
0.0770.2120.131Dual specificity phosphatase 3 inhibitor

0.131 0.115 DBMET00675

DBMET00675
0.0420.1770.073Glycine receptor agonist

0.073 0.049 DBMET00675

DBMET00675
0.0450.1820.098Chymotrypsin inhibitor

0.098 0.037 DBMET00675

DBMET00675
0.1350.2760.218Antithrombotic

0.218 0.156 DBMET00675

DBMET00675
0.0790.220.141Mannose-6-phosphate isomerase inhibitor

0.141 0.073 DBMET00675

DBMET00675
0.1630.3040.199Ca2+/calmodulin-dependent kinase IV inhibitor

0.199 0.168 DBMET00675

DBMET00675
0.0520.1980.093GABA C receptor rho-1 antagonist

0.093 0.073 DBMET00675

DBMET00675
0.1050.2570.15Death-associated protein kinase 2 inhibitor

0.15 0.105 DBMET00675

DBMET00675
0.0460.1990.16Ferrochelatase inhibitor

0.16 0.034 DBMET00675

DBMET00675
0.0120.1670.09NMDA 2A receptor antagonist

0.09 0.016 DBMET00675

DBMET00675
0.0350.1950.101Secretase beta inhibitor

0.101 0.018 DBMET00675

DBMET00675
0.0350.1990.098Histamine N-methyltransferase inhibitor

0.098 0.048 DBMET00675

DBMET00675
0.0290.1930.104Cathepsin G inhibitor

0.104 0.032 DBMET00675

DBMET00675
0.0290.1930.053Dihydroorotate oxidase inhibitor

0.053 0.043 DBMET00675

DBMET00675
0.020.1850.056Biliverdin reductase inhibitor

0.056 0.045 DBMET00675

DBMET00675
0.0290.1940.084Phospholipase D inhibitor

0.084 0.029 DBMET00675

DBMET00675
0.0180.1840.046Histamine H1 receptor agonist

0.046 0.025 DBMET00675

DBMET00675
0.1260.2930.248Alpha-glucosidase inhibitor

0.248 0.189 DBMET00675

DBMET00675
0.1360.3030.249Tyrosine 3 hydroxylase inhibitor

0.249 0.069 DBMET00675

DBMET00675
0.0480.2170.094Protein kinase C zeta inhibitor

0.094 0.059 DBMET00675

DBMET00675
0.0460.2160.07MDM2 inhibitor

0.07 0.038 DBMET00675

DBMET00675
0.1080.280.141Ca2+-transporting ATPase inhibitor

0.141 0.068 DBMET00675

DBMET00675
0.0430.2180.141GABA C receptor agonist

0.141 0.038 DBMET00675

DBMET00675
0.0630.2390.221Anticoagulant

0.221 0.046 DBMET00675

DBMET00675
0.0280.2070.118MAO A inhibitor

0.118 0.053 DBMET00675

DBMET00675
0.0520.2340.145Alpha-N-acetylglucosaminidase inhibitor

0.145 0.058 DBMET00675

DBMET00675
0.0490.2340.092Electrolyte absorption antagonist

0.092 0.07 DBMET00675

DBMET00675
0.0640.2560.211Diuretic

0.211 0.04 DBMET00675

DBMET00675
0.0420.2350.1275 Hydroxytryptamine 3A agonist

0.127 0.05 DBMET00675

DBMET00675
0.1210.3150.216Ca2+/calmodulin-dependent kinase II alpha inhibitor

0.216 0.14 DBMET00675

DBMET00675
0.020.2160.0463-Hydroxyanthranilate 3,4-dioxygenase inhibitor

0.046 0.02 DBMET00675

DBMET00675
0.0680.2650.151Thiol protease inhibitor

0.151 0.067 DBMET00675

DBMET00675
0.0430.2420.08Triose-phosphate isomerase inhibitor

0.08 0.076 DBMET00675

DBMET00675
0.0110.2150.096NMDA 2 receptor antagonist

0.096 0.034 DBMET00675

DBMET00675
0.020.2310.06Phenylalanine 4-hydroxylase inhibitor

0.06 0.058 DBMET00675

DBMET00675
0.1370.3480.2235 Hydroxytryptamine uptake stimulant

0.223 0.113 DBMET00675

DBMET00675
0.0290.2460.108MAO inhibitor

0.108 0.083 DBMET00675

DBMET00675
0.0520.270.177Nav1.5 sodium channel blocker

0.177 0.017 DBMET00675

DBMET00675
0.0140.2410.058Argininosuccinate synthase inhibitor

0.058 0.039 DBMET00675

DBMET00675
0.0360.2670.099UDP-glucose 4-epimerase inhibitor

0.099 0.062 DBMET00675

DBMET00675
0.0430.2750.127Beta amyloid protein antagonist

0.127 0.06 DBMET00675

DBMET00675
0.0330.2640.125Glycogen synthase kinase-3 alpha inhibitor

0.125 0.081 DBMET00675

DBMET00675
0.060.2960.145Anticonvulsant

0.145 0.135 DBMET00675

DBMET00675
0.0180.2570.076Nicotinic alpha4beta2 receptor antagonist

0.076 0.054 DBMET00675

DBMET00675
0.0270.2680.09Alcohol dehydrogenase inhibitor

0.09 0.064 DBMET00675

DBMET00675
0.0880.3310.18412-Lipoxygenase inhibitor

0.184 0.169 DBMET00675

DBMET00675
0.0380.2830.085GABA B receptor agonist

0.085 0.033 DBMET00675

DBMET00675
0.0210.2670.105NMDA receptor antagonist

0.105 0.044 DBMET00675

DBMET00675
0.0720.3310.144Succinate dehydrogenase inhibitor

0.144 0.123 DBMET00675

DBMET00675
0.0230.2890.185Inducible nitric-oxide synthase inhibitor

0.185 0.01 DBMET00675

DBMET00675
0.0310.2990.096Cystathionine beta-synthase inhibitor

0.096 0.081 DBMET00675

DBMET00675
0.0380.3080.275Psychostimulant

0.275 0.05 DBMET00675

DBMET00675
0.0360.3090.082UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor

0.082 0.077 DBMET00675

DBMET00675
0.0280.3020.115Glutamate receptor antagonist

0.115 0.08 DBMET00675

DBMET00675
0.0380.3170.061Calcium channel P-type blocker

0.061 0.054 DBMET00675

DBMET00675
0.0560.3390.248Interleukin agonist

0.248 0.08 DBMET00675

DBMET00675
0.0340.3310.148Sodium channel blocker

0.148 0.06 DBMET00675

DBMET00675
0.0260.3490.171Nitric-oxide synthase inhibitor

0.171 0.016 DBMET00675

DBMET00675
0.0810.4040.154Neurotensin receptor agonist

0.154 0.092 DBMET00675

DBMET00675
0.0310.3620.156Nav1.6 sodium channel blocker

0.156 0.047 DBMET00675

DBMET00675
0.0830.4140.1875 Hydroxytryptamine release stimulant

0.187 0.133 DBMET00675

DBMET00675
0.0240.3830.145Sodium channel (voltage-gated) blocker

0.145 0.058 DBMET00675

DBMET00675
0.0240.3910.059Trypsin inhibitor

0.059 0.05 DBMET00675

DBMET00675
0.0370.4180.219Nav1.2 sodium channel blocker

0.219 0.028 DBMET00675

DBMET00675
0.0240.410.067Cathepsin E inhibitor

0.067 0.032 DBMET00675

DBMET00675
0.0040.4110.058Protease activated receptor 1 antagonist

0.058 0.028 DBMET00675

DBMET00675
0.0290.4640.13Cell wall synthesis inhibitor

0.13 0.086 DBMET00675

DBMET00675
0.0090.860.127Insulin secretagoues

0.127 0.101 DBMET00675

DBMET00675
Ext Pa Pi Pmax Activity Other Results ID Pa_max