Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.6850.0150.777Analgesic

0.777 0.007 DBMET00836

DBMET00836
0.6140.0170.614Aldehyde oxidase inhibitor

0.209 0.1 DBMET00836

0.5290.0080.529Platelet aggregation inhibitor

0.522 0.008 DBMET00836

0.5150.0270.515Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.42 0.083 DBMET00836

0.4890.0120.489Psychostimulant

0.27 0.051 DBMET00836

0.4860.030.486GABA C receptor rho-3 antagonist

0.289 0.124 DBMET00836

0.4420.0050.442Platelet activating factor antagonist

0.394 0.005 DBMET00836

0.4490.0210.449HERG channel blocker
0.4590.0340.4595 Hydroxytryptamine release stimulant

0.178 0.142 DBMET00836

0.4190.0090.632Cholinergic

0.632 0.004 DBMET00836

DBMET00836
0.4250.0180.425Sigma receptor agonist

0.169 0.074 DBMET00836

0.4230.0250.423Cardiotonic

0.413 0.027 DBMET00836

0.4220.0330.422Nootropic
0.4050.020.405Ca2+/calmodulin-dependent kinase II alpha inhibitor
0.3930.0160.3935 Hydroxytryptamine uptake stimulant

0.243 0.088 DBMET00836

0.3850.0110.486Tyrosine-protein kinase receptor FLT3 inhibitor

0.486 0.006 DBMET00836

DBMET00836
0.3980.0270.398Potassium channel (Voltage-sensitive) blocker
0.360.0140.36Tyrosine 3 hydroxylase inhibitor

0.279 0.045 DBMET00836

0.3410.0040.496Substance P antagonist

0.496 0.003 DBMET00836

DBMET00836
0.3510.0240.351Anesthetic general

0.135 0.131 DBMET00836

0.3640.0490.364Vasodilator, coronary

0.235 0.149 DBMET00836

0.3040.0050.396Acetylcholine agonist

0.396 0.004 DBMET00836

DBMET00836
0.2990.0040.381Acetylcholine muscarinic agonist

0.381 0.003 DBMET00836

DBMET00836
0.330.0410.33Superoxide dismutase inhibitor

0.218 0.099 DBMET00836

0.3090.0240.3095 Hydroxytryptamine 1E antagonist

0.184 0.15 DBMET00836

0.3050.0290.305Gastrin inhibitor
0.2760.0130.276TRKB antagonist
0.2660.0040.335Neurokinin 1 antagonist

0.335 0.003 DBMET00836

DBMET00836
0.2640.0040.318Neurokinin antagonist

0.318 0.004 DBMET00836

DBMET00836
0.2570.0050.257Platelet growth factor antagonist

0.084 0.053 DBMET00836

0.310.0660.31Spasmolytic

0.287 0.075 DBMET00836

0.2850.0450.285Anticonvulsant
0.2560.0160.256Calcium channel blocker

0.115 0.093 DBMET00836

0.2780.0510.278Cyclic AMP phosphodiesterase inhibitor
0.2390.0150.274Antihistaminic

0.274 0.012 DBMET00836

DBMET00836
0.2310.0150.269Histamine antagonist

0.269 0.012 DBMET00836

DBMET00836
0.2180.0040.288Kinesin-like protein 1 inhibitor

0.288 0.003 DBMET00836

DBMET00836
0.2180.0040.288Kinesin antagonist

0.288 0.003 DBMET00836

DBMET00836
0.2180.0050.218Smo receptor antagonist
0.2590.050.259MAP kinase kinase 2 inhibitor
0.2330.0260.233Alpha-N-acetylglucosaminidase inhibitor

0.139 0.061 DBMET00836

0.2050.0050.298Acetylcholine M1 receptor agonist

0.298 0.004 DBMET00836

DBMET00836
0.2180.0190.246Butyrylcholinesterase inhibitor

0.246 0.015 DBMET00836

DBMET00836
0.2260.0310.2265 Hydroxytryptamine 3E antagonist

0.185 0.093 DBMET00836

0.2540.0640.254Potassium channel blocker
0.2220.0330.276Acetylcholine M1 receptor antagonist

0.276 0.019 DBMET00836

DBMET00836
0.2090.0220.296Acetylcholine muscarinic antagonist

0.296 0.009 DBMET00836

DBMET00836
0.2890.1020.289Vasodilator, peripheral
0.1920.010.192Prolactin inhibitor

0.098 0.057 DBMET00836

0.1850.0040.185Nicotinamide phosphoribosyltransferase inhibitor

0.066 0.01 DBMET00836

0.2090.0320.209Toll-Like receptor 9 antagonist
0.2460.0690.246DNA synthesis inhibitor

0.189 0.141 DBMET00836

0.2360.0590.236RNA-directed DNA polymerase inhibitor
0.2370.0650.237Antimitotic

0.149 0.122 DBMET00836

0.3320.1610.332Caspase 9 stimulant
0.1780.010.178Acetylcholine nicotinic agonist

0.078 0.06 DBMET00836

0.2230.0560.223Glyceraldehyde-3-phosphate dehydrogenase inhibitor
0.2990.1330.29915-Lipoxygenase inhibitor
0.1990.0320.303Cholinergic antagonist

0.303 0.014 DBMET00836

DBMET00836
0.1680.0030.168Ryanodine receptor antagonist

0.098 0.004 DBMET00836

0.1880.0250.188Ferrochelatase inhibitor
0.210.050.21Lipocortins synthesis antagonist
0.1920.0330.28Acetylcholine antagonist

0.28 0.016 DBMET00836

DBMET00836
0.180.0220.18Calcium channel (voltage-sensitive) blocker
0.1930.0350.303Acetylcholinesterase inhibitor

0.303 0.013 DBMET00836

DBMET00836
0.1780.0220.1785 Hydroxytryptamine 3A agonist
0.190.0350.19GABA C receptor rho-2 antagonist
0.1740.0180.285Histamine H1 receptor antagonist

0.285 0.007 DBMET00836

DBMET00836
0.1670.0160.167Ca2+-transporting ATPase inhibitor

0.136 0.09 DBMET00836

0.1910.0410.191Activin receptor-like kinase 2 inhibitor
0.1720.0260.172Calcium channel N-type blocker
0.2130.0680.213Ca2+/calmodulin-dependent kinase II beta inhibitor
0.1490.0050.149Histamine H3 receptor agonist

0.027 0.019 DBMET00836

0.2020.0580.202Peroxidase inhibitor
0.1670.0240.167Sphingosine 1-phosphate receptor 2 antagonist

0.12 0.098 DBMET00836

0.2330.0920.233Interleukin agonist
0.1640.030.164Falcipain 3 inhibitor
0.1440.0120.19Acetylcholine M2 receptor antagonist

0.19 0.007 DBMET00836

DBMET00836
0.1370.0050.137Histamine agonist
0.2630.1310.263Calcium channel activator
0.1710.0410.171Anesthetic local
0.2380.1110.238Hypoxia-inducible factor 1 alpha inhibitor
0.250.1250.25Cholesterol antagonist
0.1310.0150.1315 Hydroxytryptamine 1B antagonist
0.1320.0160.132Phosphodiesterase 6D inhibitor
0.120.0050.12Tryptase inhibitor

0.044 0.018 DBMET00836

0.1380.0250.138Acetylcholine release stimulant
0.260.1480.26Histamine release inhibitor
0.1830.0710.183Ca2+/calmodulin-dependent kinase II gamma inhibitor
0.1290.0170.129Glutamate release inhibitor
0.1770.0670.177Antipruritic
0.1460.0360.146GABA C receptor agonist

0.086 0.084 DBMET00836

0.1320.0230.132NADH dehydrogenase inhibitor

0.092 0.054 DBMET00836

0.1570.050.157Sphingosine 1-phosphate receptor 5 antagonist
0.1310.0290.131Electrolyte absorption antagonist
0.1110.0090.111Protein kinase C beta inhibitor
0.1140.0130.1145 Hydroxytryptamine 5A antagonist
0.1170.0170.117Calcium channel L-type blocker
0.1840.0840.184Non-steroidal antiinflammatory agent
0.1030.0040.103Acetylcholine M4 receptor agonist
0.1120.0140.112Acetylcholine M5 receptor agonist
0.1190.0230.119Analgesic, opioid

0.103 0.029 DBMET00836

0.1120.0190.1125 Hydroxytryptamine 1D antagonist
0.1050.0140.1055 Hydroxytryptamine 5 antagonist
0.1250.0360.125GABA C receptor rho-1 antagonist
0.130.0430.13GABA C receptor antagonist
0.1780.0910.178I kappa B kinase epsilon inhibitor
0.1570.070.157Cytidine deaminase inhibitor
0.1370.0510.137Beta amyloid protein antagonist
0.110.0240.11Alpha adrenoreceptor agonist
0.1340.0490.1825 Hydroxytryptamine 2B antagonist

0.182 0.03 DBMET00836

DBMET00836
0.10.0160.15 Hydroxytryptamine 3A antagonist
0.0930.010.093Purinergic P2Y antagonist
0.1070.0240.159Acetylcholine M4 receptor antagonist

0.159 0.009 DBMET00836

DBMET00836
0.1120.0310.112Porphobilinogen synthase inhibitor

0.065 0.061 DBMET00836

0.0960.0150.096Melanin-concentrating hormone receptor 1 antagonist
0.0880.0070.088CC chemokine receptor 2B antagonist
0.1220.0420.122Adenylate kinase inhibitor

0.097 0.073 DBMET00836

0.120.0410.12Creatine kinase inhibitor
0.1450.0680.145Ca2+/calmodulin-dependent kinase II delta inhibitor
0.0870.0110.087Oleamide hydrolase inhibitor
0.10.0240.1Amidase inhibitor
0.110.0340.11Acetylcholine nicotinic antagonist

0.076 0.06 DBMET00836

0.0880.0130.088Phosphodiesterase 1A inhibitor
0.0790.0050.079Angiotensin AT2 receptor antagonist

0.053 0.009 DBMET00836

0.1040.0290.1045 Hydroxytryptamine 1F antagonist
0.1350.0610.135Antibacterial (Helicobacter pylori)
0.1140.0410.114MAP kinase kinase 1 inhibitor
0.0950.0210.095Vanilloid 4 agonist
0.110.0370.11Histamine N-methyltransferase inhibitor
0.0820.010.082Prolactin release inhibitor

0.062 0.043 DBMET00836

0.0910.020.0915 Hydroxytryptamine 3 agonist
0.1370.0660.137Toll-Like receptor antagonist
0.1140.0460.114Sphingomyelinase inhibitor
0.0880.0190.088Acyl-CoA dehydrogenase inhibitor

0.05 0.043 DBMET00836

0.0870.020.087Potassium channel (Tandem pore domain) blocker
0.070.0050.07Delayed rectifier potassium channel blocker
0.1220.0560.122TRPA1 agonist
0.0950.0310.095Estrogen-related receptor beta agonist
0.0810.0170.081Nicotinic receptor alpha7 subunit antagonist
0.0940.030.094Dopamine agonist
0.070.0060.07Vascular adhesion protein 1 inhibitor
0.2180.1550.218Ca(v)3.3 blocker
0.0850.0220.0855 Hydroxytryptamine 3 antagonist
0.0860.0230.135Acetylcholine M3 receptor antagonist

0.135 0.013 DBMET00836

DBMET00836
0.0670.0050.067Purinergic P2Y12 antagonist
0.0710.010.071Cholesterol esterase inhibitor
0.0810.020.081Mannitol-1-phosphate 5-dehydrogenase inhibitor

0.052 0.045 DBMET00836

0.1040.0430.1045 Hydroxytryptamine 2C antagonist
0.1780.1160.178Antiamyloidogenic
0.1390.0780.139Heat shock protein 70 antagonist
0.080.020.08MDM2 inhibitor
0.150.090.15Tyrosine kinase inhibitor

0.115 0.113 DBMET00836

0.0820.0230.126Acetylcholine M5 receptor antagonist

0.126 0.011 DBMET00836

DBMET00836
0.0940.0380.094Glycine receptor antagonist
0.1250.0690.125Nav1.3 sodium channel blocker
0.2640.2080.2645 Hydroxytryptamine release inhibitor
0.060.0040.06Adenosine uptake inhibitor

0.037 0.018 DBMET00836

0.0870.0320.087Phosphodiesterase VI inhibitor
0.0810.0280.081Carbamoyl phosphate synthetase inhibitor
0.070.0170.075 Hydroxytryptamine 4 antagonist
0.090.0370.095 Hydroxytryptamine agonist
0.190.1380.19Neuropeptide Y2 antagonist
0.1230.0710.123Cathepsin H inhibitor
0.1820.1320.182DNA damaging
0.1740.1250.174ErbB-1 antagonist
0.0990.0490.099Alpha 2 adrenoreceptor antagonist
0.0590.0090.059Phosphodiesterase 6C inhibitor
0.090.0410.09Caspase 7 inhibitor
0.0980.0490.098Calcium antagonist
0.0920.0440.092Histamine H2 receptor antagonist
0.1250.0780.125Nav1.2 sodium channel blocker
0.0580.0120.0585 Hydroxytryptamine 3B antagonist
0.0710.0250.071Fatty acid synthase inhibitor
0.0810.0350.081Neuronal nicotinic receptor antagonist
0.1030.0580.103UDP-glucose 4-epimerase inhibitor
0.0740.0290.074Purinergic P2X1 antagonist
0.0710.0260.071Corticotropin releasing factor 2 receptor antagonist
0.0710.0270.071Calcium channel T-type blocker
0.1160.0720.116Alkylator
0.0520.010.052Calcitonin gene-related peptide antagonist
0.1090.0670.109Alpha 2b adrenoreceptor antagonist

0.1 0.074 DBMET00836

0.1040.0630.104Alpha 2c adrenoreceptor antagonist

0.091 0.074 DBMET00836

0.0850.0440.085Interferon agonist
0.0570.0160.057Neuraminidase (Influenza A) inhibitor
0.0920.0520.092Bromodomain-containing protein 2 inhibitor
0.0440.0040.044Estrogen-related receptor gamma antagonist

0.027 0.024 DBMET00836

0.0470.0080.047Phosphodiesterase 6B inhibitor
0.0870.0490.087Adrenaline agonist
0.1170.0790.117DNA repair enzyme inhibitor
0.0580.020.058Histamine H4 receptor antagonist
0.1060.070.211GABA receptor agonist

0.211 0.015 DBMET00836

DBMET00836
0.0920.0560.092Phosphodiesterase I inhibitor
0.060.0250.06Dipeptidyl peptidase inhibitor
0.0430.0090.043Nicotinic alpha3beta4 receptor agonist
0.0380.0040.038Acid ceramidase inhibitor
0.130.0960.13Thiol protease inhibitor
0.0510.0170.051Histamine H1 receptor agonist
0.0650.0320.065Nicotinic neuronal receptor agonist
0.0660.0320.066Heat shock protein 90 beta antagonist
0.1060.0730.1065 Hydroxytryptamine antagonist

0.106 0.074 DBMET00836

0.0820.050.082Cell adhesion molecule inhibitor
0.1020.070.1435 Hydroxytryptamine 2 antagonist

0.143 0.047 DBMET00836

DBMET00836
0.0980.0660.098Anabolic
0.0540.0230.054Dopamine beta hydroxylase inhibitor
0.1230.0920.123Nav1.6 sodium channel blocker
0.040.0090.04Epoxide hydrolase 2 inhibitor
0.0590.0280.0595 Hydroxytryptamine 1B agonist
0.0550.0240.055Histamine H3 receptor antagonist
0.060.0290.06Epithelial sodium channel blocker
0.0770.0470.077Glutamate decarboxylase inhibitor
0.0650.0350.065Carbonic anhydrase stimulant
0.0390.0080.039Nicotinic alpha4beta2 receptor agonist
0.0530.0220.053Toll-Like receptor 2 agonist
0.0470.0180.047Factor XIIIa inhibitor
0.0340.0050.0345 Hydroxytryptamine 4 agonist

0.027 0.011 DBMET00836

0.0520.0230.052Oxytocin agonist
0.0660.0380.066Calcium channel P-type blocker
0.050.0210.05Dipeptidyl peptidase IV inhibitor
0.0770.0490.077Catalase inhibitor
0.0430.0170.0432,3-Oxidosqualene-lanosterol cyclase inhibitor

0.036 0.026 DBMET00836

0.1040.0790.104Interleukin 2 antagonist
0.1090.0840.109Aldehyde dehydrogenase inhibitor
0.0510.0260.051Adenylate cyclase 1 inhibitor
0.0490.0250.049CC chemokine 3 receptor antagonist
0.0820.0580.082CC chemokine 5 receptor agonist
0.0530.0290.053Squalene epoxidase inhibitor
0.0310.0070.031Phosphodiesterase 6G inhibitor
0.0310.0070.031Phosphodiesterase 6H inhibitor
0.1170.0930.117Interleukin 1 antagonist
0.0590.0350.059Human rhinovirus A protease inhibitor
0.1280.1060.128Adenylate cyclase stimulant
0.0370.0150.037GHS receptor antagonist
0.0650.0430.065Interferon inducer
0.0710.050.071Benzodiazepine agonist
0.0630.0420.0635 Hydroxytryptamine 7 antagonist
0.0360.0150.036Protein kinase C beta II inhibitor
0.0910.070.15Platelet activating factor beta antagonist

0.15 0.038 DBMET00836

DBMET00836
0.1440.1240.144Succinate dehydrogenase inhibitor
0.0280.0080.028Phosphodiesterase 6A inhibitor
0.0450.0260.045Nerve growth factor antagonist
0.0360.0170.036CXC chemokine 3 receptor antagonist
0.0350.0160.035Trypsin II inhibitor
0.0530.0350.053mTOR inhibitor
0.0570.0390.0575 Hydroxytryptamine 6 antagonist
0.0860.0690.122Polo-like kinase-1 inhibitor

0.122 0.029 DBMET00836

DBMET00836
0.0540.0370.054Alpha-mannosidase inhibitor
0.0660.050.066Glutamate (mGluR7) antagonist
0.0630.0460.093Dopamine D1 antagonist

0.093 0.027 DBMET00836

DBMET00836
0.0740.0570.074Nicotinic alpha4beta2 receptor antagonist
0.0590.0440.059Cyclin D1 inhibitor
0.0840.0690.084Triose-phosphate isomerase inhibitor
0.0550.040.0555 Hydroxytryptamine 7 agonist
0.0740.0590.074Fibroblast growth factor 3 antagonist
0.0610.0470.061Purinergic P2 antagonist
0.0430.030.043Dopamine D5 antagonist

0.036 0.035 DBMET00836

0.0610.0480.061Cannabinoid receptor agonist
0.0210.0080.021Calcitonin gene-related peptide 1 receptor antagonist
0.0620.0490.062Fibroblast growth factor 2 antagonist
0.110.0970.11Tyrosine-protein kinase receptor antagonist
0.0910.0780.091Nav1.1 sodium channel blocker
0.040.0270.04AMPA 4 receptor antagonist
0.0680.0560.068Aminopeptidase I inhibitor
0.0680.0570.068Phospholipase D inhibitor
0.0480.0360.048Cytokine production stimulant
0.1190.1080.119Aurora-C kinase inhibitor
0.0460.0340.046CC chemokine 4 receptor antagonist
0.1340.1240.134DNA methyltransferase I inhibitor
0.0310.020.031Purinergic P2Y14 antagonist
0.0520.0430.052Alcohol oxidase inhibitor
0.0460.0370.046Benzodiazepine antagonist
0.0270.0180.027Myristoyl transferase inhibitor
0.050.0420.05Cannabinoid CB2 receptor agonist
0.1380.1290.138DNA methylase inhibitor
0.0990.0910.099Cell adhesion inhibitor
0.0770.0690.077Bcr-Abl kinase inhibitor
0.0140.0070.014Cyclin D2 inhibitor
0.1230.1160.123Neuropeptide Y1 antagonist
0.0230.0160.023Dopamine D1 agonist
0.0670.0610.067Glutamate dehydrogenase inhibitor
0.0360.030.036DNA gyrase subunit B inhibitor
0.0550.0490.055Collagenase 3 inhibitor
0.050.0430.05Nicotinic alpha7 receptor agonist
0.0620.0560.062Phenylalanine 4-hydroxylase inhibitor
0.0250.0190.0255 Hydroxytryptamine 1F agonist
0.0210.0150.021Neuraminidase (Influenza B) inhibitor
0.0380.0320.038Glutamate (mGluR1a) antagonist
0.0240.0190.024Lysophosphatidic acid receptor 1 agonist
0.0180.0130.018Estrogen-related receptor gamma agonist
0.0710.0660.0925 Hydroxytryptamine 2A antagonist

0.092 0.052 DBMET00836

DBMET00836
0.0210.0170.021Geranylgeranyltransferase inhibitor
0.0510.0470.051Glutamate (mGluR1) antagonist
0.0270.0240.0275 Hydroxytryptamine 6 agonist
0.0660.0640.066ErbB-4 antagonist
0.0710.080.205Antiadrenergic

0.205 0.023 DBMET00836

DBMET00836
0.0710.0810.121Alpha adrenoreceptor antagonist

0.121 0.047 DBMET00836

DBMET00836
0.0720.0840.217Fibroblast growth factor 1 antagonist

0.217 0.013 DBMET00836

DBMET00836
0.0650.0850.197Adrenaline antagonist

0.197 0.024 DBMET00836

DBMET00836
0.0440.0790.098Alpha 1b adrenoreceptor antagonist

0.098 0.036 DBMET00836

DBMET00836
0.0240.0630.153Poly(ADP-ribose) polymerase 1 inhibitor

0.153 0.005 DBMET00836

DBMET00836
0.030.0750.136Poly(ADP-ribose) polymerase inhibitor

0.136 0.005 DBMET00836

DBMET00836
0.0440.0930.175Macrophage colony-stimulating factor 1 receptor antagonist

0.175 0.01 DBMET00836

DBMET00836
0.060.130.101Granulocyte macrophage colony stimulating factor antagonist

0.101 0.07 DBMET00836

DBMET00836
0.0340.1110.077Alpha 1 adrenoreceptor antagonist

0.077 0.055 DBMET00836

DBMET00836
0.0890.2020.469Polo-like kinase-3 inhibitor

0.469 0.004 DBMET00836

DBMET00836
0.030.1910.077Proto-oncogene tyrosine-protein kinase Kit inhibitor

0.077 0.076 DBMET00836

DBMET00836
0.0240.1850.063Phosphodiesterase V inhibitor

0.063 0.06 DBMET00836

DBMET00836
0.0230.1970.063Phosphodiesterase 5A inhibitor

0.063 0.058 DBMET00836

DBMET00836
0.0220.3390.134Abl kinase inhibitor

0.134 0.057 DBMET00836

DBMET00836
0.0220.340.134Protein-tyrosine kinase (PTK, not ETK, WZC) inhibitor

0.134 0.057 DBMET00836

DBMET00836
0.0190.3870.122Protein kinase C delta inhibitor

0.122 0.036 DBMET00836

DBMET00836
0.0130.5920.19Ephrin antagonist

0.19 0.027 DBMET00836

DBMET00836
0.0070.6940.226Bronchodilator

0.226 0.015 DBMET00836

DBMET00836
Ext Pa Pi Pmax Activity Other Results ID Pa_max