Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.560.0020.56Chemokine receptor agonist

0.278 0.003 DBMET01768

0.5090.0020.509CXC chemokine receptor agonist

0.214 0.003 DBMET01768

0.4430.0120.443Anesthetic general

0.417 0.014 DBMET01768

0.4330.0040.433Check point kinase 2 inhibitor

0.34 0.005 DBMET01768

0.4230.0050.423Cyclin-dependent kinase 1 inhibitor

0.308 0.011 DBMET01768

0.3950.0030.395Transforming growth factor antagonist

0.222 0.004 DBMET01768

0.4060.0220.406Calcium channel activator

0.402 0.024 DBMET01768

0.3890.0050.389MAP kinase 9 inhibitor

0.188 0.025 DBMET01768

0.4220.0470.429Angiogenesis inhibitor

0.429 0.045 DBMET01768

DBMET01768
0.3370.0040.337Histone deacetylase stimulant

0.308 0.004 DBMET01768

0.3370.0040.337Histone deacetylase SIRT1 stimulant

0.308 0.004 DBMET01768

0.330.0140.33Protein kinase (CK1) inhibitor

0.183 0.047 DBMET01768

0.3220.0080.325I kappa B kinase epsilon inhibitor

0.325 0.008 DBMET01768

DBMET01768
0.3110.0140.311Dual specificity tyrosine-phosphorylation regulated kinase 1B inhibitor

0.305 0.015 DBMET01768

0.3990.1070.399MAP kinase 1 inhibitor

0.38 0.119 DBMET01768

0.320.0290.32MAP kinase kinase 2 inhibitor

0.313 0.031 DBMET01768

0.3010.0150.301Growth factor agonist

0.279 0.02 DBMET01768

0.3020.0350.302Platelet aggregation inhibitor

0.3 0.036 DBMET01768

0.2890.0280.289Dual specificity tyrosine-phosphorylation-regulated kinase 4 inhibitor

0.225 0.043 DBMET01768

0.270.0140.27Platelet activating factor antagonist

0.224 0.021 DBMET01768

0.2580.0020.258Methionyl aminopeptidase 1 inhibitor

0.203 0.003 DBMET01768

0.290.0460.316Antimitotic

0.316 0.04 DBMET01768

DBMET01768
0.2440.010.244MAP kinase 8 inhibitor

0.13 0.038 DBMET01768

0.3640.1360.364Ca2+/calmodulin-dependent protein kinase kinase A inhibitor
0.250.0280.253C-like protease (Human coronavirus) inhibitor

0.168 0.077 DBMET01768

0.2640.0430.264Interleukin-1 receptor-associated protein kinase 1 inhibitor

0.187 0.072 DBMET01768

0.2680.0490.268MAP-kinase-activated kinase 5 inhibitor

0.261 0.053 DBMET01768

0.2350.0190.235Protein kinase (CK1) delta inhibitor

0.146 0.055 DBMET01768

0.2320.020.232Vascular endothelial growth factor 1 antagonist

0.151 0.04 DBMET01768

0.2710.0590.34Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor

0.34 0.038 DBMET01768

DBMET01768
0.230.0210.23Cyclin-dependent kinase 3 inhibitor

0.211 0.028 DBMET01768

0.2340.0260.234Phosphodiesterase inhibitor

0.152 0.057 DBMET01768

0.2570.0520.257Clk dual-specificity kinase inhibitor

0.196 0.082 DBMET01768

0.2080.0040.208Glutamate (mGluR1) antagonist

0.124 0.01 DBMET01768

0.2120.0090.212Stem cell growth factor agonist

0.139 0.023 DBMET01768

0.2670.0640.326Dyrk kinase inhibitor

0.326 0.044 DBMET01768

DBMET01768
0.2130.0130.213Insulin receptor antagonist

0.171 0.022 DBMET01768

0.250.0510.25Ca2+/calmodulin-dependent kinase II beta inhibitor

0.207 0.072 DBMET01768

0.2020.0040.202Transforming growth factor beta 1 antagonist

0.121 0.007 DBMET01768

0.2540.0560.254Anticonvulsant
0.1990.0060.199MAP kinase kinase 8 inhibitor

0.123 0.014 DBMET01768

0.2440.0530.27RNA-directed DNA polymerase inhibitor

0.27 0.04 DBMET01768

DBMET01768
0.2250.0350.225Protein kinase (CK1) gamma 1 inhibitor

0.148 0.07 DBMET01768

0.2610.0740.261Aryl hydrocarbon receptor agonist

0.25 0.079 DBMET01768

0.2140.0280.214Aurora-B kinase inhibitor

0.164 0.041 DBMET01768

0.2340.050.234Ca2+/calmodulin-dependent kinase II gamma inhibitor

0.184 0.071 DBMET01768

0.2220.0410.222Growth factor antagonist

0.188 0.05 DBMET01768

0.1850.0090.185Glutamate (mGluR group I) antagonist

0.084 0.035 DBMET01768

0.2950.1190.356GABA C receptor rho-3 antagonist

0.356 0.082 DBMET01768

DBMET01768
0.2080.0320.208Insulin secretagoues

0.197 0.037 DBMET01768

0.2070.030.207Protein kinase (CK1) gamma 2 inhibitor

0.119 0.066 DBMET01768

0.2530.0780.295DNA damaging

0.295 0.059 DBMET01768

DBMET01768
0.1870.0150.187Protein kinase (CaMK, MLCK, PhK, SNF, KIN, NIM1, MAPKAP, POLO, CHK, ULK, RSK-2nd domain) inhibitor

0.157 0.018 DBMET01768

0.3030.1330.351Antibacterial

0.351 0.101 DBMET01768

DBMET01768
0.210.0410.21Protein kinase (CK1) gamma inhibitor

0.125 0.085 DBMET01768

0.1940.0270.194Aurora-A kinase inhibitor

0.121 0.054 DBMET01768

0.2090.0420.209Protein kinase (CK1) gamma 3 inhibitor

0.164 0.075 DBMET01768

0.1880.0210.188Protein kinase (CK2) inhibitor

0.179 0.023 DBMET01768

0.1890.0270.189Cyclin-dependent kinase 2 inhibitor

0.118 0.054 DBMET01768

0.180.0180.18Activin receptor-like kinase 4 inhibitor

0.12 0.052 DBMET01768

0.1730.0120.173MAP kinase 10 inhibitor

0.084 0.046 DBMET01768

0.1870.0270.187MAP kinase 12 inhibitor

0.13 0.058 DBMET01768

0.1860.0280.186Protein kinase (CK2) alpha inhibitor

0.18 0.029 DBMET01768

0.1880.030.188Glutamate receptor antagonist

0.168 0.04 DBMET01768

0.2160.0580.216Focal adhesion kinase 2 inhibitor

0.169 0.102 DBMET01768

0.1690.0140.169Glutamate (mGluR) antagonist

0.075 0.054 DBMET01768

0.1990.0460.199Protein-tyrosine kinase Lyn inhibitor

0.125 0.081 DBMET01768

0.1960.0430.196Glycogen synthase kinase-3 alpha inhibitor

0.184 0.047 DBMET01768

0.2120.060.212CDC-like kinase 2 inhibitor

0.147 0.095 DBMET01768

0.2930.1420.293MAP kinase kinase 6 inhibitor

0.255 0.184 DBMET01768

0.190.040.19Cyclin-dependent kinase inhibitor

0.119 0.074 DBMET01768

0.210.0620.21CDC-like kinase 4 inhibitor

0.135 0.114 DBMET01768

0.160.0140.16I kappa B kinase inhibitor

0.143 0.018 DBMET01768

0.1760.0310.176Nav1.6 sodium channel blocker

0.133 0.076 DBMET01768

0.2180.0720.332Pyruvate kinase inhibitor

0.332 0.039 DBMET01768

DBMET01768
0.1860.0420.186Vascular endothelial growth factor antagonist

0.142 0.058 DBMET01768

0.1620.0190.209Carbonic anhydrase XIII inhibitor

0.209 0.013 DBMET01768

DBMET01768
0.2170.0820.217Potassium channel blocker
0.1760.0410.176Vascular endothelial growth factor 2 antagonist

0.13 0.056 DBMET01768

0.1420.0110.142Phosphodiesterase III inhibitor

0.123 0.014 DBMET01768

0.1340.0040.148Inosine monophosphate dehydrogenase inhibitor

0.148 0.004 DBMET01768

DBMET01768
0.1640.0340.164Cyclin-dependent kinase 5 inhibitor

0.141 0.045 DBMET01768

0.1330.0070.133Phosphodiesterase X inhibitor

0.061 0.02 DBMET01768

0.1330.0070.133Phosphodiesterase 10A inhibitor

0.061 0.02 DBMET01768

0.1280.0040.128Protein kinase (CK1) epsilon inhibitor

0.05 0.013 DBMET01768

0.1460.0220.199Carbonic anhydrase VI inhibitor

0.199 0.013 DBMET01768

DBMET01768
0.1610.0380.161Antibacterial (Helicobacter pylori)

0.16 0.038 DBMET01768

0.1280.0080.128Transforming growth factor beta 3 antagonist

0.1 0.024 DBMET01768

0.1360.0180.142Dual specificity tyrosine-phosphorylation regulated kinase 2 inhibitor

0.142 0.017 DBMET01768

DBMET01768
0.2910.1750.2915 Hydroxytryptamine release inhibitor

0.282 0.187 DBMET01768

0.1420.0260.142Nitric-oxide synthase inhibitor

0.092 0.073 DBMET01768

0.1280.0130.128MAP kinase kinase 10 inhibitor

0.07 0.039 DBMET01768

0.1240.0090.124Alpha 2 adrenoreceptor agonist

0.101 0.014 DBMET01768

0.1470.0340.149DNA repair enzyme inhibitor

0.149 0.033 DBMET01768

DBMET01768
0.1390.0270.139Protein kinase A inhibitor

0.112 0.038 DBMET01768

0.1170.0050.117Glucosylceramidase inhibitor

0.096 0.009 DBMET01768

0.1670.0570.173CDC-like kinase 1 inhibitor

0.173 0.053 DBMET01768

DBMET01768
0.1390.0310.201Beta glucuronidase inhibitor

0.201 0.013 DBMET01768

DBMET01768
0.1350.0280.135Interleukin-1 receptor-associated protein kinase 4 inhibitor

0.093 0.053 DBMET01768

0.1280.0220.128Inducible nitric-oxide synthase inhibitor

0.087 0.052 DBMET01768

0.1080.0040.108Fructose-1,6-bisphosphatase inhibitor

0.105 0.004 DBMET01768

0.1720.0690.172Src kinase inhibitor

0.166 0.073 DBMET01768

0.1590.0580.159Ribosomal protein S6 kinase inhibitor

0.132 0.079 DBMET01768

0.1150.0160.115MAP3K7 inhibitor

0.094 0.026 DBMET01768

0.1590.0610.174CF transmembrane conductance regulator agonist

0.174 0.042 DBMET01768

DBMET01768
0.1390.0420.139MAP kinase 13 inhibitor

0.096 0.088 DBMET01768

0.1510.0540.151Sodium channel (voltage-gated) blocker
0.110.0140.11Neuropeptide Y5 antagonist
0.1120.0170.112Purinergic P2 antagonist
0.190.0970.19HERG channel blocker
0.1050.0120.105Transcription factor AP-1 inhibitor

0.083 0.019 DBMET01768

0.1280.0370.128CDK2/cyclin A inhibitor

0.095 0.062 DBMET01768

0.1510.0610.151RET inhibitor

0.146 0.063 DBMET01768

0.1440.0550.171MAP kinase kinase inhibitor

0.171 0.041 DBMET01768

DBMET01768
0.1170.0310.117Neuropeptide Y antagonist

0.078 0.062 DBMET01768

0.1030.0210.103I kappa B kinase 1 inhibitor

0.07 0.048 DBMET01768

0.0980.0180.0985 Hydroxytryptamine 3A antagonist
0.1210.0420.121Gastric antisecretory

0.109 0.054 DBMET01768

0.0880.0120.088Glutamate (mGluR group III) agonist

0.065 0.017 DBMET01768

0.1110.0360.111Leucine-rich repeat kinase 2 inhibitor
0.1020.0270.102Syk tyrosine kinase inhibitor

0.08 0.04 DBMET01768

0.090.0160.09I kappa B kinase 2 inhibitor

0.079 0.023 DBMET01768

0.1180.0450.118Fibroblast growth factor 1 antagonist

0.088 0.067 DBMET01768

0.0790.0070.079Heparanase inhibitor

0.076 0.008 DBMET01768

0.0830.0120.083H+/K+-transporting ATPase inhibitor

0.068 0.019 DBMET01768

0.0760.0060.076Glutamate (mGluR4) agonist

0.064 0.008 DBMET01768

0.1380.0680.138Aurora-C kinase inhibitor

0.125 0.093 DBMET01768

0.0890.0190.09Carbonic anhydrase VB inhibitor

0.09 0.019 DBMET01768

DBMET01768
0.1050.0380.105TIE antagonist
0.0890.0220.089Protein kinase C iota inhibitor

0.055 0.045 DBMET01768

0.1030.0370.103TIE-2 antagonist
0.1780.1130.178Potassium channel (Voltage-sensitive) blocker
0.0790.0160.079MAP kinase kinase 9 inhibitor

0.054 0.041 DBMET01768

0.1230.0590.123Glycogen synthase kinase-3 inhibitor
0.0970.0340.097Phosphodiesterase 3A inhibitor

0.092 0.04 DBMET01768

0.0930.0310.093Alpha adrenoreceptor agonist

0.089 0.032 DBMET01768

0.2070.1460.207Ca2+/calmodulin-dependent kinase IV inhibitor
0.0830.0220.083Prostaglandin antagonist

0.052 0.038 DBMET01768

0.1160.0560.119Protein kinase C gamma inhibitor

0.119 0.053 DBMET01768

DBMET01768
0.0920.0330.092Polo-like kinase-2 inhibitor

0.064 0.06 DBMET01768

0.0890.030.096Carbonic anhydrase VA inhibitor

0.096 0.027 DBMET01768

DBMET01768
0.1170.0590.117Polo-like kinase-4 inhibitor

0.092 0.086 DBMET01768

0.1520.0950.152LIM domain kinase 1 inhibitor
0.160.1030.16Ca2+/calmodulin-dependent protein kinase inhibitor
0.2340.1780.32515-Lipoxygenase inhibitor

0.325 0.115 DBMET01768

DBMET01768
0.130.0740.13Sodium channel blocker
0.2430.1890.243Analgesic
0.0750.0220.088Fatty acid synthase inhibitor

0.088 0.015 DBMET01768

DBMET01768
0.1650.1120.169Proto-oncogene tyrosine-protein kinase Fyn inhibitor

0.169 0.108 DBMET01768

DBMET01768
0.0830.030.083Phosphodiesterase VIII inhibitor
0.0780.0260.083Purinergic P2X1 antagonist

0.083 0.024 DBMET01768

DBMET01768
0.0780.0280.0785 Hydroxytryptamine 3 agonist

0.058 0.052 DBMET01768

0.2040.1540.204Prostaglandin dehydrogenase inhibitor

0.203 0.154 DBMET01768

0.0620.0130.062Guanylate cyclase stimulant

0.043 0.03 DBMET01768

0.0890.040.089Fibroblast growth factor 3 antagonist
0.0670.0190.067Purinergic P2X antagonist
0.0580.010.058Purinergic P2X7 antagonist
0.050.0050.05Guanylate cyclase 1 stimulant

0.023 0.01 DBMET01768

0.0640.020.064Glutamate (mGluR5) antagonist
0.0830.0390.083Adenosine A3 receptor antagonist

0.069 0.06 DBMET01768

0.1090.0650.113DNA intercalator

0.113 0.062 DBMET01768

DBMET01768
0.1130.0730.113TRKA antagonist
0.0770.0370.086Carbonic anhydrase V inhibitor

0.086 0.032 DBMET01768

DBMET01768
0.1090.070.109Nav1.5 sodium channel blocker
0.1070.0680.1075 Hydroxytryptamine 3A agonist
0.0410.0050.041Alpha 2d adrenoreceptor agonist

0.026 0.011 DBMET01768

0.0750.0390.075CDC7 inhibitor
0.0870.0520.087GABA A receptor agonist
0.0680.0340.068Adenosine A1 receptor antagonist

0.058 0.041 DBMET01768

0.0450.0130.045Potassium channel small-conductance Ca-activated activator
0.0950.0630.095Lanosterol 14 alpha demethylase inhibitor
0.0360.0040.036Alpha 2c adrenoreceptor agonist

0.017 0.015 DBMET01768

0.1180.0870.118Lck kinase inhibitor
0.0430.0120.043Endothelial nitric-oxide synthase inhibitor
0.0320.0010.032CXC chemokine 3 receptor agonist

0.024 0.001 DBMET01768

0.0570.0260.057AMPA receptor antagonist

0.047 0.034 DBMET01768

0.0880.0570.088Acetylcholine agonist
0.1690.1390.1695 Hydroxytryptamine 3E antagonist
0.1510.1210.151Death-associated protein kinase 3 inhibitor
0.0880.0590.088NADH dehydrogenase inhibitor

0.088 0.06 DBMET01768

0.1920.1620.249Hypoxia-inducible factor 1 alpha inhibitor

0.249 0.102 DBMET01768

DBMET01768
0.0420.0140.042Purinergic P2Y2 antagonist

0.036 0.02 DBMET01768

0.0330.0060.033Fructose-1,6-bisphosphatase 1 inhibitor

0.031 0.007 DBMET01768

0.0450.0190.045TRPM8 blocker
0.1010.0750.101GABA receptor agonist
0.050.0250.062Phosphodiesterase 3B inhibitor

0.062 0.019 DBMET01768

DBMET01768
0.0860.0610.087Granulocyte macrophage colony stimulating factor agonist

0.087 0.058 DBMET01768

DBMET01768
0.0740.050.074S-adenosyl-L-methionine decarboxylase inhibitor
0.070.0460.075Check point kinase 1 inhibitor

0.075 0.041 DBMET01768

DBMET01768
0.0890.0660.108Protein kinase C zeta inhibitor

0.108 0.042 DBMET01768

DBMET01768
0.0330.0110.033HCV NS5A inhibitor
0.0340.0140.034CDK4/cyclin D3 inhibitor
0.060.0410.06Potassium channel (Ca-activated) blocker
0.1690.150.169Calpain inhibitor
0.110.0920.11Ca2+/calmodulin-dependent kinase II delta inhibitor
0.0460.0280.046Stearoyl-CoA desaturase inhibitor
0.0660.0490.066Nav1.7 sodium channel blocker
0.0210.0050.021CDK2/cyclin A3 inhibitor
0.070.0540.07Orexin receptor 1 antagonist
0.0540.0390.054Acetylcholine muscarinic agonist
0.0480.0340.051Dopamine beta hydroxylase inhibitor

0.051 0.028 DBMET01768

DBMET01768
0.0440.0320.044Poly(ADP-ribose) polymerase inhibitor
0.0210.0090.021Alpha 2b adrenoreceptor agonist
0.0580.0460.058Adenosine A2a receptor antagonist
0.0260.0150.026Complement factor 1s inhibitor
0.0510.040.051GABA A receptor antagonist
0.0410.0310.041Acetylcholine M1 receptor agonist
0.0850.0750.085Platelet activating factor beta antagonist

0.085 0.075 DBMET01768

0.1090.0990.109Toll-Like receptor 9 antagonist
0.0860.0770.086MAP kinase kinase 1 inhibitor

0.084 0.08 DBMET01768

0.060.0530.06Aryl hydrocarbon receptor antagonist
0.0640.0560.064ZAP-70 protein tyrosine kinase inhibitor

0.063 0.058 DBMET01768

0.0730.0650.099Platelet growth factor antagonist

0.099 0.041 DBMET01768

DBMET01768
0.0690.0610.069ErbB-2 antagonist

0.067 0.065 DBMET01768

0.0570.050.057Cyclin A2 inhibitor
0.0510.0450.051Tyrosine-protein kinase EMT inhibitor
0.0570.0510.057Adenosine A2 receptor antagonist
0.1930.1870.193Antithrombotic
0.0610.0550.061Orexin receptor antagonist
0.0910.0850.11EphA2 antagonist

0.11 0.065 DBMET01768

DBMET01768
0.0350.030.035Poly(ADP-ribose) polymerase 1 inhibitor
0.050.0440.05GABA receptor antagonist
0.0370.0320.037AMPA 4 receptor antagonist
0.0170.0120.017O6-alkylguanine-DNA alkyltransferase inhibitor
0.0390.0340.039Guanylate cyclase inhibitor
0.0280.0250.028Lysophosphatidic acid 2 receptor antagonist
0.0840.0830.084MAP kinase kinase kinase inhibitor
0.0180.0170.018Hexokinase stimulant
0.1210.1230.124GABA C receptor rho-2 antagonist

0.124 0.117 DBMET01768

DBMET01768
0.1180.1210.146Hexokinase inhibitor

0.146 0.084 DBMET01768

DBMET01768
0.0710.0760.091MAP kinase kinase 7 inhibitor

0.091 0.024 DBMET01768

DBMET01768
0.0640.0680.109Topoisomerase II alpha inhibitor

0.109 0.034 DBMET01768

DBMET01768
0.0880.0970.102Nav1.4 sodium channel blocker

0.102 0.073 DBMET01768

DBMET01768
0.1640.1780.183DNA synthesis inhibitor

0.183 0.149 DBMET01768

DBMET01768
0.0880.1050.119DOPA decarboxylase inhibitor

0.119 0.046 DBMET01768

DBMET01768
0.2430.2620.32Caspase 9 stimulant

0.32 0.173 DBMET01768

DBMET01768
0.050.0750.07Phenylalanine 4-hydroxylase inhibitor

0.07 0.046 DBMET01768

DBMET01768
0.0610.0920.106Adrenaline agonist

0.106 0.033 DBMET01768

DBMET01768
0.1690.2030.2Tyrosine 3 hydroxylase inhibitor

0.2 0.135 DBMET01768

DBMET01768
0.1240.1680.202Aldehyde oxidase inhibitor

0.202 0.104 DBMET01768

DBMET01768
0.080.1320.101Epidermal growth factor receptor kinase inhibitor

0.101 0.096 DBMET01768

DBMET01768
0.140.2160.213Lipoxygenase inhibitor

0.213 0.128 DBMET01768

DBMET01768
0.0830.1610.14Peroxidase inhibitor

0.14 0.084 DBMET01768

DBMET01768
0.1980.2790.255Cyclophilin D inhibitor

0.255 0.207 DBMET01768

DBMET01768
0.1090.1990.135MAP kinase kinase 4 inhibitor

0.135 0.097 DBMET01768

DBMET01768
0.0930.1850.135NOS3 expression enhancer

0.135 0.09 DBMET01768

DBMET01768
0.0580.1740.085Xanthine oxidase inhibitor

0.085 0.081 DBMET01768

DBMET01768
0.090.2110.131Dual specificity phosphatase inhibitor

0.131 0.119 DBMET01768

DBMET01768
0.0560.1790.126Tubulin antagonist

0.126 0.074 DBMET01768

DBMET01768
0.0360.1860.074Macrophage migration inhibitory factor inhibitor

0.074 0.059 DBMET01768

DBMET01768
0.0150.1820.052Alpha tubulin antagonist

0.052 0.038 DBMET01768

DBMET01768
0.0420.2090.106Topoisomerase II inhibitor

0.106 0.08 DBMET01768

DBMET01768
0.0340.2080.11M18 aspartyl aminopeptidase inhibitor

0.11 0.08 DBMET01768

DBMET01768
0.1190.310.176ErbB-1 antagonist

0.176 0.122 DBMET01768

DBMET01768
0.1330.4540.367Calcium channel L-type activator

0.367 0.105 DBMET01768

DBMET01768
0.0040.9640.103Estrogen antagonist

0.103 0.091 DBMET01768

DBMET01768
0.0040.9660.093Estrogen receptor beta antagonist

0.093 0.078 DBMET01768

DBMET01768
Ext Pa Pi Pmax Activity Other Results ID Pa_max