Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.8640.0030.864Bronchodilator

0.558 0.004 DBMET00975

0.8280.0040.828Antiadrenergic

0.509 0.005 DBMET00975

0.8250.0040.825Adrenaline antagonist

0.507 0.005 DBMET00975

0.8250.0040.825Spasmolytic

0.788 0.004 DBMET00975

0.7850.0060.785Antiobesity

0.783 0.006 DBMET00975

0.6840.0040.684Psychostimulant

0.16 0.107 DBMET00975

0.6680.0030.668Calcium channel L-type activator

0.591 0.007 DBMET00975

0.6740.010.674Toll-Like receptor 7 agonist

0.328 0.094 DBMET00975

0.6710.010.671Toll-Like receptor agonist

0.359 0.078 DBMET00975

0.6420.0060.642Vasodilator, coronary

0.368 0.047 DBMET00975

0.6360.0120.636Vasodilator, peripheral
0.6410.0210.641Cyclophilin D inhibitor

0.616 0.025 DBMET00975

0.6090.0040.609Peroxidase inhibitor

0.404 0.02 DBMET00975

0.6090.0180.609Aldehyde oxidase inhibitor
0.6040.0140.6045 Hydroxytryptamine release stimulant
0.5880.0330.588Transcription factor NF kappa B inhibitor

0.447 0.054 DBMET00975

0.5270.0020.527Phenylalanine 4-hydroxylase inhibitor

0.269 0.004 DBMET00975

0.5240.0130.524Cardiotonic

0.28 0.065 DBMET00975

0.5080.0040.508Anesthetic local

0.137 0.055 DBMET00975

0.5060.0020.506Adrenaline agonist

0.293 0.004 DBMET00975

0.4870.0020.487Beta adrenoreceptor antagonist

0.185 0.004 DBMET00975

0.4910.0090.491Interleukin agonist

0.197 0.124 DBMET00975

0.4730.0020.473Beta 2 adrenoreceptor antagonist

0.177 0.004 DBMET00975

0.4770.0170.477Hypoxia-inducible factor 1 alpha inhibitor

0.271 0.083 DBMET00975

0.4730.0140.473Vasodilator

0.272 0.058 DBMET00975

0.4860.0370.4865 Hydroxytryptamine release inhibitor
0.4380.0090.4385 Hydroxytryptamine uptake stimulant

0.204 0.143 DBMET00975

0.4130.0140.413Sodium/bile acid cotransporter inhibitor

0.39 0.02 DBMET00975

0.4040.0160.404Cyclic AMP phosphodiesterase inhibitor
0.4060.0230.406Calcium channel activator

0.247 0.151 DBMET00975

0.3830.0020.383Beta 1 adrenoreceptor antagonist

0.146 0.005 DBMET00975

0.3820.0020.382Beta 3 adrenoreceptor antagonist

0.212 0.004 DBMET00975

0.4260.0480.426Calpain 2 inhibitor
0.3650.0020.365Beta adrenoreceptor agonist

0.135 0.003 DBMET00975

0.4240.0630.424Histamine release inhibitor

0.358 0.096 DBMET00975

0.4420.0870.442Caspase 9 stimulant
0.3660.0130.366Tyrosine 3 hydroxylase inhibitor

0.195 0.145 DBMET00975

0.3490.0120.349Peptidyltransferase inhibitor

0.271 0.038 DBMET00975

0.3380.0020.338Adenylate cyclase stimulant

0.325 0.002 DBMET00975

0.3850.0530.602Antithrombotic

0.602 0.016 DBMET00975

DBMET00975
0.3940.0640.394GABA C receptor rho-3 antagonist
0.380.0540.538Cholesterol antagonist

0.538 0.027 DBMET00975

DBMET00975
0.330.0060.33Nitric-oxide synthase stimulant

0.176 0.139 DBMET00975

0.3360.0130.336Alpha-N-acetylglucosaminidase inhibitor
0.3570.0360.357Hypoglycemic
0.3440.0380.459Superoxide dismutase inhibitor

0.459 0.018 DBMET00975

DBMET00975
0.3160.0120.316Acetylcholine M1 receptor antagonist

0.163 0.064 DBMET00975

0.310.0080.31Acetylcholine muscarinic antagonist

0.155 0.041 DBMET00975

0.3450.0480.45Antioxidant

0.45 0.027 DBMET00975

DBMET00975
0.3060.0130.306Adenylate cyclase inhibitor

0.126 0.062 DBMET00975

0.3550.0630.423Immunostimulant

0.423 0.043 DBMET00975

DBMET00975
0.2930.0040.293Glutamate decarboxylase inhibitor

0.155 0.012 DBMET00975

0.3030.0140.303Cholinergic antagonist

0.124 0.07 DBMET00975

0.3350.0520.335Interleukin 2 agonist

0.222 0.154 DBMET00975

0.2940.0140.294Acetylcholine antagonist

0.122 0.069 DBMET00975

0.3210.0460.321Free radical scavenger

0.252 0.068 DBMET00975

0.2840.020.284Insulin sensitizer

0.226 0.05 DBMET00975

0.2670.0050.267Acetylcholine M3 receptor antagonist
0.2660.0110.266Expectorant

0.127 0.046 DBMET00975

0.2590.0050.259Mucolytic

0.156 0.029 DBMET00975

0.2790.0310.279Glyceraldehyde-3-phosphate dehydrogenase inhibitor
0.2470.0020.247Beta 2 adrenoreceptor agonist

0.144 0.003 DBMET00975

0.2830.040.283Calpain inhibitor
0.2390.0060.239Creatine kinase inhibitor

0.14 0.028 DBMET00975

0.2510.0210.251M18 aspartyl aminopeptidase inhibitor
0.2310.0060.231Alpha adrenoreceptor agonist
0.2730.0540.273DNA synthesis inhibitor

0.175 0.16 DBMET00975

0.2150.0020.215Beta 1 adrenoreceptor agonist

0.054 0.004 DBMET00975

0.220.0090.22Aminoacyl-tRNA synthetase inhibitor

0.147 0.02 DBMET00975

0.230.0340.23Amylase inhibitor
0.210.0150.236Carbonic anhydrase III inhibitor

0.236 0.011 DBMET00975

DBMET00975
0.2250.0330.225Melanin inhibitor
0.1940.0020.194Beta 3 adrenoreceptor agonist

0.027 0.004 DBMET00975

0.2560.0680.256Antiamyloidogenic
0.2140.030.214Monophenol monooxygenase inhibitor

0.149 0.047 DBMET00975

0.1820.0080.182Somatostatin 1 agonist

0.125 0.021 DBMET00975

0.3050.1310.474Antibacterial

0.474 0.048 DBMET00975

DBMET00975
0.1770.0080.189Anabolic

0.189 0.005 DBMET00975

DBMET00975
0.1990.030.366Cell wall synthesis inhibitor

0.366 0.007 DBMET00975

DBMET00975
0.2010.0320.525Hemostatic

0.525 0.004 DBMET00975

DBMET00975
0.1820.0140.182Sphingomyelinase inhibitor
0.240.0720.24Hypolipemic

0.147 0.14 DBMET00975

0.1820.0220.182Carbonic anhydrase XV inhibitor

0.118 0.048 DBMET00975

0.1790.0320.179Nav1.3 sodium channel blocker
0.2380.0930.238Gastrin inhibitor
0.1750.0320.175Interleukin 4 antagonist
0.2590.1190.259Apoptosis antagonist
0.1560.0180.156Histidine decarboxylase inhibitor
0.1590.0250.159Mediator release inhibitor
0.1690.0370.169Alkylator

0.138 0.053 DBMET00975

0.1420.0120.142Carbonic anhydrase stimulant

0.057 0.044 DBMET00975

0.1490.0210.149Electron transport complex I inhibitor
0.2020.0740.202Neurotrophic factor enhancer
0.1640.0380.224Cholesterol synthesis inhibitor

0.224 0.022 DBMET00975

DBMET00975
0.1830.0580.216Phospholipase C inhibitor

0.216 0.035 DBMET00975

DBMET00975
0.1620.0390.162Cyclooxygenase 3 inhibitor
0.1760.0540.176Neurotensin receptor agonist
0.1460.0270.146Transcription factor STAT6 inhibitor
0.1450.0270.181Catalase inhibitor

0.181 0.019 DBMET00975

DBMET00975
0.1280.0150.128Acetylcholine M2 receptor antagonist
0.1470.0350.147GABA C receptor agonist
0.1510.040.151Cystathionine beta-synthase inhibitor
0.1850.0740.185Nitric oxide antagonist

0.148 0.096 DBMET00975

0.2290.1180.229Insulysin inhibitor
0.2030.0930.435Angiogenesis stimulant

0.435 0.017 DBMET00975

DBMET00975
0.1380.0290.138DOPA decarboxylase inhibitor
0.1460.0390.179Aminopeptidase B inhibitor

0.179 0.027 DBMET00975

DBMET00975
0.1520.0460.152Proteasome inhibitor
0.160.0620.16Lipid peroxidase inhibitor

0.158 0.063 DBMET00975

0.1170.020.117Aminopeptidase I inhibitor
0.1210.0250.121Ornithine decarboxylase inhibitor
0.1070.0130.107Alpha 2 adrenoreceptor agonist
0.1350.0410.176Nav1.4 sodium channel blocker

0.176 0.025 DBMET00975

DBMET00975
0.1080.0150.108Alpha 1 adrenoreceptor agonist
0.1640.0710.245Thrombolytic

0.245 0.035 DBMET00975

DBMET00975
0.1460.0530.146Ca2+-transporting ATPase inhibitor
0.1470.0540.147Toll-Like receptor 2 antagonist
0.1070.0140.107Maillard reaction inhibitor
0.1960.1060.256RNA-directed DNA polymerase inhibitor

0.256 0.046 DBMET00975

DBMET00975
0.1030.0150.161Neuraminidase (influenza) inhibitor

0.161 0.006 DBMET00975

DBMET00975
0.130.0430.13GABA C receptor antagonist
0.1230.0360.123Prolactin inhibitor
0.1470.0610.147Neurotrophic factor
0.1560.070.156Interferon gamma antagonist
0.1310.0450.131Photosensitizer
0.1520.0670.152Protein kinase stimulant
0.1010.0160.101GABA B receptor agonist
0.1290.0460.129Chelator
0.1140.0320.114NADH dehydrogenase inhibitor
0.1030.0220.103Estrogen-related receptor beta agonist
0.2390.1580.239Immunosuppressant
0.1620.0820.162ATPase inhibitor
0.1230.0420.123Urease inhibitor
0.1150.0360.115Glutamate (mGluR7) agonist
0.1180.0410.118Factor V inhibitor
0.1240.0480.124Estrogen antagonist
0.1250.050.125Ferrochelatase inhibitor
0.1640.0890.164Succinate dehydrogenase inhibitor
0.1940.120.194DNA damaging
0.0780.0050.078Alpha 1d adrenoreceptor agonist
0.1490.0750.149GABA C receptor rho-2 antagonist
0.0910.0190.114Neuraminidase inhibitor

0.114 0.011 DBMET00975

DBMET00975
0.1730.1010.173Interleukin antagonist
0.1160.0440.116GABA C receptor rho-1 antagonist
0.0830.0120.083Myc inhibitor
0.0930.0230.093Secretase beta inhibitor
0.210.1410.2112-Lipoxygenase inhibitor
0.1160.0470.116Adenylate kinase inhibitor
0.1240.0560.124Microtubule formation inhibitor
0.1660.0980.166Anesthetic general
0.1040.0370.104Glutamate release inhibitor
0.0880.0210.088Acetylcholine M5 receptor antagonist
0.0760.0090.076Alpha 1b adrenoreceptor agonist

0.048 0.042 DBMET00975

0.1110.0450.111Estrogen receptor beta antagonist

0.09 0.083 DBMET00975

0.1040.0420.108Bile acid receptor antagonist

0.108 0.035 DBMET00975

DBMET00975
0.2630.2010.263Apoptosis agonist
0.1290.0680.129Vanilloid 1 agonist
0.0990.040.114Carbonic anhydrase VI inhibitor

0.114 0.032 DBMET00975

DBMET00975
0.0860.0270.091Phospholipase D inhibitor

0.091 0.021 DBMET00975

DBMET00975
0.0730.0150.089Alpha-mannosidase inhibitor

0.089 0.008 DBMET00975

DBMET00975
0.1060.0470.106Lanosterol 14 alpha demethylase inhibitor
0.0650.0080.065Diamine oxidase inhibitor
0.130.0740.13Sphingosine 1-phosphate receptor 2 antagonist
0.1910.1360.191Neuropeptide Y2 antagonist
0.1370.0810.137Pregnane X receptor agonist
0.1330.0770.133Farnesoid X receptor antagonist
0.0770.0230.077Heat shock protein 90 beta antagonist
0.1040.0510.104HIV-1 integrase (Overall Integration) inhibitor
0.0760.0260.076Alcohol oxidase inhibitor
0.1570.1070.157P-glycoprotein inhibitor
0.1380.0880.138Phospholipase A2 inhibitor
0.1240.0760.124Antibacterial (Helicobacter pylori)

0.116 0.087 DBMET00975

0.1040.0560.104UDP-glucose 4-epimerase inhibitor
0.1530.1060.153Amyloid beta aggregation inhibitor
0.150.1040.15DNA methyltransferase I inhibitor
0.1110.0650.111Alpha 2b adrenoreceptor antagonist
0.050.0050.05Alpha 1a adrenoreceptor agonist
0.0850.040.085Glutamate dehydrogenase inhibitor
0.0610.0160.078Mannosidase inhibitor

0.078 0.009 DBMET00975

DBMET00975
0.0860.0420.086Keratolytic
0.0820.040.082MAP kinase kinase 7 inhibitor
0.0860.0440.097Na+ K+ transporting ATPase inhibitor

0.097 0.035 DBMET00975

DBMET00975
0.0570.0150.057Neuraminidase (Influenza A) inhibitor
0.0550.0140.055Dopamine D5 agonist
0.0580.0190.058Oxytocin agonist
0.0430.0040.043Alpha 2a adrenoreceptor agonist
0.0480.0090.048Lysophosphatidic acid 2 receptor antagonist
0.090.0520.09Granulocyte macrophage colony stimulating factor agonist
0.0630.0280.063Sphingosine kinase 2 inhibitor
0.0670.0320.067Cathepsin E inhibitor
0.0690.0340.07NMDA 2C receptor antagonist

0.07 0.033 DBMET00975

DBMET00975
0.1510.1170.151DNA methylase inhibitor
0.090.0560.09Alpha 2 adrenoreceptor antagonist
0.0520.0190.052Somatostatin 1 antagonist
0.0850.0540.085Histamine H2 receptor antagonist
0.0890.0580.089Opioid antagonist
0.0880.0580.088Interleukin 5 antagonist
0.1450.1150.197Hepatoprotectant

0.197 0.067 DBMET00975

DBMET00975
0.0340.0040.034Neuraminidase (Influenza B) inhibitor
0.0340.0050.034Calcium-sensing receptor antagonist
0.0560.0280.056Lysophosphatidic acid 3 receptor antagonist
0.0350.0070.0461,3-Beta-glucan synthase inhibitor

0.046 0.003 DBMET00975

DBMET00975
0.0420.0140.042Ceramide glucosyltransferase inhibitor

0.037 0.021 DBMET00975

0.0930.0670.093Phosphodiesterase 6D inhibitor
0.0610.0340.061Ribonucleoside-diphosphate reductase inhibitor
0.1290.1020.129Neuropeptide Y1 antagonist
0.0620.0350.062Argininosuccinate synthase inhibitor
0.0960.070.131Gastric antisecretory

0.131 0.036 DBMET00975

DBMET00975
0.0610.0360.061Ribonucleotide reductase inhibitor
0.1270.1010.127Insulin secretagoues
0.0460.0210.0463-Hydroxyanthranilate 3,4-dioxygenase inhibitor
0.0640.0390.064Purinergic P2X1 antagonist
0.0590.0340.059Acetyl-CoA transferase 2 inhibitor
0.0640.0390.064Carbamoyl phosphate synthetase inhibitor
0.0430.020.043Arginase inhibitor
0.0620.0390.062Androgen agonist

0.054 0.049 DBMET00975

0.130.1070.13Growth hormone agonist
0.0560.0340.056Ornithine carbamoyltransferase inhibitor
0.0530.0330.122Factor IXa inhibitor

0.122 0.005 DBMET00975

DBMET00975
0.0560.0360.056Glucosylceramidase inhibitor
0.0860.0660.218Triose-phosphate isomerase inhibitor

0.218 0.009 DBMET00975

DBMET00975
0.0710.0520.071Glycine receptor agonist
0.0670.0470.067Purinergic P2X2 antagonist
0.0590.040.085Sphingosine kinase inhibitor

0.085 0.013 DBMET00975

DBMET00975
0.0510.0330.051Potassium channel (Inward rectifier) blocker
0.0590.040.059Sphingosine 1-phosphate receptor 3 antagonist
0.0250.0060.025Ileal bile acid transport inhibitor
0.0620.0450.062Opioid delta receptor antagonist
0.0620.0450.077NMDA receptor agonist

0.077 0.031 DBMET00975

DBMET00975
0.0790.0620.079Glutathione S-transferase inhibitor
0.0310.0150.031Purinergic P2Y15 antagonist
0.1010.0850.101DNA polymerase I inhibitor
0.1240.1080.124Thiol protease inhibitor
0.0720.0560.287Carbonic anhydrase XIII inhibitor

0.287 0.006 DBMET00975

DBMET00975
0.0490.0340.049Bombesin 2 receptor antagonist
0.0710.0560.071Alpha 2a adrenoreceptor antagonist
0.080.0660.103NMDA receptor antagonist

0.103 0.045 DBMET00975

DBMET00975
0.0220.0080.022Antibiotic Anthracycline-like
0.0360.0230.039Phosphoglycerate kinase inhibitor

0.039 0.02 DBMET00975

DBMET00975
0.050.0380.05NMDA 2A receptor antagonist
0.090.0780.09Nitric-oxide synthase inhibitor
0.0680.0560.208Cathepsin G inhibitor

0.208 0.015 DBMET00975

DBMET00975
0.0590.0480.0595 Hydroxytryptamine 2A agonist
0.0510.040.051Cathepsin D inhibitor
0.0710.060.071Vanilloid 4 agonist
0.0790.0690.079Myeloperoxidase inhibitor
0.0740.0630.074Interferon agonist
0.0420.0330.042Geranyltranstransferase inhibitor
0.0260.0160.026Lysophosphatidic acid receptor 1 agonist
0.0730.0640.073Acetylcholine nicotinic antagonist
0.0540.0460.054Fibroblast growth factor 4 antagonist
0.0830.0750.083UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor
0.0520.0450.052Cathepsin B inhibitor
0.0250.0180.025Vanilloid 2 agonist

0.023 0.022 DBMET00975

0.1120.1050.112Papain-like protease (SARS coronavirus) inhibitor
0.0820.0760.082Alcohol dehydrogenase inhibitor
0.060.0540.06Interferon inducer
0.0890.0830.089Falcipain 3 inhibitor
0.050.0440.059Leukotriene B4 antagonist

0.059 0.029 DBMET00975

DBMET00975
0.0270.0230.027Vasopressin 1A agonist
0.0270.0240.027Plasmepsin I inhibitor
0.1290.1260.129Heat shock protein 70 antagonist
0.0980.0950.098Caspase 3 inhibitor
0.0840.0810.084Protease inhibitor
0.0290.0280.029Calcitonin receptor agonist
0.0220.0270.029Thyroid hormone agonist

0.029 0.014 DBMET00975

DBMET00975
0.0420.0480.062Aldose reductase inhibitor

0.062 0.031 DBMET00975

DBMET00975
0.0710.0790.074Inducible nitric-oxide synthase inhibitor

0.074 0.073 DBMET00975

DBMET00975
0.0490.0610.214Selectin antagonist

0.214 0.01 DBMET00975

DBMET00975
0.0170.0310.118Estrogen receptor beta agonist

0.118 0.009 DBMET00975

DBMET00975
0.020.0350.024Glutamate (mGluR1) agonist

0.024 0.018 DBMET00975

DBMET00975
0.0320.0530.19Estrogen agonist

0.19 0.009 DBMET00975

DBMET00975
0.030.0690.094Carbonic anhydrase VB inhibitor

0.094 0.017 DBMET00975

DBMET00975
0.0120.0520.02Glutamate (mGluR1a) agonist

0.02 0.019 DBMET00975

DBMET00975
0.0220.0670.081Dopamine D2 agonist

0.081 0.014 DBMET00975

DBMET00975
0.0230.0740.683Cholecystokinin B agonist

0.683 0.001 DBMET00975

DBMET00975
0.0960.1470.382Diuretic

0.382 0.014 DBMET00975

DBMET00975
0.040.0930.197HIV-1 integrase (3'-Processing) inhibitor

0.197 0.01 DBMET00975

DBMET00975
0.0430.0960.078Adenine nucleotide translocase inhibitor

0.078 0.01 DBMET00975

DBMET00975
0.0390.0940.187Carbonic anhydrase V inhibitor

0.187 0.008 DBMET00975

DBMET00975
0.0420.10.132Carbonic anhydrase VA inhibitor

0.132 0.015 DBMET00975

DBMET00975
0.0350.1010.09NMDA 2 receptor antagonist

0.09 0.037 DBMET00975

DBMET00975
0.0480.1160.096HIV-1 integrase inhibitor

0.096 0.027 DBMET00975

DBMET00975
0.0240.0920.116Leukocyte elastase inhibitor

0.116 0.008 DBMET00975

DBMET00975
0.0470.1250.14CDC25A inhibitor

0.14 0.014 DBMET00975

DBMET00975
0.0250.1270.148HIV-1 integrase (Strand Transfer) inhibitor

0.148 0.013 DBMET00975

DBMET00975
0.060.1640.085Protein kinase C zeta inhibitor

0.085 0.076 DBMET00975

DBMET00975
0.0470.160.165Protein-tyrosine phosphatase 1B inhibitor

0.165 0.04 DBMET00975

DBMET00975
0.0430.160.075Glycine receptor antagonist

0.075 0.065 DBMET00975

DBMET00975
0.0260.1460.247NMDA 2B receptor antagonist

0.247 0.005 DBMET00975

DBMET00975
0.0870.2080.327Platelet adhesion inhibitor

0.327 0.026 DBMET00975

DBMET00975
0.0760.1970.469Anticoagulant

0.469 0.012 DBMET00975

DBMET00975
0.0050.1340.717Cholecystokinin agonist

0.717 0.002 DBMET00975

DBMET00975
0.0350.1630.103Thrombin inhibitor

0.103 0.024 DBMET00975

DBMET00975
0.0050.1580.661Cholecystokinin A agonist

0.661 0.002 DBMET00975

DBMET00975
0.0420.1980.071Chymotrypsin inhibitor

0.071 0.068 DBMET00975

DBMET00975
0.0630.2280.277Protein-tyrosine phosphatase inhibitor

0.277 0.024 DBMET00975

DBMET00975
0.0040.1780.115Estrone sulfatase inhibitor

0.115 0.004 DBMET00975

DBMET00975
0.0170.210.091Elastase inhibitor

0.091 0.012 DBMET00975

DBMET00975
0.0090.2290.06NMDA 2D receptor antagonist

0.06 0.005 DBMET00975

DBMET00975
0.0040.2260.343Cholecystokinin A antagonist

0.343 0.004 DBMET00975

DBMET00975
0.0140.2510.029Toll-Like receptor 4 agonist

0.029 0.014 DBMET00975

DBMET00975
0.0050.2650.288Cholecystokinin antagonist

0.288 0.004 DBMET00975

DBMET00975
0.0040.2770.252Cholecystokinin B antagonist

0.252 0.004 DBMET00975

DBMET00975
0.0390.3760.266Dual specificity phosphatase inhibitor

0.266 0.035 DBMET00975

DBMET00975
0.0370.5690.227Angiogenesis inhibitor

0.227 0.141 DBMET00975

DBMET00975
0.0160.5820.192Multidrug resistance-associated protein 1 inhibitor

0.192 0.012 DBMET00975

DBMET00975
0.0160.590.219Dual specificity phosphatase 3 inhibitor

0.219 0.052 DBMET00975

DBMET00975
0.0090.5930.037Purinergic P2Y2 antagonist

0.037 0.019 DBMET00975

DBMET00975
Ext Pa Pi Pmax Activity Other Results ID Pa_max