Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.6170.0020.6175 Hydroxytryptamine 3 antagonist

0.315 0.004 DBMET01834

0.307 0.004 DBMET01835

0.257 0.004 DBMET01836

0.50.0020.55 Hydroxytryptamine 3B antagonist

0.196 0.003 DBMET01834

0.191 0.003 DBMET01835

0.118 0.004 DBMET01836

0.4390.0090.4395 Hydroxytryptamine antagonist

0.242 0.026 DBMET01834

0.226 0.029 DBMET01835

0.279 0.021 DBMET01836

0.3930.010.393Cholinergic

0.345 0.014 DBMET01834

0.326 0.015 DBMET01835

0.304 0.018 DBMET01836

0.3610.0060.3615 Hydroxytryptamine 2C antagonist

0.23 0.014 DBMET01834

0.226 0.014 DBMET01835

0.189 0.019 DBMET01836

0.350.0110.355 Hydroxytryptamine 2B antagonist

0.223 0.022 DBMET01834

0.23 0.022 DBMET01835

0.152 0.04 DBMET01836

0.3410.0130.3415 Hydroxytryptamine 2 antagonist

0.208 0.029 DBMET01834

0.204 0.029 DBMET01835

0.198 0.031 DBMET01836

0.3310.010.331Acetylcholinesterase inhibitor

0.31 0.012 DBMET01834

0.292 0.014 DBMET01835

0.27 0.017 DBMET01836

0.3790.0710.427GABA C receptor rho-3 antagonist

0.367 0.077 DBMET01834

0.427 0.05 DBMET01835

0.276 0.133 DBMET01836

DBMET01835
0.2570.0230.257Acetylcholine M1 receptor antagonist

0.251 0.025 DBMET01834

0.246 0.026 DBMET01835

0.256 0.024 DBMET01836

0.2720.0590.272Potassium channel (Voltage-sensitive) blocker

0.152 0.135 DBMET01834

0.154 0.134 DBMET01835

0.2290.0170.2295 Hydroxytryptamine 2A antagonist

0.126 0.035 DBMET01834

0.125 0.035 DBMET01835

0.124 0.036 DBMET01836

0.2660.0560.297Cyclic AMP phosphodiesterase inhibitor

0.297 0.043 DBMET01834

0.259 0.059 DBMET01835

0.174 0.118 DBMET01836

DBMET01834
0.2110.020.211Butyrylcholinesterase inhibitor

0.184 0.024 DBMET01834

0.164 0.029 DBMET01835

0.149 0.034 DBMET01836

0.2050.0170.205GABA receptor agonist

0.153 0.034 DBMET01834

0.145 0.039 DBMET01835

0.143 0.04 DBMET01836

0.1760.0180.176Histamine H1 receptor antagonist

0.094 0.045 DBMET01834

0.09 0.048 DBMET01835

0.096 0.043 DBMET01836

0.160.0080.16GABA A receptor antagonist

0.111 0.014 DBMET01834

0.1 0.016 DBMET01835

0.071 0.025 DBMET01836

0.2210.0790.221HERG channel blocker
0.1510.0090.151GABA receptor antagonist

0.103 0.015 DBMET01834

0.093 0.017 DBMET01835

0.066 0.028 DBMET01836

0.1720.0330.179Acetylcholine muscarinic antagonist

0.161 0.038 DBMET01834

0.161 0.038 DBMET01835

0.179 0.031 DBMET01836

DBMET01836
0.1630.0380.191DNA intercalator

0.161 0.038 DBMET01834

0.156 0.04 DBMET01835

0.191 0.028 DBMET01836

DBMET01836
0.1510.0270.151Alpha 2 adrenoreceptor antagonist

0.119 0.037 DBMET01834

0.124 0.035 DBMET01835

0.087 0.058 DBMET01836

0.1280.0080.1285 Hydroxytryptamine 3A antagonist

0.066 0.048 DBMET01834

0.066 0.047 DBMET01835

0.1240.0040.1245 Hydroxytryptamine 4 antagonist

0.093 0.008 DBMET01834

0.093 0.008 DBMET01835

0.085 0.011 DBMET01836

0.1920.0850.217Psychostimulant

0.168 0.102 DBMET01834

0.183 0.09 DBMET01835

0.217 0.071 DBMET01836

DBMET01836
0.1560.0490.156Cholinergic antagonist

0.143 0.057 DBMET01834

0.145 0.055 DBMET01835

0.155 0.049 DBMET01836

0.1150.0180.115Benzodiazepine agonist
0.1480.0510.148Acetylcholine antagonist

0.136 0.058 DBMET01834

0.138 0.057 DBMET01835

0.148 0.051 DBMET01836

0.1070.0110.107Protein kinase C beta inhibitor

0.106 0.011 DBMET01834

0.1 0.013 DBMET01835

0.073 0.041 DBMET01836

0.1160.0260.116GABA A receptor agonist

0.082 0.059 DBMET01834

0.08 0.064 DBMET01835

0.083 0.058 DBMET01836

0.1460.060.146Pregnane X receptor agonist

0.14 0.074 DBMET01834

0.128 0.106 DBMET01835

0.1810.1060.181Potassium channel blocker
0.1270.0530.127Alpha 2b adrenoreceptor antagonist

0.099 0.076 DBMET01834

0.105 0.071 DBMET01835

0.0880.0180.119NMDA 2B receptor antagonist

0.114 0.013 DBMET01834

0.119 0.012 DBMET01835

0.097 0.016 DBMET01836

DBMET01835
0.080.0170.08Corticotropin releasing factor 2 receptor antagonist
0.0880.0290.0885 Hydroxytryptamine 1B antagonist
0.090.0320.09Alpha adrenoreceptor agonist

0.076 0.041 DBMET01834

0.086 0.034 DBMET01835

0.07 0.046 DBMET01836

0.1830.1270.188MAP-kinase-activated kinase 5 inhibitor

0.188 0.12 DBMET01834

0.187 0.121 DBMET01835

DBMET01834
0.0860.0320.086Cannabinoid receptor agonist
0.2420.190.242Analgesic

0.228 0.205 DBMET01834

0.0850.0320.085Neuronal nicotinic receptor antagonist

0.067 0.047 DBMET01834

0.072 0.043 DBMET01835

0.1120.060.181Topoisomerase I inhibitor

0.164 0.036 DBMET01834

0.155 0.039 DBMET01835

0.181 0.031 DBMET01836

DBMET01836
0.10.0510.101Phosphodiesterase 6D inhibitor

0.101 0.049 DBMET01834

0.1 0.051 DBMET01835

0.089 0.08 DBMET01836

DBMET01834
0.0720.0230.072Melanin-concentrating hormone receptor 1 antagonist
0.0870.0430.087Transforming growth factor beta 3 antagonist

0.077 0.074 DBMET01835

0.0830.0430.083Acetylcholine M4 receptor antagonist
0.0870.0480.087Acetylcholine nicotinic antagonist

0.071 0.067 DBMET01834

0.073 0.064 DBMET01835

0.0410.0070.041CYP24 inhibitor

0.04 0.007 DBMET01834

0.037 0.008 DBMET01835

0.033 0.009 DBMET01836

0.0940.0610.094Alpha 2d adrenoreceptor antagonist
0.0860.0570.086Hematopoietic

0.085 0.06 DBMET01834

0.085 0.059 DBMET01835

0.1540.1250.154Anticonvulsant
0.1730.1490.1815 Hydroxytryptamine release stimulant

0.181 0.14 DBMET01834

DBMET01834
0.0630.0390.083Aromatase inhibitor

0.083 0.026 DBMET01834

0.078 0.029 DBMET01835

0.075 0.031 DBMET01836

DBMET01834
0.0370.0150.037Protein kinase C beta II inhibitor

0.037 0.014 DBMET01834

0.036 0.016 DBMET01835

0.03 0.028 DBMET01836

0.1290.1080.129GABA C receptor rho-2 antagonist

0.129 0.108 DBMET01835

0.0590.0380.059Alpha 1 adrenoreceptor agonist

0.054 0.045 DBMET01835

0.0480.0270.058Dopamine D5 antagonist

0.058 0.02 DBMET01834

0.051 0.024 DBMET01835

0.042 0.03 DBMET01836

DBMET01834
0.0550.0350.055Nicotinic receptor alpha7 subunit antagonist
0.140.1210.152Lipocortins synthesis antagonist

0.152 0.102 DBMET01834

0.136 0.128 DBMET01836

DBMET01834
0.0550.0360.055Thromboxane synthase inhibitor

0.052 0.043 DBMET01834

0.051 0.047 DBMET01835

0.070.0520.07Telomerase inhibitor
0.0850.0670.085Phosphodiesterase I inhibitor

0.08 0.076 DBMET01834

0.083 0.071 DBMET01836

0.0670.0490.067Protein kinase C alpha inhibitor
0.1350.1210.283Amyloid beta aggregation inhibitor

0.224 0.066 DBMET01834

0.208 0.074 DBMET01835

0.283 0.048 DBMET01836

DBMET01836
0.0720.0580.072Phosphodiesterase VI inhibitor

0.069 0.065 DBMET01834

0.071 0.059 DBMET01835

0.1940.1830.198Vasodilator, peripheral

0.198 0.179 DBMET01834

0.196 0.18 DBMET01836

DBMET01834
0.1930.1850.193Ca2+/calmodulin-dependent kinase IV inhibitor
0.0510.0440.051Bromodomain-containing protein 4 inhibitor
0.0580.0530.089Dopamine D1 antagonist

0.089 0.029 DBMET01834

0.078 0.034 DBMET01835

0.071 0.039 DBMET01836

DBMET01834
0.0280.0230.028Glutamate (mGluR2) antagonist
0.0550.0520.0555 Hydroxytryptamine 2A agonist
0.0540.0510.054Alpha 2 adrenoreceptor agonist
0.080.0780.08Antihistaminic
0.0310.0320.032Protein kinase C beta I inhibitor

0.032 0.029 DBMET01834

DBMET01834
0.1260.130.149Antipruritic

0.13 0.123 DBMET01834

0.149 0.096 DBMET01836

DBMET01836
0.0450.0520.051Protein kinase C eta inhibitor

0.051 0.042 DBMET01834

0.049 0.044 DBMET01835

DBMET01834
0.090.0970.096Protein kinase C gamma inhibitor

0.096 0.084 DBMET01834

DBMET01834
0.0530.0620.088Opioid mu receptor antagonist

0.088 0.036 DBMET01834

0.082 0.039 DBMET01835

DBMET01834
0.0720.0810.103Opioid antagonist

0.103 0.046 DBMET01834

0.098 0.049 DBMET01835

0.081 0.068 DBMET01836

DBMET01834
0.0280.0460.033Tubulin agonist

0.033 0.026 DBMET01836

DBMET01836
0.0840.1030.138Topoisomerase II inhibitor

0.136 0.057 DBMET01834

0.124 0.064 DBMET01835

0.138 0.055 DBMET01836

DBMET01836
0.0640.0890.09Opioid kappa receptor antagonist

0.09 0.046 DBMET01834

0.084 0.052 DBMET01835

DBMET01834
0.0220.050.039Catechol O-methyltransferase inhibitor

0.033 0.022 DBMET01834

0.033 0.022 DBMET01835

0.039 0.014 DBMET01836

DBMET01836
0.0510.0940.085Topoisomerase II alpha inhibitor

0.085 0.049 DBMET01834

0.075 0.057 DBMET01835

DBMET01834
0.120.1760.142Platelet aggregation inhibitor

0.142 0.139 DBMET01835

DBMET01835
0.2060.2640.349Calcium channel L-type activator

0.266 0.188 DBMET01834

0.349 0.118 DBMET01835

0.24 0.217 DBMET01836

DBMET01835
0.1430.2180.198DNA synthesis inhibitor

0.175 0.161 DBMET01834

0.176 0.159 DBMET01835

0.198 0.126 DBMET01836

DBMET01836
0.040.1140.057Heat shock protein 90 beta antagonist

0.056 0.047 DBMET01834

0.057 0.045 DBMET01835

DBMET01835
0.1110.190.135MAP kinase kinase 4 inhibitor

0.135 0.1 DBMET01834

DBMET01834
0.1760.2610.262Antibacterial

0.239 0.188 DBMET01834

0.227 0.199 DBMET01835

0.262 0.166 DBMET01836

DBMET01836
0.0480.1670.1Bronchodilator

0.1 0.064 DBMET01836

DBMET01836
0.0340.1570.072NAD(P)H dehydrogenase (quinone) inhibitor

0.072 0.059 DBMET01836

DBMET01836
0.1740.3140.258Apoptosis agonist

0.258 0.205 DBMET01834

0.257 0.207 DBMET01835

0.248 0.216 DBMET01836

DBMET01834
0.0510.2020.076MAP kinase kinase 7 inhibitor

0.076 0.06 DBMET01834

DBMET01834
0.1840.3460.258Caspase 9 stimulant

0.258 0.243 DBMET01835

DBMET01835
0.0090.2420.042Cathepsin L2 inhibitor

0.042 0.027 DBMET01836

DBMET01836
0.1060.3710.214Sodium/bile acid cotransporter inhibitor

0.214 0.17 DBMET01834

DBMET01834
Ext Pa Pi Pmax Activity Other Results ID Pa_max