Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.8890.0050.931Antiinflammatory

0.931 0.005 DBMET00589

DBMET00589
0.7790.0030.779Cyclooxygenase 1 inhibitor

0.493 0.005 DBMET00589

0.6770.0040.882Non-steroidal antiinflammatory agent

0.882 0.003 DBMET00589

DBMET00589
0.6680.010.793Cholesterol antagonist

0.793 0.004 DBMET00589

DBMET00589
0.6580.0050.658Superoxide dismutase inhibitor
0.640.0140.64Aldehyde oxidase inhibitor
0.620.0040.62Amyloid beta precursor protein antagonist

0.163 0.087 DBMET00589

0.6290.0220.629Analgesic

0.35 0.109 DBMET00589

0.5840.0040.584Cyclooxygenase inhibitor

0.37 0.009 DBMET00589

0.5580.0110.558Calcium channel L-type activator

0.412 0.073 DBMET00589

0.5480.0030.548Calcium channel activator

0.337 0.059 DBMET00589

0.5060.0080.506Anesthetic general

0.434 0.013 DBMET00589

0.4820.0140.482Hypolipemic

0.448 0.018 DBMET00589

0.4640.0050.464Interleukin 6 antagonist

0.284 0.017 DBMET00589

0.5010.050.759Cyclophilin D inhibitor

0.759 0.009 DBMET00589

DBMET00589
0.4790.0320.703Antithrombotic

0.703 0.008 DBMET00589

DBMET00589
0.4860.0460.844Transcription factor NF kappa B inhibitor

0.844 0.01 DBMET00589

DBMET00589
0.450.0260.45Lipoxygenase inhibitor
0.4330.010.433Sodium/bile acid cotransporter inhibitor

0.417 0.013 DBMET00589

0.4470.0250.447Interleukin antagonist

0.172 0.102 DBMET00589

0.4260.0080.502Alpha-N-acetylglucosaminidase inhibitor

0.502 0.005 DBMET00589

DBMET00589
0.4190.0040.419Gastrin inhibitor

0.308 0.028 DBMET00589

0.4190.0220.538Interleukin 2 agonist

0.538 0.005 DBMET00589

DBMET00589
0.4160.0250.609Hypoglycemic

0.609 0.008 DBMET00589

DBMET00589
0.3870.0060.387Interleukin 1 antagonist

0.183 0.041 DBMET00589

0.3820.0060.382Cyclooxygenase 2 inhibitor

0.245 0.021 DBMET00589

0.4310.060.487Histamine release inhibitor

0.487 0.033 DBMET00589

DBMET00589
0.3690.0040.369Interleukin 8 antagonist

0.1 0.096 DBMET00589

0.380.0210.38Platelet aggregation inhibitor
0.3860.040.582Vasodilator, coronary

0.582 0.009 DBMET00589

DBMET00589
0.3520.0080.352Chelator

0.119 0.054 DBMET00589

0.3710.030.371Amyloid beta aggregation inhibitor

0.213 0.071 DBMET00589

0.3730.040.709Antioxidant

0.709 0.005 DBMET00589

DBMET00589
0.3970.0640.567Immunosuppressant

0.567 0.018 DBMET00589

DBMET00589
0.3570.0320.357Insulysin inhibitor
0.340.0180.34Tyrosine 3 hydroxylase inhibitor
0.3430.0310.478Interleukin agonist

0.478 0.01 DBMET00589

DBMET00589
0.3590.050.55Spasmolytic

0.55 0.018 DBMET00589

DBMET00589
0.3110.0050.346ATPase inhibitor

0.346 0.004 DBMET00589

DBMET00589
0.3220.020.339Thrombolytic

0.339 0.018 DBMET00589

DBMET00589
0.3010.0040.301HIV-1 integrase (Overall Integration) inhibitor
0.3020.0060.563Cyclooxygenase 3 inhibitor

0.563 0.003 DBMET00589

DBMET00589
0.3020.0130.302Phospholipase A2 inhibitor

0.233 0.028 DBMET00589

0.3550.0720.355Thyroid hormone antagonist
0.2870.010.287GABA C receptor agonist
0.3280.0530.328Hypoxia-inducible factor 1 alpha inhibitor

0.255 0.096 DBMET00589

0.320.0460.599Free radical scavenger

0.599 0.009 DBMET00589

DBMET00589
0.390.1170.561Caspase 9 stimulant

0.561 0.042 DBMET00589

DBMET00589
0.2770.0050.277ABCA1 expression enhancer
0.2740.0030.274Arachidonic acid antagonist

0.22 0.017 DBMET00589

0.2770.0150.277Succinate dehydrogenase inhibitor
0.2620.0030.262Glycine receptor agonist

0.232 0.003 DBMET00589

0.2680.0110.268Ferrochelatase inhibitor
0.260.0030.26Bile acid receptor antagonist

0.118 0.021 DBMET00589

0.30.0450.35 Hydroxytryptamine uptake stimulant
0.260.0090.26Adenylate kinase inhibitor

0.152 0.026 DBMET00589

0.2530.0030.253Liver X receptor alpha agonist
0.2840.040.284Peroxidase inhibitor
0.2680.0250.268Insulin sensitizer

0.201 0.072 DBMET00589

0.2450.0040.245Peroxisome proliferator-activated receptor gamma antagonist

0.07 0.052 DBMET00589

0.2480.0070.26Mucolytic

0.26 0.005 DBMET00589

DBMET00589
0.2520.0110.252Farnesoid X receptor antagonist

0.136 0.071 DBMET00589

0.2470.0070.337Triose-phosphate isomerase inhibitor

0.337 0.004 DBMET00589

DBMET00589
0.2470.0080.247Alcohol dehydrogenase inhibitor

0.109 0.043 DBMET00589

0.3520.1130.3525 Hydroxytryptamine release inhibitor

0.307 0.157 DBMET00589

0.290.0550.551Antiamyloidogenic

0.551 0.011 DBMET00589

DBMET00589
0.2370.0090.237Porphobilinogen synthase inhibitor
0.3070.0780.485Immunomodulator

0.485 0.025 DBMET00589

DBMET00589
0.2540.0270.485Amylase inhibitor

0.485 0.006 DBMET00589

DBMET00589
0.2330.0150.515Expectorant

0.515 0.004 DBMET00589

DBMET00589
0.2340.0160.249Mannose-6-phosphate isomerase inhibitor

0.249 0.012 DBMET00589

DBMET00589
0.2180.0060.218Peroxisome proliferator-activated receptor gamma agonist

0.064 0.055 DBMET00589

0.2140.0040.214Ornithine decarboxylase inhibitor

0.128 0.021 DBMET00589

0.3470.140.72Apoptosis agonist

0.72 0.027 DBMET00589

DBMET00589
0.2680.0620.733Angiogenesis stimulant

0.733 0.004 DBMET00589

DBMET00589
0.2280.0230.267Hexokinase inhibitor

0.267 0.014 DBMET00589

DBMET00589
0.2680.0650.376Platelet antagonist

0.376 0.032 DBMET00589

DBMET00589
0.2230.0190.297Cell adhesion inhibitor

0.297 0.01 DBMET00589

DBMET00589
0.2350.0330.235Histone acetyltransferase inhibitor
0.3090.1090.309Calpain 2 inhibitor
0.2310.0320.372Interferon gamma antagonist

0.372 0.012 DBMET00589

DBMET00589
0.2120.0130.212Catalase inhibitor
0.2460.0520.246RNA-directed DNA polymerase inhibitor

0.217 0.078 DBMET00589

0.1980.0040.198CXC chemokine 1 receptor antagonist
0.2010.0090.212Cell adhesion molecule inhibitor

0.212 0.009 DBMET00589

DBMET00589
0.2860.0950.434Apoptosis antagonist

0.434 0.03 DBMET00589

DBMET00589
0.2310.040.231Lipocortins synthesis antagonist

0.167 0.084 DBMET00589

0.3040.1130.304GABA C receptor rho-3 antagonist
0.2020.0120.202GABA C receptor antagonist
0.2430.0540.508Nitric oxide antagonist

0.508 0.015 DBMET00589

DBMET00589
0.1920.0040.192Peroxisome proliferator-activated receptor alpha agonist
0.1910.0080.191DOPA decarboxylase inhibitor
0.1930.0170.193UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor

0.18 0.019 DBMET00589

0.1890.0150.212Photosensitizer

0.212 0.01 DBMET00589

DBMET00589
0.1880.0150.188Uric acid excretion stimulant

0.188 0.015 DBMET00589

0.2050.0330.237Insulin secretagoues

0.237 0.022 DBMET00589

DBMET00589
0.1840.0130.184Sphingosine 1-phosphate receptor 2 antagonist
0.1980.0290.202DNA polymerase I inhibitor

0.202 0.028 DBMET00589

DBMET00589
0.1870.0190.187Sphingosine 1-phosphate receptor 5 antagonist
0.2070.040.207Phospholipase C inhibitor

0.17 0.073 DBMET00589

0.2760.110.28Vasodilator, peripheral

0.28 0.108 DBMET00589

DBMET00589
0.1890.0220.189Interleukin 1b antagonist

0.098 0.083 DBMET00589

0.1870.0270.1875-Lipoxygenase inhibitor
0.1790.0190.179Pregnane X receptor agonist
0.2190.060.219Neurotrophic factor enhancer

0.193 0.084 DBMET00589

0.1880.0290.188Toll-Like receptor 2 antagonist
0.1610.0040.161Aconitate hydratase inhibitor
0.1860.0290.186Adenylate cyclase inhibitor

0.135 0.056 DBMET00589

0.1610.0040.161Liver X receptor beta agonist
0.330.1740.33Ca2+/calmodulin-dependent protein kinase kinase A inhibitor
0.2450.0910.2455 Hydroxytryptamine release stimulant

0.182 0.138 DBMET00589

0.1550.0040.155GABA B receptor agonist
0.1590.0090.159Leukotriene antagonist

0.102 0.021 DBMET00589

0.2560.1060.25612-Lipoxygenase inhibitor
0.1540.0030.154Peroxisome proliferator-activated receptor alpha antagonist
0.160.010.16Aldose reductase inhibitor

0.073 0.026 DBMET00589

0.1570.0090.157Alcohol oxidase inhibitor
0.1670.0210.167TRPA1 agonist
0.170.0230.17Vanilloid 1 agonist

0.153 0.036 DBMET00589

0.1640.0170.164Prolactin inhibitor
0.1640.0190.174Ca2+-transporting ATPase inhibitor

0.174 0.01 DBMET00589

DBMET00589
0.2080.0650.304DNA methyltransferase I inhibitor

0.304 0.025 DBMET00589

DBMET00589
0.1440.0030.144Retinoid X alpha receptor agonist
0.1720.0320.172Cystathionine beta-synthase inhibitor
0.1690.0290.241Microtubule formation inhibitor

0.241 0.011 DBMET00589

DBMET00589
0.1460.0070.1465-Alpha-reductase inhibitor
0.1830.0460.183Neurotensin receptor agonist
0.2080.0740.36DNA methylase inhibitor

0.36 0.015 DBMET00589

DBMET00589
0.1480.0130.148Glutamate decarboxylase inhibitor
0.1370.0050.137Estrogen-related receptor beta agonist
0.1680.0380.168Aldehyde dehydrogenase inhibitor

0.11 0.083 DBMET00589

0.1470.0160.147Glutamate dehydrogenase inhibitor

0.074 0.051 DBMET00589

0.2010.0710.201Glyceraldehyde-3-phosphate dehydrogenase inhibitor

0.154 0.139 DBMET00589

0.1470.0180.147Thioredoxin inhibitor

0.137 0.021 DBMET00589

0.1650.0380.165Cholesterol synthesis inhibitor

0.113 0.071 DBMET00589

0.1580.030.158Nav1.1 sodium channel blocker
0.1680.0410.462Monophenol monooxygenase inhibitor

0.462 0.009 DBMET00589

DBMET00589
0.1650.040.165Protein-tyrosine phosphatase 1B inhibitor

0.155 0.043 DBMET00589

0.180.0560.18Protein-tyrosine phosphatase inhibitor

0.153 0.075 DBMET00589

0.1360.0140.15Glutamate release inhibitor

0.15 0.01 DBMET00589

DBMET00589
0.1410.020.212Phosphofructokinase-1 inhibitor

0.212 0.01 DBMET00589

DBMET00589
0.1560.0350.156Aminopeptidase B inhibitor
0.1240.0040.124DNA helicase inhibitor

0.058 0.03 DBMET00589

0.1830.0630.1833C-like protease (Human coronavirus) inhibitor
0.1220.0040.122Urate transporter 1 inhibitor
0.1710.0550.219Protein kinase stimulant

0.219 0.035 DBMET00589

DBMET00589
0.1320.0160.132CDC25A inhibitor

0.067 0.063 DBMET00589

0.120.0050.12Peroxisome proliferator-activated receptor delta agonist
0.1610.0460.161Adenylate cyclase stimulant
0.1560.0410.156Antibacterial (Helicobacter pylori)

0.145 0.051 DBMET00589

0.160.0450.16MAP kinase kinase 4 inhibitor
0.1180.0040.118Retinoid X receptor agonist
0.1690.060.225Melanin inhibitor

0.225 0.033 DBMET00589

DBMET00589
0.1420.0330.248Mediator release inhibitor

0.248 0.01 DBMET00589

DBMET00589
0.1980.0920.198Nitric-oxide synthase stimulant

0.185 0.117 DBMET00589

0.1830.0770.433Hepatoprotectant

0.433 0.011 DBMET00589

DBMET00589
0.1340.0320.134Creatine kinase inhibitor
0.1060.0040.106Liver X receptor beta antagonist
0.1180.0150.118Argininosuccinate synthase inhibitor
0.1210.0190.121Aminopeptidase I inhibitor
0.120.0190.127ATPase (Vacuolar H+) inhibitor

0.127 0.015 DBMET00589

DBMET00589
0.1120.0150.112Prostaglandin antagonist
0.1110.0160.111Biliverdin reductase inhibitor
0.0960.0020.096Retinoid X beta receptor antagonist
0.1130.0190.113GABA aminotransferase inhibitor

0.107 0.022 DBMET00589

0.10.0060.1Thromboxane synthase inhibitor
0.1290.0380.39UDP-glucose 4-epimerase inhibitor

0.39 0.006 DBMET00589

DBMET00589
0.0930.0020.093Retinoid X receptor antagonist
0.1190.0290.244NADH dehydrogenase inhibitor

0.244 0.008 DBMET00589

DBMET00589
0.0970.0080.097MDM2 inhibitor
0.1140.0260.114Glutathione S-transferase inhibitor
0.2580.170.626Antibacterial

0.626 0.016 DBMET00589

DBMET00589
0.1070.0230.107Phenylalanine 4-hydroxylase inhibitor
0.1490.0660.305Cell wall synthesis inhibitor

0.305 0.01 DBMET00589

DBMET00589
0.130.0470.13Caspase 3 inhibitor
0.0910.0080.091Liver X receptor agonist
0.220.1380.22Thyroid hormone beta antagonist
0.0920.010.092CD45 antagonist
0.0940.0130.094Glutamate (mGluR6) antagonist
0.090.010.09Diacylglycerol O-acyltransferase inhibitor
0.0820.0020.082Retinoid X alpha receptor antagonist
0.0920.0130.106Nitric oxide donor

0.106 0.006 DBMET00589

DBMET00589
0.1040.0250.104Prostaglandin-E synthase inhibitor
0.1090.030.109Cathepsin G inhibitor
0.0920.0140.092Thromboxane antagonist
0.1960.1180.286DNA damaging

0.286 0.063 DBMET00589

DBMET00589
0.0840.0060.084Peroxisome proliferator-activated receptor delta antagonist
0.1740.0970.194Psychostimulant

0.194 0.084 DBMET00589

DBMET00589
0.1770.1010.177Anticonvulsant
0.1240.0480.124Estrogen antagonist
0.1940.1190.194Calpain inhibitor
0.0870.0120.087NMDA receptor subunit 3B antagonist
0.1410.0670.141Bone formation stimulant

0.134 0.073 DBMET00589

0.080.0060.08AMPA 4 receptor antagonist
0.0960.0220.096Elastase 1 inhibitor
0.10.0260.1Leukotriene synthesis inhibitor
0.0890.0160.101Transcription factor AP-1 inhibitor

0.101 0.013 DBMET00589

DBMET00589
0.0940.0220.094Carbamoyl phosphate synthetase inhibitor
0.1150.0440.115Anabolic
0.120.0490.136Acetylcholine release stimulant

0.136 0.027 DBMET00589

DBMET00589
0.0790.0080.079AICAR transformylase inhibitor
0.1360.0660.136NADPH oxidase inhibitor
0.1280.0590.128Sphingosine 1-phosphate receptor 4 antagonist
0.1140.0450.114Folate antagonist
0.0770.0080.077Cholesterol esterase inhibitor

0.045 0.038 DBMET00589

0.1120.0430.112Estrogen receptor beta antagonist
0.0970.0290.097Estrogen receptor alpha antagonist
0.1110.0440.111Electrolyte absorption antagonist
0.0870.020.087Glutamate (mGluR7) antagonist
0.1020.0350.102Inducible nitric-oxide synthase inhibitor
0.0850.0190.085Exportin-1 inhibitor
0.0780.0130.078Leukocyte elastase inhibitor
0.0770.0120.077Dihydroorotate oxidase inhibitor
0.070.0060.075-Alpha-reductase 2 inhibitor
0.0960.0330.096Keratolytic
0.1620.0990.221P-glycoprotein inhibitor

0.221 0.052 DBMET00589

DBMET00589
0.0860.0230.086CDC25B inhibitor

0.061 0.049 DBMET00589

0.0740.0130.074NMDA receptor subunit 3A antagonist
0.0770.0160.077Thromboxane A2 antagonist
0.0640.0040.064Thyroid hormone agonist
0.0710.0120.085Glucose-6-phosphate isomerase inhibitor

0.085 0.007 DBMET00589

DBMET00589
0.0680.0090.068Fumarate hydratase inhibitor
0.0760.0170.076Leukotriene B4 antagonist

0.076 0.017 DBMET00589

0.0670.010.067Glutamate (mGluR group III) antagonist
0.0720.0150.072Oleamide hydrolase inhibitor
0.0840.0270.084NMDA receptor agonist
0.1380.0820.138Heat shock protein 70 antagonist
0.120.0650.12Proteasome inhibitor
0.060.0050.06Free fatty acid receptor 1 antagonist
0.1050.0510.105Interleukin 1 beta converting enzyme inhibitor
0.1840.130.471Immunostimulant

0.471 0.033 DBMET00589

DBMET00589
0.0940.0410.094Vanilloid agonist
0.0770.0230.077Acyl-CoA dehydrogenase inhibitor
0.0910.040.116Na+ K+ transporting ATPase inhibitor

0.116 0.018 DBMET00589

DBMET00589
0.1040.0530.104Glutamate (mGluR7) agonist
0.0940.0440.094Granulocyte macrophage colony stimulating factor agonist
0.0820.0320.082Phospholipase D inhibitor
0.0650.0160.065Macrophage elastase inhibitor
0.0560.0070.0565-Alpha-reductase 1 inhibitor
0.1890.140.299DNA synthesis inhibitor

0.299 0.044 DBMET00589

DBMET00589
0.0620.0130.062Glutamate (mGluR4) antagonist
0.0540.0050.054Cholesterol ester transfer protein antagonist
0.0860.0380.086Histidine decarboxylase inhibitor
0.0570.0090.057Glutamate (mGluR3) antagonist
0.0830.0360.083HIV-1 integrase inhibitor
0.0660.0180.066Leukotriene C antagonist
0.1170.0690.117Anesthetic local
0.0880.0410.101T cell inhibitor

0.101 0.023 DBMET00589

DBMET00589
0.0710.0240.071Acetyl-CoA transferase inhibitor
0.0680.0230.068Elastase inhibitor
0.0540.010.054Kainate receptor agonist
0.0590.0140.059Geranyltranstransferase inhibitor
0.0490.0050.049Elastase 2B inhibitor

0.031 0.02 DBMET00589

0.0490.0050.049Elastase 3B inhibitor

0.031 0.02 DBMET00589

0.0490.0050.049Elastase 3A inhibitor

0.031 0.02 DBMET00589

0.0830.040.083Sphingosine 1-phosphate receptor antagonist
0.0530.010.053Glutamate (mGluR8) agonist
0.1010.0590.101Nitric-oxide synthase inhibitor
0.0720.030.072Purinergic P2X1 antagonist
0.0530.0120.053p53 inhibitor
0.0470.0060.047Liver X receptor alpha antagonist
0.0450.0040.045Retinoid X gamma receptor antagonist

0.027 0.018 DBMET00589

0.0980.0580.098Lanosterol 14 alpha demethylase inhibitor
0.0860.0460.086NAD(P)H dehydrogenase (quinone) inhibitor
0.0490.010.049Liver X receptor antagonist
0.1990.160.199Nootropic
0.0580.020.058Carbonic anhydrase IV inhibitor
0.0970.0580.097Potassium channel (Ca-activated) activator
0.0460.0080.046Lysine carboxypeptidase inhibitor
0.0710.0340.071Aromatase inhibitor
0.0440.0070.044Prostaglandin D2 antagonist
0.0440.0080.044Kynurenine 3 monooxygenase inhibitor
0.0710.0360.071NMDA receptor glycine site agonist
0.0980.0640.098GABA C receptor rho-1 antagonist
0.0590.0250.129Glucose-6-phosphate translocase inhibitor

0.129 0.004 DBMET00589

DBMET00589
0.0410.0090.041Glutamate (mGluR3) agonist
0.1390.1070.139Antipruritic
0.1280.0960.148Diuretic

0.148 0.079 DBMET00589

DBMET00589
0.0440.0130.044AMPA receptor agonist
0.070.040.07Neutrophil collagenase inhibitor
0.0850.0550.085D-Ala-D-Ala ligase inhibitor
0.050.0210.05Guanylate cyclase inhibitor

0.043 0.028 DBMET00589

0.0620.0330.065Mannitol-1-phosphate 5-dehydrogenase inhibitor

0.065 0.03 DBMET00589

DBMET00589
0.0470.0190.0473-Hydroxyanthranilate 3,4-dioxygenase inhibitor
0.0580.0310.058NMDA 2A receptor antagonist
0.1080.080.216Alkylator

0.216 0.022 DBMET00589

DBMET00589
0.0590.0320.059Ornithine carbamoyltransferase inhibitor
0.0410.0130.041Melatonin receptor 1A agonist
0.0440.0170.044Leukotriene C4 antagonist
0.0360.0090.036CXC chemokine 2 receptor antagonist
0.0710.0450.071Purinergic P2X2 antagonist
0.0560.030.114Heparanase inhibitor

0.114 0.003 DBMET00589

DBMET00589
0.0390.0140.039Carboxypeptidase B inhibitor
0.0410.0150.041Glutamate (mGluR8) antagonist
0.0430.0170.043Integrin alpha2 antagonist
0.0340.0090.034Prostaglandin H2 antagonist
0.0280.0030.028Thyroid hormone beta agonist
0.0460.0220.046Acetyl-CoA transferase 1 inhibitor
0.0780.0540.078Metalloproteinase-2 inhibitor
0.0380.0140.038Diacylglycerol O-acyltransferase 1 inhibitor
0.0290.0060.029Free fatty acid receptor 1 agonist
0.0380.0150.038ATP citrate lysase inhibitor
0.1290.1060.129GABA C receptor rho-2 antagonist
0.0390.0160.039HMG CoA reductase inhibitor
0.0990.0770.099Nav1.4 sodium channel blocker
0.0310.010.031Retinoid X gamma receptor agonist
0.0630.0420.063Caspase 9 inhibitor
0.0550.0340.055Sphingosine 1-phosphate receptor 5 agonist
0.1430.1220.143Pyruvate kinase inhibitor
0.0410.020.041Nicotinic acid receptor agonist
0.0240.0030.0244-Hydroxyphenylpyruvate dioxygenase inhibitor
0.0390.0190.039Prostacyclin antagonist
0.0280.0080.028Retinoic acid alpha receptor antagonist
0.0250.0050.025Thyroid hormone alpha antagonist
0.0240.0050.024Thyroid hormone alpha agonist
0.0420.0230.042Membrane dipeptidase inhibitor
0.0230.0040.023Human herpes virus 5 capsid protein P40 inhibitor
0.110.0910.11Tubulin antagonist
0.0590.0410.059Ryanodine receptor antagonist
0.0460.0290.046Integrin antagonist
0.0360.0190.036Estrogen-related receptor alpha antagonist
0.1380.1210.47Platelet adhesion inhibitor

0.47 0.006 DBMET00589

DBMET00589
0.0590.0420.059HIV-1 integrase (Strand Transfer) inhibitor
0.0510.0340.051Lysophosphatidic acid 3 receptor antagonist
0.0540.0390.054Matrix metalloproteinase (membrane-type) inhibitor
0.0490.0340.049Plasminogen activator inhibitor antagonist
0.0260.0120.026Prostaglandin F2 alpha agonist
0.060.0460.06Prostaglandin F2 alpha antagonist
0.0230.0090.023Retinoic acid receptor antagonist
0.0320.0180.032Glucagon receptor antagonist
0.0490.0350.049Bombesin 2 receptor antagonist
0.040.0260.04Retinoic acid alpha receptor agonist
0.0240.0120.024Retinoid X beta receptor agonist
0.0460.0340.046Potassium channel Kv1.3 blocker
0.0520.040.0523(or 17)beta-hydroxysteroid dehydrogenase inhibitor
0.0620.050.062Calcium channel P-type blocker
0.0270.0160.027Integrin alpha2beta1 antagonist
0.0290.0180.029Estrogen-related receptor gamma antagonist
0.0410.0310.041Angiotensin AT1 receptor antagonist
0.020.0090.02CXC chemokine 5 receptor antagonist
0.0530.0420.053Epithelial sodium channel blocker
0.040.030.04Integrin alpha5beta1 antagonist
0.0380.0280.038MAP3K5 inhibitor
0.0550.0450.055Pregnane X receptor antagonist
0.030.0210.03Factor VII inhibitor
0.0740.0650.074Carbonic anhydrase VI inhibitor
0.1120.1030.362Lipid peroxidase inhibitor

0.362 0.012 DBMET00589

DBMET00589
0.0550.0470.055Sphingosine 1-phosphate receptor 3 antagonist
0.0230.0150.023ICAM 1 antagonist
0.0550.0470.055Carbonic anhydrase stimulant
0.0380.0310.038Dopamine D5 agonist
0.0170.0090.017Calcium-sensing receptor antagonist
0.0240.0170.024Glutamate (mGluR1) agonist
0.0930.0860.093GABA receptor agonist
0.0180.0110.018G-protein-coupled receptor 120 agonist
0.0490.0420.049Alpha tubulin antagonist
0.0150.0090.015Integrin beta6 antagonist
0.0170.0110.018Vitamin D receptor agonist

0.018 0.009 DBMET00589

DBMET00589
0.0210.0160.021Integrin alphaVbeta3 antagonist
0.0520.0480.099Adenine nucleotide translocase inhibitor

0.099 0.005 DBMET00589

DBMET00589
0.0220.0170.022Retinoic acid gamma receptor agonist
0.0870.0820.087Urease inhibitor
0.0240.020.033Vanilloid 2 agonist

0.033 0.007 DBMET00589

DBMET00589
0.0360.0330.036GABA uptake inhibitor
0.0240.020.024Lysophosphatidic acid receptor 1 agonist
0.0210.0170.021Glutamate (mGluR1a) agonist
0.0570.0540.057Heme oxygenase stimulant
0.0340.0310.0342,3-Oxidosqualene-lanosterol cyclase inhibitor
0.0110.0080.011Thromboxane agonist
0.0070.0040.007Integrin alpha5beta6 antagonist
0.020.0170.02Neuraminidase (Influenza B) inhibitor
0.0120.0090.012Glutamate (mGluR6) agonist
0.0250.0220.025Nicotinic acid receptor 2 antagonist
0.1520.1490.199Cyclic AMP phosphodiesterase inhibitor

0.199 0.095 DBMET00589

DBMET00589
0.030.0280.03Catechol O-methyltransferase inhibitor
0.0230.0210.023Leukotriene D4 antagonist
0.0310.0290.0311-Alkyl-2-acetylglycerophosphocholine esterase inhibitor
0.0110.010.011Retinoic acid beta receptor antagonist
0.0170.0160.017Estrogen-related receptor gamma agonist
0.0110.010.011Retinoic acid receptor gamma antagonist
0.020.020.024Vitamin D receptor antagonist

0.024 0.012 DBMET00589

DBMET00589
0.0480.0490.078Alpha-mannosidase inhibitor

0.078 0.012 DBMET00589

DBMET00589
0.0150.0170.021Telomerase stimulant

0.021 0.007 DBMET00589

DBMET00589
0.0710.0730.096Glycine receptor antagonist

0.096 0.036 DBMET00589

DBMET00589
0.0820.0870.114Xanthine oxidase inhibitor

0.114 0.051 DBMET00589

DBMET00589
0.0130.0180.022Ileal bile acid transport inhibitor

0.022 0.008 DBMET00589

DBMET00589
0.0160.0240.033Antibiotic Anthracycline-like

0.033 0.003 DBMET00589

DBMET00589
0.1110.1240.214Anticoagulant

0.214 0.048 DBMET00589

DBMET00589
0.0340.050.047Estrogen agonist

0.047 0.037 DBMET00589

DBMET00589
0.0350.0520.072Mannosidase inhibitor

0.072 0.011 DBMET00589

DBMET00589
0.0970.1240.153Interleukin 4 antagonist

0.153 0.047 DBMET00589

DBMET00589
0.0170.0470.079Sodium/glucose cotransporter 2 inhibitor

0.079 0.004 DBMET00589

DBMET00589
0.0180.0520.067Sodium/glucose cotransporter inhibitor

0.067 0.004 DBMET00589

DBMET00589
0.0480.0850.067Lipocortins synthesis agonist

0.067 0.025 DBMET00589

DBMET00589
0.040.080.048Factor III inhibitor

0.048 0.041 DBMET00589

DBMET00589
0.0810.1210.206Beta amyloid protein antagonist

0.206 0.015 DBMET00589

DBMET00589
0.0350.0810.101Factor IXa inhibitor

0.101 0.009 DBMET00589

DBMET00589
0.0290.0760.058Carbonic anhydrase XIV inhibitor

0.058 0.026 DBMET00589

DBMET00589
0.0350.0850.05Protein kinase C eta inhibitor

0.05 0.044 DBMET00589

DBMET00589
0.010.0640.034Squalene synthetase inhibitor

0.034 0.021 DBMET00589

DBMET00589
0.010.0660.021Corticosteroid-like

0.021 0.016 DBMET00589

DBMET00589
0.0280.0860.099Protein 50S ribosomal subunit inhibitor

0.099 0.013 DBMET00589

DBMET00589
0.1030.1610.273Hemostatic

0.273 0.019 DBMET00589

DBMET00589
0.1460.2060.359Peptidyltransferase inhibitor

0.359 0.011 DBMET00589

DBMET00589
0.0240.0870.033Protein kinase C beta I inhibitor

0.033 0.025 DBMET00589

DBMET00589
0.0180.0830.035Toll-Like receptor 4 agonist

0.035 0.007 DBMET00589

DBMET00589
0.0020.0710.013Antibiotic Macrolide-like

0.013 0.011 DBMET00589

DBMET00589
0.0680.1450.177AMP-activated protein kinase stimulant

0.177 0.015 DBMET00589

DBMET00589
0.030.1260.201Antineoplastic antibiotic

0.201 0.021 DBMET00589

DBMET00589
0.0680.1660.096Phosphodiesterase 6D inhibitor

0.096 0.06 DBMET00589

DBMET00589
0.1560.2580.235Caspase 3 stimulant

0.235 0.126 DBMET00589

DBMET00589
0.0870.1910.167DNA repair enzyme inhibitor

0.167 0.019 DBMET00589

DBMET00589
0.0250.1340.353Selectin antagonist

0.353 0.004 DBMET00589

DBMET00589
0.0230.1350.052Microtubule stabilization

0.052 0.026 DBMET00589

DBMET00589
0.0570.1860.191Beta glucuronidase inhibitor

0.191 0.014 DBMET00589

DBMET00589
0.020.1530.05Neuraminidase (Influenza A) inhibitor

0.05 0.024 DBMET00589

DBMET00589
0.060.1950.166Toll-Like receptor 4 antagonist

0.166 0.014 DBMET00589

DBMET00589
0.0720.2730.243NOS3 expression enhancer

0.243 0.028 DBMET00589

DBMET00589
0.110.3140.401Alpha-glucosidase inhibitor

0.401 0.114 DBMET00589

DBMET00589
0.020.2440.072Neuraminidase (influenza) inhibitor

0.072 0.032 DBMET00589

DBMET00589
0.0120.2540.06Neuraminidase inhibitor

0.06 0.044 DBMET00589

DBMET00589
0.0210.2930.081Topoisomerase II alpha inhibitor

0.081 0.053 DBMET00589

DBMET00589
0.0420.330.126Transcription factor NF kappa B stimulant

0.126 0.023 DBMET00589

DBMET00589
0.0430.440.282Vasodilator

0.282 0.055 DBMET00589

DBMET00589
0.0170.4160.226Topoisomerase I inhibitor

0.226 0.021 DBMET00589

DBMET00589
0.0240.4350.13Multidrug resistance-associated protein 1 inhibitor

0.13 0.038 DBMET00589

DBMET00589
0.0160.4660.112Topoisomerase II inhibitor

0.112 0.074 DBMET00589

DBMET00589
0.0120.4780.066Antibiotic Aminoglycoside-like

0.066 0.007 DBMET00589

DBMET00589
0.0360.5040.394Tumour necrosis factor alpha release inhibitor

0.394 0.028 DBMET00589

DBMET00589
0.0450.5150.228Angiogenesis inhibitor

0.228 0.14 DBMET00589

DBMET00589
0.0730.6340.135CC chemokine 6 receptor antagonist

0.135 0.054 DBMET00589

DBMET00589
0.0040.5820.033Protein 30S ribosomal subunit inhibitor

0.033 0.012 DBMET00589

DBMET00589
Ext Pa Pi Pmax Activity Other Results ID Pa_max