Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.7350.0090.735Antiobesity

0.318 0.104 DBMET00909

0.5940.0020.594Mineralocorticoid receptor antagonist
0.6030.0270.603Cyclophilin D inhibitor

0.264 0.197 DBMET00909

0.5570.0020.557CYP2A6 inhibitor

0.183 0.01 DBMET00909

0.5660.0120.566Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.525 0.023 DBMET00909

0.5370.0030.537Gonadotropin-releasing hormone receptor antagonist

0.147 0.005 DBMET00909

0.5010.0040.501Aldehyde dehydrogenase inhibitor

0.15 0.047 DBMET00909

0.4890.0040.489Hedgehog signaling inhibitor

0.21 0.01 DBMET00909

0.4840.030.484GABA C receptor rho-3 antagonist

0.368 0.076 DBMET00909

0.4230.0070.423Protein-tyrosine phosphatase inhibitor
0.4080.0050.408Protein-tyrosine phosphatase 1B inhibitor
0.4210.0230.421Superoxide dismutase inhibitor

0.302 0.05 DBMET00909

0.4370.0570.4625 Hydroxytryptamine release inhibitor

0.462 0.046 DBMET00909

DBMET00909
0.3870.0520.515Cholesterol antagonist

0.515 0.03 DBMET00909

DBMET00909
0.3960.0780.437Histamine release inhibitor

0.437 0.056 DBMET00909

DBMET00909
0.3240.0070.35Nitric-oxide synthase stimulant

0.35 0.005 DBMET00909

DBMET00909
0.3140.0040.31411-Beta-hydroxysteroid dehydrogenase 1 inhibitor
0.3190.0190.319Diuretic
0.3010.0440.3015 Hydroxytryptamine uptake stimulant

0.238 0.094 DBMET00909

0.2870.040.461Peroxidase inhibitor

0.461 0.013 DBMET00909

DBMET00909
0.3710.1290.371Caspase 9 stimulant

0.363 0.136 DBMET00909

0.2310.0090.231Porphobilinogen synthase inhibitor

0.208 0.011 DBMET00909

0.2430.0390.243MAP kinase kinase 3 inhibitor

0.225 0.065 DBMET00909

0.2420.0430.242Neurotrophic factor enhancer

0.235 0.048 DBMET00909

0.1860.0040.186Aldosterone antagonist
0.220.0410.223C-like protease (Human coronavirus) inhibitor
0.280.1070.418Vasodilator, peripheral

0.418 0.05 DBMET00909

DBMET00909
0.1710.0080.171Acetylcholine release stimulant

0.143 0.021 DBMET00909

0.2010.040.201Interferon gamma antagonist

0.178 0.051 DBMET00909

0.1970.0360.197Arachidonic acid antagonist

0.185 0.048 DBMET00909

0.2730.120.317Calcium channel activator

0.317 0.075 DBMET00909

DBMET00909
0.1740.0290.313Ferrochelatase inhibitor

0.313 0.006 DBMET00909

DBMET00909
0.1820.040.182GABA C receptor rho-2 antagonist

0.151 0.073 DBMET00909

0.230.090.274Aldehyde oxidase inhibitor

0.274 0.074 DBMET00909

DBMET00909
0.2430.1110.243Ca(v)3.3 blocker
0.1720.0440.237Alpha-N-acetylglucosaminidase inhibitor

0.237 0.025 DBMET00909

DBMET00909
0.1720.0470.172Cytokine production inhibitor
0.1530.0280.153Protease inhibitor
0.220.1040.22Tyrosine 3 hydroxylase inhibitor

0.18 0.177 DBMET00909

0.1510.0380.151Death-associated protein kinase 1 inhibitor
0.180.0680.18Succinate dehydrogenase inhibitor

0.166 0.086 DBMET00909

0.2190.1070.2195 Hydroxytryptamine release stimulant

0.209 0.114 DBMET00909

0.1880.0810.199Anesthetic general

0.199 0.075 DBMET00909

DBMET00909
0.2020.0960.202RNA-directed DNA polymerase inhibitor

0.2 0.1 DBMET00909

0.1490.0450.155Ca2+-transporting ATPase inhibitor

0.155 0.032 DBMET00909

DBMET00909
0.1460.0430.329Interleukin 1b antagonist

0.329 0.007 DBMET00909

DBMET00909
0.1580.0580.158Mannose-6-phosphate isomerase inhibitor

0.124 0.094 DBMET00909

0.1370.0380.139GABA C receptor antagonist

0.139 0.037 DBMET00909

DBMET00909
0.1210.030.195Lanosterol 14 alpha demethylase inhibitor

0.195 0.005 DBMET00909

DBMET00909
0.1850.0930.1855 Hydroxytryptamine 3E antagonist
0.1110.020.111Epoxide hydrolase inhibitor
0.1060.0170.132Alcohol oxidase inhibitor

0.132 0.012 DBMET00909

DBMET00909
0.1110.0230.111Granulocyte macrophage colony stimulating factor agonist

0.081 0.072 DBMET00909

0.1110.0230.111Nicotinic alpha4beta2 receptor antagonist

0.088 0.042 DBMET00909

0.1260.0390.126UDP-glucose 4-epimerase inhibitor

0.115 0.047 DBMET00909

0.1360.050.136CC chemokine 6 receptor antagonist

0.132 0.063 DBMET00909

0.090.0070.09Glutamate (mGluR4) antagonist
0.1470.0670.179Adenylate cyclase stimulant

0.179 0.027 DBMET00909

DBMET00909
0.0840.0060.084Estradiol 17 beta-dehydrogenase 2 inhibitor
0.1170.040.117UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor

0.102 0.052 DBMET00909

0.1240.0470.125GABA C receptor agonist

0.125 0.046 DBMET00909

DBMET00909
0.0950.0190.095Tyrosine-protein kinase EMT inhibitor
0.130.0560.25Cholesterol synthesis inhibitor

0.25 0.018 DBMET00909

DBMET00909
0.1180.0470.118DOPA decarboxylase inhibitor

0.101 0.074 DBMET00909

0.1020.0320.102p38 MAP kinase inhibitor
0.1230.0550.123TRPA1 agonist
0.0860.0190.086Exportin-1 inhibitor

0.082 0.023 DBMET00909

0.0730.0060.073Potassium channel Kv1.1 blocker
0.140.0740.177Pregnane X receptor agonist

0.177 0.02 DBMET00909

DBMET00909
0.0940.0290.267Vanilloid 1 antagonist

0.267 0.007 DBMET00909

DBMET00909
0.120.0580.12Cystathionine beta-synthase inhibitor

0.101 0.076 DBMET00909

0.1450.0840.145Cyclin-dependent kinase 8 inhibitor
0.0760.0150.087Aconitate hydratase inhibitor

0.087 0.011 DBMET00909

DBMET00909
0.0710.0130.075Pregnane X receptor antagonist

0.075 0.01 DBMET00909

DBMET00909
0.0790.0210.099Mannitol-1-phosphate 5-dehydrogenase inhibitor

0.099 0.014 DBMET00909

DBMET00909
0.0730.0160.073Nicotinic alpha3beta2 receptor antagonist
0.0670.010.067Glutamate (mGluR group III) antagonist
0.1070.0530.107GABA C receptor rho-1 antagonist

0.104 0.056 DBMET00909

0.1230.0710.123Cathepsin H inhibitor
0.1490.1010.149Tumour necrosis factor antagonist
0.1020.0540.102Electrolyte absorption antagonist

0.097 0.062 DBMET00909

0.0890.0420.089Glutamate (mGluR) antagonist
0.0830.0350.083Glycine receptor agonist

0.077 0.042 DBMET00909

0.0780.030.078Glutamate (mGluR7) antagonist

0.071 0.041 DBMET00909

0.1270.080.276Interleukin 1 antagonist

0.276 0.014 DBMET00909

DBMET00909
0.0730.0270.073Cathepsin B inhibitor
0.0790.0370.079Neuronal nicotinic receptor antagonist
0.0840.0430.094Keratolytic

0.094 0.034 DBMET00909

DBMET00909
0.0790.0380.178Phenylalanine 4-hydroxylase inhibitor

0.178 0.009 DBMET00909

DBMET00909
0.0870.0480.087Acetylcholine nicotinic antagonist
0.0870.0480.087Estrogen-related receptor beta agonist

0.083 0.058 DBMET00909

0.0480.010.048Vanilloid 3 antagonist

0.041 0.019 DBMET00909

0.0570.0190.057Dopamine beta hydroxylase inhibitor

0.055 0.022 DBMET00909

0.0910.0540.112Ornithine decarboxylase inhibitor

0.112 0.032 DBMET00909

DBMET00909
0.0820.0450.097Vanilloid antagonist

0.097 0.037 DBMET00909

DBMET00909
0.0540.0190.055Geranyltranstransferase inhibitor

0.055 0.017 DBMET00909

DBMET00909
0.0950.0590.102Toll-Like receptor 3 antagonist

0.102 0.047 DBMET00909

DBMET00909
0.0690.0350.069Aromatase inhibitor

0.069 0.035 DBMET00909

0.060.0250.06Immunoglobulin Fc receptor antagonist

0.054 0.043 DBMET00909

0.0660.0340.066Histone deacetylase SIRT3 inhibitor
0.10.0680.122Adenylate kinase inhibitor

0.122 0.042 DBMET00909

DBMET00909
0.1350.1040.135Heat shock protein 90 alpha antagonist
0.0590.0280.06Thromboxane synthase inhibitor

0.06 0.028 DBMET00909

DBMET00909
0.0970.0670.117Anabolic

0.117 0.043 DBMET00909

DBMET00909
0.1350.1050.153Melanin inhibitor

0.153 0.077 DBMET00909

DBMET00909
0.1240.0960.124Cytidine deaminase inhibitor
0.0480.020.048Nerve growth factor antagonist

0.04 0.035 DBMET00909

0.0580.0310.058Nicotinic receptor alpha7 subunit antagonist
0.0690.0420.069Potassium channel (ATP-sensitive) blocker
0.0750.0490.075Nav1.8 sodium channel blocker
0.090.0650.098HIV-1 integrase (Overall Integration) inhibitor

0.098 0.056 DBMET00909

DBMET00909
0.0330.0080.087Steroid 17-alpha-hydroxylase/17,20 lyase inhibitor

0.087 0.005 DBMET00909

DBMET00909
0.0620.0380.062Potassium channel intermediate-conductance Ca-activated blocker
0.1040.080.116Photosensitizer

0.116 0.063 DBMET00909

DBMET00909
0.0340.0120.034Nicotinic alpha4beta2 receptor agonist
0.0350.0140.035Nicotinic alpha3beta4 receptor agonist
0.0640.0440.064Transcription factor RelA inhibitor
0.0240.0050.024CC chemokine 9 receptor antagonist

0.018 0.011 DBMET00909

0.2330.2140.233MAP kinase kinase 6 inhibitor
0.0710.0520.083Aminopeptidase I inhibitor

0.083 0.04 DBMET00909

DBMET00909
0.0480.0290.048Glutamate (mGluR5) agonist
0.0710.0530.092Glutamate decarboxylase inhibitor

0.092 0.034 DBMET00909

DBMET00909
0.050.0340.05Squalene epoxidase inhibitor
0.0720.0560.072S-adenosyl-L-methionine decarboxylase inhibitor
0.1750.160.1755 Hydroxytryptamine 1E antagonist
0.0530.0390.0533(or 17)beta-hydroxysteroid dehydrogenase inhibitor
0.1050.0920.109Transcription factor STAT6 inhibitor

0.109 0.083 DBMET00909

DBMET00909
0.0570.0440.074Biliverdin reductase inhibitor

0.074 0.029 DBMET00909

DBMET00909
0.080.0670.08Histamine N-methyltransferase inhibitor
0.0470.0340.047Glutamate (mGluR group I) agonist
0.1850.1720.185Gastrin inhibitor
0.1410.1290.141Death-associated protein kinase 2 inhibitor
0.0370.0260.037Factor XIIIa inhibitor
0.0650.0540.065MDM2 inhibitor
0.0390.0270.062Alpha 1d adrenoreceptor agonist

0.062 0.01 DBMET00909

DBMET00909
0.0530.0420.053Bombesin 3 receptor antagonist
0.0530.0430.053Argininosuccinate synthase inhibitor
0.0430.0330.043Histamine H1 receptor agonist
0.0420.0330.044Heme oxygenase inhibitor

0.044 0.025 DBMET00909

DBMET00909
0.0360.0280.036Delayed rectifier potassium channel blocker
0.0810.0730.102Triose-phosphate isomerase inhibitor

0.102 0.045 DBMET00909

DBMET00909
0.0390.0310.039Glutamate (mGluR1a) antagonist
0.1260.1180.126MAP kinase 3 inhibitor
0.0250.0180.031Prostaglandin H2 antagonist

0.031 0.012 DBMET00909

DBMET00909
0.0670.0610.067Phospholipase D inhibitor
0.120.1150.122NOS3 expression enhancer

0.122 0.112 DBMET00909

DBMET00909
0.0270.0220.027Glucosylceramidase stimulant
0.0130.0090.013Cyclin D2 inhibitor
0.0480.0440.058Acyl-CoA dehydrogenase inhibitor

0.058 0.034 DBMET00909

DBMET00909
0.0150.0130.015Nicotinic alpha4 receptor agonist
0.0450.0440.045Nicotinic receptor alpha4 subunit antagonist
0.0060.0050.006CC chemokine 6 receptor agonist
0.0790.0770.092NADH dehydrogenase inhibitor

0.092 0.054 DBMET00909

DBMET00909
0.190.1910.243Vasodilator, coronary

0.243 0.141 DBMET00909

DBMET00909
0.0380.0390.04Kainate receptor agonist

0.04 0.031 DBMET00909

DBMET00909
0.0860.0880.095Phosphodiesterase 6D inhibitor

0.095 0.062 DBMET00909

DBMET00909
0.0160.020.02Alpha 2b adrenoreceptor agonist

0.02 0.01 DBMET00909

DBMET00909
0.1680.1720.21DNA synthesis inhibitor

0.21 0.108 DBMET00909

DBMET00909
0.0630.0680.073Glutamate dehydrogenase inhibitor

0.073 0.053 DBMET00909

DBMET00909
0.1450.1520.152Growth factor agonist

0.152 0.137 DBMET00909

DBMET00909
0.050.0570.056Botulinum neurotoxin type A inhibitor

0.056 0.045 DBMET00909

DBMET00909
0.0540.0630.072Phosphofructokinase-1 inhibitor

0.072 0.046 DBMET00909

DBMET00909
0.0410.0520.054Lysophosphatidic acid 3 receptor antagonist

0.054 0.03 DBMET00909

DBMET00909
0.050.0630.057Purinergic P2X1 antagonist

0.057 0.049 DBMET00909

DBMET00909
0.0780.0910.107Sphingomyelinase inhibitor

0.107 0.052 DBMET00909

DBMET00909
0.0390.0540.045Glucose-6-phosphate isomerase inhibitor

0.045 0.04 DBMET00909

DBMET00909
0.0540.0730.081Catalase inhibitor

0.081 0.047 DBMET00909

DBMET00909
0.0430.0680.055Carbamoyl phosphate synthetase inhibitor

0.055 0.049 DBMET00909

DBMET00909
0.0250.0510.044Diamine oxidase inhibitor

0.044 0.019 DBMET00909

DBMET00909
0.0210.050.029Purinergic P2Y15 antagonist

0.029 0.019 DBMET00909

DBMET00909
0.0250.0560.04Ceramide glucosyltransferase inhibitor

0.04 0.018 DBMET00909

DBMET00909
0.050.0840.079Na+ K+ transporting ATPase inhibitor

0.079 0.052 DBMET00909

DBMET00909
0.0980.1420.141Cell wall synthesis inhibitor

0.141 0.074 DBMET00909

DBMET00909
0.0380.0870.058Carbonic anhydrase stimulant

0.058 0.042 DBMET00909

DBMET00909
0.080.130.103Microtubule formation inhibitor

0.103 0.086 DBMET00909

DBMET00909
0.0960.1490.124Neurotrophic factor

0.124 0.089 DBMET00909

DBMET00909
0.0240.0770.039Membrane dipeptidase inhibitor

0.039 0.029 DBMET00909

DBMET00909
0.0730.1310.098Mucolytic

0.098 0.08 DBMET00909

DBMET00909
0.1670.2250.24Antithrombotic

0.24 0.134 DBMET00909

DBMET00909
0.0290.0980.088Beta 1 adrenoreceptor antagonist

0.088 0.014 DBMET00909

DBMET00909
0.0280.10.051Potassium channel (Inward rectifier) blocker

0.051 0.032 DBMET00909

DBMET00909
0.1120.1870.166Insulin sensitizer

0.166 0.112 DBMET00909

DBMET00909
0.0250.110.075Beta 2 adrenoreceptor antagonist

0.075 0.014 DBMET00909

DBMET00909
0.0270.1270.05Alpha-mannosidase inhibitor

0.05 0.044 DBMET00909

DBMET00909
0.0330.1410.05Glucosylceramidase inhibitor

0.05 0.049 DBMET00909

DBMET00909
0.0320.1560.087Beta adrenoreceptor antagonist

0.087 0.023 DBMET00909

DBMET00909
0.0650.2020.13Electron transport complex I inhibitor

0.13 0.035 DBMET00909

DBMET00909
0.0270.170.049Beta adrenoreceptor agonist

0.049 0.019 DBMET00909

DBMET00909
0.0890.2520.159Spasmolytic

0.159 0.155 DBMET00909

DBMET00909
0.0380.2120.15Protein-tyrosine kinase (PTK, not ETK, WZC) inhibitor

0.15 0.047 DBMET00909

DBMET00909
0.0370.2110.15Abl kinase inhibitor

0.15 0.047 DBMET00909

DBMET00909
0.0340.2080.067Beta 3 adrenoreceptor antagonist

0.067 0.038 DBMET00909

DBMET00909
0.1280.3130.265Sodium/bile acid cotransporter inhibitor

0.265 0.113 DBMET00909

DBMET00909
0.0730.2670.175Interleukin agonist

0.175 0.144 DBMET00909

DBMET00909
0.0590.2530.111Interleukin 4 antagonist

0.111 0.099 DBMET00909

DBMET00909
0.0360.2320.062Beta 2 adrenoreceptor agonist

0.062 0.04 DBMET00909

DBMET00909
0.030.2420.119Adrenaline agonist

0.119 0.026 DBMET00909

DBMET00909
0.0390.4140.31Interleukin antagonist

0.31 0.046 DBMET00909

DBMET00909
0.0210.4370.08Somatostatin 1 agonist

0.08 0.052 DBMET00909

DBMET00909
0.0310.5480.162Tumour necrosis factor alpha release inhibitor

0.162 0.142 DBMET00909

DBMET00909
0.0990.6250.44Calcium channel L-type activator

0.44 0.056 DBMET00909

DBMET00909
0.0770.6310.24Peptidyltransferase inhibitor

0.24 0.058 DBMET00909

DBMET00909
0.0090.630.264Bronchodilator

0.264 0.012 DBMET00909

DBMET00909
0.0280.7780.658Antiinflammatory

0.658 0.039 DBMET00909

DBMET00909
0.0480.8420.206Interleukin 2 agonist

0.206 0.178 DBMET00909

DBMET00909
0.0040.9050.105Adrenaline antagonist

0.105 0.051 DBMET00909

DBMET00909
0.0040.9070.107Antiadrenergic

0.107 0.052 DBMET00909

DBMET00909
0.0050.9370.476Cardiotonic

0.476 0.018 DBMET00909

DBMET00909
Ext Pa Pi Pmax Activity Other Results ID Pa_max