Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.6460.0130.646Aldehyde oxidase inhibitor

0.482 0.035 DBMET00322

0.5960.0040.596Sigma receptor agonist

0.312 0.037 DBMET00322

0.5720.0110.572GABA C receptor rho-3 antagonist
0.550.0090.55Superoxide dismutase inhibitor

0.339 0.039 DBMET00322

0.540.0220.545 Hydroxytryptamine release inhibitor

0.325 0.138 DBMET00322

0.5130.0040.513Tyrosine 3 hydroxylase inhibitor

0.326 0.023 DBMET00322

0.4940.0160.494Cardiotonic

0.256 0.078 DBMET00322

0.460.0050.46Anesthetic local

0.096 0.087 DBMET00322

0.4570.0060.457MAP kinase kinase 2 inhibitor
0.4470.0150.447Peroxidase inhibitor

0.427 0.017 DBMET00322

0.4340.0730.434Ca2+/calmodulin-dependent protein kinase kinase A inhibitor
0.3790.0260.379Psychostimulant
0.3560.0130.356Lipocortins synthesis antagonist

0.19 0.063 DBMET00322

0.350.010.35Nav1.2 sodium channel blocker
0.3360.0120.336Ca2+/calmodulin-dependent kinase II delta inhibitor
0.3180.0090.318Chelator

0.263 0.015 DBMET00322

0.3580.050.358Spasmolytic
0.3140.0110.314DNA intercalator

0.159 0.039 DBMET00322

0.3350.0340.335Interleukin agonist
0.3320.0340.332Ca2+/calmodulin-dependent protein kinase inhibitor
0.3050.0170.305Neuropeptide Y2 antagonist

0.204 0.112 DBMET00322

0.320.0330.32Ca2+/calmodulin-dependent kinase I alpha inhibitor
0.330.0450.33Ca2+/calmodulin-dependent kinase II alpha inhibitor
0.2950.0130.295Nitric-oxide synthase stimulant
0.2960.0260.296Peptidyltransferase inhibitor

0.288 0.029 DBMET00322

0.3180.0480.318Insulysin inhibitor
0.2820.0120.282MAP kinase kinase 3 inhibitor
0.280.0230.28I kappa B kinase epsilon inhibitor
0.3090.0540.309DNA damaging
0.2890.0360.289Anesthetic general

0.187 0.082 DBMET00322

0.350.10.35Histamine release inhibitor

0.224 0.177 DBMET00322

0.2880.0380.2885 Hydroxytryptamine 1E antagonist
0.2690.0280.269Focal adhesion kinase 2 inhibitor
0.2480.0120.248GABA C receptor rho-2 antagonist
0.2470.0140.247Nav1.3 sodium channel blocker
0.2350.0030.235Topoisomerase II beta inhibitor

0.062 0.021 DBMET00322

0.2650.0360.265Glyceraldehyde-3-phosphate dehydrogenase inhibitor

0.166 0.115 DBMET00322

0.2720.0560.272Gastrin inhibitor
0.2330.0210.233Adenylate cyclase inhibitor
0.2970.090.297Vasodilator, coronary
0.2250.020.225Death-associated protein kinase 2 inhibitor

0.164 0.077 DBMET00322

0.2850.0850.285Interleukin 2 agonist
0.250.0520.25ErbB-1 antagonist
0.2650.0670.2655 Hydroxytryptamine uptake stimulant

0.206 0.14 DBMET00322

0.2270.0310.227Phospholipase C inhibitor

0.151 0.105 DBMET00322

0.2380.0440.238LIM domain kinase 1 inhibitor
0.2510.0590.251MAP-kinase-activated kinase 5 inhibitor
0.2050.0130.205Telomerase inhibitor

0.104 0.032 DBMET00322

0.2710.0880.271Immunostimulant
0.1930.0090.193GABA C receptor rho-1 antagonist
0.2070.0240.207Alkylator
0.2250.0530.225Ca2+/calmodulin-dependent kinase II gamma inhibitor
0.2260.0570.226DNA methyltransferase I inhibitor
0.2290.0610.229DNA methylase inhibitor
0.1990.0330.199Catenin beta inhibitor
0.1820.0170.182GABA C receptor antagonist
0.1790.0150.222Porphobilinogen synthase inhibitor

0.222 0.01 DBMET00322

DBMET00322
0.1950.0350.195Acetylcholinesterase inhibitor
0.1740.0160.174Sphingomyelinase inhibitor

0.094 0.067 DBMET00322

0.1720.0140.172NADH dehydrogenase inhibitor

0.144 0.019 DBMET00322

0.1670.0090.167Acetylcholine release stimulant
0.1570.0030.157Epithelial sodium channel blocker
0.170.0160.17Folate antagonist
0.1930.0410.193Heat shock protein 90 antagonist
0.1640.0150.164Electrolyte absorption antagonist
0.2650.1170.265Transcription factor NF kappa B inhibitor
0.1510.0050.151Heat shock protein 90 beta antagonist
0.1940.0490.194Cholinergic
0.1740.0310.174Cyclooxygenase 3 inhibitor
0.1770.0350.177Aldehyde dehydrogenase inhibitor

0.13 0.061 DBMET00322

0.2270.0880.227Calpain inhibitor
0.1720.0330.172Adenylate cyclase stimulant

0.129 0.104 DBMET00322

0.2110.0720.211Amyloid beta aggregation inhibitor

0.205 0.075 DBMET00322

0.1420.0040.142Phospholipase D inhibitor
0.1690.0320.169Alpha 2b adrenoreceptor antagonist
0.1630.0260.163Carbonic anhydrase XV inhibitor
0.2970.160.297Calcium channel L-type activator
0.1810.0450.181Toll-Like receptor 9 antagonist
0.2250.0880.225DNA synthesis inhibitor
0.160.0250.16Potassium channel (Ca-activated) activator
0.1440.0110.144Histamine H2 receptor antagonist
0.2640.1310.264Calcium channel activator
0.1590.0270.159Papain-like protease (SARS coronavirus) inhibitor
0.2680.1370.268Calpain 2 inhibitor
0.2040.0740.204Ca2+/calmodulin-dependent kinase II beta inhibitor
0.1380.0090.138Histone deacetylase inhibitor
0.1710.0420.171Toll-Like receptor antagonist
0.1320.0060.132Estrogen-related receptor beta agonist

0.093 0.035 DBMET00322

0.1560.0320.156Butyrylcholinesterase inhibitor
0.1750.0550.175Acetylcholine M1 receptor antagonist
0.1380.0190.138Toll-Like receptor 3 antagonist
0.1750.0570.175Diuretic
0.1410.030.141Adenylate kinase inhibitor

0.1 0.068 DBMET00322

0.1570.0460.157Nav1.6 sodium channel blocker
0.1530.0440.153Cathepsin H inhibitor
0.30.1940.3Caspase 9 stimulant

0.262 0.239 DBMET00322

0.1610.0560.161Hemostatic
0.160.0550.16Ca2+/calmodulin-dependent protein kinase kinase B inhibitor
0.1230.0190.123Myeloperoxidase inhibitor
0.1080.0040.108Dihydropteroate synthase inhibitor
0.1840.0810.184Growth factor agonist
0.1370.0350.137Platelet activating factor alpha antagonist
0.1290.0270.129MAP kinase kinase 1 inhibitor
0.1050.0040.105Ryanodine receptor antagonist
0.160.060.16CF transmembrane conductance regulator agonist
0.1490.050.149Topoisomerase II inhibitor
0.1520.0540.152Alpha-N-acetylglucosaminidase inhibitor

0.13 0.069 DBMET00322

0.1660.0690.166Interleukin 6 antagonist
0.1390.0420.139Falcipain 3 inhibitor
0.1630.0670.163Cyclin-dependent kinase 8 inhibitor
0.1150.020.165Phenylalanine 4-hydroxylase inhibitor

0.165 0.01 DBMET00322

DBMET00322
0.1230.0280.123Polo-like kinase-1 inhibitor
0.170.0770.17Tumour necrosis factor antagonist
0.1720.080.172MAP kinase kinase 5 inhibitor
0.2650.1720.265MAP kinase kinase 6 inhibitor
0.1270.0360.127Interleukin 2 antagonist
0.1850.0930.1855 Hydroxytryptamine 3E antagonist
0.1250.0350.125Nitric-oxide synthase inhibitor
0.0940.0060.094Sodium/calcium exchanger inhibitor
0.1510.0640.151Ribosomal protein S6 kinase inhibitor
0.1180.0310.118Histamine N-methyltransferase inhibitor
0.1610.0760.161Heat shock protein 90 alpha antagonist
0.1370.0530.137Acetylcholine muscarinic antagonist
0.0880.0040.088Delayed rectifier potassium channel blocker
0.190.1060.19Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase inhibitor
0.0910.0090.091Histone deacetylase class I inhibitor
0.1890.1070.189Antiamyloidogenic
0.1110.0310.111I kappa B kinase inhibitor
0.0870.0090.087Carbonic anhydrase IV inhibitor
0.0920.0150.092CC chemokine 2 receptor antagonist
0.0820.0070.082Adenylate cyclase 1 inhibitor
0.1230.0480.123GABA C receptor agonist
0.0930.0190.093S-adenosyl-L-methionine decarboxylase inhibitor
0.080.0080.08Thymidylate synthase inhibitor
0.1630.0910.163TRKC antagonist
0.1450.0730.145Neuropeptide Y1 antagonist
0.0990.030.099Interferon agonist
0.0980.0290.098Aminopeptidase I inhibitor
0.1280.0590.128Proteasome inhibitor
0.0810.0130.0815 Hydroxytryptamine 4 antagonist
0.1210.0530.121Ferrochelatase inhibitor
0.0830.020.083I kappa B kinase 2 inhibitor
0.080.0180.08Gonadotropin-releasing hormone receptor agonist
0.1070.0450.107Lanosterol 14 alpha demethylase inhibitor
0.080.0180.08Histone deacetylase SIRT3 inhibitor
0.0660.0050.066Dopamine autoreceptor agonist
0.1170.0570.117Mucolytic
0.0690.0080.069Plasmepsin II inhibitor
0.190.130.195 Hydroxytryptamine release stimulant
0.1150.0550.115Aminopeptidase B inhibitor
0.10.0410.1Bcr-Abl kinase inhibitor
0.0970.0390.097Granulocyte macrophage colony stimulating factor agonist
0.0830.0270.083Potassium channel (Tandem pore domain) blocker
0.1040.0480.104Potassium channel (Voltage-sensitive) activator
0.0930.0380.093D-Ala-D-Ala ligase inhibitor
0.0740.0190.074Glycine transporter 2 inhibitor
0.1260.0710.126Toll-Like receptor 2 antagonist
0.0860.0320.086MAP kinase kinase 7 inhibitor
0.1320.0780.132Histone deacetylase SIRT1 inhibitor
0.0810.0280.081Adenosine A1 receptor antagonist
0.0710.0180.071Beta 2 adrenoreceptor agonist
0.0890.0370.089Glutamate dehydrogenase inhibitor

0.069 0.058 DBMET00322

0.1040.0530.104Glutamate (mGluR7) agonist
0.0530.0020.053Estrogen-related receptor gamma agonist

0.021 0.01 DBMET00322

0.1080.0580.108Urease inhibitor
0.0760.0270.076Carbonic anhydrase I inhibitor
0.1080.0590.108Alpha 2c adrenoreceptor antagonist
0.1350.0870.135Cytidine deaminase inhibitor
0.1580.110.158Death-associated protein kinase 3 inhibitor
0.0730.0250.073Acyl-CoA dehydrogenase inhibitor
0.0680.0210.068Phosphorylase inhibitor
0.1650.1190.165Histone acetyltransferase inhibitor
0.060.0140.06Growth hormone secretagogue receptor antagonist
0.060.0140.06AICAR transformylase inhibitor
0.0950.050.095Glutamate release inhibitor
0.0790.0360.079Carbonic anhydrase inhibitor
0.1180.0750.118Cholinergic antagonist
0.0890.0470.089Topoisomerase II alpha inhibitor
0.0490.0080.049Lysine carboxypeptidase inhibitor
0.0480.0070.048Methionyl aminopeptidase 2 inhibitor
0.0750.0340.075Potassium channel (ATP-sensitive) blocker
0.0590.0190.059Factor III inhibitor
0.0530.0140.053Histone deacetylase 9 inhibitor
0.0960.0570.096Alcohol dehydrogenase inhibitor

0.095 0.058 DBMET00322

0.1140.0760.114Acetylcholine antagonist
0.0820.0440.082GABA aminotransferase inhibitor
0.0670.0290.067Acetylcholine muscarinic agonist
0.070.0310.075 Hydroxytryptamine 5A antagonist
0.0620.0240.062Alpha-mannosidase inhibitor
0.0920.0550.092Pim-3 kinase inhibitor
0.0670.0310.067Carbonic anhydrase II inhibitor
0.1030.0670.103Topoisomerase I inhibitor
0.130.0950.13Thiol protease inhibitor
0.0820.0480.082Fibroblast growth factor 3 antagonist
0.0850.050.085CC chemokine 5 receptor agonist
0.0660.0310.066Prolactin release inhibitor
0.0540.0190.054Geranyltranstransferase inhibitor
0.070.0350.07Interferon inducer
0.1260.0920.126Aurora-C kinase inhibitor
0.0850.0520.085Platelet growth factor antagonist
0.0840.0520.084Adrenaline agonist
0.0660.0340.066Carbonic anhydrase stimulant
0.0390.0070.039Purinergic P2Y15 antagonist
0.0690.0370.069NMDA receptor agonist
0.1150.0840.115DNA repair enzyme inhibitor
0.0460.0150.046Opioid delta receptor agonist
0.0880.0570.088Acetylcholine agonist
0.0680.0380.068Adenosine A2a receptor antagonist
0.0980.0680.098Nav1.1 sodium channel blocker
0.1120.0820.112MAP kinase kinase inhibitor
0.0450.0150.045Glucose-6-phosphate dehydrogenase inhibitor
0.070.040.07Adenosine A2 receptor antagonist
0.1190.0890.119Calcium channel blocker
0.0970.0680.097Check point kinase 2 inhibitor
0.1220.0940.122Activin receptor-like kinase 2 inhibitor
0.0460.0180.046Factor XIIIa inhibitor
0.0670.0390.067Beta 3 adrenoreceptor antagonist
0.0920.0650.092Prolactin inhibitor
0.1420.1160.142ATPase inhibitor
0.1220.0960.122Protein kinase (CK1) gamma 1 inhibitor
0.1550.130.155Neurotrophic factor enhancer
0.0610.0360.0615 Hydroxytryptamine 5 antagonist
0.1070.0820.107Calcium channel N-type blocker
0.0450.0210.045Membrane dipeptidase inhibitor
0.1130.090.113Cyclin-dependent kinase 7 inhibitor
0.0740.0520.074Rho-associated kinase I inhibitor
0.0370.0150.037GHS receptor antagonist
0.0410.0190.041Integrin alpha2 antagonist
0.0460.0250.046Histamine H1 receptor agonist
0.0460.0260.046Histamine H2 receptor agonist
0.0570.0370.057Mannitol-1-phosphate 5-dehydrogenase inhibitor
0.0230.0040.023CDK2/cyclin A3 inhibitor
0.0620.0420.062Corticotropin releasing factor 2 receptor antagonist
0.1580.1390.158Cyclic AMP phosphodiesterase inhibitor
0.0320.0130.032Estrogen-related receptor gamma antagonist

0.032 0.012 DBMET00322

0.1490.130.149Anticonvulsant
0.0470.0290.047Mannosidase inhibitor
0.0440.0260.044Glutamate (mGluR1a) antagonist
0.1140.0960.114Cytokine production inhibitor
0.0450.0280.045Dihydrofolate reductase inhibitor
0.0610.0440.061Acetylcholine M2 receptor antagonist
0.1120.0950.112Antibacterial (Helicobacter pylori)
0.130.1130.13Protein kinase (CK1) gamma 3 inhibitor
0.0320.0160.032CDK4/cyclin D3 inhibitor
0.1430.1270.143Succinate dehydrogenase inhibitor
0.0270.0110.0275 Hydroxytryptamine 4 agonist
0.030.0150.03Histone deacetylase 1 inhibitor
0.0770.0620.077Carbonic anhydrase VI inhibitor
0.0390.0240.039Diamine oxidase inhibitor
0.0710.0560.071Adenosine A3 receptor antagonist
0.0870.0730.087Platelet activating factor beta antagonist
0.0410.0280.041Thymidine kinase inhibitor
0.0650.0510.065Potassium channel large-conductance Ca-activated activator
0.0210.0080.021Adenosine A2a receptor agonist
0.0570.0440.057Biliverdin reductase inhibitor
0.0380.0250.038Histone deacetylase 7 inhibitor
0.0320.0190.032AMPA 3 receptor antagonist
0.0990.0860.099Calcium channel (voltage-sensitive) blocker
0.0350.0230.035Adenosine uptake inhibitor
0.1270.1140.127Polo-like kinase-3 inhibitor
0.0590.0470.059NMDA 2C receptor antagonist
0.0880.0760.088Interleukin 1 beta converting enzyme inhibitor
0.0240.0130.024ICAM 1 antagonist
0.10.0890.1CDK3/cyclin E inhibitor
0.0490.0390.049NMDA 2A receptor antagonist
0.0190.0090.019Adenosine A2 receptor agonist
0.0820.0720.082Fibroblast growth factor 1 antagonist
0.0550.0460.055Botulinum neurotoxin type A inhibitor
0.0280.0190.028Hypoxanthine phosphoribosyltransferase inhibitor
0.20.1920.2Ca(v)3.3 blocker
0.0570.0490.057NMDA receptor glycine site agonist
0.0210.0130.021Factor XIII inhibitor
0.1380.130.138Cyclin-dependent kinase 3 inhibitor
0.1050.0980.105Lck kinase inhibitor
0.0450.0390.045Benzodiazepine antagonist
0.0440.0380.044Beta adrenoreceptor agonist
0.0750.070.075Glutathione S-transferase inhibitor
0.0530.0470.053Immunoglobulin Fc receptor antagonist
0.0920.0860.092Platelet activating factor antagonist
0.0550.0510.055Purinergic P2X1 antagonist
0.020.0160.02Neuraminidase (Influenza B) inhibitor
0.0060.0020.006Reverse transcriptase (HBV) inhibitor
0.080.0760.08Potassium channel activator
0.0440.0410.044Transforming growth factor beta 1 antagonist
0.1420.1390.142Platelet aggregation inhibitor
0.0710.0670.071Acetylcholine nicotinic antagonist
0.0780.0750.078Proto-oncogene tyrosine-protein kinase Kit inhibitor
0.0360.0340.036AMPA 4 receptor antagonist
0.0370.0360.037Acetylcholine M1 receptor agonist
0.0960.0950.096MAO inhibitor
0.0470.0460.047Toll-Like receptor 8 antagonist
0.0340.0330.034ATM kinase inhibitor
0.0960.0950.096TRKA antagonist
0.180.2550.269Antibacterial

0.269 0.16 DBMET00322

DBMET00322
0.0340.20.076Epidermal growth factor antagonist

0.076 0.071 DBMET00322

DBMET00322
0.0670.2680.127Dual specificity phosphatase inhibitor

0.127 0.125 DBMET00322

DBMET00322
0.070.3060.163Free radical scavenger

0.163 0.131 DBMET00322

DBMET00322
0.0740.3250.184Antioxidant

0.184 0.128 DBMET00322

DBMET00322
0.0230.30.146M18 aspartyl aminopeptidase inhibitor

0.146 0.054 DBMET00322

DBMET00322
0.0150.5140.11Cyclooxygenase 1 inhibitor

0.11 0.09 DBMET00322

DBMET00322
Ext Pa Pi Pmax Activity Other Results ID Pa_max