Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.5730.010.601Hypoglycemic

0.601 0.008 DBMET00289

DBMET00289
0.4840.0020.484Carbonic anhydrase stimulant

0.356 0.003 DBMET00289

0.4790.0090.479Diuretic

0.366 0.015 DBMET00289

0.4530.020.453Cardiotonic

0.416 0.026 DBMET00289

0.4390.0210.466Platelet antagonist

0.466 0.017 DBMET00289

DBMET00289
0.3630.0040.363Carbonic anhydrase XII inhibitor

0.332 0.004 DBMET00289

0.4040.0480.537Antithrombotic

0.537 0.024 DBMET00289

DBMET00289
0.4110.0560.411Calpain 2 inhibitor

0.344 0.09 DBMET00289

0.3560.0080.356Insulin secretagoues

0.346 0.009 DBMET00289

0.3660.0290.366Insulysin inhibitor

0.318 0.048 DBMET00289

0.3540.0230.354Anesthetic general

0.343 0.025 DBMET00289

0.3430.0210.343Platelet adhesion inhibitor

0.342 0.022 DBMET00289

0.3210.0040.321Carbonic anhydrase inhibitor

0.315 0.004 DBMET00289

0.3130.0040.313Carbonic anhydrase IX inhibitor

0.293 0.005 DBMET00289

0.3080.0110.396Aldehyde dehydrogenase inhibitor

0.396 0.005 DBMET00289

DBMET00289
0.2910.0040.291Carbonic anhydrase I inhibitor

0.268 0.004 DBMET00289

0.2660.0040.266Carbonic anhydrase II inhibitor

0.251 0.005 DBMET00289

0.2660.0040.266Electrolyte absorption antagonist

0.209 0.007 DBMET00289

0.2660.0110.378Carbonic anhydrase XV inhibitor

0.378 0.004 DBMET00289

DBMET00289
0.2530.0040.323Carbonic anhydrase V inhibitor

0.323 0.003 DBMET00289

DBMET00289
0.250.0030.354Thromboxane antagonist

0.354 0.002 DBMET00289

DBMET00289
0.3140.0670.321Sodium/bile acid cotransporter inhibitor

0.321 0.061 DBMET00289

DBMET00289
0.2870.0430.287Gastrin inhibitor

0.246 0.084 DBMET00289

0.2440.0020.244Carbonic anhydrase II stimulant

0.196 0.002 DBMET00289

0.2420.0010.242Carbonic anhydrase I stimulant

0.206 0.002 DBMET00289

0.2380.0030.35Thromboxane A2 antagonist

0.35 0.002 DBMET00289

DBMET00289
0.2760.0420.276Platelet aggregation inhibitor

0.238 0.057 DBMET00289

0.2360.0030.236Potassium channel (ATP-sensitive) blocker

0.184 0.004 DBMET00289

0.2760.0440.276Calpain inhibitor

0.258 0.057 DBMET00289

0.2350.0070.235Metalloproteinase-2 inhibitor

0.234 0.007 DBMET00289

0.2260.0040.268Carbonic anhydrase VA inhibitor

0.268 0.003 DBMET00289

DBMET00289
0.2720.0520.2725 Hydroxytryptamine 1E antagonist
0.2270.010.359Carbonic anhydrase VI inhibitor

0.359 0.005 DBMET00289

DBMET00289
0.2750.060.2755 Hydroxytryptamine uptake stimulant

0.265 0.068 DBMET00289

0.2030.0020.203Bombesin 3 receptor antagonist

0.191 0.002 DBMET00289

0.2040.0050.204Carbonic anhydrase VII inhibitor

0.188 0.005 DBMET00289

0.2070.0080.212Metalloproteinase-9 inhibitor

0.212 0.007 DBMET00289

DBMET00289
0.2510.0550.251Neuropeptide Y2 antagonist

0.214 0.097 DBMET00289

0.2070.0140.207Neuropeptide Y antagonist

0.078 0.062 DBMET00289

0.2120.0210.212Nav1.3 sodium channel blocker

0.19 0.028 DBMET00289

0.2420.0570.247Peptidyltransferase inhibitor

0.247 0.053 DBMET00289

DBMET00289
0.2020.0220.202Cathepsin H inhibitor

0.17 0.034 DBMET00289

0.2010.0210.201Aminopeptidase B inhibitor

0.199 0.021 DBMET00289

0.1830.0060.237Prostaglandin E2 antagonist

0.237 0.005 DBMET00289

DBMET00289
0.1780.0040.331Carbonic anhydrase XIV inhibitor

0.331 0.003 DBMET00289

DBMET00289
0.2730.1030.273Thyroid hormone beta antagonist
0.2690.1120.269Thyroid hormone antagonist
0.290.1380.29Beta lactamase inhibitor
0.1620.0110.195Neutrophil collagenase inhibitor

0.195 0.008 DBMET00289

DBMET00289
0.1960.0460.301Phospholipase C inhibitor

0.301 0.018 DBMET00289

DBMET00289
0.140.0030.14Potassium channel Kv1.1 blocker

0.055 0.011 DBMET00289

0.1410.0050.174Beta 1 adrenoreceptor antagonist

0.174 0.004 DBMET00289

DBMET00289
0.1790.0430.179Alkaline phosphatase inhibitor

0.126 0.079 DBMET00289

0.1410.0060.141Bcl2 antagonist

0.13 0.008 DBMET00289

0.1380.0040.141Vanilloid 4 agonist

0.141 0.004 DBMET00289

DBMET00289
0.1540.0210.257Carbonic anhydrase XIII inhibitor

0.257 0.008 DBMET00289

DBMET00289
0.1690.0360.182Adenylate cyclase stimulant

0.182 0.024 DBMET00289

DBMET00289
0.1350.0030.135Fructose-1,6-bisphosphatase inhibitor

0.097 0.004 DBMET00289

0.1310.0010.131Carbonic anhydrase IV stimulant

0.104 0.001 DBMET00289

0.1990.0720.214Non-steroidal antiinflammatory agent

0.214 0.061 DBMET00289

DBMET00289
0.1420.0150.152Matrix metalloproteinase inhibitor

0.152 0.013 DBMET00289

DBMET00289
0.1310.0040.16Thromboxane synthase inhibitor

0.16 0.004 DBMET00289

DBMET00289
0.1510.0280.23Carbonic anhydrase III inhibitor

0.23 0.012 DBMET00289

DBMET00289
0.1560.0340.156Sphingosine 1-phosphate receptor 2 antagonist

0.151 0.039 DBMET00289

0.1320.0110.189Carbonic anhydrase VB inhibitor

0.189 0.005 DBMET00289

DBMET00289
0.1260.0060.159Beta 2 adrenoreceptor antagonist

0.159 0.004 DBMET00289

DBMET00289
0.1670.0480.167Nav1.2 sodium channel blocker

0.108 0.099 DBMET00289

0.130.0150.13Epoxide hydrolase inhibitor

0.097 0.027 DBMET00289

0.2660.1530.26615-Lipoxygenase inhibitor
0.1460.0340.146Chemokine receptor antagonist

0.102 0.061 DBMET00289

0.1270.0160.127Thrombin inhibitor

0.108 0.022 DBMET00289

0.1140.0060.18Glucosylceramidase inhibitor

0.18 0.003 DBMET00289

DBMET00289
0.1130.0040.211Prostaglandin EP4 antagonist

0.211 0.003 DBMET00289

DBMET00289
0.1080.0020.108Fructose-1,6-bisphosphatase 1 inhibitor

0.06 0.003 DBMET00289

0.1270.0230.228Adrenaline agonist

0.228 0.005 DBMET00289

DBMET00289
0.1490.0470.149Proteasome inhibitor

0.146 0.049 DBMET00289

0.1120.010.112Matrix metalloproteinase 1 inhibitor

0.109 0.011 DBMET00289

0.1110.0130.143Beta adrenoreceptor antagonist

0.143 0.006 DBMET00289

DBMET00289
0.1550.0570.155Neuropeptide Y1 antagonist

0.123 0.117 DBMET00289

0.120.0230.12Glutathione S-transferase inhibitor

0.116 0.025 DBMET00289

0.1030.0060.103Carbonic anhydrase IV inhibitor

0.103 0.007 DBMET00289

0.1060.0120.106Acetyl-CoA transferase inhibitor

0.071 0.024 DBMET00289

0.1170.0230.117Cannabinoid receptor antagonist

0.062 0.06 DBMET00289

0.1990.1050.199Aldehyde oxidase inhibitor

0.177 0.118 DBMET00289

0.10.0060.1Bcl-xL inhibitor

0.092 0.008 DBMET00289

0.1070.0140.107Cannabinoid CB1 receptor antagonist

0.068 0.037 DBMET00289

0.0980.0060.098Collagenase inhibitor

0.076 0.008 DBMET00289

0.1050.0130.126Beta 3 adrenoreceptor antagonist

0.126 0.009 DBMET00289

DBMET00289
0.0960.0080.096Potassium channel (Inward rectifier) blocker

0.08 0.013 DBMET00289

0.1340.0460.134Interleukin 8 antagonist

0.1 0.096 DBMET00289

0.0920.0040.092Angiotensin AT2 receptor antagonist

0.087 0.004 DBMET00289

0.0920.0060.096Prostaglandin EP3 antagonist

0.096 0.006 DBMET00289

DBMET00289
0.1020.0160.102Trypsin inhibitor

0.093 0.02 DBMET00289

0.1440.0610.144Nav1.6 sodium channel blocker

0.115 0.104 DBMET00289

0.1010.020.113Sphingosine 1-phosphate receptor antagonist

0.113 0.015 DBMET00289

DBMET00289
0.0910.010.091Purinergic P2Y antagonist

0.085 0.011 DBMET00289

0.0830.0040.102Angiotensin II receptor antagonist

0.102 0.003 DBMET00289

DBMET00289
0.20.1210.2MAP kinase kinase 3 inhibitor
0.0850.0060.085Potassium channel (Inward rectifier) activator

0.057 0.024 DBMET00289

0.2080.1320.249Lipoxygenase inhibitor

0.249 0.101 DBMET00289

DBMET00289
0.0860.0120.113Sphingosine 1-phosphate receptor 1 antagonist

0.113 0.007 DBMET00289

DBMET00289
0.080.0070.08Potassium channel (ATP-sensitive) activator

0.053 0.024 DBMET00289

0.0730.0040.082Angiotensin AT1 receptor antagonist

0.082 0.003 DBMET00289

DBMET00289
0.1690.1010.169Focal adhesion kinase 2 inhibitor
0.0970.030.097Aminopeptidase I inhibitor

0.089 0.035 DBMET00289

0.10.0340.1Histamine H2 receptor antagonist
0.0840.020.084Prostaglandin F2 alpha antagonist

0.078 0.024 DBMET00289

0.0840.0210.131Prostaglandin antagonist

0.131 0.012 DBMET00289

DBMET00289
0.1110.0490.111Factor V inhibitor

0.109 0.052 DBMET00289

0.0930.0320.093GABA aminotransferase inhibitor

0.081 0.046 DBMET00289

0.1120.0510.138Adenylate kinase inhibitor

0.138 0.032 DBMET00289

DBMET00289
0.0650.0050.065Bombesin agonist

0.036 0.006 DBMET00289

0.0730.0150.111Beta 2 adrenoreceptor agonist

0.111 0.004 DBMET00289

DBMET00289
0.1730.1150.173Ca2+/calmodulin-dependent kinase I alpha inhibitor
0.0960.0370.096CC chemokine receptor antagonist

0.07 0.064 DBMET00289

0.0920.0330.092Ca(v)3.1 blocker
0.1380.080.138Pregnane X receptor agonist
0.1440.0860.169Hexokinase inhibitor

0.169 0.058 DBMET00289

DBMET00289
0.1960.1390.196Transcription factor STAT3 inhibitor

0.179 0.166 DBMET00289

0.080.0240.085Collagenase 3 inhibitor

0.085 0.022 DBMET00289

DBMET00289
0.1170.0650.128Caspase 3 inhibitor

0.128 0.049 DBMET00289

DBMET00289
0.0560.0050.056Bombesin 3 receptor agonist

0.033 0.005 DBMET00289

0.0690.0190.069Metalloproteinase-3 inhibitor

0.064 0.022 DBMET00289

0.0620.0120.088Cytokine production stimulant

0.088 0.005 DBMET00289

DBMET00289
0.0580.0090.063Aggrecanase 1 inhibitor

0.063 0.008 DBMET00289

DBMET00289
0.1280.0790.128CC chemokine 6 receptor antagonist

0.122 0.108 DBMET00289

0.0570.0080.061Integrin alpha2 antagonist

0.061 0.007 DBMET00289

DBMET00289
0.0580.010.058Acetyl-CoA transferase 1 inhibitor

0.047 0.02 DBMET00289

0.0470.0020.047Angiotensin AT2 receptor agonist

0.029 0.002 DBMET00289

0.0560.0130.056Dihydropteroate synthase inhibitor

0.047 0.019 DBMET00289

0.1330.0910.134Thiol protease inhibitor

0.134 0.089 DBMET00289

DBMET00289
0.0830.0420.111Cathepsin G inhibitor

0.111 0.029 DBMET00289

DBMET00289
0.0530.0130.096Beta adrenoreceptor agonist

0.096 0.004 DBMET00289

DBMET00289
0.0440.0040.044Angiotensin AT1A receptor antagonist

0.039 0.004 DBMET00289

0.0660.0270.076Matrix metalloproteinase (membrane-type) inhibitor

0.076 0.022 DBMET00289

DBMET00289
0.1960.1560.19612-Lipoxygenase inhibitor
0.0690.030.069Potassium channel Kv1.5 blocker
0.0660.0270.066Neuropeptide Y5 antagonist
0.0810.0430.091Glutamate dehydrogenase inhibitor

0.091 0.036 DBMET00289

DBMET00289
0.0570.0210.057Bombesin antagonist

0.053 0.026 DBMET00289

0.0430.0060.043Calcium-sensing receptor agonist

0.04 0.007 DBMET00289

0.0380.0030.042Angiotensin AT1B receptor antagonist

0.042 0.003 DBMET00289

DBMET00289
0.120.0870.127Vanilloid 1 agonist

0.127 0.072 DBMET00289

DBMET00289
0.0810.0470.081Viral attachment inhibitor

0.076 0.058 DBMET00289

0.0370.0050.098Beta 1 adrenoreceptor agonist

0.098 0.003 DBMET00289

DBMET00289
0.0520.0220.052Leukocyte elastase inhibitor

0.047 0.026 DBMET00289

0.170.1390.292Immunostimulant

0.292 0.081 DBMET00289

DBMET00289
0.0540.0250.054Potassium channel Kv1.3 blocker

0.043 0.038 DBMET00289

0.1580.1290.158Histone acetyltransferase inhibitor
0.0340.0060.034Protease (Human cytomegalovirus) inhibitor

0.021 0.017 DBMET00289

0.1280.1020.137Anticoagulant

0.137 0.092 DBMET00289

DBMET00289
0.2740.2490.274Ca2+/calmodulin-dependent protein kinase kinase A inhibitor
0.0320.0080.032Vanilloid 2 agonist

0.029 0.011 DBMET00289

0.0840.060.088Vanilloid agonist

0.088 0.05 DBMET00289

DBMET00289
0.1140.0920.114Sodium channel blocker
0.0330.0110.033CXC chemokine 2 receptor antagonist

0.028 0.016 DBMET00289

0.0330.0120.033Epoxide hydrolase 2 inhibitor
0.1060.0850.106Sphingosine 1-phosphate receptor 2 agonist
0.0650.0440.097Interferon inducer

0.097 0.014 DBMET00289

DBMET00289
0.0470.0270.051Macrophage elastase inhibitor

0.051 0.024 DBMET00289

DBMET00289
0.0860.0660.107Aminoacyl-tRNA synthetase inhibitor

0.107 0.039 DBMET00289

DBMET00289
0.0310.0110.035Integrin alpha2beta1 antagonist

0.035 0.008 DBMET00289

DBMET00289
0.0690.050.069CXC chemokine receptor antagonist
0.0410.0220.053Farnesoid X receptor agonist

0.053 0.013 DBMET00289

DBMET00289
0.0230.0040.023CC chemokine 10 receptor antagonist

0.019 0.005 DBMET00289

0.0450.0260.045Histamine H2 receptor agonist
0.0420.0240.042Phenylethanolamine N methyltransferase inhibitor

0.042 0.025 DBMET00289

0.1390.1220.139ATPase inhibitor
0.0290.0140.029Prostaglandin H2 antagonist

0.029 0.014 DBMET00289

0.0620.0470.062Transcription factor RelA inhibitor
0.0750.060.114Interferon agonist

0.114 0.02 DBMET00289

DBMET00289
0.1690.1540.1765 Hydroxytryptamine release stimulant

0.176 0.146 DBMET00289

DBMET00289
0.2390.2250.402Cyclophilin D inhibitor

0.402 0.09 DBMET00289

DBMET00289
0.0320.0180.032Trypsin II inhibitor

0.027 0.025 DBMET00289

0.0520.0380.071Ornithine carbamoyltransferase inhibitor

0.071 0.025 DBMET00289

DBMET00289
0.1750.1610.234DNA synthesis inhibitor

0.234 0.079 DBMET00289

DBMET00289
0.0990.0860.099Nav1.5 sodium channel blocker
0.0790.0660.079CC chemokine 5 receptor agonist
0.0230.010.023Factor XIII inhibitor

0.019 0.018 DBMET00289

0.090.0780.09Urease inhibitor
0.1480.1360.187Insulin sensitizer

0.187 0.087 DBMET00289

DBMET00289
0.1650.1540.1655 Hydroxytryptamine 3E antagonist
0.2080.1970.208GABA C receptor rho-3 antagonist
0.0560.0450.084Prostaglandin EP2 antagonist

0.084 0.025 DBMET00289

DBMET00289
0.20.190.331Interleukin 2 agonist

0.331 0.055 DBMET00289

DBMET00289
0.0450.0350.045Glycine transporter inhibitor
0.1060.0970.106Cyclooxygenase 2 inhibitor
0.0520.0430.054Epithelial sodium channel blocker

0.054 0.039 DBMET00289

DBMET00289
0.0830.0750.091Thioredoxin inhibitor

0.091 0.061 DBMET00289

DBMET00289
0.0270.0190.027Myristoyl transferase inhibitor
0.050.0420.05Neuropeptide agonist
0.0250.0180.025Complement factor 1s inhibitor
0.0390.0330.039Oxytocin agonist
0.0130.0070.055Beta 3 adrenoreceptor agonist

0.055 0.004 DBMET00289

DBMET00289
0.0460.0410.046HCV NS3/NS4A protease inhibitor
0.1390.1340.147Succinate dehydrogenase inhibitor

0.147 0.117 DBMET00289

DBMET00289
0.0160.0120.016Carbonic anhydrase VIII inhibitor
0.0160.0120.016Carbonic anhydrase X inhibitor
0.0210.0180.021Purinergic P2Y12 antagonist
0.0070.0040.007Bone morphogenic protein 1 inhibitor

0.007 0.003 DBMET00289

0.0480.0450.048Elastase inhibitor
0.0280.0260.028Epoxide hydrolase 1 inhibitor
0.1360.1340.163Cyclin-dependent kinase 3 inhibitor

0.163 0.07 DBMET00289

DBMET00289
0.0250.0230.025Bradykinin B1 receptor antagonist
0.0240.0220.024Acid ceramidase inhibitor
0.0460.0450.046Alpha 1b adrenoreceptor agonist
0.0330.0320.033Bradykinin antagonist
0.0310.030.038Melatonin receptor 1A agonist

0.038 0.016 DBMET00289

DBMET00289
0.0790.0790.11Triose-phosphate isomerase inhibitor

0.11 0.039 DBMET00289

DBMET00289
0.0130.0170.023Ileal bile acid transport inhibitor

0.023 0.007 DBMET00289

DBMET00289
0.0410.0450.053CC chemokine 4 receptor antagonist

0.053 0.023 DBMET00289

DBMET00289
0.1160.1220.138Phospholipase A2 inhibitor

0.138 0.089 DBMET00289

DBMET00289
0.0770.0860.11Prolactin inhibitor

0.11 0.046 DBMET00289

DBMET00289
0.180.190.224Transcription factor NF kappa B inhibitor

0.224 0.147 DBMET00289

DBMET00289
0.0640.0750.092Somatostatin 1 agonist

0.092 0.039 DBMET00289

DBMET00289
0.0180.0330.022Isoleucine-tRNA ligase inhibitor

0.022 0.017 DBMET00289

DBMET00289
0.0940.1160.148Toll-Like receptor 2 antagonist

0.148 0.054 DBMET00289

DBMET00289
0.040.0630.051Argininosuccinate synthase inhibitor

0.051 0.045 DBMET00289

DBMET00289
0.0480.0750.067Lipase inhibitor

0.067 0.057 DBMET00289

DBMET00289
0.0680.1030.094Protease inhibitor

0.094 0.07 DBMET00289

DBMET00289
0.0290.0670.053Ribonucleoside-diphosphate reductase inhibitor

0.053 0.039 DBMET00289

DBMET00289
0.0280.0680.054Ribonucleotide reductase inhibitor

0.054 0.04 DBMET00289

DBMET00289
0.0760.1290.144Amylase inhibitor

0.144 0.067 DBMET00289

DBMET00289
0.0130.0710.031Liver X receptor beta antagonist

0.031 0.018 DBMET00289

DBMET00289
0.1550.2150.301Cholesterol antagonist

0.301 0.091 DBMET00289

DBMET00289
0.0730.1350.095Nav1.4 sodium channel blocker

0.095 0.084 DBMET00289

DBMET00289
0.0310.1170.06Phosphofructokinase-1 inhibitor

0.06 0.057 DBMET00289

DBMET00289
0.0610.1680.108Alkylator

0.108 0.079 DBMET00289

DBMET00289
0.0570.1690.09Transcription factor NF kappa B stimulant

0.09 0.05 DBMET00289

DBMET00289
0.0460.1660.062Prolactin release inhibitor

0.062 0.045 DBMET00289

DBMET00289
0.0240.1460.051Alpha-mannosidase inhibitor

0.051 0.041 DBMET00289

DBMET00289
0.0910.2290.145Hypolipemic

0.145 0.142 DBMET00289

DBMET00289
0.0450.1840.127Bronchodilator

0.127 0.04 DBMET00289

DBMET00289
0.0590.20.113Alpha-N-acetylglucosaminidase inhibitor

0.113 0.085 DBMET00289

DBMET00289
Ext Pa Pi Pmax Activity Other Results ID Pa_max