Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.9090.0020.964Phosphodiesterase IV inhibitor

0.964 0.001 DBMET00997

DBMET00997
0.910.0040.959Toll-Like receptor 7 agonist

0.959 0.004 DBMET00997

DBMET00997
0.9080.0040.96Toll-Like receptor agonist

0.96 0.004 DBMET00997

DBMET00997
0.8620.0020.927Phosphodiesterase 4D inhibitor

0.927 0.002 DBMET00997

DBMET00997
0.8490.0020.936Phosphodiesterase 4B inhibitor

0.936 0.002 DBMET00997

DBMET00997
0.8330.0030.957Phosphodiesterase inhibitor

0.957 0.003 DBMET00997

DBMET00997
0.7610.0040.825Tumour necrosis factor alpha release inhibitor

0.825 0.004 DBMET00997

DBMET00997
0.6910.0020.868Phosphodiesterase 4A inhibitor

0.868 0.002 DBMET00997

DBMET00997
0.6470.0030.761Phosphodiesterase 4C inhibitor

0.761 0.002 DBMET00997

DBMET00997
0.5710.0040.665Tumour necrosis factor antagonist

0.665 0.003 DBMET00997

DBMET00997
0.610.0510.614Antiinflammatory

0.614 0.05 DBMET00997

DBMET00997
0.4740.0050.62Bronchodilator

0.62 0.004 DBMET00997

DBMET00997
0.3940.040.394Nootropic

0.246 0.112 DBMET00997

0.4290.0760.429Cyclophilin D inhibitor

0.36 0.115 DBMET00997

0.4060.0820.406Analgesic

0.28 0.158 DBMET00997

0.3440.0540.344Calcium channel activator

0.284 0.108 DBMET00997

0.2970.0310.2975 Hydroxytryptamine 1E antagonist

0.264 0.06 DBMET00997

0.2560.0040.256Janus tyrosine kinase 1 inhibitor

0.18 0.006 DBMET00997

0.2520.0060.252CF transmembrane conductance regulator agonist

0.217 0.014 DBMET00997

0.2910.0450.291Tyrosine kinase inhibitor
0.2610.0230.2613C-like protease (Human coronavirus) inhibitor

0.136 0.129 DBMET00997

0.2430.0080.243Janus tyrosine kinase 2 inhibitor

0.106 0.033 DBMET00997

0.2320.0090.232Nav1.5 sodium channel blocker

0.119 0.056 DBMET00997

0.2320.0190.232Sodium channel (voltage-gated) blocker

0.11 0.097 DBMET00997

0.2380.0440.238I kappa B kinase epsilon inhibitor
0.20.0080.2Nav1.8 sodium channel blocker

0.126 0.019 DBMET00997

0.2060.0340.248Cytokine production inhibitor

0.248 0.024 DBMET00997

DBMET00997
0.2030.0310.203Sodium channel blocker
0.1760.0070.176Interleukin 5 antagonist

0.153 0.01 DBMET00997

0.220.060.256Nitric-oxide synthase stimulant

0.256 0.029 DBMET00997

DBMET00997
0.2830.1290.283Antiobesity
0.2130.0610.286Non-steroidal antiinflammatory agent

0.286 0.031 DBMET00997

DBMET00997
0.1480.0050.148Secretase beta inhibitor

0.091 0.024 DBMET00997

0.1880.0580.212Antipruritic

0.212 0.041 DBMET00997

DBMET00997
0.1390.0110.139Amidase inhibitor

0.082 0.036 DBMET00997

0.1390.0160.139Glutamate (mGluR7) agonist

0.096 0.069 DBMET00997

0.1710.0540.171Vascular endothelial growth factor 3 antagonist
0.2590.1430.291Calpain 2 inhibitor

0.291 0.12 DBMET00997

DBMET00997
0.1140.0030.114Vanilloid 3 antagonist

0.058 0.005 DBMET00997

0.1220.0170.122Nicotinic alpha4beta2 receptor antagonist
0.1170.0120.117NMDA 2B receptor antagonist

0.089 0.018 DBMET00997

0.1220.0190.122Prostaglandin-E synthase inhibitor
0.1450.0480.145Sphingosine 1-phosphate receptor 2 antagonist

0.114 0.112 DBMET00997

0.120.0290.12ALK inhibitor
0.130.0410.13Proto-oncogene tyrosine-protein kinase Kit inhibitor
0.1760.0920.176Growth factor agonist
0.0880.0050.088Farnesoid X receptor agonist

0.072 0.007 DBMET00997

0.1220.0390.122Hedgehog signaling inhibitor
0.0920.0190.092Orexin receptor 1 antagonist
0.0760.010.076Antiviral (Hepatitis D)

0.062 0.02 DBMET00997

0.0830.0230.083Orexin receptor antagonist
0.1230.0670.123Sphingosine 1-phosphate receptor 4 antagonist

0.118 0.076 DBMET00997

0.0850.030.085Nav1.7 sodium channel blocker
0.1030.050.103Potassium channel (Voltage-sensitive) activator
0.0690.020.069Diacylglycerol O-acyltransferase inhibitor
0.2840.2360.284Ca2+/calmodulin-dependent protein kinase kinase A inhibitor
0.0880.0410.088Rho-associated kinase inhibitor
0.080.0350.08Potassium channel (Tandem pore domain) blocker
0.0570.0120.057Glutamate (mGluR group II) antagonist
0.0510.0090.051Free fatty acid receptor 1 antagonist

0.037 0.019 DBMET00997

0.1410.1030.141Interleukin-1 receptor-associated protein kinase 1 inhibitor
0.1060.0690.106EphA2 antagonist
0.0880.0520.088Myeloperoxidase inhibitor
0.1260.0920.126Death-associated protein kinase 1 inhibitor
0.2080.1750.208Ca(v)3.3 blocker
0.0410.0110.041Glutamate (mGluR2) antagonist
0.0580.0310.058Melanin-concentrating hormone receptor 1 antagonist
0.0360.0120.036Prostaglandin EP4 antagonist
0.0510.0280.051Carnitine palmitoyltransferase 1B inhibitor

0.044 0.041 DBMET00997

0.0740.0510.074Rho-associated kinase II inhibitor
0.0750.0570.075Sphingosine 1-phosphate receptor antagonist
0.1030.0850.103Beta amyloid protein antagonist
0.0540.0370.054Protein kinase C epsilon inhibitor
0.0240.0080.024Cyclin T1 inhibitor
0.0210.0050.021Prokineticin receptor 1 antagonist

0.02 0.007 DBMET00997

0.0380.0220.038Orexin receptor 2 antagonist
0.0850.0710.085Polo-like kinase-1 inhibitor
0.0880.0740.088Toll-Like receptor 3 antagonist
0.0670.0540.096NMDA 2 receptor antagonist

0.096 0.034 DBMET00997

DBMET00997
0.0370.0250.037Delayed rectifier potassium channel activator
0.0370.0250.037Potassium channel KCNQ activator
0.0340.0210.034Calcium release-activated channel blocker
0.0320.020.032Prostaglandin agonist

0.028 0.026 DBMET00997

0.0490.0370.049Prostaglandin E2 antagonist
0.020.0090.02Complement factor D inhibitor
0.0860.0770.086Sphingomyelinase inhibitor
0.0230.0160.023Prostaglandin E2 agonist
0.0410.0350.041Phosphodiesterase 3B inhibitor
0.0760.0710.076Stem cell growth factor agonist
0.0320.0270.032Carnitine palmitoyltransferase 1 inhibitor
0.0540.0490.054Sphingosine 1-phosphate receptor 3 antagonist
0.0550.050.055TRPA1 antagonist
0.0550.0510.055Ca(v)3.2 blocker
0.0310.0280.031Carnitine palmitoyltransferase inhibitor
0.1120.1090.112Vanilloid 1 agonist
0.0260.0240.026Carnitine palmitoyltransferase 1A inhibitor
0.0550.0540.055Protease activated receptor antagonist
0.0640.0630.064Vanilloid antagonist
0.0820.0890.098Gastric antisecretory

0.098 0.069 DBMET00997

DBMET00997
0.1850.2010.217Apoptosis antagonist

0.217 0.159 DBMET00997

DBMET00997
0.040.070.053Phosphodiesterase 7A inhibitor

0.053 0.033 DBMET00997

DBMET00997
0.0530.1130.07Phosphodiesterase VIII inhibitor

0.07 0.053 DBMET00997

DBMET00997
0.0270.1170.067Acetylcholine M3 receptor antagonist

0.067 0.034 DBMET00997

DBMET00997
Ext Pa Pi Pmax Activity Other Results ID Pa_max