Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.7290.0040.729Protein kinase (CaMK, MLCK, PhK, SNF, KIN, NIM1, MAPKAP, POLO, CHK, ULK, RSK-2nd domain) inhibitor

0.554 0.004 DBMET01498

0.554 0.004 DBMET01500

0.6580.0030.658Check point kinase 1 inhibitor

0.468 0.004 DBMET01498

0.472 0.004 DBMET01500

0.6140.0040.614EphB2 antagonist

0.423 0.014 DBMET01498

0.438 0.012 DBMET01500

0.5570.0050.557Glycogen synthase kinase-3 inhibitor

0.356 0.011 DBMET01498

0.413 0.008 DBMET01500

0.5750.0270.619MAP kinase 1 inhibitor

0.619 0.016 DBMET01498

0.476 0.063 DBMET01500

DBMET01498
0.5250.0040.541Xanthine oxidase inhibitor

0.541 0.003 DBMET01498

0.367 0.005 DBMET01500

DBMET01498
0.5170.0050.517Glycogen synthase kinase-3 beta inhibitor

0.304 0.013 DBMET01498

0.365 0.009 DBMET01500

0.4930.0040.493Ribosomal protein S6 kinase inhibitor

0.387 0.005 DBMET01498

0.449 0.004 DBMET01500

0.4870.0060.487RET inhibitor

0.302 0.022 DBMET01498

0.263 0.029 DBMET01500

0.480.0020.587Xanthine dehydrogenase inhibitor

0.587 0.002 DBMET01498

0.352 0.003 DBMET01500

DBMET01498
0.470.0040.47Protein kinase (CK2) alpha inhibitor

0.467 0.004 DBMET01498

0.242 0.017 DBMET01500

0.4690.0050.469MAP kinase 9 inhibitor

0.232 0.018 DBMET01498

0.32 0.01 DBMET01500

0.4630.0050.463Glycogen synthase kinase-3 alpha inhibitor

0.374 0.008 DBMET01498

0.325 0.013 DBMET01500

0.4640.0290.47MAP kinase kinase 6 inhibitor

0.356 0.088 DBMET01498

0.47 0.027 DBMET01500

DBMET01500
0.4610.0370.461Angiogenesis inhibitor

0.306 0.09 DBMET01498

0.431 0.044 DBMET01500

0.4190.0030.419Protein kinase C delta inhibitor

0.283 0.004 DBMET01498

0.28 0.004 DBMET01500

0.4070.0140.407CDC-like kinase 4 inhibitor

0.19 0.073 DBMET01498

0.284 0.036 DBMET01500

0.4020.0190.402Clk dual-specificity kinase inhibitor

0.211 0.073 DBMET01498

0.258 0.052 DBMET01500

0.3760.0040.376Uric acid excretion stimulant

0.359 0.004 DBMET01498

0.271 0.005 DBMET01500

0.3920.0280.392Dyrk kinase inhibitor

0.307 0.05 DBMET01498

0.234 0.079 DBMET01500

0.3610.0030.361Protein kinase B beta inhibitor

0.242 0.004 DBMET01498

0.324 0.004 DBMET01500

0.3910.0410.391Nootropic

0.215 0.139 DBMET01498

0.265 0.095 DBMET01500

0.360.0130.36Vascular endothelial growth factor 3 antagonist

0.231 0.032 DBMET01498

0.159 0.06 DBMET01500

0.360.0160.36Dual specificity tyrosine-phosphorylation regulated kinase 3 inhibitor

0.214 0.066 DBMET01498

0.214 0.066 DBMET01500

0.3440.0050.369Protein kinase (CK2) inhibitor

0.369 0.004 DBMET01498

0.175 0.024 DBMET01500

DBMET01498
0.3420.0030.342Protein kinase C theta inhibitor

0.18 0.004 DBMET01498

0.221 0.004 DBMET01500

0.3520.0160.352TRKC antagonist

0.196 0.069 DBMET01498

0.239 0.052 DBMET01500

0.3440.0220.344CDC-like kinase 2 inhibitor

0.142 0.099 DBMET01498

0.157 0.089 DBMET01500

0.3280.0090.328Protein-tyrosine kinase (PTK, not ETK, WZC) inhibitor

0.178 0.034 DBMET01498

0.248 0.018 DBMET01500

0.3270.0090.327Abl kinase inhibitor

0.178 0.034 DBMET01498

0.247 0.018 DBMET01500

0.3160.0040.316Protein kinase B alpha inhibitor

0.19 0.005 DBMET01498

0.239 0.004 DBMET01500

0.3280.0170.328Cyclin-dependent kinase inhibitor

0.197 0.038 DBMET01498

0.209 0.035 DBMET01500

0.3310.0310.331Cyclic AMP phosphodiesterase inhibitor

0.206 0.089 DBMET01498

0.159 0.137 DBMET01500

0.3050.0080.305Cyclin-dependent kinase 8 inhibitor

0.198 0.037 DBMET01498

0.233 0.02 DBMET01500

0.3220.0310.322Ca2+/calmodulin-dependent kinase II gamma inhibitor

0.174 0.076 DBMET01498

0.3040.0150.304Dual specificity tyrosine-phosphorylation regulated kinase 1B inhibitor

0.169 0.06 DBMET01498

0.245 0.027 DBMET01500

0.2990.0120.299Protein kinase (CK1) delta inhibitor

0.166 0.044 DBMET01498

0.13 0.066 DBMET01500

0.3020.0170.302Protein kinase (CK1) inhibitor

0.162 0.059 DBMET01498

0.121 0.091 DBMET01500

0.3090.0320.309MAP kinase kinase 2 inhibitor

0.164 0.108 DBMET01498

0.165 0.108 DBMET01500

0.280.0040.28Protein kinase C alpha inhibitor

0.215 0.005 DBMET01498

0.211 0.005 DBMET01500

0.3170.0450.317Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor

0.252 0.067 DBMET01498

0.2810.0130.281Cyclin-dependent kinase 1 inhibitor

0.175 0.032 DBMET01498

0.189 0.028 DBMET01500

0.2770.0140.277MAP kinase kinase 3 inhibitor

0.22 0.074 DBMET01498

0.223 0.068 DBMET01500

0.2670.0090.267MAP kinase 8 inhibitor

0.145 0.031 DBMET01498

0.168 0.023 DBMET01500

0.2750.0220.275Tyrosine-protein kinase receptor FLT3 inhibitor

0.103 0.078 DBMET01498

0.125 0.065 DBMET01500

0.2950.0450.295Ca2+/calmodulin-dependent protein kinase inhibitor

0.154 0.108 DBMET01498

0.2650.0250.265Cytidine deaminase inhibitor

0.147 0.078 DBMET01498

0.153 0.073 DBMET01500

0.260.020.589Phosphodiesterase inhibitor

0.264 0.02 DBMET01498

0.589 0.004 DBMET01500

DBMET01500
0.3150.0780.315Calcium channel activator

0.213 0.194 DBMET01500

0.2430.0060.243MAP kinase 10 inhibitor

0.142 0.018 DBMET01498

0.127 0.021 DBMET01500

0.2430.0080.243Rho-associated kinase II inhibitor

0.084 0.042 DBMET01498

0.097 0.033 DBMET01500

0.2790.0470.279Tyrosine kinase inhibitor

0.126 0.104 DBMET01498

0.122 0.107 DBMET01500

0.2590.0270.259Protein kinase (CK1) gamma inhibitor

0.119 0.091 DBMET01498

0.2470.0210.247Activin receptor-like kinase 2 inhibitor

0.131 0.084 DBMET01498

0.133 0.082 DBMET01500

0.3420.1230.3425 Hydroxytryptamine release inhibitor
0.2310.0120.231Platelet activating factor alpha antagonist

0.157 0.028 DBMET01498

0.129 0.039 DBMET01500

0.2320.0180.263Glutamate receptor antagonist

0.263 0.014 DBMET01498

0.232 0.018 DBMET01500

DBMET01498
0.2470.0370.247Dual specificity tyrosine-phosphorylation-regulated kinase 4 inhibitor

0.115 0.105 DBMET01498

0.2190.010.219Rho-associated kinase inhibitor

0.082 0.045 DBMET01498

0.107 0.031 DBMET01500

0.2390.030.239Vascular endothelial growth factor antagonist

0.146 0.056 DBMET01498

0.141 0.058 DBMET01500

0.2170.0090.217MAP kinase kinase 4 inhibitor

0.185 0.021 DBMET01498

0.172 0.031 DBMET01500

0.220.0130.22Check point kinase 2 inhibitor

0.148 0.032 DBMET01498

0.142 0.034 DBMET01500

0.2220.0170.222MAP kinase 12 inhibitor

0.175 0.031 DBMET01498

0.15 0.042 DBMET01500

0.2590.0540.263Ca2+/calmodulin-dependent kinase IV inhibitor

0.263 0.051 DBMET01498

0.196 0.177 DBMET01500

DBMET01498
0.2060.0060.206Death-associated protein kinase 1 inhibitor

0.178 0.014 DBMET01498

0.164 0.023 DBMET01500

0.2510.0520.251Death-associated protein kinase 3 inhibitor

0.144 0.132 DBMET01498

0.2120.0180.212MAP kinase 13 inhibitor

0.158 0.032 DBMET01498

0.121 0.055 DBMET01500

0.2230.030.223Vascular endothelial growth factor 2 antagonist

0.134 0.055 DBMET01498

0.122 0.06 DBMET01500

0.1980.0080.198Protein kinase B gamma inhibitor

0.107 0.029 DBMET01498

0.098 0.033 DBMET01500

0.2170.0270.321Hemostatic

0.321 0.014 DBMET01498

0.183 0.041 DBMET01500

DBMET01498
0.2040.0170.204Protein kinase (Mos, Mil/Raf, MEKK, RIPK, TESK, LIMK, IRAK, ILK, Activin/TGF-beta) inhibitor

0.098 0.055 DBMET01498

0.107 0.048 DBMET01500

0.1870.0050.187Phosphodiesterase X inhibitor

0.145 0.006 DBMET01498

0.075 0.015 DBMET01500

0.1870.0050.187Phosphodiesterase 10A inhibitor

0.145 0.006 DBMET01498

0.075 0.015 DBMET01500

0.2090.0290.209Cyclin-dependent kinase 3 inhibitor

0.164 0.069 DBMET01498

0.157 0.081 DBMET01500

0.2030.0250.203Aurora-A kinase inhibitor

0.087 0.077 DBMET01498

0.128 0.05 DBMET01500

0.1830.0060.183CDC7 inhibitor

0.161 0.008 DBMET01498

0.083 0.033 DBMET01500

0.1990.0220.203Granulocyte macrophage colony stimulating factor antagonist

0.105 0.066 DBMET01498

0.203 0.021 DBMET01500

DBMET01500
0.1870.0110.187Glutamate (mGluR) antagonist

0.131 0.022 DBMET01498

0.14 0.019 DBMET01500

0.2240.0520.224LIM domain kinase 1 inhibitor
0.2370.0680.237MAP-kinase-activated kinase 5 inhibitor

0.231 0.073 DBMET01498

0.3350.1680.335Ca2+/calmodulin-dependent protein kinase kinase A inhibitor
0.2270.060.227Ca2+/calmodulin-dependent kinase II beta inhibitor

0.158 0.118 DBMET01498

0.2010.0340.201Death-associated protein kinase 2 inhibitor

0.201 0.034 DBMET01498

0.167 0.072 DBMET01500

0.190.0250.19Ca2+/calmodulin-dependent protein kinase kinase B inhibitor

0.175 0.037 DBMET01498

0.152 0.069 DBMET01500

0.1980.0360.198c-Src kinase inhibitor

0.097 0.092 DBMET01498

0.151 0.055 DBMET01500

0.1950.0330.195Mannose-6-phosphate isomerase inhibitor

0.173 0.047 DBMET01498

0.14 0.074 DBMET01500

0.2050.0440.205Protein-tyrosine kinase Lyn inhibitor
0.1640.0050.164MAP kinase kinase 9 inhibitor

0.072 0.019 DBMET01498

0.062 0.029 DBMET01500

0.1810.0230.181Beta amyloid protein antagonist

0.135 0.052 DBMET01498

0.1770.0190.177Pim-1 kinase inhibitor

0.091 0.067 DBMET01498

0.170.0130.17Pim-3 kinase inhibitor

0.127 0.027 DBMET01498

0.088 0.062 DBMET01500

0.2150.060.215Interleukin-1 receptor-associated protein kinase 1 inhibitor
0.1660.0160.166Raf kinase inhibitor

0.077 0.048 DBMET01498

0.085 0.041 DBMET01500

0.2020.0530.202Src kinase inhibitor

0.119 0.108 DBMET01498

0.134 0.096 DBMET01500

0.1610.0120.161MAP-kinase-activated kinase inhibitor

0.118 0.027 DBMET01498

0.1 0.039 DBMET01500

0.1870.0380.187Alkaline phosphatase inhibitor

0.162 0.052 DBMET01498

0.1820.0330.194MAP kinase 3 inhibitor

0.194 0.027 DBMET01498

DBMET01498
0.1730.0260.198MAP kinase kinase kinase inhibitor

0.096 0.071 DBMET01498

0.198 0.019 DBMET01500

DBMET01500
0.1750.030.175Cyclin-dependent kinase 2 inhibitor

0.114 0.057 DBMET01498

0.131 0.046 DBMET01500

0.1590.0170.159Leucine-rich repeat kinase 2 inhibitor

0.099 0.043 DBMET01498

0.1690.0280.169Proto-oncogene tyrosine-protein kinase Kit inhibitor

0.087 0.065 DBMET01500

0.1550.0180.212MAP kinase 14 inhibitor

0.212 0.01 DBMET01500

DBMET01500
0.20.0630.2Growth factor agonist

0.184 0.081 DBMET01498

0.168 0.106 DBMET01500

0.1550.0190.155ALK inhibitor

0.098 0.042 DBMET01498

0.078 0.063 DBMET01500

0.1740.0390.174MAP kinase kinase inhibitor

0.119 0.074 DBMET01498

0.116 0.078 DBMET01500

0.1490.0140.149Tyk2 inhibitor

0.089 0.032 DBMET01498

0.1740.040.174Protein kinase (CK1) gamma 2 inhibitor
0.1360.0030.136Bombesin agonist

0.116 0.004 DBMET01498

0.115 0.004 DBMET01500

0.1650.0330.165Cyclin-dependent kinase 5 inhibitor

0.113 0.064 DBMET01498

0.142 0.045 DBMET01500

0.1430.0120.143MAP-kinase-activated kinase 2 inhibitor

0.098 0.029 DBMET01498

0.085 0.039 DBMET01500

0.1860.0560.186Protein kinase (CK1) gamma 3 inhibitor
0.1790.0490.179Tyrosine-protein kinase receptor antagonist

0.109 0.097 DBMET01498

0.1660.040.166Aurora-B kinase inhibitor

0.097 0.086 DBMET01498

0.129 0.058 DBMET01500

0.140.0170.14Fibroblast growth factor 3 antagonist

0.08 0.051 DBMET01498

0.073 0.06 DBMET01500

0.1630.0430.163TRKA antagonist

0.11 0.077 DBMET01498

0.1310.0130.131MAP kinase kinase 10 inhibitor

0.063 0.053 DBMET01498

0.067 0.045 DBMET01500

0.1460.030.146Activin receptor-like kinase 4 inhibitor

0.096 0.095 DBMET01498

0.1980.0820.198Pyruvate kinase inhibitor

0.16 0.107 DBMET01498

0.194 0.084 DBMET01500

0.2370.1210.237Ca(v)3.3 blocker
0.2040.0880.204Ca2+/calmodulin-dependent kinase I alpha inhibitor
0.1230.0080.185AMPA receptor antagonist

0.132 0.007 DBMET01498

0.185 0.005 DBMET01500

DBMET01500
0.1620.0480.162Toll-Like receptor antagonist

0.115 0.092 DBMET01500

0.1150.0030.115Bombesin 3 receptor agonist

0.097 0.004 DBMET01498

0.096 0.004 DBMET01500

0.1380.0270.138Interleukin-1 receptor-associated protein kinase 4 inhibitor

0.098 0.047 DBMET01498

0.094 0.052 DBMET01500

0.1250.0180.125Raf kinase B inhibitor

0.057 0.043 DBMET01500

0.1230.0180.123Glutamate (mGluR) agonist

0.064 0.041 DBMET01498

0.1260.0240.126MAP kinase 11 inhibitor

0.072 0.053 DBMET01498

0.108 0.031 DBMET01500

0.1120.010.112mTOR inhibitor

0.076 0.019 DBMET01498

0.051 0.037 DBMET01500

0.1160.0160.116I kappa B kinase 1 inhibitor

0.064 0.057 DBMET01500

0.1160.0170.116Phosphatidylinositol kinase inhibitor

0.073 0.031 DBMET01498

0.054 0.048 DBMET01500

0.110.0150.11Toll-Like receptor 7 antagonist
0.1090.0150.109Phosphatidylinositol 3-kinase alpha inhibitor

0.067 0.026 DBMET01498

0.049 0.038 DBMET01500

0.1340.0390.187Cyclin-dependent kinase 9 inhibitor

0.187 0.025 DBMET01500

DBMET01500
0.1160.0230.116Adenosine A2 receptor antagonist

0.076 0.037 DBMET01498

0.087 0.031 DBMET01500

0.1410.050.32Platelet activating factor antagonist

0.32 0.009 DBMET01500

DBMET01500
0.1630.0720.163Polo-like kinase-3 inhibitor
0.0980.0070.098DNA-dependent protein kinase inhibitor

0.053 0.019 DBMET01498

0.073 0.01 DBMET01500

0.1140.0240.114Macrophage colony-stimulating factor 1 receptor antagonist

0.11 0.025 DBMET01500

0.1060.0170.106Protein kinase C iota inhibitor

0.057 0.044 DBMET01498

0.075 0.029 DBMET01500

0.1090.0210.109Fibroblast growth factor 2 antagonist

0.073 0.039 DBMET01498

0.1180.0310.118mTOR complex 1 inhibitor

0.095 0.073 DBMET01498

0.1070.020.107Janus tyrosine kinase 1 inhibitor

0.049 0.047 DBMET01498

0.0910.0040.091Vascular adhesion protein 1 inhibitor

0.038 0.028 DBMET01498

0.037 0.03 DBMET01500

0.1540.0670.154Growth factor antagonist
0.1220.0360.15DNA directed RNA polymerase inhibitor

0.103 0.053 DBMET01498

0.15 0.024 DBMET01500

DBMET01500
0.1210.0350.121Hepatocyte growth factor antagonist

0.085 0.068 DBMET01498

0.0890.0040.089Alpha 1d adrenoreceptor agonist

0.037 0.029 DBMET01498

0.042 0.023 DBMET01500

0.0970.0130.097Protein kinase C epsilon inhibitor
0.1570.0740.157Peroxidase inhibitor

0.117 0.103 DBMET01498

0.0950.0120.095Exportin-1 inhibitor
0.0950.0120.095Cyclin-dependent kinase 6 inhibitor

0.094 0.012 DBMET01498

0.075 0.026 DBMET01500

0.1080.0270.204Phosphodiesterase 3A inhibitor

0.204 0.008 DBMET01498

0.081 0.054 DBMET01500

DBMET01498
0.1750.0940.175I kappa B kinase epsilon inhibitor
0.1360.0570.136TRKB antagonist
0.0960.0190.096DNA gyrase inhibitor

0.075 0.031 DBMET01498

0.08 0.026 DBMET01500

0.0890.0130.089Toll-Like receptor 8 antagonist
0.1110.0350.112Polo-like kinase-1 inhibitor

0.112 0.035 DBMET01500

DBMET01500
0.0990.0230.099Adenosine A1 receptor antagonist

0.06 0.039 DBMET01498

0.071 0.032 DBMET01500

0.1080.0330.108Janus tyrosine kinase 2 inhibitor
0.110.0370.11Stem cell growth factor agonist

0.085 0.059 DBMET01500

0.1030.030.103Rho-associated kinase I inhibitor

0.07 0.056 DBMET01500

0.1980.1260.198DNA synthesis inhibitor

0.182 0.15 DBMET01500

0.1390.0680.139Cyclin-dependent kinase 7 inhibitor

0.121 0.084 DBMET01500

0.1020.0320.104p38 MAP kinase inhibitor

0.104 0.031 DBMET01500

DBMET01500
0.0950.0250.095MAP kinase kinase 8 inhibitor

0.062 0.059 DBMET01498

0.1350.0650.275M17 leucyl aminopeptidase inhibitor

0.275 0.016 DBMET01498

DBMET01498
0.1050.0370.105Bcr-Abl kinase inhibitor

0.098 0.043 DBMET01500

0.0720.0060.072DNA gyrase subunit B inhibitor

0.046 0.016 DBMET01498

0.0830.0170.102Fatty acid synthase inhibitor

0.102 0.01 DBMET01498

0.095 0.012 DBMET01500

DBMET01498
0.1330.070.133Sodium channel (voltage-gated) blocker
0.1090.0460.109CDK/cyclin complex inhibitor
0.10.0380.1I kappa B kinase inhibitor
0.0840.0240.084Protein kinase C beta inhibitor

0.067 0.054 DBMET01498

0.1340.0740.134Ca2+/calmodulin-dependent kinase II delta inhibitor
0.0860.0270.086S-adenosyl-L-methionine decarboxylase inhibitor
0.0870.0290.087Cyclin E inhibitor
0.0680.010.068Glutamate (mGluR group II) agonist

0.036 0.023 DBMET01498

0.0730.0170.075Adenosine A2b receptor antagonist

0.062 0.023 DBMET01498

0.075 0.016 DBMET01500

DBMET01500
0.0650.010.065Glutamate (mGluR2) agonist

0.031 0.023 DBMET01498

0.1050.0530.105Protein kinase C mu inhibitor

0.096 0.06 DBMET01498

0.0810.0310.081Adenosine A2a receptor antagonist
0.1330.0840.133Protein kinase (CK1) gamma 1 inhibitor
0.0850.0370.085Adenosine A3 receptor antagonist

0.075 0.05 DBMET01498

0.0510.0070.051ATR kinase inhibitor

0.033 0.022 DBMET01498

0.03 0.029 DBMET01500

0.0810.0370.081Glutamate (mGluR group I) antagonist

0.063 0.059 DBMET01498

0.067 0.053 DBMET01500

0.0710.0270.071Heat shock protein 90 beta antagonist

0.063 0.035 DBMET01498

0.1250.0810.142Toll-Like receptor 9 antagonist

0.142 0.068 DBMET01500

DBMET01500
0.050.0070.05Carnitine palmitoyltransferase 1A inhibitor

0.034 0.013 DBMET01498

0.031 0.016 DBMET01500

0.0840.0420.084Janus tyrosine kinase 3 inhibitor
0.0990.0580.099Fibroblast growth factor 1 antagonist
0.0610.0210.061Glutamate (mGluR5) antagonist

0.043 0.037 DBMET01498

0.0660.0270.066Phosphatidylinositol 3-kinase gamma inhibitor
0.1590.1210.159HERG channel blocker
0.120.0820.12Proto-oncogene tyrosine-protein kinase Yes inhibitor
0.0860.0480.086Glutamate receptor agonist
0.0620.0250.062Transforming growth factor beta 1 antagonist
0.130.0940.13MAP3K9 inhibitor
0.0850.050.085Transforming growth factor beta 3 antagonist
0.120.0850.12Lck kinase inhibitor
0.0760.0440.113Benzodiazepine agonist

0.113 0.019 DBMET01500

DBMET01500
0.0750.0430.075Orexin receptor 1 antagonist
0.1350.1060.135CF transmembrane conductance regulator agonist
0.0730.0440.073Transforming growth factor antagonist
0.0460.0180.046Glutamate (mGluR group II) antagonist
0.0630.0350.063Phosphatidylinositol 3-kinase delta inhibitor

0.053 0.044 DBMET01498

0.0570.030.057Factor IXa inhibitor

0.057 0.029 DBMET01500

0.0770.0510.077CYP2A6 inhibitor
0.0730.0470.073Phosphodiesterase VIII inhibitor

0.073 0.047 DBMET01500

0.0920.0660.092CDK2/cyclin A inhibitor

0.081 0.079 DBMET01500

0.0570.0340.057Pim-2 kinase inhibitor
0.0680.0460.068Nav1.7 sodium channel blocker
0.0810.0590.081Protein kinase A inhibitor
0.0380.0170.038Carnitine palmitoyltransferase 1 inhibitor
0.1070.0860.107Transcription factor STAT6 inhibitor
0.1530.1340.153Potassium channel (Voltage-sensitive) blocker
0.0410.0230.043CF transmembrane conductance regulator antagonist

0.039 0.03 DBMET01498

0.043 0.017 DBMET01500

DBMET01500
0.0370.0190.037Carnitine palmitoyltransferase inhibitor
0.0620.0440.073Phosphodiesterase 1C inhibitor

0.073 0.026 DBMET01498

DBMET01498
0.0330.0160.033Glutamate (mGluR2) antagonist
0.0510.0340.051Alpha 1b adrenoreceptor agonist
0.080.0640.08GABA A receptor agonist
0.0880.0750.136Vascular endothelial growth factor 1 antagonist

0.136 0.046 DBMET01498

DBMET01498
0.0170.0050.028Egl nine homolog 2 inhibitor

0.028 0.004 DBMET01498

DBMET01498
0.0590.0480.059I kappa B kinase 2 inhibitor
0.0520.0410.052Myc inhibitor
0.0190.0090.027CC chemokine 9 receptor antagonist

0.027 0.004 DBMET01500

DBMET01500
0.0730.0640.073Proto-oncogene tyrosine-protein kinase c-hck inhibitor
0.0270.0190.042Protocollagen prolyl hydroxylase inhibitor

0.042 0.007 DBMET01498

DBMET01498
0.060.0520.06Cyclin-dependent kinase 4 inhibitor
0.0360.0290.036Poly(ADP-ribose) polymerase 1 inhibitor
0.0420.0350.042Poly(ADP-ribose) polymerase inhibitor
0.0960.090.096CDC-like kinase 3 inhibitor
0.0510.0450.051Bombesin 3 receptor antagonist
0.0080.0030.008CC chemokine 6 receptor agonist
0.0720.0670.072Platelet growth factor antagonist
0.0620.0580.062Syk tyrosine kinase inhibitor
0.0540.050.058Cyclin A inhibitor

0.058 0.045 DBMET01500

DBMET01500
0.0280.0240.033MAP3K8 inhibitor

0.033 0.012 DBMET01500

DBMET01500
0.0330.0290.033Orexin receptor 2 antagonist
0.0420.0380.042Glutamate (mGluR5) agonist
0.0530.050.053CDK2/cyclin E inhibitor
0.060.0570.06Orexin receptor antagonist
0.0350.0340.035MAP3K5 inhibitor
0.2040.2030.204GABA C receptor rho-3 antagonist
0.0530.0550.059Cyclin A2 inhibitor

0.059 0.048 DBMET01500

DBMET01500
0.0530.0590.113Phosphodiesterase III inhibitor

0.113 0.018 DBMET01498

DBMET01498
0.0290.0360.055Factor XI inhibitor

0.055 0.008 DBMET01498

0.039 0.016 DBMET01500

DBMET01498
0.0420.050.045Potassium channel (ATP-sensitive) activator

0.045 0.041 DBMET01500

DBMET01500
0.0430.0520.047Potassium channel (Inward rectifier) activator

0.047 0.043 DBMET01500

DBMET01500
0.0190.0320.026CXC chemokine 2 receptor antagonist

0.026 0.019 DBMET01498

DBMET01498
0.0720.0850.08Factor XII inhibitor

0.08 0.066 DBMET01500

DBMET01500
0.0370.0640.055Benzodiazepine inverse agonist

0.055 0.019 DBMET01500

DBMET01500
0.0520.0850.086CXC chemokine receptor antagonist

0.086 0.033 DBMET01500

DBMET01500
0.0060.0490.013Egl nine homolog 1 inhibitor

0.013 0.012 DBMET01498

DBMET01498
0.0240.0720.057Factor XIa inhibitor

0.057 0.014 DBMET01498

DBMET01498
0.0250.0740.101Phosphodiesterase 3B inhibitor

0.101 0.011 DBMET01498

DBMET01498
0.0610.120.092Potassium channel activator

0.092 0.058 DBMET01500

DBMET01500
0.030.0930.202Phosphodiesterase 4C inhibitor

0.202 0.005 DBMET01500

DBMET01500
0.0570.1250.236Bronchodilator

0.236 0.014 DBMET01500

DBMET01500
0.0990.1740.124Heat shock protein 90 alpha antagonist

0.124 0.12 DBMET01500

DBMET01500
0.0350.1230.079Phosphodiesterase 4B inhibitor

0.079 0.037 DBMET01500

DBMET01500
0.0190.1270.384Phosphodiesterase 4A inhibitor

0.384 0.004 DBMET01500

DBMET01500
0.0350.150.124Phosphodiesterase IV inhibitor

0.124 0.031 DBMET01500

DBMET01500
0.1380.2560.181Nitric-oxide synthase stimulant

0.181 0.125 DBMET01500

DBMET01500
0.0960.2260.28Platelet aggregation inhibitor

0.28 0.041 DBMET01500

DBMET01500
0.0240.1550.074Farnesyltransferase inhibitor

0.074 0.014 DBMET01500

DBMET01500
0.1780.3090.236Cyclophilin D inhibitor

0.236 0.229 DBMET01498

DBMET01498
0.0240.190.237Phosphodiesterase 4D inhibitor

0.237 0.008 DBMET01500

DBMET01500
0.0220.190.064HIV-1 reverse transcriptase inhibitor

0.064 0.055 DBMET01498

DBMET01498
0.0360.2060.114Chemokine receptor antagonist

0.114 0.052 DBMET01500

DBMET01500
0.1190.3040.209Vasodilator, peripheral

0.209 0.166 DBMET01500

DBMET01500
0.10.3890.637Toll-Like receptor 7 agonist

0.637 0.013 DBMET01500

DBMET01500
0.0630.3540.328Tumour necrosis factor alpha release inhibitor

0.328 0.044 DBMET01500

DBMET01500
0.0930.4080.627Toll-Like receptor agonist

0.627 0.014 DBMET01500

DBMET01500
0.0490.4090.29Vasodilator

0.29 0.052 DBMET01500

DBMET01500
0.0050.3840.065Dopamine D4 agonist

0.065 0.025 DBMET01500

DBMET01500
Ext Pa Pi Pmax Activity Other Results ID Pa_max