Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.6950.0010.695O6-alkylguanine-DNA alkyltransferase inhibitor

0.062 0.001 DBMET00499

0.037 0.002 DBMET00498

0.6750.0030.675Cyclin B1 inhibitor

0.274 0.004 DBMET00499

0.650.0030.65Cyclin B2 inhibitor

0.25 0.004 DBMET00499

0.6370.0040.637Cyclin-dependent kinase 1 inhibitor

0.308 0.011 DBMET00499

0.6030.0030.603DNA polymerase I inhibitor

0.444 0.005 DBMET00499

0.17 0.039 DBMET00498

0.5980.0030.598Cyclin B inhibitor

0.231 0.004 DBMET00499

0.5520.0040.552CDK1/cyclin B inhibitor

0.094 0.027 DBMET00499

0.5330.0090.533RNA-directed DNA polymerase inhibitor

0.473 0.012 DBMET00499

0.337 0.026 DBMET00498

0.331 0.026 DB11100

0.510.0130.51DNA synthesis inhibitor

0.416 0.02 DBMET00499

0.279 0.051 DBMET00498

0.25 0.066 DB11100

0.4780.0320.478GABA C receptor rho-3 antagonist

0.454 0.04 DBMET00499

0.378 0.072 DBMET00498

0.274 0.134 DB11100

0.4060.0040.406CDK1/cyclin B1 inhibitor

0.093 0.031 DBMET00499

0.062 0.058 DBMET00498

0.3920.0040.392Check point kinase 2 inhibitor

0.089 0.075 DBMET00499

0.4270.050.556Toll-Like receptor agonist

0.556 0.023 DBMET00499

DBMET00499
0.3790.010.379Glycogen synthase kinase-3 inhibitor

0.187 0.034 DBMET00499

0.4330.0740.473Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.473 0.047 DBMET00499

0.344 0.158 DBMET00498

0.405 0.096 DB11100

DBMET00499
0.4090.0560.566Toll-Like receptor 7 agonist

0.566 0.021 DBMET00499

DBMET00499
0.3570.0050.397Protein kinase (CaMK, MLCK, PhK, SNF, KIN, NIM1, MAPKAP, POLO, CHK, ULK, RSK-2nd domain) inhibitor

0.397 0.005 DBMET00499

0.121 0.027 DB11100

DBMET00499
0.3450.0050.345Nitric-oxide synthase stimulant

0.277 0.018 DBMET00499

0.206 0.079 DBMET00498

0.3480.010.348Glycogen synthase kinase-3 beta inhibitor

0.178 0.034 DBMET00499

0.3420.0050.354Adenosine A1 receptor antagonist

0.354 0.005 DBMET00499

0.112 0.021 DBMET00498

DBMET00499
0.3560.0230.476EphB2 antagonist

0.476 0.009 DBMET00499

DBMET00499
0.3380.0080.338CDK/cyclin complex inhibitor
0.3140.0090.314GABA C receptor agonist

0.26 0.013 DBMET00499

0.257 0.013 DBMET00498

0.177 0.025 DB11100

0.3340.030.734Cyclic AMP phosphodiesterase inhibitor

0.734 0.003 DBMET00499

0.291 0.045 DBMET00498

DBMET00499
0.3070.0030.307Folate antagonist
0.310.0090.509Bronchodilator

0.509 0.004 DBMET00499

DBMET00499
0.3080.010.431Ribosomal protein S6 kinase inhibitor

0.431 0.005 DBMET00499

DBMET00499
0.2910.0050.291MAP kinase 3 inhibitor

0.176 0.037 DBMET00499

0.2990.0150.299Growth factor agonist
0.2750.0050.347Check point kinase 1 inhibitor

0.347 0.005 DBMET00499

0.06 0.059 DBMET00498

0.121 0.02 DB11100

DBMET00499
0.2790.010.408Protein kinase (Mos, Mil/Raf, MEKK, RIPK, TESK, LIMK, IRAK, ILK, Activin/TGF-beta) inhibitor

0.408 0.005 DBMET00499

DBMET00499
0.2690.0050.311Phosphodiesterase 7B inhibitor

0.311 0.004 DBMET00499

DBMET00499
0.2710.010.556Xanthine oxidase inhibitor

0.306 0.007 DBMET00499

0.556 0.003 DBMET00498

DBMET00498
0.2690.0080.269CDK2/cyclin A inhibitor

0.115 0.046 DBMET00499

0.3330.0780.333Angiogenesis inhibitor
0.2590.0050.259DNA repair enzyme inhibitor

0.237 0.006 DBMET00499

0.199 0.009 DBMET00498

0.2540.0010.254Purine nucleoside phosphorylase inhibitor

0.035 0.002 DBMET00499

0.021 0.003 DBMET00498

0.2650.0150.265Cyclin-dependent kinase 2 inhibitor

0.159 0.034 DBMET00499

0.2570.0080.456NADH dehydrogenase inhibitor

0.456 0.004 DBMET00499

0.223 0.009 DBMET00498

0.118 0.03 DB11100

DBMET00499
0.2690.0240.269Cyclin-dependent kinase inhibitor

0.155 0.054 DBMET00499

0.2510.0070.319Adenosine A2 receptor antagonist

0.319 0.005 DBMET00499

0.068 0.041 DBMET00498

DBMET00499
0.2410.0050.241Phenylalanine 4-hydroxylase inhibitor

0.082 0.036 DBMET00499

0.126 0.016 DBMET00498

0.2380.0050.974Phosphodiesterase III inhibitor

0.736 0.002 DBMET00499

0.974 0.001 DBMET00498

DBMET00498
0.2350.0040.235Myeloperoxidase inhibitor

0.115 0.022 DBMET00499

0.2320.0020.232Thymidine kinase inhibitor

0.189 0.003 DBMET00499

0.098 0.006 DBMET00498

0.037 0.035 DB11100

0.3270.0990.327Immunosuppressant
0.2940.0680.692Aldehyde oxidase inhibitor

0.692 0.009 DBMET00499

0.178 0.118 DB11100

DBMET00499
0.3590.1340.5DNA directed DNA polymerase inhibitor

0.328 0.149 DBMET00499

0.5 0.082 DBMET00498

DBMET00498
0.2540.0350.254Src kinase inhibitor

0.181 0.064 DBMET00499

0.3410.1230.3415 Hydroxytryptamine release inhibitor

0.243 0.238 DBMET00499

0.2270.010.383Raf kinase inhibitor

0.383 0.005 DBMET00499

DBMET00499
0.2250.0080.308Phosphodiesterase I inhibitor

0.308 0.005 DBMET00499

0.12 0.027 DBMET00498

0.131 0.022 DB11100

DBMET00499
0.2580.0460.294Peroxidase inhibitor

0.136 0.086 DBMET00499

0.142 0.082 DBMET00498

0.294 0.038 DB11100

DB11100
0.2320.0210.346Adenylate cyclase inhibitor

0.346 0.01 DBMET00499

DBMET00499
0.2380.0270.238c-Src kinase inhibitor

0.195 0.037 DBMET00499

0.2590.0550.266Ca2+/calmodulin-dependent kinase IV inhibitor

0.249 0.067 DBMET00499

0.266 0.048 DBMET00498

DBMET00498
0.2330.030.233Protein kinase (CK1) inhibitor

0.149 0.068 DBMET00499

0.260.0630.26Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor

0.215 0.084 DBMET00499

0.2020.0070.202Mannitol-1-phosphate 5-dehydrogenase inhibitor

0.182 0.007 DBMET00499

0.136 0.009 DBMET00498

0.064 0.031 DB11100

0.2150.0220.215Protein kinase (CK2) alpha inhibitor

0.116 0.064 DBMET00499

0.2010.0090.201Antimetabolite

0.191 0.01 DBMET00499

0.168 0.011 DBMET00498

0.05 0.031 DB11100

0.1970.0090.348Adenosine A3 receptor antagonist

0.348 0.004 DBMET00499

0.148 0.013 DBMET00498

DBMET00499
0.1960.010.248Adenosine A2a receptor antagonist

0.248 0.007 DBMET00499

0.065 0.04 DBMET00498

DBMET00499
0.2530.070.253Dyrk kinase inhibitor

0.214 0.091 DBMET00499

0.1890.0070.189Cyclin B3 inhibitor
0.1860.0090.2Argininosuccinate synthase inhibitor

0.2 0.008 DBMET00499

0.064 0.034 DBMET00498

0.077 0.026 DB11100

DBMET00499
0.1820.0050.224Phosphodiesterase 4C inhibitor

0.144 0.008 DBMET00499

0.224 0.005 DBMET00498

0.117 0.011 DB11100

DBMET00498
0.1990.0220.199CF transmembrane conductance regulator agonist

0.171 0.046 DBMET00499

0.2160.040.2275 Hydroxytryptamine 3E antagonist

0.227 0.03 DBMET00499

DBMET00499
0.1980.0290.198MAP kinase kinase inhibitor

0.166 0.043 DBMET00499

0.1710.0020.171AICAR transformylase inhibitor

0.147 0.003 DBMET00499

0.072 0.009 DBMET00498

0.1680.0010.168Hypoxanthine phosphoribosyltransferase inhibitor

0.133 0.001 DBMET00499

0.07 0.006 DBMET00498

0.029 0.018 DB11100

0.1760.0110.176Cyclin A2 inhibitor

0.065 0.043 DBMET00499

0.1890.0250.189Cyclin-dependent kinase 5 inhibitor

0.124 0.055 DBMET00499

0.1670.0030.167Dihydropteroate synthase inhibitor

0.059 0.012 DBMET00498

0.1840.0260.186Ferrochelatase inhibitor

0.159 0.034 DBMET00499

0.146 0.039 DBMET00498

0.186 0.026 DB11100

DB11100
0.260.1070.439Immunomodulator

0.192 0.174 DBMET00499

0.439 0.034 DBMET00498

DBMET00498
0.1650.0130.165Glutamate dehydrogenase inhibitor

0.139 0.018 DBMET00499

0.081 0.043 DBMET00498

0.097 0.032 DB11100

0.1620.0120.162MAP kinase kinase 1 inhibitor

0.114 0.041 DBMET00499

0.103 0.053 DBMET00498

0.2810.1340.281Histamine release inhibitor

0.28 0.135 DBMET00499

0.1810.0360.181Protein kinase (CK1) delta inhibitor
0.1490.0050.207Nicotinic acid receptor 1 agonist

0.207 0.004 DBMET00499

DBMET00499
0.1560.0120.192Proto-oncogene tyrosine-protein kinase c-hck inhibitor

0.192 0.006 DBMET00499

DBMET00499
0.1510.0090.151mTOR complex 2 inhibitor

0.09 0.047 DBMET00499

0.1590.020.159TIE-2 antagonist
0.1510.0130.151Cyclin A inhibitor

0.055 0.048 DBMET00499

0.1590.0210.159TIE antagonist
0.1590.0230.163Adenylate kinase inhibitor

0.163 0.022 DBMET00499

0.122 0.042 DBMET00498

0.144 0.029 DB11100

DBMET00499
0.1460.0120.199Carbamoyl phosphate synthetase inhibitor

0.199 0.007 DBMET00499

0.109 0.018 DBMET00498

0.132 0.014 DB11100

DBMET00499
0.1530.020.153Telomerase inhibitor
0.1440.0120.144Phosphatidylinositol 3-kinase delta inhibitor

0.073 0.028 DBMET00499

0.150.0190.15Phosphodiesterase 4D inhibitor

0.138 0.022 DBMET00499

0.094 0.04 DBMET00498

0.133 0.023 DB11100

0.1970.070.197Tyrosine kinase inhibitor
0.1630.0370.163Aurora-C kinase inhibitor
0.1490.0240.168DNA directed RNA polymerase inhibitor

0.168 0.019 DBMET00499

0.095 0.063 DBMET00498

DBMET00499
0.1280.0030.128Adenosine deaminase inhibitor

0.085 0.008 DBMET00499

0.061 0.02 DBMET00498

0.1470.0230.156GABA C receptor rho-1 antagonist

0.156 0.019 DBMET00499

0.091 0.076 DBMET00498

DBMET00499
0.150.0270.15CDK3/cyclin E inhibitor
0.1270.0060.127Histamine agonist

0.05 0.039 DBMET00499

0.1720.0510.28RET inhibitor

0.28 0.026 DBMET00499

DBMET00499
0.1540.0330.154MAP kinase kinase kinase inhibitor

0.112 0.056 DBMET00499

0.1520.0320.214Protein kinase (CK2) inhibitor

0.214 0.016 DBMET00499

DBMET00499
0.1270.0070.973Phosphodiesterase 3B inhibitor

0.266 0.004 DBMET00499

0.973 0.001 DBMET00498

DBMET00498
0.1880.0690.202LIM domain kinase 1 inhibitor

0.202 0.062 DBMET00499

DBMET00499
0.1210.0040.121Thymidylate synthase inhibitor

0.075 0.009 DBMET00499

0.081 0.007 DBMET00498

0.1950.0780.195Proto-oncogene tyrosine-protein kinase Fyn inhibitor

0.144 0.143 DBMET00499

0.1520.0360.152Death-associated protein kinase 1 inhibitor

0.143 0.052 DBMET00498

0.1340.0170.134mTOR complex 1 inhibitor

0.12 0.029 DBMET00499

0.1340.0190.487Phosphodiesterase 3A inhibitor

0.185 0.01 DBMET00499

0.487 0.003 DBMET00498

DBMET00498
0.1230.0080.332Adenosine A2b receptor antagonist

0.332 0.003 DBMET00499

0.045 0.04 DBMET00498

DBMET00499
0.2180.1040.218Interleukin agonist
0.1620.0480.162Tyrosine-protein kinase receptor FLT3 inhibitor
0.1710.0570.171Protein-tyrosine kinase Lyn inhibitor

0.139 0.072 DBMET00499

0.130.0170.142Alpha 2d adrenoreceptor antagonist

0.142 0.011 DBMET00499

DBMET00499
0.1630.050.805Phosphodiesterase inhibitor

0.625 0.004 DBMET00499

0.805 0.004 DBMET00498

DBMET00498
0.140.0270.14Protein kinase A inhibitor

0.077 0.063 DBMET00499

0.1910.0790.191I kappa B kinase epsilon inhibitor
0.1660.0550.195GABA C receptor rho-2 antagonist

0.195 0.032 DBMET00499

0.14 0.087 DBMET00498

DBMET00499
0.1440.0330.152GABA C receptor antagonist

0.152 0.029 DBMET00499

0.124 0.049 DBMET00498

DBMET00499
0.1460.0350.146Nav1.4 sodium channel blocker
0.1150.0050.115Histamine H3 receptor agonist

0.102 0.006 DBMET00499

0.120.0110.295Xanthine dehydrogenase inhibitor

0.154 0.007 DBMET00499

0.295 0.003 DBMET00498

DBMET00498
0.1130.0070.113Factor IXa inhibitor
0.1220.0180.237Phosphodiesterase V inhibitor

0.237 0.005 DBMET00499

0.209 0.005 DBMET00498

DBMET00499
0.1260.0230.142Phosphofructokinase-1 inhibitor

0.142 0.02 DBMET00499

0.083 0.039 DBMET00498

0.074 0.045 DB11100

DBMET00499
0.1960.0930.196Ca2+/calmodulin-dependent kinase I alpha inhibitor

0.177 0.111 DB11100

0.1490.0470.149Alkylator

0.128 0.061 DBMET00499

0.1070.0050.107CDK5/p25 inhibitor

0.042 0.027 DBMET00499

0.1650.0650.301Diuretic

0.301 0.022 DBMET00499

DBMET00499
0.1080.0080.108MAP kinase kinase 7 inhibitor

0.085 0.034 DBMET00499

0.081 0.044 DBMET00498

0.1140.0150.232Biliverdin reductase inhibitor

0.232 0.004 DBMET00499

0.129 0.012 DBMET00498

0.112 0.015 DB11100

DBMET00499
0.1430.0470.296MAP kinase 12 inhibitor

0.296 0.007 DBMET00499

0.166 0.034 DBMET00498

DBMET00499
0.1060.010.106S-adenosyl-L-methionine decarboxylase inhibitor

0.078 0.04 DBMET00499

0.0970.0020.097Thymidine kinase (Herpes simplex virus 1) inhibitor

0.078 0.003 DBMET00499

0.047 0.004 DBMET00498

0.1560.0620.156Lck kinase inhibitor

0.103 0.099 DBMET00499

0.1170.0240.117Hematopoietic
0.0970.0040.097Histamine H2 receptor agonist

0.058 0.016 DBMET00499

0.1350.0430.135Platelet activating factor beta antagonist

0.085 0.075 DBMET00499

0.1090.0190.109CDC7 inhibitor

0.069 0.045 DBMET00499

0.1290.0410.129Cyclin-dependent kinase 9 inhibitor
0.1040.020.104MAP3K7 inhibitor
0.0990.0160.1Ornithine carbamoyltransferase inhibitor

0.1 0.016 DBMET00499

0.047 0.043 DBMET00498

0.073 0.024 DB11100

DBMET00499
0.1190.0370.123Electrolyte absorption antagonist

0.113 0.043 DBMET00499

0.123 0.034 DB11100

DB11100
0.1490.0680.194Glycogen synthase kinase-3 alpha inhibitor

0.194 0.043 DBMET00499

DBMET00499
0.2150.1340.215Hypoxia-inducible factor 1 alpha inhibitor

0.188 0.167 DBMET00499

0.0950.0180.095Acyl-CoA dehydrogenase inhibitor

0.081 0.022 DBMET00499

0.049 0.043 DBMET00498

0.0960.020.096Carbonic anhydrase stimulant

0.059 0.041 DBMET00499

0.20.1230.2MAP kinase kinase 3 inhibitor
0.1910.1160.223MAP-kinase-activated kinase 5 inhibitor

0.223 0.08 DBMET00499

DBMET00499
0.1120.0370.112Interleukin 12 antagonist
0.1010.0280.112Interferon agonist

0.112 0.021 DBMET00498

DBMET00498
0.0990.0260.12Protein kinase B beta inhibitor

0.12 0.015 DBMET00499

0.069 0.058 DBMET00498

DBMET00499
0.0980.0280.232Phosphodiesterase 5A inhibitor

0.232 0.005 DBMET00499

0.211 0.005 DBMET00498

DBMET00499
0.0960.0280.096T cell inhibitor
0.120.0520.12Protein kinase C gamma inhibitor
0.0720.0060.072Dihydrofolate reductase inhibitor
0.0960.0290.096CDK2/cyclin E2 inhibitor
0.0850.0190.085Phosphodiesterase 4A inhibitor

0.085 0.019 DBMET00499

0.0840.0230.128Phosphodiesterase VII inhibitor

0.128 0.005 DBMET00499

DBMET00499
0.0820.0220.096Interferon inducer

0.096 0.014 DBMET00498

DBMET00498
0.1880.1280.32Immunostimulant

0.159 0.147 DBMET00499

0.32 0.073 DBMET00498

DBMET00498
0.1030.0430.103Histamine N-methyltransferase inhibitor

0.077 0.07 DBMET00499

0.0620.0020.062Phosphoribosylglycinamide formyltransferase inhibitor

0.007 0.006 DBMET00498

0.1410.0810.141MAP kinase kinase 4 inhibitor
0.1160.0560.116Aurora-A kinase inhibitor
0.1240.0650.124Protein-tyrosine kinase (PTK, not ETK, WZC) inhibitor
0.1240.0650.124Abl kinase inhibitor
0.1680.1110.244Glyceraldehyde-3-phosphate dehydrogenase inhibitor

0.222 0.057 DBMET00499

0.244 0.045 DBMET00498

DBMET00498
0.0580.0040.058Histamine H4 receptor agonist
0.0670.0140.067Histamine H4 receptor antagonist
0.0730.0210.117Phosphodiesterase 1A inhibitor

0.117 0.007 DBMET00499

0.062 0.036 DB11100

DBMET00499
0.0660.0140.067Alpha 1b adrenoreceptor agonist

0.067 0.014 DBMET00499

DBMET00499
0.0870.0350.087Syk tyrosine kinase inhibitor
0.1750.1240.175ErbB-1 antagonist
0.0720.0220.394Phosphodiesterase II inhibitor

0.117 0.008 DBMET00499

0.394 0.002 DBMET00498

DBMET00498
0.0870.0380.087Histidine decarboxylase inhibitor

0.079 0.043 DBMET00499

0.074 0.047 DB11100

0.1610.1120.161MAP kinase kinase 5 inhibitor
0.1570.1080.199Clk dual-specificity kinase inhibitor

0.199 0.08 DBMET00499

DBMET00499
0.1340.0860.149MAP3K9 inhibitor

0.149 0.061 DBMET00499

DBMET00499
0.0570.010.057Histamine H1 receptor agonist

0.053 0.015 DBMET00499

0.1310.0850.131CDC-like kinase 1 inhibitor
0.1590.1130.159MAP kinase kinase 2 inhibitor

0.158 0.114 DBMET00499

0.0720.0260.072Cyclin H inhibitor
0.0450.0040.091DNA polymerase III inhibitor

0.062 0.003 DBMET00499

0.091 0.002 DBMET00498

DBMET00498
0.080.0420.08GABA B receptor agonist
0.0990.0610.099Nitric-oxide synthase inhibitor
0.060.0230.06Carbonic anhydrase II stimulant

0.054 0.032 DBMET00499

0.070.0340.371Raf kinase B inhibitor

0.371 0.005 DBMET00499

DBMET00499
0.0980.0620.098Creatine kinase inhibitor
0.0450.0090.069Phosphodiesterase 6B inhibitor

0.069 0.004 DBMET00499

0.069 0.004 DBMET00498

DBMET00498
0.0490.0140.058Fumarate hydratase inhibitor

0.058 0.011 DBMET00499

0.033 0.026 DB11100

DBMET00499
0.1060.0710.151Polo-like kinase-4 inhibitor

0.151 0.035 DBMET00499

DBMET00499
0.2080.1750.235Vasodilator, coronary

0.235 0.149 DBMET00499

DBMET00499
0.1130.080.113Epidermal growth factor receptor kinase inhibitor
0.0580.0250.385Phosphodiesterase 2A inhibitor

0.096 0.009 DBMET00499

0.385 0.002 DBMET00498

DBMET00498
0.1230.0930.123Activin receptor-like kinase 2 inhibitor
0.0920.0620.13Alcohol dehydrogenase inhibitor

0.13 0.029 DBMET00499

DBMET00499
0.0460.0160.046Phosphoglycerate kinase inhibitor

0.033 0.027 DBMET00499

0.050.0210.074Phosphodiesterase 6C inhibitor

0.064 0.006 DBMET00499

0.074 0.004 DBMET00498

DBMET00498
0.0370.0080.037Purinergic P2Y15 antagonist

0.033 0.012 DBMET00499

0.028 0.02 DBMET00498

0.0330.0040.066Thymidine kinase (Herpes simplex virus 2) inhibitor

0.066 0.002 DBMET00499

0.034 0.004 DBMET00498

DBMET00499
0.0490.0220.105Glutamate (mGluR4) antagonist

0.105 0.005 DBMET00499

DBMET00499
0.0930.0690.196UDP-glucose 4-epimerase inhibitor

0.196 0.019 DBMET00499

0.116 0.046 DBMET00498

0.143 0.031 DB11100

DBMET00499
0.0450.020.057Alpha 1d adrenoreceptor agonist

0.057 0.012 DBMET00499

DBMET00499
0.0330.010.157Thymidine phosphorylase inhibitor

0.11 0.003 DBMET00499

0.157 0.002 DBMET00498

0.049 0.005 DB11100

DBMET00498
0.0430.0210.043MAP3K5 inhibitor
0.0620.040.062Alpha 2 adrenoreceptor agonist
0.030.0090.035Alpha 2d adrenoreceptor agonist

0.035 0.007 DBMET00499

DBMET00499
0.0570.0380.106Alcohol oxidase inhibitor

0.082 0.023 DBMET00499

0.053 0.042 DBMET00498

0.106 0.017 DB11100

DB11100
0.060.0410.06Raf kinase C inhibitor
0.0230.0040.023CDK2/cyclin A3 inhibitor
0.0410.0230.041Diamine oxidase inhibitor
0.0360.0180.036Potassium channel small-conductance Ca-activated activator
0.0830.0660.083Granulocyte macrophage colony stimulating factor agonist
0.060.0430.143Purinergic P2X1 antagonist

0.083 0.023 DBMET00499

0.143 0.008 DBMET00498

DBMET00498
0.0860.0690.086Fibroblast growth factor 1 antagonist
0.190.1730.205Insulysin inhibitor

0.205 0.149 DBMET00499

DBMET00499
0.0790.0620.079AXL receptor tyrosine kinase inhibitor
0.0670.0510.08Exportin-1 inhibitor

0.08 0.025 DBMET00499

DBMET00499
0.0630.0480.063Fibroblast growth factor 2 antagonist
0.0980.0840.098Vascular endothelial growth factor antagonist
0.0360.0230.041Tryptophan 5 hydroxylase inhibitor

0.034 0.032 DBMET00499

0.041 0.014 DBMET00498

DBMET00498
0.0170.0040.031DNA polymerase III polC-type inhibitor

0.031 0.003 DBMET00499

DBMET00499
0.0790.0670.081Histamine H2 receptor antagonist

0.081 0.063 DB11100

DB11100
0.0130.0030.035DNA polymerase III subunit alpha inhibitor

0.018 0.002 DBMET00499

0.035 0.001 DBMET00498

DBMET00498
0.0310.0210.031Endothelial nitric-oxide synthase inhibitor
0.0190.010.019Granulocyte colony stimulating factor receptor agonist
0.020.0110.02Alpha 2c adrenoreceptor agonist
0.1240.1150.144Adenylate cyclase stimulant

0.144 0.073 DBMET00499

0.128 0.105 DBMET00498

DBMET00499
0.0240.0150.034Phosphodiesterase 6A inhibitor

0.034 0.005 DBMET00499

0.028 0.008 DBMET00498

DBMET00499
0.0340.0250.034Purinergic P2X3 antagonist
0.0320.0240.032ATR kinase inhibitor
0.110.1030.11Growth factor antagonist
0.0190.0120.019Methylmalonyl-CoA mutase inhibitor

0.017 0.015 DBMET00499

0.0230.0170.04Phosphodiesterase 6H inhibitor

0.031 0.007 DBMET00499

0.04 0.004 DBMET00498

DBMET00498
0.0230.0170.04Phosphodiesterase 6G inhibitor

0.031 0.007 DBMET00499

0.04 0.004 DBMET00498

DBMET00498
0.0630.0570.063Protein kinase B alpha inhibitor
0.1030.0980.203Alpha-N-acetylglucosaminidase inhibitor

0.133 0.066 DBMET00499

0.203 0.033 DBMET00498

0.159 0.05 DB11100

DBMET00498
0.0090.0040.019DNA topoisomerase III inhibitor

0.011 0.003 DBMET00499

0.019 0.002 DBMET00498

0.008 0.004 DB11100

DBMET00498
0.0170.0120.017Tryptophan hydroxylase 1 inhibitor
0.0550.050.134Phosphodiesterase 1B inhibitor

0.134 0.008 DBMET00499

0.068 0.032 DBMET00498

DBMET00499
0.0580.0530.058Purinergic P2X2 antagonist
0.0630.0590.063Janus tyrosine kinase 3 inhibitor
0.0170.0130.017Adenosine A3 receptor agonist
0.0180.0150.018Alpha 2b adrenoreceptor agonist
0.0750.0730.075Epidermal growth factor antagonist
0.010.0080.01Purinergic P2Y2 agonist
0.0490.0470.049Bruton tyrosine kinase inhibitor
0.020.0180.031Glutaminyl-peptide cyclotransferase inhibitor

0.031 0.006 DBMET00499

DBMET00499
0.0330.0320.033Carbonic anhydrase I stimulant
0.040.040.055Glutamate (mGluR group III) antagonist

0.055 0.016 DBMET00499

DBMET00499
0.0630.0640.072Porphobilinogen synthase inhibitor

0.072 0.054 DBMET00499

DBMET00499
0.030.0350.059Protein kinase (CK2) beta inhibitor

0.059 0.005 DBMET00499

0.031 0.028 DBMET00498

0.032 0.026 DB11100

DBMET00499
0.0090.0140.024Egl nine homolog 2 inhibitor

0.024 0.004 DBMET00499

DBMET00499
0.1270.1360.132Ca2+-transporting ATPase inhibitor

0.13 0.122 DBMET00499

0.132 0.108 DBMET00498

DBMET00498
0.0410.0520.05mTOR inhibitor

0.05 0.038 DBMET00499

DBMET00499
0.0540.0680.089Phosphodiesterase 1C inhibitor

0.089 0.014 DBMET00499

0.082 0.018 DBMET00498

0.064 0.039 DB11100

DBMET00499
0.0720.0910.158HIV-1 integrase (Overall Integration) inhibitor

0.158 0.022 DBMET00498

DBMET00498
0.090.1110.13Nav1.3 sodium channel blocker

0.13 0.064 DBMET00499

DBMET00499
0.0070.0290.031Egl nine homolog 3 inhibitor

0.031 0.003 DBMET00499

0.025 0.004 DBMET00498

DBMET00499
0.1120.140.262Interleukin-1 receptor-associated protein kinase 1 inhibitor

0.262 0.044 DBMET00499

DBMET00499
0.0770.1060.097Granulocyte macrophage colony stimulating factor antagonist

0.097 0.075 DBMET00499

DBMET00499
0.0490.080.076Corticotropin releasing factor 2 receptor antagonist

0.076 0.021 DBMET00499

DBMET00499
0.0590.0950.086Phosphodiesterase VI inhibitor

0.086 0.033 DBMET00499

DBMET00499
0.020.0570.082Nicotinic acid receptor agonist

0.082 0.006 DBMET00499

DBMET00499
0.0050.0510.019Egl nine homolog 1 inhibitor

0.018 0.006 DBMET00499

0.019 0.006 DBMET00498

DBMET00498
0.0240.0730.034Transforming growth factor beta 2 antagonist

0.034 0.021 DBMET00499

DBMET00499
0.0510.10.203Protein kinase B gamma inhibitor

0.076 0.051 DBMET00499

0.203 0.008 DBMET00498

DBMET00498
0.0880.1390.117Protein kinase (CK1) gamma inhibitor

0.117 0.093 DBMET00499

DBMET00499
0.0660.1170.105Ephrin antagonist

0.105 0.059 DBMET00499

DBMET00499
0.0660.1190.318Uric acid excretion stimulant

0.222 0.01 DBMET00499

0.318 0.005 DBMET00498

DBMET00498
0.2050.260.31MAP kinase kinase 6 inhibitor

0.31 0.126 DBMET00498

DBMET00498
0.1630.2180.215Tyrosine 3 hydroxylase inhibitor

0.215 0.11 DBMET00498

0.189 0.157 DB11100

DBMET00498
0.050.1050.191Phosphodiesterase IV inhibitor

0.191 0.014 DBMET00499

0.117 0.034 DBMET00498

0.084 0.057 DB11100

DBMET00499
0.1010.1570.144Cyclin-dependent kinase 8 inhibitor

0.144 0.086 DBMET00499

DBMET00499
0.0330.0890.052EphB4 antagonist

0.052 0.047 DBMET00499

DBMET00499
0.0990.1570.18CDC-like kinase 4 inhibitor

0.18 0.079 DBMET00499

DBMET00499
0.1280.1920.572Vasodilator

0.572 0.007 DBMET00499

DBMET00499
0.060.1260.083Pim-3 kinase inhibitor

0.083 0.071 DBMET00499

DBMET00499
0.1360.2120.262Superoxide dismutase inhibitor

0.195 0.123 DBMET00499

0.262 0.067 DB11100

DB11100
0.0740.1510.094DOPA decarboxylase inhibitor

0.094 0.089 DBMET00498

DBMET00498
0.0890.1660.123Cell wall synthesis inhibitor

0.117 0.103 DBMET00499

0.123 0.095 DB11100

DB11100
0.1090.1880.165Ca2+/calmodulin-dependent protein kinase inhibitor

0.165 0.099 DBMET00499

DBMET00499
0.0290.110.044Glucose-6-phosphate isomerase inhibitor

0.044 0.04 DBMET00498

DBMET00498
0.0150.0960.026Acid ceramidase inhibitor

0.026 0.017 DBMET00499

DBMET00499
0.0510.1340.095Aminopeptidase B inhibitor

0.095 0.069 DB11100

DB11100
0.0790.170.194Cytidine deaminase inhibitor

0.155 0.072 DBMET00499

0.194 0.05 DBMET00498

DBMET00498
0.0570.1490.086Triose-phosphate isomerase inhibitor

0.086 0.065 DB11100

DB11100
0.0260.1180.049Kainate receptor agonist

0.039 0.035 DBMET00498

0.049 0.014 DB11100

DB11100
0.060.1530.125 Hydroxytryptamine 3A agonist

0.12 0.055 DB11100

DB11100
0.030.1270.118HIV-1 reverse transcriptase inhibitor

0.118 0.023 DBMET00498

DBMET00498
0.1110.2070.161Succinate dehydrogenase inhibitor

0.161 0.093 DBMET00498

DBMET00498
0.0580.1570.115M18 aspartyl aminopeptidase inhibitor

0.115 0.075 DBMET00499

DBMET00499
0.1980.2970.458MAP kinase 1 inhibitor

0.25 0.233 DBMET00499

0.458 0.073 DBMET00498

DBMET00498
0.0150.1170.053Inosine monophosphate dehydrogenase inhibitor

0.053 0.013 DBMET00498

DBMET00498
0.0270.1310.055Aconitate hydratase inhibitor

0.055 0.031 DB11100

DB11100
0.0240.1320.043CC chemokine 4 receptor antagonist

0.043 0.04 DBMET00499

DBMET00499
0.0890.2010.193Polo-like kinase-3 inhibitor

0.193 0.049 DBMET00499

DBMET00499
0.0450.1580.106MAP-kinase-activated kinase inhibitor

0.106 0.034 DBMET00499

DBMET00499
0.0530.1720.134UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor

0.099 0.055 DBMET00499

0.134 0.032 DB11100

DB11100
0.0070.1260.056Uridine phosphorylase inhibitor

0.033 0.015 DBMET00499

0.056 0.006 DBMET00498

0.04 0.012 DB11100

DBMET00498
0.0340.1570.073Sirtuin 1 inhibitor

0.073 0.041 DBMET00499

DBMET00499
0.0340.1590.081Phospholipase D inhibitor

0.073 0.048 DBMET00499

0.081 0.033 DBMET00498

DBMET00498
0.0320.1580.083Glutamate decarboxylase inhibitor

0.083 0.041 DB11100

DB11100
0.0630.190.1Phosphodiesterase 6D inhibitor

0.1 0.053 DBMET00499

DBMET00499
0.0670.1980.119Protein kinase C nu inhibitor

0.119 0.094 DBMET00499

DBMET00499
0.0150.1510.046Glutamate (mGluR3) antagonist

0.046 0.015 DBMET00498

DBMET00498
0.0520.1890.38Proto-oncogene tyrosine-protein kinase Yes inhibitor

0.38 0.009 DBMET00498

DBMET00498
0.070.210.103Interleukin 8 antagonist

0.103 0.09 DBMET00499

DBMET00499
0.0090.1610.032Nicotinic acid receptor 2 antagonist

0.032 0.011 DBMET00499

DBMET00499
0.0140.1680.042Stearoyl-CoA desaturase inhibitor

0.042 0.033 DBMET00499

DBMET00499
0.0320.190.083MAP-kinase-activated kinase 2 inhibitor

0.083 0.041 DBMET00499

DBMET00499
0.0290.1890.062Dihydroorotate oxidase inhibitor

0.062 0.026 DBMET00499

0.061 0.027 DB11100

DBMET00499
0.0490.2120.088Polo-like kinase-1 inhibitor

0.088 0.065 DBMET00499

DBMET00499
0.020.1880.076GABA A receptor antagonist

0.076 0.023 DBMET00498

DBMET00498
0.0080.1780.165Somatostatin 4 antagonist

0.165 0.004 DB11100

DB11100
0.0210.1910.214Purinergic P2 antagonist

0.055 0.053 DBMET00499

0.214 0.006 DBMET00498

DBMET00498
0.010.1810.126AMPA receptor antagonist

0.059 0.025 DBMET00499

0.126 0.008 DBMET00498

DBMET00498
0.0730.2470.123Hexokinase inhibitor

0.123 0.114 DBMET00499

DBMET00499
0.0180.1970.075GABA receptor antagonist

0.075 0.024 DBMET00498

DBMET00498
0.0270.2090.063NMDA receptor agonist

0.063 0.043 DB11100

DB11100
0.0140.1990.058Dihydroorotate dehydrogenase inhibitor

0.058 0.03 DBMET00499

DBMET00499
0.0160.2070.073NMDA receptor glycine site agonist

0.073 0.034 DB11100

DB11100
0.0410.2320.128Cystathionine beta-synthase inhibitor

0.128 0.052 DBMET00498

DBMET00498
0.0510.2450.138Ca2+/calmodulin-dependent kinase II delta inhibitor

0.138 0.072 DBMET00499

DBMET00499
0.0050.2040.086Calcitonin gene-related peptide antagonist

0.086 0.003 DBMET00499

0.066 0.005 DBMET00498

0.073 0.004 DB11100

DBMET00499
0.0230.2460.057I kappa B kinase 2 inhibitor

0.057 0.054 DB11100

DB11100
0.0780.3090.421Prostaglandin dehydrogenase inhibitor

0.421 0.061 DBMET00498

DBMET00498
0.0730.3080.275Tumour necrosis factor antagonist

0.231 0.037 DBMET00499

0.275 0.024 DB11100

DB11100
0.070.3050.429Growth hormone agonist

0.204 0.057 DBMET00499

0.429 0.012 DB11100

DB11100
0.0050.2460.118Calcitonin gene-related peptide 1 receptor antagonist

0.118 0.003 DBMET00499

0.115 0.004 DBMET00498

0.114 0.004 DB11100

DBMET00499
0.0570.3080.146Mannose-6-phosphate isomerase inhibitor

0.146 0.068 DBMET00498

DBMET00498
0.0050.2620.208Somatostatin 2 antagonist

0.208 0.004 DB11100

DB11100
0.0190.280.137NMDA receptor antagonist

0.137 0.029 DBMET00498

DBMET00498
0.0070.2840.088Purinergic P2Y antagonist

0.052 0.025 DBMET00499

0.088 0.011 DBMET00498

DBMET00498
0.0760.3550.123Sphingosine 1-phosphate receptor 5 antagonist

0.123 0.118 DBMET00498

DBMET00498
0.0050.2980.041NMDA receptor subunit 3A antagonist

0.041 0.024 DBMET00498

DBMET00498
0.0450.3390.313Anesthetic general

0.135 0.131 DBMET00499

0.313 0.03 DB11100

DB11100
0.0230.3290.064Glucosylceramidase inhibitor

0.064 0.026 DBMET00498

DBMET00498
0.050.360.23Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase inhibitor

0.23 0.085 DBMET00498

DBMET00498
0.0280.340.515Keratolytic

0.515 0.002 DB11100

DB11100
0.0070.3410.062NMDA receptor subunit 3B antagonist

0.062 0.018 DBMET00498

DBMET00498
0.0080.350.033Somatostatin agonist

0.033 0.021 DB11100

DB11100
0.0750.4240.324Gastrin inhibitor

0.324 0.019 DB11100

DB11100
0.070.430.35115-Lipoxygenase inhibitor

0.351 0.099 DBMET00498

DBMET00498
0.0550.430.31DNA polymerase beta inhibitor

0.31 0.16 DBMET00498

DBMET00498
0.0310.4070.086Bromodomain-containing protein 2 inhibitor

0.086 0.064 DBMET00499

0.08 0.076 DB11100

DBMET00499
0.0520.4360.186Thyroid hormone antagonist

0.186 0.174 DBMET00498

DBMET00498
0.0510.4460.41Cardiotonic

0.41 0.027 DBMET00499

0.215 0.106 DB11100

DBMET00499
0.0070.4060.06Somatostatin 1 antagonist

0.06 0.015 DB11100

DB11100
0.0040.410.672Purinergic P2Y12 antagonist

0.055 0.006 DBMET00499

0.672 0.002 DBMET00498

DBMET00498
0.050.4580.178Thyroid hormone beta antagonist

0.178 0.175 DBMET00498

DBMET00498
0.0050.4140.08Nicotinic acid receptor 2 agonist

0.08 0.008 DBMET00499

DBMET00499
0.0220.4460.148AMP-activated protein kinase stimulant

0.148 0.029 DBMET00498

DBMET00498
0.0050.4350.089Somatostatin 3 antagonist

0.089 0.004 DB11100

DB11100
0.0340.4730.17Platelet aggregation inhibitor

0.17 0.107 DBMET00499

DBMET00499
0.0320.4720.245Interleukin antagonist

0.245 0.064 DBMET00498

DBMET00498
0.0170.4620.086Caspase 7 inhibitor

0.086 0.049 DBMET00498

DBMET00498
0.0830.5740.26Peptidyltransferase inhibitor

0.26 0.044 DBMET00499

0.24 0.058 DB11100

DBMET00499
0.0180.5220.333Somatostatin 1 agonist

0.333 0.002 DB11100

DB11100
0.0260.5580.165Interleukin 5 antagonist

0.165 0.008 DBMET00498

DBMET00498
0.030.5970.565Interleukin 4 antagonist

0.565 0.004 DBMET00498

DBMET00498
0.0080.6080.188Glutamate receptor antagonist

0.188 0.03 DBMET00498

DBMET00498
0.0210.6280.115Interleukin 1 antagonist

0.115 0.096 DBMET00498

DBMET00498
0.0130.6540.248Alpha-glucosidase inhibitor

0.248 0.188 DBMET00498

DBMET00498
0.0030.6650.027Kainate receptor 4 antagonist

0.027 0.016 DBMET00498

DBMET00498
0.0020.7770.909Cholecystokinin B antagonist

0.909 0.001 DB11100

DB11100
0.0030.7960.925Cholecystokinin A antagonist

0.925 0.001 DB11100

DB11100
0.0060.8060.314Potassium channel blocker

0.314 0.042 DB11100

DB11100
0.0030.8630.946Cholecystokinin antagonist

0.946 0.001 DB11100

DB11100
0.0070.8690.31Streptokinase A inhibitor

0.31 0.075 DBMET00498

DBMET00498
0.0040.8670.047Bromodomain-containing protein 3 inhibitor

0.047 0.039 DB11100

DB11100
0.0020.8780.015Thyroid hormone alpha agonist

0.015 0.014 DB11100

DB11100
0.0080.8930.142Interleukin 6 antagonist

0.142 0.101 DB11100

DB11100
0.0050.8970.113M17 leucyl aminopeptidase inhibitor

0.113 0.084 DBMET00498

DBMET00498
0.0040.9180.06Mineralocorticoid receptor antagonist

0.06 0.02 DB11100

DB11100
0.0020.9190.048Somatostatin 5 antagonist

0.048 0.014 DB11100

DB11100
0.0050.9220.367Thioredoxin glutathione reductase inhibitor

0.367 0.07 DBMET00498

DBMET00498
0.0020.9320.049Cholecystokinin agonist

0.049 0.007 DB11100

DB11100
0.0020.9480.033Bradykinin antagonist

0.033 0.032 DB11100

DB11100
0.010.9840.191Heme oxygenase stimulant

0.191 0.002 DBMET00498

DBMET00498
0.0020.9770.054Kinesin antagonist

0.054 0.015 DB11100

DB11100
0.0020.9770.054Kinesin-like protein 1 inhibitor

0.054 0.015 DB11100

DB11100
0.0040.9840.369Antiobesity

0.369 0.078 DB11100

DB11100
Ext Pa Pi Pmax Activity Other Results ID Pa_max