Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.8130.0030.8135 Hydroxytryptamine release stimulant

0.243 0.093 DBMET00900

0.215 0.11 DBMET00927

0.8010.0050.801Antiobesity

0.486 0.04 DBMET00900

0.786 0.006 DBMET00927

0.7970.0020.7975 Hydroxytryptamine 2C agonist

0.222 0.004 DBMET00900

0.087 0.009 DBMET00927

0.7870.0010.7875 Hydroxytryptamine 2B agonist

0.075 0.005 DBMET00900

0.7670.0040.7675 Hydroxytryptamine agonist

0.1 0.033 DBMET00900

0.7230.0020.7235 Hydroxytryptamine 2 agonist

0.061 0.025 DBMET00900

0.660.0020.665 Hydroxytryptamine 2A agonist

0.062 0.045 DBMET00900

0.5240.0430.524Analgesic
0.470.0050.475 Hydroxytryptamine uptake stimulant

0.216 0.123 DBMET00900

0.450.0420.45GABA C receptor rho-3 antagonist
0.420.0190.42Psychostimulant
0.4140.020.414Calcium channel activator

0.254 0.142 DBMET00900

0.3860.0050.3865 Hydroxytryptamine uptake inhibitor
0.3830.0240.383Sigma receptor agonist
0.3390.0040.339GABA C receptor antagonist

0.146 0.032 DBMET00900

0.4060.0770.406Calcium channel L-type activator
0.3250.0050.325NMDA receptor antagonist
0.3240.0080.3245 Hydroxytryptamine 2C antagonist
0.3290.0140.3295 Hydroxytryptamine 2 antagonist
0.3280.0220.328Tyrosine 3 hydroxylase inhibitor
0.3170.0170.3175 Hydroxytryptamine antagonist
0.3180.020.3185 Hydroxytryptamine 1E antagonist

0.219 0.109 DBMET00900

0.3080.0130.308Acetylcholine M1 receptor antagonist

0.12 0.109 DBMET00900

0.2860.0040.286MAP-kinase-activated kinase inhibitor
0.2790.0040.279Adrenaline uptake inhibitor
0.3690.10.3695 Hydroxytryptamine release inhibitor

0.249 0.229 DBMET00927

0.3430.0770.343Vasodilator, peripheral
0.3090.0470.309HERG channel blocker
0.2630.0040.263MAP-kinase-activated kinase 2 inhibitor
0.2970.0410.297Anticonvulsant
0.2920.0520.292Potassium channel (Voltage-sensitive) blocker
0.2340.0030.234Nicotinic alpha3beta2 receptor antagonist
0.2720.0410.272Anesthetic general
0.2310.0070.231HIV-1 integrase (Overall Integration) inhibitor

0.121 0.039 DBMET00900

0.2340.0170.234Alpha 2b adrenoreceptor antagonist
0.2320.0210.2325 Hydroxytryptamine 2B antagonist
0.250.0390.25Neurotrophic factor enhancer

0.149 0.139 DBMET00927

0.2210.0120.221Alpha 2a adrenoreceptor antagonist
0.2010.0040.201Nicotinic alpha4beta2 receptor antagonist
0.2230.0270.223Cholinergic antagonist
0.2190.0240.256ATPase inhibitor

0.256 0.012 DBMET00927

DBMET00927
0.220.0260.22Acetylcholine antagonist
0.2110.0180.2115 Hydroxytryptamine 2A antagonist
0.1910.0070.191Dopamine uptake inhibitor
0.220.0370.22Antipruritic
0.2070.0250.207GABA C receptor rho-2 antagonist
0.2010.020.201GABA C receptor agonist
0.2550.0750.255Interleukin agonist
0.1850.0050.185NMDA 2C receptor antagonist
0.2370.0580.237RNA-directed DNA polymerase inhibitor
0.1840.0070.184Acetylcholine M4 receptor antagonist
0.1840.0110.184NMDA 2 receptor antagonist
0.1990.0260.199Glutamate receptor antagonist
0.1910.020.191GABA receptor agonist
0.1880.0190.188Alpha 2 adrenoreceptor antagonist
0.1930.0260.193Acetylcholine muscarinic antagonist
0.1750.0120.175Dopamine D1 antagonist
0.1840.020.1845 Hydroxytryptamine 3A agonist
0.1580.0060.158Glycine receptor antagonist

0.106 0.027 DBMET00900

0.088 0.046 DBMET00927

0.1680.0150.168GABA C receptor rho-1 antagonist
0.1810.0310.181Alpha adrenoreceptor antagonist
0.1560.0090.156Lanosterol 14 alpha demethylase inhibitor
0.2620.1170.287Antithrombotic

0.287 0.097 DBMET00927

DBMET00927
0.1610.0160.161Dopamine D4 antagonist
0.1850.0480.185Protein kinase stimulant

0.177 0.051 DBMET00927

0.1670.0290.167Pregnane X receptor agonist
0.1450.0080.1455 Hydroxytryptamine 5A antagonist
0.1440.0080.1445 Hydroxytryptamine 5 antagonist
0.1350.0050.135NMDA receptor subunit 3A antagonist
0.1390.0090.139Acetylcholine M5 receptor antagonist
0.2230.0930.223Aldehyde oxidase inhibitor
0.3110.1820.311Caspase 9 stimulant
0.1450.0170.145Inducible nitric-oxide synthase inhibitor
0.1350.0080.135Alpha 2 adrenoreceptor agonist
0.1330.0090.133Glycine receptor agonist

0.084 0.033 DBMET00900

0.077 0.042 DBMET00927

0.1660.0440.166Neuropeptide Y1 antagonist
0.1950.0730.195Focal adhesion kinase 2 inhibitor
0.130.0090.135 Hydroxytryptamine 6 antagonist
0.1450.0250.145Nitric-oxide synthase inhibitor
0.1760.0580.176Arachidonic acid antagonist

0.152 0.086 DBMET00900

0.1620.0440.162Adenylate cyclase stimulant
0.1440.0280.144Acetylcholine agonist
0.1420.0270.142Dopamine antagonist
0.1340.0230.1345 Hydroxytryptamine 1A antagonist
0.1340.0270.1345 Hydroxytryptamine 1 antagonist
0.1270.020.1275 Hydroxytryptamine 7 antagonist
0.2150.1080.215Spasmolytic
0.120.0140.12Acetylcholine muscarinic agonist
0.1140.0090.114Nicotinic receptor alpha3 subunit antagonist
0.3070.2040.307Ca2+/calmodulin-dependent protein kinase kinase A inhibitor
0.170.0670.17Catenin beta inhibitor
0.1560.0540.156Nav1.2 sodium channel blocker
0.1420.0410.142Sphingosine 1-phosphate receptor 4 antagonist
0.1550.0540.155Sphingosine 1-phosphate receptor 5 antagonist
0.1070.0060.107Somatostatin 4 agonist
0.110.010.11Glycine transporter inhibitor
0.1970.0960.197Cyclic AMP phosphodiesterase inhibitor
0.1110.0110.111Acetylcholine M1 receptor agonist
0.1270.0280.127Acetylcholine nicotinic antagonist
0.120.0220.12Alpha adrenoreceptor agonist
0.1020.0040.102Dopamine D5 agonist
0.10.0030.1Phenylethanolamine N methyltransferase inhibitor

0.047 0.017 DBMET00900

0.2080.1110.208DNA synthesis inhibitor
0.1470.0510.147Ca2+-transporting ATPase inhibitor

0.141 0.069 DBMET00927

0.1060.010.106NMDA receptor subunit 3B antagonist
0.1350.040.135Alpha 2c adrenoreceptor antagonist
0.1220.0270.122Dopamine D2 antagonist
0.1010.0080.101Myc inhibitor
0.1070.0130.107Dopamine D4 agonist
0.1060.0130.106Androgen agonist
0.1690.0760.1693C-like protease (Human coronavirus) inhibitor
0.1220.0290.122Glutamate (mGluR7) agonist
0.0980.0050.098Kainate receptor 2 antagonist
0.1130.0220.113Dopamine agonist
0.1010.0110.101Dopamine transporter inhibitor
0.1230.0330.123Acetylcholine M3 receptor agonist
0.1030.0140.103GABA B receptor agonist
0.0960.0080.0965 Hydroxytryptamine 7 agonist
0.130.0420.13Antiadrenergic
0.0940.0060.094Glycine transporter 1 inhibitor

0.053 0.014 DBMET00900

0.1080.0210.108Neuronal nicotinic receptor antagonist
0.1220.0360.122Alpha 1 adrenoreceptor antagonist
0.1320.0460.132TRPA1 agonist

0.115 0.064 DBMET00927

0.1260.0420.126Adrenaline antagonist
0.2130.1290.213Gastrin inhibitor
0.1430.060.143Sodium channel (voltage-gated) blocker
0.1120.030.112Acetylcholine nicotinic agonist
0.1110.030.111Bromodomain-containing protein 2 inhibitor
0.1560.0750.194Anticoagulant

0.194 0.055 DBMET00927

DBMET00927
0.1810.1020.1815 Hydroxytryptamine 3E antagonist
0.0960.0170.0965 Hydroxytryptamine 3 agonist
0.1110.0320.111Alpha 1a adrenoreceptor antagonist
0.0880.010.088Glutamate (mGluR group I) agonist
0.0830.0080.083Histamine H4 receptor antagonist
0.0790.0050.079Endothelial nitric-oxide synthase inhibitor
0.1180.0440.118Antihistaminic
0.1440.070.144MAP3K9 inhibitor
0.0850.0130.085Corticotropin releasing factor 2 receptor antagonist
0.0760.0040.076Alpha 1L adrenoreceptor agonist

0.046 0.023 DBMET00900

0.1090.040.109Androgen antagonist
0.1560.0870.156Neurotensin receptor agonist
0.1240.0570.124Interleukin 8 antagonist
0.0870.0230.087Acetylcholine M3 receptor antagonist
0.1290.0650.129Nav1.3 sodium channel blocker
0.2240.160.224Vasodilator, coronary
0.0720.0080.072GABA B receptor antagonist
0.1740.1120.174Potassium channel blocker
0.1290.0680.129Cyclooxygenase 3 inhibitor
0.0690.0080.069AMPA 4 receptor antagonist
0.0830.0220.083Exportin-1 inhibitor
0.1430.0820.143Cholinergic
0.190.1290.19Superoxide dismutase inhibitor
0.0830.0230.0835 Hydroxytryptamine 3 antagonist
0.1220.0630.122Cholesterol synthesis inhibitor

0.113 0.072 DBMET00900

0.103 0.084 DBMET00927

0.0740.0150.074Nicotinic receptor alpha4 subunit antagonist
0.0890.0290.0895 Hydroxytryptamine 1B antagonist
0.0770.0180.077Kallikrein 7 inhibitor
0.0870.0290.088Vanilloid 4 agonist

0.088 0.028 DBMET00900

DBMET00900
0.0730.0160.073Lysine-specific demethylase 1A inhibitor
0.130.0740.13Sodium channel blocker
0.0690.0130.069Kainate receptor antagonist
0.1330.0770.133Aurora-C kinase inhibitor
0.1810.1260.181Nitric-oxide synthase stimulant
0.0970.0430.097ALK inhibitor
0.1050.0510.105Electrolyte absorption antagonist
0.0960.0450.096ATPase (Vacuolar H+) inhibitor

0.09 0.055 DBMET00927

0.1380.0890.138MAP kinase 3 inhibitor
0.0670.0180.067Pregnane X receptor antagonist
0.0520.0040.052Imidazoline I1 receptor antagonist
0.0750.0270.075MDM2 inhibitor
0.0720.0250.072GABA receptor antagonist
0.0860.0390.0865 Hydroxytryptamine 1F antagonist
0.0770.0310.077Acetylcholine M2 receptor antagonist
0.0960.050.096Histamine N-methyltransferase inhibitor
0.0510.0040.051Nicotinic alpha4beta2 receptor agonist
0.0670.0210.067Histamine agonist
0.0680.0230.0685 Hydroxytryptamine 1A agonist
0.050.0050.05Nicotinic alpha3beta4 receptor agonist
0.0580.0130.058Guanylate cyclase inhibitor

0.04 0.033 DBMET00900

0.042 0.03 DBMET00927

0.0680.0240.068Glucosylceramidase inhibitor
0.0790.0360.079Phospholipase D inhibitor
0.0990.0560.099Prolactin inhibitor
0.1870.1440.187Neuropeptide Y2 antagonist
0.0870.0440.087CC chemokine 5 receptor agonist
0.070.0280.07Nicotinic neuronal receptor agonist
0.0980.0560.098UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor
0.0890.0480.089Neuropeptide Y antagonist
0.0740.0330.074Glutamate (mGluR6) antagonist
0.0550.0150.055Factor XIa inhibitor
0.0580.0190.058Potassium channel small-conductance Ca-activated blocker
0.0930.0550.093Glutamate release inhibitor
0.0610.0240.061AMPA receptor antagonist
0.0470.010.047AMPA 3 receptor antagonist
0.0550.0190.055Purinergic P2X4 antagonist
0.0590.0240.0595 Hydroxytryptamine 4 antagonist
0.0510.0170.051Histamine H1 receptor agonist
0.0630.0290.063NMDA 2B receptor antagonist
0.0820.0480.082Focal adhesion kinase 1 inhibitor
0.0610.0270.061Sigma receptor antagonist
0.0670.0340.067Calcium channel P-type blocker
0.0980.0650.098Anabolic
0.0410.0070.0415 Hydroxytryptamine 6 agonist
0.0440.010.04411-Beta-hydroxysteroid dehydrogenase 2 inhibitor

0.025 0.021 DBMET00927

0.1210.0870.121Calcium channel blocker

0.12 0.088 DBMET00900

0.0480.0150.048p53 inhibitor
0.1360.1040.136CF transmembrane conductance regulator agonist
0.0870.0570.087Histamine antagonist
0.0350.0040.035NMDA receptor phencyclidine site antagonist
0.0530.0230.053Adenylate cyclase 1 inhibitor
0.0950.0660.095Sphingomyelinase inhibitor
0.0330.0040.033Nicotinic alpha4 receptor agonist
0.060.0310.06GABA A receptor antagonist
0.1470.1180.147Succinate dehydrogenase inhibitor
0.0670.0390.067Dopamine D3 antagonist
0.0370.010.037LFA antagonist

0.029 0.018 DBMET00900

0.0520.0250.052CC chemokine 4 receptor antagonist
0.070.0430.07Nav1.7 sodium channel blocker
0.0520.0260.075Carnitine palmitoyltransferase 1B inhibitor

0.075 0.009 DBMET00900

DBMET00900
0.0640.0390.064Phosphodiesterase 1C inhibitor
0.1070.0810.107Sphingosine 1-phosphate receptor 2 agonist
0.1180.0930.118Ribosomal protein S6 kinase inhibitor
0.0890.0660.089Protein kinase C zeta inhibitor
0.0840.0610.084Calcium antagonist
0.0720.0490.072Benzodiazepine agonist
0.0770.0540.077Estrogen receptor alpha antagonist
0.0940.0710.094Check point kinase 2 inhibitor
0.0720.0490.072Calcium channel L-type blocker
0.0630.0410.063I kappa B kinase 2 inhibitor
0.0440.0220.044Acid-sensing ion channel blocker
0.0490.0270.049Glutamate (mGluR5) agonist
0.0310.010.031Kainate receptor 1 antagonist
0.0350.0150.035Complement C5a chemotactic receptor antagonist
0.0430.0230.043GABA uptake inhibitor
0.080.060.08I kappa B kinase inhibitor
0.0760.0570.076Glutamate receptor agonist
0.0460.0280.046Dopamine D5 antagonist
0.0430.0250.043Kainate receptor agonist
0.0450.0290.045Dipeptidyl peptidase IV inhibitor
0.0520.0360.052NMDA 2A receptor antagonist
0.0230.0080.023Histone-lysine N-methyltransferase EZH2 inhibitor
0.0330.0180.033AMPA 1 receptor antagonist
0.0520.0380.052Dipeptidyl peptidase inhibitor
0.0380.0240.038Integrin alpha2 antagonist
0.0430.0290.043Nerve growth factor antagonist
0.1120.0980.112Toll-Like receptor antagonist
0.0890.0760.089Bile acid receptor antagonist
0.0290.0160.029Myristoyl transferase inhibitor
0.0660.0560.066Alpha 1b adrenoreceptor antagonist
0.0740.0640.074Histamine H1 receptor antagonist
0.0560.0460.056Heat shock protein 90 beta antagonist
0.0440.0340.044Phosphorylase inhibitor
0.0340.0240.034Factor XI inhibitor
0.0320.0220.032ATP citrate lysase inhibitor
0.0250.0160.025Glutamate (mGluR1) agonist
0.050.0410.05Toll-Like receptor 8 antagonist
0.0510.0430.051CC chemokine 2 receptor antagonist
0.0580.050.058NMDA receptor agonist
0.0330.0260.033Progesterone antagonist
0.050.0430.05Nicotinic receptor alpha7 subunit antagonist
0.0190.0130.019Alpha 2c adrenoreceptor agonist
0.0810.0750.081Pim-3 kinase inhibitor
0.0180.0120.018Cyclin T1 inhibitor
0.0330.0280.033Arginase inhibitor
0.020.0150.02Thymidine kinase (Herpes simplex virus 2) inhibitor
0.0680.0630.068Protein kinase (CaMK, MLCK, PhK, SNF, KIN, NIM1, MAPKAP, POLO, CHK, ULK, RSK-2nd domain) inhibitor
0.0670.0620.067Na+ K+ transporting ATPase inhibitor
0.040.0350.04GHS receptor agonist
0.0180.0130.018Histamine H4 receptor agonist
0.0220.0170.022Motilin receptor agonist
0.0290.0250.029Epoxide hydrolase 1 inhibitor
0.0370.0320.037Integrin alpha1beta1 antagonist
0.0910.0870.091Cystathionine beta-synthase inhibitor
0.0610.0570.061Check point kinase 1 inhibitor
0.0560.0530.056Enoyl-[acyl-carrier-protein] reductase inhibitor
0.0730.070.073Opioid kappa receptor antagonist
0.0230.0190.023Kainate receptor 4 antagonist
0.0510.0490.051Alpha 1 adrenoreceptor agonist
0.0780.0760.0783C-Like protease (SARS coronavirus) inhibitor
0.0560.0550.056Bcl-xL inhibitor
0.0540.0530.054Ca(v)3.2 blocker
0.0830.0820.083MAP kinase kinase 1 inhibitor
0.0430.0420.0435 Hydroxytryptamine 1 agonist
0.0090.0080.009Progesterone receptor A antagonist
0.030.0310.036ADAM10 endopeptidase inhibitor

0.036 0.019 DBMET00927

DBMET00927
0.1120.1130.179Cell wall synthesis inhibitor

0.179 0.041 DBMET00900

DBMET00900
0.0310.0390.082Glutamate (mGluR8) antagonist

0.082 0.003 DBMET00927

DBMET00927
0.1410.1550.205Platelet antagonist

0.205 0.098 DBMET00927

DBMET00927
0.1860.2150.262Interleukin 2 agonist

0.262 0.106 DBMET00927

DBMET00927
0.0310.0750.109Protein 50S ribosomal subunit inhibitor

0.109 0.011 DBMET00927

DBMET00927
0.0740.1370.104Toll-Like receptor 4 antagonist

0.104 0.063 DBMET00927

DBMET00927
0.1460.260.288Immunosuppressant

0.288 0.123 DBMET00927

DBMET00927
0.0490.1660.076Cell adhesion molecule inhibitor

0.076 0.059 DBMET00927

DBMET00927
0.0690.1990.157Cell adhesion inhibitor

0.157 0.043 DBMET00927

DBMET00927
0.1560.290.428Antibacterial

0.371 0.091 DBMET00900

0.428 0.065 DBMET00927

DBMET00927
0.0830.2270.135Nitric oxide antagonist

0.135 0.112 DBMET00927

DBMET00927
0.0160.1590.035Purinergic P2Y2 antagonist

0.035 0.021 DBMET00900

DBMET00900
0.0050.1560.058Squalene synthetase inhibitor

0.058 0.012 DBMET00927

DBMET00927
0.0040.1590.045Estrone sulfatase inhibitor

0.045 0.008 DBMET00900

DBMET00900
0.0050.1780.244Urotensin II antagonist

0.244 0.004 DBMET00900

DBMET00900
0.1420.3760.351Apoptosis agonist

0.351 0.138 DBMET00927

DBMET00927
0.030.2820.059Adenine nucleotide translocase inhibitor

0.059 0.03 DBMET00927

DBMET00927
0.0770.3710.186Hypoglycemic

0.186 0.127 DBMET00927

DBMET00927
0.120.4250.483Cyclophilin D inhibitor

0.483 0.055 DBMET00927

DBMET00927
0.1030.4080.282Peptidyltransferase inhibitor

0.282 0.032 DBMET00927

DBMET00927
0.0560.3850.146Hepatoprotectant

0.146 0.114 DBMET00927

DBMET00927
0.0410.3930.362Hypolipemic

0.362 0.032 DBMET00900

0.282 0.055 DBMET00927

DBMET00900
0.0130.4220.037Antibiotic Aminoglycoside-like

0.037 0.025 DBMET00927

DBMET00927
0.0270.4760.24Angiogenesis stimulant

0.24 0.075 DBMET00927

DBMET00927
0.0270.5030.18DNA polymerase I inhibitor

0.18 0.035 DBMET00927

DBMET00927
0.0230.5240.371Beta lactamase inhibitor

0.371 0.109 DBMET00900

DBMET00900
0.0290.5440.206Antioxidant

0.206 0.11 DBMET00927

DBMET00927
0.0220.5460.172Free radical scavenger

0.172 0.122 DBMET00927

DBMET00927
0.0050.5550.055Selectin antagonist

0.055 0.054 DBMET00927

DBMET00927
0.010.7560.163Amyloid beta precursor protein antagonist

0.163 0.087 DBMET00927

DBMET00927
Ext Pa Pi Pmax Activity Other Results ID Pa_max