Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.8990.0030.8995 Hydroxytryptamine antagonist

0.837 0.003 DBMET03491

0.724 0.004 DBMET03492

0.890.0030.895 Hydroxytryptamine 2 antagonist

0.817 0.003 DBMET03491

0.684 0.004 DBMET03492

0.880.0030.88Dopamine D2 antagonist

0.742 0.004 DBMET03491

0.664 0.004 DBMET03492

0.8720.0030.872Dopamine antagonist

0.779 0.003 DBMET03491

0.661 0.004 DBMET03492

0.8540.0020.8545 Hydroxytryptamine 2A antagonist

0.749 0.003 DBMET03491

0.638 0.004 DBMET03492

0.8120.0020.812Dopamine D3 antagonist

0.744 0.002 DBMET03491

0.669 0.003 DBMET03492

0.7370.0030.737Dopamine D2 agonist

0.53 0.004 DBMET03491

0.594 0.003 DBMET03492

0.730.0030.73Dopamine agonist

0.583 0.004 DBMET03491

0.625 0.004 DBMET03492

0.6420.0040.6425 Hydroxytryptamine 2B antagonist

0.504 0.005 DBMET03491

0.372 0.01 DBMET03492

0.5680.0050.568Alpha adrenoreceptor antagonist

0.39 0.01 DBMET03491

0.368 0.011 DBMET03492

0.5270.0040.5275 Hydroxytryptamine 2C antagonist

0.439 0.005 DBMET03491

0.298 0.009 DBMET03492

0.5250.0040.525Dopamine D4 antagonist

0.286 0.008 DBMET03491

0.265 0.008 DBMET03492

0.4980.0030.498Dopamine D3 agonist

0.373 0.003 DBMET03491

0.419 0.003 DBMET03492

0.4970.0160.497HERG channel blocker

0.48 0.017 DBMET03491

0.478 0.017 DBMET03492

0.4850.0050.4855 Hydroxytryptamine 1 antagonist

0.373 0.007 DBMET03491

0.27 0.012 DBMET03492

0.4820.0040.482Alpha 2 adrenoreceptor antagonist

0.308 0.008 DBMET03491

0.237 0.013 DBMET03492

0.4510.0030.4515 Hydroxytryptamine 5A antagonist

0.311 0.004 DBMET03491

0.24 0.004 DBMET03492

0.4570.0190.457Potassium channel (Voltage-sensitive) blocker

0.453 0.019 DBMET03491

0.441 0.021 DBMET03492

0.4360.0050.436Alpha 1a adrenoreceptor antagonist

0.323 0.008 DBMET03491

0.31 0.009 DBMET03492

0.4230.0050.4235 Hydroxytryptamine 1A antagonist

0.279 0.01 DBMET03491

0.237 0.012 DBMET03492

0.4730.0570.488Analgesic

0.488 0.053 DBMET03491

0.403 0.083 DBMET03492

DBMET03491
0.4120.0060.412Alpha 1 adrenoreceptor antagonist

0.31 0.01 DBMET03491

0.305 0.01 DBMET03492

0.4010.0040.401Neuropeptide Y antagonist

0.395 0.004 DBMET03491

0.4 0.004 DBMET03492

0.4160.0190.416Sigma receptor agonist

0.375 0.026 DBMET03491

0.363 0.028 DBMET03492

0.40.0050.4Alpha 2a adrenoreceptor antagonist

0.334 0.005 DBMET03491

0.255 0.009 DBMET03492

0.3790.0030.3795 Hydroxytryptamine 5 antagonist

0.283 0.004 DBMET03491

0.213 0.005 DBMET03492

0.3680.0040.368Dopamine D4 agonist

0.347 0.004 DBMET03491

0.353 0.004 DBMET03492

0.3580.0050.3585 Hydroxytryptamine 1 agonist

0.273 0.008 DBMET03491

0.264 0.008 DBMET03492

0.3520.0050.3525 Hydroxytryptamine 1A agonist

0.293 0.006 DBMET03491

0.288 0.006 DBMET03492

0.3530.0060.353Alpha 1b adrenoreceptor antagonist

0.274 0.009 DBMET03491

0.236 0.011 DBMET03492

0.3510.0050.351Dopamine D1 antagonist

0.19 0.011 DBMET03491

0.154 0.014 DBMET03492

0.3510.010.3515 Hydroxytryptamine 1E antagonist

0.341 0.012 DBMET03491

0.327 0.016 DBMET03492

0.3450.0050.345Alpha 2c adrenoreceptor antagonist

0.297 0.007 DBMET03491

0.217 0.015 DBMET03492

0.3370.0050.337Alpha 1d adrenoreceptor antagonist

0.236 0.007 DBMET03491

0.231 0.008 DBMET03492

0.3250.0040.3315 Hydroxytryptamine 1B antagonist

0.331 0.004 DBMET03491

0.179 0.01 DBMET03492

DBMET03491
0.3250.0050.3355 Hydroxytryptamine 7 antagonist

0.335 0.005 DBMET03491

0.32 0.005 DBMET03492

DBMET03491
0.3240.0120.324Neuropeptide Y2 antagonist

0.299 0.019 DBMET03491

0.323 0.012 DBMET03492

0.2980.0090.298Alpha 2b adrenoreceptor antagonist

0.246 0.015 DBMET03491

0.194 0.025 DBMET03492

0.3010.0130.301Antiadrenergic

0.267 0.016 DBMET03491

0.249 0.017 DBMET03492

0.2970.0130.297Adrenaline antagonist

0.262 0.016 DBMET03491

0.245 0.017 DBMET03492

0.2860.0050.348Neuropeptide Y1 antagonist

0.348 0.004 DBMET03491

0.318 0.004 DBMET03492

DBMET03491
0.2870.0090.2875 Hydroxytryptamine agonist

0.239 0.011 DBMET03491

0.234 0.012 DBMET03492

0.3040.0280.304MAP-kinase-activated kinase 5 inhibitor

0.164 0.159 DBMET03491

0.173 0.144 DBMET03492

0.2780.0190.313Acetylcholine M1 receptor antagonist

0.313 0.012 DBMET03491

0.243 0.027 DBMET03492

DBMET03491
0.2960.0480.329Potassium channel blocker

0.329 0.038 DBMET03491

0.276 0.055 DBMET03492

DBMET03491
0.2280.0050.2445 Hydroxytryptamine 1D antagonist

0.244 0.005 DBMET03491

0.145 0.013 DBMET03492

DBMET03491
0.230.0090.2565 Hydroxytryptamine uptake inhibitor

0.256 0.008 DBMET03491

0.155 0.015 DBMET03492

DBMET03491
0.270.0570.287Gastrin inhibitor

0.287 0.043 DBMET03491

0.273 0.054 DBMET03492

DBMET03491
0.2150.0040.354CC chemokine 3 receptor antagonist

0.354 0.003 DBMET03491

0.178 0.005 DBMET03492

DBMET03491
0.2220.0190.222Acetylcholine muscarinic antagonist

0.211 0.022 DBMET03491

0.142 0.049 DBMET03492

0.20.0050.2Melanin-concentrating hormone receptor 1 antagonist

0.13 0.008 DBMET03491

0.066 0.026 DBMET03492

0.2050.0170.229Chemokine receptor antagonist

0.226 0.014 DBMET03491

0.229 0.014 DBMET03492

DBMET03492
0.2990.1170.299Antiobesity

0.269 0.14 DBMET03491

0.281 0.131 DBMET03492

0.2010.030.201Acetylcholine antagonist

0.196 0.032 DBMET03491

0.124 0.067 DBMET03492

0.2020.0320.202Cholinergic antagonist

0.197 0.033 DBMET03491

0.124 0.07 DBMET03492

0.1730.0070.296Amidase inhibitor

0.249 0.005 DBMET03491

0.296 0.004 DBMET03492

DBMET03492
0.1510.0030.151Dopamine autoreceptor agonist

0.112 0.004 DBMET03491

0.096 0.004 DBMET03492

0.1530.0090.1695 Hydroxytryptamine 3 antagonist

0.169 0.008 DBMET03491

0.144 0.01 DBMET03492

DBMET03491
0.1470.0050.147Oleamide hydrolase inhibitor

0.143 0.005 DBMET03491

0.115 0.007 DBMET03492

0.1530.0160.255Alpha adrenoreceptor agonist

0.255 0.005 DBMET03491

0.177 0.011 DBMET03492

DBMET03491
0.1410.0120.141Sigma receptor antagonist

0.118 0.014 DBMET03491

0.115 0.014 DBMET03492

0.1380.0090.138Acetylcholine M5 receptor antagonist

0.112 0.014 DBMET03491

0.108 0.015 DBMET03492

0.1830.0580.183Protein kinase (CK1) gamma 3 inhibitor
0.1340.0120.134Dopamine uptake inhibitor

0.134 0.012 DBMET03491

0.088 0.022 DBMET03492

0.1320.0220.166CC chemokine receptor antagonist

0.166 0.015 DBMET03491

0.154 0.017 DBMET03492

DBMET03491
0.1890.0830.195 Hydroxytryptamine 3E antagonist

0.19 0.082 DBMET03491

0.179 0.109 DBMET03492

DBMET03491
0.1130.0110.186Alpha 2 adrenoreceptor agonist

0.186 0.005 DBMET03491

0.143 0.007 DBMET03492

DBMET03491
0.1640.0680.164Dual specificity tyrosine-phosphorylation-regulated kinase 4 inhibitor
0.1090.0130.109Calcium channel T-type blocker

0.065 0.032 DBMET03491

0.052 0.051 DBMET03492

0.1020.0130.12CC chemokine 2 receptor antagonist

0.12 0.009 DBMET03491

0.07 0.024 DBMET03492

DBMET03491
0.1060.020.106Acetylcholine M2 receptor antagonist

0.083 0.028 DBMET03491

0.1310.0470.1915 Hydroxytryptamine 3A agonist

0.174 0.024 DBMET03491

0.191 0.018 DBMET03492

DBMET03492
0.10.0170.108Alpha 1 adrenoreceptor agonist

0.108 0.015 DBMET03491

0.071 0.027 DBMET03492

DBMET03491
0.1050.0220.105CXC chemokine receptor antagonist

0.085 0.034 DBMET03491

0.104 0.022 DBMET03492

0.1020.020.102Ca(v)3.1 blocker

0.082 0.055 DBMET03491

0.078 0.067 DBMET03492

0.1550.0730.155Cholinergic
0.1220.0420.158Antihistaminic

0.158 0.03 DBMET03491

0.095 0.059 DBMET03492

DBMET03491
0.1170.0370.165NMDA receptor antagonist

0.109 0.042 DBMET03491

0.165 0.02 DBMET03492

DBMET03492
0.0970.0190.111Adrenaline uptake inhibitor

0.111 0.016 DBMET03491

0.066 0.038 DBMET03492

DBMET03491
0.1160.040.153Histamine antagonist

0.153 0.029 DBMET03491

0.088 0.056 DBMET03492

DBMET03491
0.1040.030.1045 Hydroxytryptamine 1F antagonist

0.101 0.031 DBMET03491

0.120.0490.12Multidrug resistance-associated protein 1 inhibitor
0.1510.0830.151Polo-like kinase-3 inhibitor
0.1050.0390.105Histamine H1 receptor antagonist

0.097 0.043 DBMET03491

0.089 0.049 DBMET03492

0.170.1040.17Ca2+/calmodulin-dependent kinase II beta inhibitor

0.15 0.128 DBMET03491

0.151 0.127 DBMET03492

0.0910.0260.102Purinergic P2 antagonist

0.102 0.021 DBMET03491

0.097 0.023 DBMET03492

DBMET03491
0.0770.0140.077Prolactin release inhibitor
0.0860.0230.0895 Hydroxytryptamine 2A agonist

0.069 0.038 DBMET03491

0.089 0.02 DBMET03492

DBMET03492
0.170.1070.299Anticonvulsant

0.299 0.041 DBMET03491

0.295 0.042 DBMET03492

DBMET03491
0.0690.0060.069Sigma 2 receptor antagonist

0.049 0.01 DBMET03491

0.04 0.013 DBMET03492

0.0760.0140.0795 Hydroxytryptamine 4 antagonist

0.079 0.013 DBMET03491

0.074 0.015 DBMET03492

DBMET03491
0.0740.0150.074Neurokinin 2 antagonist

0.043 0.027 DBMET03491

0.04 0.03 DBMET03492

0.1270.0720.127Acetylcholinesterase inhibitor
0.080.0260.13Acetylcholine M3 receptor antagonist

0.13 0.013 DBMET03491

0.064 0.037 DBMET03492

DBMET03491
0.2850.2340.336Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.336 0.167 DBMET03491

0.286 0.233 DBMET03492

DBMET03491
0.0640.0160.07Histamine H4 receptor antagonist

0.067 0.014 DBMET03491

0.07 0.012 DBMET03492

DBMET03492
0.1010.0540.101Prolactin inhibitor
0.0780.0330.085 Hydroxytryptamine 3A antagonist

0.08 0.031 DBMET03491

0.074 0.037 DBMET03492

DBMET03491
0.090.0460.09Acetylcholine nicotinic agonist

0.087 0.048 DBMET03491

0.1390.0970.139Ca2+/calmodulin-dependent kinase II gamma inhibitor
0.0810.0390.109Cannabinoid receptor antagonist

0.109 0.025 DBMET03491

0.066 0.054 DBMET03492

DBMET03491
0.0670.0260.067Acetyl-CoA transferase inhibitor
0.0770.0370.077Cannabinoid receptor agonist

0.069 0.042 DBMET03491

0.072 0.04 DBMET03492

0.0510.0140.053Purinergic P2X7 antagonist

0.053 0.013 DBMET03491

0.052 0.013 DBMET03492

DBMET03491
0.0820.0450.082Analgesic, opioid

0.07 0.062 DBMET03491

0.076 0.053 DBMET03492

0.0430.0080.053Epoxide hydrolase 2 inhibitor

0.053 0.005 DBMET03491

0.046 0.007 DBMET03492

DBMET03491
0.0590.0240.063Purinergic P2X antagonist

0.061 0.023 DBMET03491

0.063 0.021 DBMET03492

DBMET03492
0.0420.0080.163CC chemokine 1 receptor antagonist

0.141 0.004 DBMET03491

0.163 0.004 DBMET03492

DBMET03492
0.0840.0520.085Opioid kappa receptor antagonist

0.08 0.058 DBMET03491

0.085 0.052 DBMET03492

DBMET03492
0.0760.0460.103Epoxide hydrolase inhibitor

0.103 0.023 DBMET03491

0.09 0.033 DBMET03492

DBMET03491
0.0420.0120.042Sigma 1 receptor antagonist

0.036 0.014 DBMET03491

0.033 0.015 DBMET03492

0.0550.0280.055Antiviral (Hepatitis D)
0.0580.0310.058Neuropeptide Y5 antagonist
0.0650.0390.106Cannabinoid CB1 receptor agonist

0.088 0.024 DBMET03491

0.106 0.018 DBMET03492

DBMET03492
0.0560.030.061Chemokine receptor agonist

0.043 0.041 DBMET03491

0.061 0.026 DBMET03492

DBMET03492
0.0390.0140.041CXC chemokine 3 receptor antagonist

0.041 0.013 DBMET03491

0.036 0.016 DBMET03492

DBMET03491
0.0520.0320.052Neurokinin antagonist
0.0440.0240.044Acetyl-CoA transferase 1 inhibitor
0.1430.1230.158Psychostimulant

0.158 0.109 DBMET03491

0.158 0.11 DBMET03492

DBMET03492
0.1110.0920.111Ca2+/calmodulin-dependent kinase II delta inhibitor
0.0420.0240.042Substance P antagonist
0.1420.1230.184Phospholipase C inhibitor

0.184 0.056 DBMET03492

DBMET03492
0.0430.0250.056Nicotinic acid receptor 1 agonist

0.056 0.018 DBMET03491

0.05 0.02 DBMET03492

DBMET03491
0.0610.0440.071Corticotropin releasing factor 2 receptor antagonist

0.058 0.05 DBMET03491

0.071 0.027 DBMET03492

DBMET03492
0.0550.040.0565 Hydroxytryptamine 7 agonist

0.056 0.038 DBMET03491

0.052 0.048 DBMET03492

DBMET03491
0.1760.160.176DNA synthesis inhibitor
0.0510.0360.051Cannabinoid CB2 receptor antagonist
0.0390.0240.041Integrin alpha1beta1 antagonist

0.04 0.021 DBMET03491

0.041 0.02 DBMET03492

DBMET03492
0.0340.0190.034Acetylcholine M4 receptor agonist
0.0520.0370.057Histamine agonist

0.047 0.045 DBMET03491

0.057 0.03 DBMET03492

DBMET03492
0.0580.0440.058Ca(v)3.2 blocker

0.055 0.052 DBMET03491

0.0480.0350.051CC chemokine receptor 2B antagonist

0.047 0.037 DBMET03491

0.051 0.03 DBMET03492

DBMET03492
0.0210.010.021Apolipoprotein B-100 inhibitor
0.0250.0150.0255 Hydroxytryptamine 4 agonist

0.025 0.016 DBMET03491

0.024 0.017 DBMET03492

0.0440.0370.044Glycine transporter inhibitor

0.042 0.038 DBMET03491

0.0960.090.096Calcium channel (voltage-sensitive) blocker
0.0670.0610.067Acetylcholine M4 receptor antagonist
0.0460.0410.054CC chemokine 5 receptor antagonist

0.054 0.031 DBMET03491

0.046 0.043 DBMET03492

DBMET03491
0.0430.0390.044Dopamine transporter inhibitor

0.044 0.038 DBMET03491

DBMET03491
0.090.0860.098EphA2 antagonist

0.095 0.081 DBMET03491

0.098 0.078 DBMET03492

DBMET03492
0.0760.0720.076Acetylcholine agonist
0.0510.0480.0515 Hydroxytryptamine 6 antagonist
0.0330.030.033Adenosine uptake inhibitor
0.0340.0310.0342,3-Oxidosqualene-lanosterol cyclase inhibitor
0.0310.0290.031Protein kinase (CK2) beta inhibitor
0.030.0290.03Nociceptin (N/OFQ) receptor antagonist

0.03 0.028 DBMET03492

0.0710.0710.117Adrenaline agonist

0.117 0.027 DBMET03491

0.101 0.036 DBMET03492

DBMET03491
0.0280.0290.033CXC chemokine receptor agonist

0.033 0.025 DBMET03492

DBMET03492
0.0530.0550.072Cannabinoid CB1 receptor antagonist

0.072 0.033 DBMET03491

DBMET03491
0.1880.1910.222Vasodilator, peripheral

0.222 0.152 DBMET03491

DBMET03491
0.0330.0370.034Delayed rectifier potassium channel blocker

0.034 0.033 DBMET03491

DBMET03491
0.0730.080.085Histamine H2 receptor antagonist

0.085 0.054 DBMET03491

DBMET03491
0.0730.080.077Opioid antagonist

0.077 0.073 DBMET03492

DBMET03492
0.0680.0750.086Cell adhesion molecule inhibitor

0.086 0.046 DBMET03491

DBMET03491
0.0230.0320.034Peptide deformylase inhibitor

0.034 0.018 DBMET03491

DBMET03491
0.0250.0350.034Epoxide hydrolase 1 inhibitor

0.034 0.016 DBMET03491

0.029 0.024 DBMET03492

DBMET03491
0.1280.140.165Anesthetic general

0.165 0.098 DBMET03492

DBMET03492
0.0240.0490.031DNA topoisomerase IV inhibitor

0.031 0.018 DBMET03491

DBMET03491
0.2310.2570.2835 Hydroxytryptamine release inhibitor

0.283 0.185 DBMET03492

DBMET03492
0.0280.0710.039Glucose-6-phosphate dehydrogenase inhibitor

0.039 0.023 DBMET03492

DBMET03492
0.1310.1840.196Spasmolytic

0.196 0.123 DBMET03491

DBMET03491
0.0340.0870.044Baculoviral IAP repeat-containing protein inhibitor

0.044 0.04 DBMET03491

DBMET03491
0.050.1090.06Beta 2 adrenoreceptor agonist

0.06 0.05 DBMET03492

DBMET03492
0.0930.1550.119Anticoagulant

0.119 0.113 DBMET03492

DBMET03492
0.0290.0940.05Nicotinic neuronal receptor agonist

0.05 0.045 DBMET03491

DBMET03491
0.0210.0870.031Carboxypeptidase B inhibitor

0.031 0.029 DBMET03492

DBMET03492
0.0730.1450.09Glutamate (mGluR7) agonist

0.09 0.084 DBMET03491

DBMET03491
0.0280.1050.048Potassium channel (Inward rectifier) blocker

0.048 0.037 DBMET03491

DBMET03491
0.1060.1910.17Antipruritic

0.155 0.089 DBMET03491

0.17 0.074 DBMET03492

DBMET03492
0.0370.1260.071DNA gyrase inhibitor

0.071 0.035 DBMET03491

DBMET03491
0.0690.160.102mTOR complex 1 inhibitor

0.102 0.057 DBMET03491

DBMET03491
0.1620.2570.343Toll-Like receptor 7 agonist

0.343 0.086 DBMET03492

DBMET03492
0.1540.270.336Toll-Like receptor agonist

0.336 0.089 DBMET03492

DBMET03492
0.1050.2250.211Tumour necrosis factor alpha release inhibitor

0.211 0.099 DBMET03492

DBMET03492
0.0350.2020.092Somatostatin 1 agonist

0.092 0.04 DBMET03492

DBMET03492
0.0650.3750.152Ca2+/calmodulin-dependent kinase I alpha inhibitor

0.152 0.142 DBMET03492

DBMET03492
Ext Pa Pi Pmax Activity Other Results ID Pa_max