Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.9610.0030.961Tyrosine kinase inhibitor

0.946 0.004 DBMET03261

0.651 0.008 DBMET03264

0.905 0.004 DBMET03262

0.919 0.004 DBMET03263

0.9110.0020.911Janus tyrosine kinase 3 inhibitor

0.851 0.003 DBMET03261

0.467 0.004 DBMET03264

0.77 0.003 DBMET03262

0.805 0.003 DBMET03263

0.8430.010.852Antiinflammatory

0.81 0.014 DBMET03261

0.798 0.015 DBMET03264

0.852 0.009 DBMET03262

0.829 0.012 DBMET03263

DBMET03262
0.8350.0050.835Toll-Like receptor 7 agonist

0.76 0.006 DBMET03261

0.486 0.034 DBMET03264

0.809 0.005 DBMET03262

0.783 0.005 DBMET03263

0.830.0050.83Toll-Like receptor agonist

0.752 0.006 DBMET03261

0.476 0.037 DBMET03264

0.802 0.005 DBMET03262

0.776 0.005 DBMET03263

0.7760.0030.776Janus tyrosine kinase 2 inhibitor

0.767 0.003 DBMET03261

0.417 0.005 DBMET03264

0.656 0.003 DBMET03262

0.673 0.003 DBMET03263

0.7180.0040.718CDC-like kinase 2 inhibitor

0.462 0.008 DBMET03261

0.373 0.017 DBMET03264

0.495 0.006 DBMET03262

0.508 0.005 DBMET03263

0.7020.0020.702I kappa B kinase epsilon inhibitor

0.42 0.003 DBMET03261

0.303 0.014 DBMET03264

0.564 0.002 DBMET03262

0.644 0.002 DBMET03263

0.6940.0040.694Death-associated protein kinase 3 inhibitor

0.523 0.005 DBMET03261

0.488 0.007 DBMET03264

0.551 0.005 DBMET03262

0.559 0.005 DBMET03263

0.680.0040.68Dual specificity tyrosine-phosphorylation regulated kinase 1B inhibitor

0.411 0.005 DBMET03261

0.338 0.009 DBMET03264

0.447 0.005 DBMET03262

0.466 0.005 DBMET03263

0.6660.0030.666Ca2+/calmodulin-dependent kinase II alpha inhibitor

0.579 0.004 DBMET03261

0.582 0.004 DBMET03264

0.596 0.003 DBMET03262

0.592 0.003 DBMET03263

0.6480.0040.648TRKC antagonist

0.534 0.005 DBMET03261

0.439 0.009 DBMET03264

0.575 0.005 DBMET03262

0.564 0.005 DBMET03263

0.6480.0050.648Ca2+/calmodulin-dependent protein kinase inhibitor

0.391 0.019 DBMET03261

0.336 0.032 DBMET03264

0.432 0.013 DBMET03262

0.437 0.013 DBMET03263

0.6190.0040.619Protein kinase C nu inhibitor

0.416 0.009 DBMET03261

0.344 0.017 DBMET03264

0.453 0.006 DBMET03262

0.434 0.007 DBMET03263

0.6180.0050.618CDC-like kinase 4 inhibitor

0.358 0.019 DBMET03261

0.206 0.064 DBMET03264

0.404 0.014 DBMET03262

0.441 0.01 DBMET03263

0.590.0050.59Clk dual-specificity kinase inhibitor

0.36 0.026 DBMET03261

0.184 0.089 DBMET03264

0.398 0.02 DBMET03262

0.427 0.015 DBMET03263

0.5880.0050.588RET inhibitor

0.312 0.02 DBMET03261

0.35 0.015 DBMET03262

0.351 0.014 DBMET03263

0.5890.0130.61Immunomodulator

0.506 0.022 DBMET03261

0.61 0.01 DBMET03262

0.513 0.021 DBMET03263

DBMET03262
0.5830.0060.583Dual specificity tyrosine-phosphorylation regulated kinase 1A inhibitor

0.357 0.034 DBMET03261

0.189 0.1 DBMET03264

0.381 0.028 DBMET03262

0.446 0.019 DBMET03263

0.5770.0080.577Dyrk kinase inhibitor

0.345 0.038 DBMET03261

0.166 0.121 DBMET03264

0.37 0.032 DBMET03262

0.426 0.022 DBMET03263

0.570.0170.636Immunosuppressant

0.597 0.014 DBMET03261

0.477 0.039 DBMET03264

0.636 0.009 DBMET03262

0.575 0.016 DBMET03263

DBMET03262
0.5460.0020.546Janus tyrosine kinase 1 inhibitor

0.48 0.002 DBMET03261

0.36 0.003 DBMET03264

0.428 0.002 DBMET03262

0.441 0.002 DBMET03263

0.5480.0040.548Proto-oncogene tyrosine-protein kinase Fyn inhibitor

0.425 0.009 DBMET03261

0.217 0.06 DBMET03264

0.446 0.007 DBMET03262

0.442 0.007 DBMET03263

0.5240.0040.524Antipruritic

0.446 0.005 DBMET03261

0.494 0.005 DBMET03262

0.501 0.004 DBMET03263

0.4860.0030.486Tyk2 inhibitor

0.337 0.004 DBMET03261

0.241 0.006 DBMET03264

0.355 0.004 DBMET03262

0.368 0.004 DBMET03263

0.4690.0040.469TRKB antagonist

0.342 0.007 DBMET03261

0.186 0.029 DBMET03264

0.379 0.005 DBMET03262

0.353 0.006 DBMET03263

0.4590.0060.459Tyrosine-protein kinase receptor antagonist

0.207 0.038 DBMET03261

0.319 0.015 DBMET03262

0.186 0.046 DBMET03263

0.4640.0130.464Growth factor antagonist

0.154 0.067 DBMET03261

0.167 0.059 DBMET03262

0.216 0.042 DBMET03263

0.430.0060.43Protein kinase (CK1) inhibitor

0.237 0.029 DBMET03261

0.119 0.092 DBMET03264

0.267 0.023 DBMET03262

0.303 0.017 DBMET03263

0.4130.0050.413Protein-tyrosine kinase (PTK, not ETK, WZC) inhibitor

0.192 0.03 DBMET03261

0.215 0.024 DBMET03262

0.205 0.027 DBMET03263

0.4120.0050.412Abl kinase inhibitor

0.191 0.03 DBMET03261

0.214 0.024 DBMET03262

0.203 0.027 DBMET03263

0.3970.0040.397Cyclin-dependent kinase 8 inhibitor

0.245 0.017 DBMET03261

0.127 0.108 DBMET03264

0.319 0.007 DBMET03262

0.223 0.024 DBMET03263

0.3750.0050.375Protein kinase A inhibitor

0.217 0.011 DBMET03261

0.082 0.059 DBMET03264

0.269 0.008 DBMET03262

0.219 0.011 DBMET03263

0.3680.0030.368Leucine-rich repeat kinase 2 inhibitor

0.179 0.013 DBMET03261

0.217 0.008 DBMET03262

0.215 0.008 DBMET03263

0.3780.020.378EphB2 antagonist

0.287 0.04 DBMET03261

0.301 0.035 DBMET03262

0.266 0.049 DBMET03263

0.3570.0050.357Fibroblast growth factor 1 antagonist

0.201 0.016 DBMET03261

0.22 0.013 DBMET03264

0.216 0.013 DBMET03262

0.237 0.01 DBMET03263

0.3920.0630.392MAP kinase kinase 6 inhibitor

0.286 0.149 DBMET03261

0.268 0.169 DBMET03262

0.256 0.182 DBMET03263

0.3370.0120.337Glycogen synthase kinase-3 alpha inhibitor

0.151 0.066 DBMET03261

0.221 0.035 DBMET03262

0.259 0.024 DBMET03263

0.350.0380.486Tumour necrosis factor alpha release inhibitor

0.433 0.022 DBMET03261

0.229 0.086 DBMET03264

0.448 0.02 DBMET03262

0.486 0.015 DBMET03263

DBMET03263
0.3120.0040.312Rho-associated kinase I inhibitor

0.086 0.041 DBMET03261

0.101 0.031 DBMET03262

0.118 0.022 DBMET03263

0.3660.0640.366Angiogenesis inhibitor

0.256 0.119 DBMET03261

0.279 0.104 DBMET03262

0.286 0.1 DBMET03263

0.3070.0050.307Rho-associated kinase inhibitor

0.107 0.032 DBMET03261

0.11 0.03 DBMET03262

0.129 0.024 DBMET03263

0.3130.0310.313MAP kinase kinase 2 inhibitor

0.165 0.108 DBMET03261

0.185 0.092 DBMET03262

0.146 0.125 DBMET03263

0.2710.0050.271I kappa B kinase inhibitor

0.143 0.018 DBMET03261

0.194 0.008 DBMET03262

0.253 0.005 DBMET03263

0.2790.0150.329Aurora-A kinase inhibitor

0.127 0.051 DBMET03261

0.329 0.01 DBMET03264

0.139 0.044 DBMET03262

0.199 0.025 DBMET03263

DBMET03264
0.2910.0290.291Ca2+/calmodulin-dependent kinase IV inhibitor

0.194 0.184 DBMET03261

0.2770.0180.277Phosphodiesterase inhibitor

0.233 0.026 DBMET03261

0.254 0.021 DBMET03262

0.255 0.021 DBMET03263

0.2750.0180.275Aurora-B kinase inhibitor

0.101 0.08 DBMET03261

0.134 0.054 DBMET03262

0.207 0.029 DBMET03263

0.2550.0230.255Lck kinase inhibitor

0.146 0.068 DBMET03261

0.166 0.056 DBMET03262

0.158 0.06 DBMET03263

0.2510.0260.251Tyrosine-protein kinase receptor FLT3 inhibitor
0.2710.0470.271MAP-kinase-activated kinase 5 inhibitor

0.186 0.122 DBMET03261

0.206 0.096 DBMET03262

0.188 0.12 DBMET03263

0.2530.0290.253MAP kinase kinase 3 inhibitor

0.191 0.151 DBMET03261

0.191 0.151 DBMET03262

0.205 0.108 DBMET03263

0.2220.0050.222Phosphodiesterase III inhibitor

0.17 0.008 DBMET03261

0.076 0.039 DBMET03264

0.164 0.009 DBMET03262

0.201 0.006 DBMET03263

0.2180.0050.218Fibroblast growth factor 3 antagonist

0.079 0.051 DBMET03261

0.099 0.033 DBMET03262

0.123 0.023 DBMET03263

0.2580.0460.258Interleukin-1 receptor-associated protein kinase 1 inhibitor
0.2410.0380.241Src kinase inhibitor

0.134 0.095 DBMET03261

0.144 0.088 DBMET03262

0.146 0.086 DBMET03263

0.2470.0530.247ErbB-1 antagonist
0.1890.0120.221Phosphodiesterase 4D inhibitor

0.221 0.009 DBMET03261

0.194 0.012 DBMET03262

0.201 0.011 DBMET03263

DBMET03261
0.2260.050.226LIM domain kinase 1 inhibitor
0.1780.0060.178Tyrosine-protein kinase EMT inhibitor

0.093 0.02 DBMET03261

0.103 0.017 DBMET03262

0.093 0.02 DBMET03263

0.1910.020.288Bronchodilator

0.288 0.01 DBMET03261

0.265 0.012 DBMET03262

0.21 0.017 DBMET03263

DBMET03261
0.180.0240.18MAP kinase kinase 4 inhibitor

0.159 0.047 DBMET03261

0.168 0.035 DBMET03262

0.143 0.078 DBMET03263

0.1510.0070.162Phosphodiesterase 4C inhibitor

0.15 0.007 DBMET03261

0.14 0.008 DBMET03262

0.162 0.006 DBMET03263

DBMET03263
0.1660.0220.166Activin receptor-like kinase 4 inhibitor

0.106 0.074 DBMET03261

0.103 0.08 DBMET03262

0.113 0.063 DBMET03263

0.160.0180.16Interleukin-1 receptor-associated protein kinase 4 inhibitor

0.112 0.037 DBMET03261

0.142 0.025 DBMET03262

0.079 0.072 DBMET03263

0.1810.0460.181Ribosomal protein S6 kinase inhibitor
0.1720.040.172MAP kinase kinase inhibitor

0.116 0.078 DBMET03261

0.12 0.074 DBMET03262

0.1560.0310.156Death-associated protein kinase 1 inhibitor

0.122 0.107 DBMET03263

0.1350.0130.135Protein kinase B alpha inhibitor
0.1270.0050.127Fibroblast growth factor 4 antagonist

0.085 0.015 DBMET03261

0.077 0.021 DBMET03264

0.086 0.015 DBMET03262

0.091 0.012 DBMET03263

0.1650.0490.165Cyclin-dependent kinase inhibitor

0.101 0.09 DBMET03262

0.1270.0120.127Phosphodiesterase 4A inhibitor

0.127 0.012 DBMET03261

0.11 0.014 DBMET03262

0.119 0.013 DBMET03263

0.1260.0130.126MAP3K7 inhibitor

0.081 0.039 DBMET03261

0.092 0.028 DBMET03262

0.074 0.048 DBMET03263

0.1680.0570.168CDC-like kinase 1 inhibitor

0.109 0.108 DBMET03263

0.1320.0210.132Protein kinase B gamma inhibitor

0.066 0.063 DBMET03262

0.1190.0160.119Protein kinase B beta inhibitor

0.077 0.046 DBMET03261

0.086 0.036 DBMET03262

0.073 0.052 DBMET03263

0.1250.0270.125ALK inhibitor

0.077 0.063 DBMET03261

0.083 0.055 DBMET03262

0.092 0.046 DBMET03263

0.1560.0630.156Protein-tyrosine kinase Lyn inhibitor
0.1540.0630.154Activin receptor-like kinase 2 inhibitor
0.1230.0330.123Hepatocyte growth factor antagonist

0.089 0.064 DBMET03263

0.1390.0490.139Glycogen synthase kinase-3 beta inhibitor

0.113 0.066 DBMET03263

0.1370.0510.137Glycogen synthase kinase-3 inhibitor

0.109 0.071 DBMET03263

0.1090.0240.109Focal adhesion kinase 1 inhibitor

0.079 0.05 DBMET03264

0.072 0.059 DBMET03262

0.096 0.033 DBMET03263

0.1230.0380.123Protein kinase (Mos, Mil/Raf, MEKK, RIPK, TESK, LIMK, IRAK, ILK, Activin/TGF-beta) inhibitor
0.1110.0280.111MAP kinase 10 inhibitor

0.071 0.063 DBMET03262

0.1020.020.102Phosphatidylinositol kinase inhibitor

0.066 0.036 DBMET03262

0.086 0.026 DBMET03263

0.0990.020.099Phosphatidylinositol 3-kinase delta inhibitor

0.05 0.046 DBMET03262

0.072 0.029 DBMET03263

0.1270.0570.127Protein kinase (CK2) alpha inhibitor

0.119 0.063 DBMET03263

0.1320.0620.132Vascular endothelial growth factor antagonist
0.0910.0220.091MAP kinase kinase 10 inhibitor
0.1030.0370.103AXL receptor tyrosine kinase inhibitor

0.076 0.067 DBMET03261

0.096 0.043 DBMET03262

0.130.0660.13Protein kinase (CK1) delta inhibitor
0.0990.0360.099Protein kinase (CaMK, MLCK, PhK, SNF, KIN, NIM1, MAPKAP, POLO, CHK, ULK, RSK-2nd domain) inhibitor

0.071 0.059 DBMET03261

0.078 0.052 DBMET03262

0.067 0.065 DBMET03263

0.0910.0280.091Cyclin A2 inhibitor
0.1280.0650.128Epidermal growth factor receptor kinase inhibitor
0.1190.0570.119Polo-like kinase-4 inhibitor
0.1070.0460.107Protein kinase C delta inhibitor

0.094 0.058 DBMET03262

0.1410.0840.284Heat shock protein 90 antagonist

0.169 0.056 DBMET03261

0.284 0.013 DBMET03262

0.17 0.055 DBMET03263

DBMET03262
0.0760.020.076Phosphodiesterase II inhibitor

0.06 0.032 DBMET03261

0.061 0.031 DBMET03262

0.055 0.039 DBMET03263

0.0880.0340.088Check point kinase 1 inhibitor

0.066 0.049 DBMET03261

0.073 0.043 DBMET03262

0.062 0.055 DBMET03263

0.0840.0290.084Cyclin A inhibitor
0.0930.0390.093Proto-oncogene tyrosine-protein kinase c-hck inhibitor
0.1440.0910.144Polo-like kinase-3 inhibitor
0.080.0290.08Raf kinase B inhibitor

0.054 0.046 DBMET03263

0.0710.0220.071Protein kinase C theta inhibitor
0.1130.0640.113Vascular endothelial growth factor 2 antagonist
0.0770.0290.077Adenosine A1 receptor antagonist

0.069 0.034 DBMET03261

0.065 0.036 DBMET03262

0.062 0.038 DBMET03263

0.0670.020.067Phosphodiesterase 2A inhibitor

0.051 0.033 DBMET03261

0.052 0.032 DBMET03262

0.047 0.04 DBMET03263

0.1310.0840.131Vascular endothelial growth factor 3 antagonist
0.1340.0880.134MAP3K9 inhibitor
0.0860.0410.086Raf kinase inhibitor
0.0690.0250.069Phosphatidylinositol 3-kinase gamma inhibitor

0.052 0.042 DBMET03262

0.059 0.034 DBMET03263

0.1240.0810.124Cyclin-dependent kinase 7 inhibitor
0.1050.0620.105MAP kinase kinase kinase inhibitor
0.0920.0510.153Phosphodiesterase IV inhibitor

0.153 0.022 DBMET03261

0.133 0.028 DBMET03262

0.151 0.022 DBMET03263

DBMET03261
0.0820.0420.082MAP kinase kinase 7 inhibitor
0.0670.0280.067Bruton tyrosine kinase inhibitor
0.0890.0530.089Bcr-Abl kinase inhibitor
0.0630.0260.063mTOR inhibitor

0.052 0.036 DBMET03262

0.046 0.044 DBMET03263

0.0920.0560.124Pim-3 kinase inhibitor

0.098 0.047 DBMET03261

0.124 0.029 DBMET03262

DBMET03262
0.1260.0920.126Aurora-C kinase inhibitor
0.0410.0090.041LIM domain kinase 2 inhibitor
0.1350.1030.135Ca2+/calmodulin-dependent protein kinase kinase B inhibitor
0.150.120.15Dual specificity tyrosine-phosphorylation regulated kinase 3 inhibitor
0.0980.0670.098Check point kinase 2 inhibitor
0.0850.0550.085ErbB-3 antagonist
0.0770.0470.093Adenosine A3 receptor antagonist

0.093 0.031 DBMET03261

0.085 0.037 DBMET03262

DBMET03261
0.070.040.07Adenosine A2 receptor antagonist
0.0850.0560.085mTOR complex 2 inhibitor
0.1020.0750.102CDC-like kinase 3 inhibitor
0.1420.1160.142Cyclin-dependent kinase 3 inhibitor
0.0690.0450.069Protein kinase C alpha inhibitor
0.0920.0710.136Protein kinase (CK2) inhibitor

0.089 0.074 DBMET03262

0.136 0.039 DBMET03263

DBMET03263
0.0770.0590.093Phosphodiesterase 3A inhibitor

0.093 0.039 DBMET03263

DBMET03263
0.0680.050.068I kappa B kinase 1 inhibitor
0.130.1140.13Protein kinase (CK1) gamma 3 inhibitor
0.0840.070.084Phosphodiesterase I inhibitor

0.08 0.077 DBMET03261

0.0590.0450.059Adenosine A2a receptor antagonist
0.0340.020.046Transforming growth factor beta 2 antagonist

0.032 0.025 DBMET03261

0.031 0.03 DBMET03262

0.046 0.008 DBMET03263

DBMET03263
0.0930.0810.093Granulocyte macrophage colony stimulating factor antagonist
0.070.060.07ErbB-4 antagonist
0.0470.0370.047Adenosine A2b receptor antagonist
0.0210.0130.021Histone-lysine N-methyltransferase EZH2 inhibitor
0.0780.0710.078Transforming growth factor beta 3 antagonist
0.0980.0910.098c-Src kinase inhibitor
0.0770.0710.077Epidermal growth factor antagonist
0.1250.1190.125MAP kinase 3 inhibitor
0.0940.090.094MAP kinase 13 inhibitor
0.0180.0160.036Integrin alphaVbeta1 antagonist

0.036 0.005 DBMET03264

0.021 0.011 DBMET03262

DBMET03264
0.0310.0290.031ATR kinase inhibitor
0.1110.1090.111Protein kinase (CK1) gamma 1 inhibitor
0.0110.010.011Purine nucleoside phosphorylase inhibitor

0.011 0.01 DBMET03262

0.0660.0650.066ErbB-2 antagonist
0.0530.0540.06Heat shock protein 90 beta antagonist

0.06 0.04 DBMET03262

DBMET03262
0.0460.0540.069Pim-2 kinase inhibitor

0.052 0.042 DBMET03261

0.069 0.025 DBMET03262

DBMET03262
0.0360.0430.039Phosphodiesterase 3B inhibitor

0.039 0.038 DBMET03263

DBMET03263
0.0590.0680.065Transforming growth factor antagonist

0.065 0.056 DBMET03263

DBMET03263
0.0740.0910.104Pim-1 kinase inhibitor

0.089 0.069 DBMET03261

0.104 0.054 DBMET03262

0.09 0.068 DBMET03263

DBMET03262
0.0540.0750.088Macrophage colony-stimulating factor 1 receptor antagonist

0.088 0.035 DBMET03264

DBMET03264
0.0830.1060.094mTOR complex 1 inhibitor

0.094 0.075 DBMET03262

DBMET03262
0.050.0750.062Syk tyrosine kinase inhibitor

0.062 0.058 DBMET03262

DBMET03262
0.1150.1470.129Pregnane X receptor agonist

0.123 0.12 DBMET03261

0.129 0.101 DBMET03262

DBMET03262
0.1330.1850.204Growth factor agonist

0.151 0.14 DBMET03262

0.204 0.059 DBMET03263

DBMET03263
0.0210.0940.049Adenosine deaminase inhibitor

0.049 0.031 DBMET03261

0.045 0.035 DBMET03262

DBMET03261
0.070.1480.098Alpha 2d adrenoreceptor antagonist

0.098 0.053 DBMET03261

0.088 0.075 DBMET03262

0.089 0.073 DBMET03263

DBMET03261
0.0470.1260.067MAP kinase kinase 8 inhibitor

0.067 0.05 DBMET03262

DBMET03262
0.0080.1120.097Somatostatin 3 antagonist

0.097 0.004 DBMET03264

DBMET03264
0.0840.2160.126Heat shock protein 90 alpha antagonist

0.126 0.118 DBMET03262

DBMET03262
0.0820.2640.131Tumour necrosis factor antagonist

0.131 0.126 DBMET03263

DBMET03263
0.10.3870.285Sodium/bile acid cotransporter inhibitor

0.241 0.138 DBMET03261

0.285 0.093 DBMET03262

DBMET03262
0.0490.3720.162Platelet antagonist

0.162 0.132 DBMET03261

DBMET03261
0.0030.7310.174Somatostatin 2 antagonist

0.174 0.004 DBMET03264

DBMET03264
0.0040.7370.151Somatostatin 1 antagonist

0.151 0.005 DBMET03264

DBMET03264
0.0040.7720.154Somatostatin 4 antagonist

0.154 0.004 DBMET03264

DBMET03264
0.0020.9020.136Somatostatin 5 antagonist

0.136 0.005 DBMET03264

DBMET03264
Ext Pa Pi Pmax Activity Other Results ID Pa_max