| Min Pa: | Min Pa(max): | Activity's type: |
| Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |
|---|---|---|---|---|---|---|
| 0.816 | 0.009 | 0.83 | Caspase 9 stimulant | 0.83 0.007 DB14219 | DB14219 | |
| 0.618 | 0.014 | 0.663 | Vasodilator, peripheral | 0.663 0.009 DB14219 | DB14219 | |
| 0.631 | 0.045 | 0.646 | Antiinflammatory | 0.646 0.042 DB14219 | DB14219 | |
| 0.565 | 0.012 | 0.565 | GABA C receptor rho-3 antagonist | 0.466 0.036 DB14219 | ||
| 0.556 | 0.003 | 0.71 | GABA C receptor agonist | 0.71 0.002 DB14219 | DB14219 | |
| 0.586 | 0.052 | 0.586 | Apoptosis agonist | 0.555 0.059 DB14219 | ||
| 0.556 | 0.024 | 0.594 | Cholesterol antagonist | 0.594 0.019 DB14219 | DB14219 | |
| 0.542 | 0.016 | 0.559 | Antioxidant | 0.559 0.014 DB14219 | DB14219 | |
| 0.535 | 0.01 | 0.647 | Platelet antagonist | 0.647 0.005 DB14219 | DB14219 | |
| 0.526 | 0.017 | 0.574 | Apoptosis antagonist | 0.574 0.012 DB14219 | DB14219 | |
| 0.519 | 0.014 | 0.519 | Free radical scavenger | 0.514 0.015 DB14219 | ||
| 0.507 | 0.005 | 0.609 | Alpha-N-acetylglucosaminidase inhibitor | 0.609 0.004 DB14219 | DB14219 | |
| 0.498 | 0.002 | 0.742 | Fumarate hydratase inhibitor | 0.742 0.001 DB14219 | DB14219 | |
| 0.499 | 0.005 | 0.506 | Platelet adhesion inhibitor | 0.506 0.005 DB14219 | DB14219 | |
| 0.508 | 0.032 | 0.568 | Aldehyde oxidase inhibitor | 0.568 0.023 DB14219 | DB14219 | |
| 0.485 | 0.014 | 0.512 | Hypolipemic | 0.512 0.012 DB14219 | DB14219 | |
| 0.489 | 0.032 | 0.489 | Calcium channel L-type activator | 0.472 0.04 DB14219 | ||
| 0.471 | 0.017 | 0.471 | Tumour necrosis factor alpha release inhibitor | 0.382 0.03 DB14219 | ||
| 0.48 | 0.039 | 0.48 | 5 Hydroxytryptamine release inhibitor | 0.466 0.045 DB14219 | ||
| 0.483 | 0.047 | 0.53 | Transcription factor NF kappa B inhibitor | 0.53 0.04 DB14219 | DB14219 | |
| 0.439 | 0.033 | 0.439 | Caspase 3 stimulant | 0.406 0.043 DB14219 | ||
| 0.424 | 0.017 | 0.424 | Calcium channel activator | 0.383 0.032 DB14219 | ||
| 0.442 | 0.04 | 0.549 | Antithrombotic | 0.549 0.022 DB14219 | DB14219 | |
| 0.403 | 0.004 | 0.598 | Succinate dehydrogenase inhibitor | 0.598 0.002 DB14219 | DB14219 | |
| 0.439 | 0.043 | 0.439 | Thioredoxin glutathione reductase inhibitor | 0.382 0.064 DB14219 | ||
| 0.432 | 0.04 | 0.432 | 5 Hydroxytryptamine release stimulant | 0.295 0.071 DB14219 | ||
| 0.409 | 0.025 | 0.409 | Nitric oxide antagonist | 0.376 0.028 DB14219 | ||
| 0.392 | 0.009 | 0.412 | Tyrosine 3 hydroxylase inhibitor | 0.412 0.007 DB14219 | DB14219 | |
| 0.399 | 0.023 | 0.399 | Vasodilator | 0.391 0.025 DB14219 | ||
| 0.401 | 0.028 | 0.409 | DNA damaging | 0.409 0.027 DB14219 | DB14219 | |
| 0.399 | 0.027 | 0.414 | Superoxide dismutase inhibitor | 0.414 0.024 DB14219 | DB14219 | |
| 0.393 | 0.022 | 0.431 | Peroxidase inhibitor | 0.431 0.016 DB14219 | DB14219 | |
| 0.38 | 0.009 | 0.38 | Protein kinase stimulant | 0.38 0.01 DB14219 | ||
| 0.386 | 0.018 | 0.465 | Anesthetic general | 0.465 0.01 DB14219 | DB14219 | |
| 0.38 | 0.018 | 0.38 | 5 Hydroxytryptamine uptake stimulant | 0.34 0.029 DB14219 | ||
| 0.432 | 0.074 | 0.432 | Ca2+/calmodulin-dependent protein kinase kinase A inhibitor | 0.353 0.147 DB14219 | ||
| 0.379 | 0.025 | 0.433 | DNA synthesis inhibitor | 0.433 0.018 DB14219 | DB14219 | |
| 0.358 | 0.009 | 0.358 | Amyloid beta precursor protein antagonist | 0.293 0.019 DB14219 | ||
| 0.346 | 0.003 | 0.346 | Human rhinovirus A protease inhibitor | 0.242 0.005 DB14219 | ||
| 0.364 | 0.03 | 0.368 | Insulysin inhibitor | 0.368 0.029 DB14219 | DB14219 | |
| 0.405 | 0.073 | 0.475 | Histamine release inhibitor | 0.475 0.038 DB14219 | DB14219 | |
| 0.337 | 0.007 | 0.383 | Cystathionine beta-synthase inhibitor | 0.383 0.005 DB14219 | DB14219 | |
| 0.373 | 0.045 | 0.373 | Vasodilator, coronary | 0.342 0.059 DB14219 | ||
| 0.339 | 0.014 | 0.374 | Gastrin inhibitor | 0.374 0.006 DB14219 | DB14219 | |
| 0.319 | 0.005 | 0.319 | Falcipain inhibitor | 0.193 0.017 DB14219 | ||
| 0.319 | 0.005 | 0.319 | Falcipain 2 inhibitor | 0.191 0.015 DB14219 | ||
| 0.318 | 0.005 | 0.318 | GABA C receptor rho-2 antagonist | 0.262 0.01 DB14219 | ||
| 0.315 | 0.005 | 0.436 | Histidine decarboxylase inhibitor | 0.436 0.003 DB14219 | DB14219 | |
| 0.325 | 0.027 | 0.325 | RNA-directed DNA polymerase inhibitor | 0.293 0.033 DB14219 | ||
| 0.298 | 0.008 | 0.337 | Ferrochelatase inhibitor | 0.337 0.005 DB14219 | DB14219 | |
| 0.309 | 0.021 | 0.338 | Glyceraldehyde-3-phosphate dehydrogenase inhibitor | 0.338 0.014 DB14219 | DB14219 | |
| 0.313 | 0.033 | 0.353 | Platelet aggregation inhibitor | 0.353 0.025 DB14219 | DB14219 | |
| 0.284 | 0.007 | 0.401 | Catalase inhibitor | 0.401 0.004 DB14219 | DB14219 | |
| 0.291 | 0.013 | 0.291 | 3C-like protease (Human coronavirus) inhibitor | 0.209 0.047 DB14219 | ||
| 0.332 | 0.057 | 0.379 | Lipoxygenase inhibitor | 0.379 0.043 DB14219 | DB14219 | |
| 0.321 | 0.046 | 0.484 | Hypoglycemic | 0.484 0.017 DB14219 | DB14219 | |
| 0.368 | 0.092 | 0.404 | Antibacterial | 0.404 0.075 DB14219 | DB14219 | |
| 0.295 | 0.02 | 0.303 | Interferon gamma antagonist | 0.303 0.019 DB14219 | DB14219 | |
| 0.274 | 0.005 | 0.283 | HIV-1 integrase (Strand Transfer) inhibitor | 0.283 0.005 DB14219 | DB14219 | |
| 0.269 | 0.005 | 0.465 | Alcohol oxidase inhibitor | 0.465 0.004 DB14219 | DB14219 | |
| 0.273 | 0.009 | 0.273 | ATPase inhibitor | 0.272 0.009 DB14219 | ||
| 0.311 | 0.048 | 0.311 | Transcription factor STAT3 inhibitor | 0.244 0.088 DB14219 | ||
| 0.28 | 0.02 | 0.326 | Phospholipase C inhibitor | 0.326 0.016 DB14219 | DB14219 | |
| 0.266 | 0.009 | 0.303 | Adenylate kinase inhibitor | 0.303 0.007 DB14219 | DB14219 | |
| 0.326 | 0.069 | 0.378 | Immunomodulator | 0.378 0.051 DB14219 | DB14219 | |
| 0.289 | 0.033 | 0.322 | Hepatoprotectant | 0.322 0.024 DB14219 | DB14219 | |
| 0.256 | 0.004 | 0.256 | Toll-Like receptor 4 antagonist | 0.218 0.005 DB14219 | ||
| 0.26 | 0.01 | 0.26 | Antibacterial (Helicobacter pylori) | 0.255 0.011 DB14219 | ||
| 0.27 | 0.021 | 0.27 | Nitric-oxide synthase stimulant | 0.24 0.04 DB14219 | ||
| 0.252 | 0.006 | 0.268 | HIV-1 integrase (3'-Processing) inhibitor | 0.268 0.006 DB14219 | DB14219 | |
| 0.291 | 0.05 | 0.345 | Pyruvate kinase inhibitor | 0.345 0.035 DB14219 | DB14219 | |
| 0.249 | 0.008 | 0.249 | Protease inhibitor | 0.185 0.018 DB14219 | ||
| 0.314 | 0.075 | 0.349 | Immunostimulant | 0.349 0.065 DB14219 | DB14219 | |
| 0.245 | 0.007 | 0.245 | GABA C receptor antagonist | 0.239 0.007 DB14219 | ||
| 0.272 | 0.035 | 0.272 | P-glycoprotein inhibitor | 0.18 0.079 DB14219 | ||
| 0.249 | 0.013 | 0.331 | Expectorant | 0.331 0.007 DB14219 | DB14219 | |
| 0.24 | 0.005 | 0.24 | GABA C receptor rho-1 antagonist | 0.232 0.005 DB14219 | ||
| 0.328 | 0.099 | 0.394 | Immunosuppressant | 0.394 0.066 DB14219 | DB14219 | |
| 0.236 | 0.007 | 0.236 | Photosensitizer | 0.236 0.007 DB14219 | ||
| 0.289 | 0.063 | 0.289 | Transcription factor STAT inhibitor | 0.212 0.122 DB14219 | ||
| 0.228 | 0.003 | 0.418 | Aconitate hydratase inhibitor | 0.418 0.002 DB14219 | DB14219 | |
| 0.243 | 0.018 | 0.321 | DNA polymerase I inhibitor | 0.321 0.01 DB14219 | DB14219 | |
| 0.256 | 0.031 | 0.314 | Insulin sensitizer | 0.314 0.013 DB14219 | DB14219 | |
| 0.228 | 0.004 | 0.228 | Acetylcholine release stimulant | 0.159 0.012 DB14219 | ||
| 0.234 | 0.01 | 0.249 | Arachidonic acid antagonist | 0.249 0.006 DB14219 | DB14219 | |
| 0.25 | 0.028 | 0.273 | Amylase inhibitor | 0.273 0.023 DB14219 | DB14219 | |
| 0.278 | 0.06 | 0.283 | Interleukin agonist | 0.283 0.057 DB14219 | DB14219 | |
| 0.225 | 0.011 | 0.253 | Carbonic anhydrase XIII inhibitor | 0.253 0.008 DB14219 | DB14219 | |
| 0.223 | 0.011 | 0.291 | Carbonic anhydrase VI inhibitor | 0.291 0.006 DB14219 | DB14219 | |
| 0.264 | 0.053 | 0.264 | Amyloid beta aggregation inhibitor | 0.25 0.058 DB14219 | ||
| 0.241 | 0.03 | 0.241 | Melanin inhibitor | 0.24 0.03 DB14219 | ||
| 0.247 | 0.04 | 0.272 | Neurotrophic factor enhancer | 0.272 0.028 DB14219 | DB14219 | |
| 0.216 | 0.009 | 0.229 | Gastric antisecretory | 0.229 0.008 DB14219 | DB14219 | |
| 0.21 | 0.004 | 0.21 | 3C-Like protease (SARS coronavirus) inhibitor | 0.146 0.01 DB14219 | ||
| 0.234 | 0.03 | 0.234 | Thiol protease inhibitor | 0.221 0.033 DB14219 | ||
| 0.246 | 0.044 | 0.282 | Non-steroidal antiinflammatory agent | 0.282 0.032 DB14219 | DB14219 | |
| 0.214 | 0.014 | 0.255 | UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor | 0.255 0.009 DB14219 | DB14219 | |
| 0.205 | 0.006 | 0.223 | DOPA decarboxylase inhibitor | 0.223 0.005 DB14219 | DB14219 | |
| 0.211 | 0.012 | 0.211 | Calcium antagonist | 0.128 0.031 DB14219 | ||
| 0.233 | 0.035 | 0.353 | Protein-tyrosine phosphatase inhibitor | 0.353 0.012 DB14219 | DB14219 | |
| 0.206 | 0.01 | 0.261 | Triose-phosphate isomerase inhibitor | 0.261 0.006 DB14219 | DB14219 | |
| 0.226 | 0.031 | 0.303 | Phospholipase A2 inhibitor | 0.303 0.013 DB14219 | DB14219 | |
| 0.2 | 0.006 | 0.226 | Heat shock protein 70 antagonist | 0.226 0.004 DB14219 | DB14219 | |
| 0.215 | 0.021 | 0.215 | Neurotrophic factor | 0.157 0.053 DB14219 | ||
| 0.202 | 0.01 | 0.346 | Glutamate dehydrogenase inhibitor | 0.346 0.005 DB14219 | DB14219 | |
| 0.211 | 0.022 | 0.221 | 5-Lipoxygenase inhibitor | 0.221 0.02 DB14219 | DB14219 | |
| 0.208 | 0.02 | 0.215 | Toll-Like receptor 2 antagonist | 0.215 0.018 DB14219 | DB14219 | |
| 0.192 | 0.004 | 0.192 | Ca2+-transporting ATPase inhibitor | 0.186 0.005 DB14219 | ||
| 0.207 | 0.02 | 0.207 | Interleukin 4 antagonist | 0.176 0.032 DB14219 | ||
| 0.238 | 0.052 | 0.244 | DNA methyltransferase I inhibitor | 0.244 0.05 DB14219 | DB14219 | |
| 0.193 | 0.009 | 0.193 | Thioredoxin inhibitor | 0.141 0.02 DB14219 | ||
| 0.197 | 0.013 | 0.197 | Vanilloid 1 agonist | 0.193 0.014 DB14219 | ||
| 0.224 | 0.04 | 0.224 | Tumour necrosis factor antagonist | 0.153 0.097 DB14219 | ||
| 0.22 | 0.036 | 0.22 | 5 Hydroxytryptamine 3E antagonist | 0.171 0.133 DB14219 | ||
| 0.187 | 0.003 | 0.187 | Granulocyte macrophage colony stimulating factor agonist | 0.161 0.004 DB14219 | ||
| 0.195 | 0.012 | 0.274 | Phosphofructokinase-1 inhibitor | 0.274 0.006 DB14219 | DB14219 | |
| 0.199 | 0.018 | 0.199 | UDP-glucose 4-epimerase inhibitor | 0.185 0.02 DB14219 | ||
| 0.194 | 0.016 | 0.196 | Adenylate cyclase stimulant | 0.196 0.015 DB14219 | DB14219 | |
| 0.185 | 0.008 | 0.286 | Glutamate decarboxylase inhibitor | 0.286 0.004 DB14219 | DB14219 | |
| 0.25 | 0.075 | 0.25 | 5 Hydroxytryptamine 1E antagonist | |||
| 0.233 | 0.058 | 0.235 | DNA methylase inhibitor | 0.235 0.057 DB14219 | DB14219 | |
| 0.189 | 0.016 | 0.212 | Mucolytic | 0.212 0.011 DB14219 | DB14219 | |
| 0.184 | 0.012 | 0.209 | NADH dehydrogenase inhibitor | 0.209 0.01 DB14219 | DB14219 | |
| 0.19 | 0.018 | 0.249 | Carbonic anhydrase III inhibitor | 0.249 0.009 DB14219 | DB14219 | |
| 0.193 | 0.021 | 0.193 | Microtubule formation inhibitor | 0.192 0.022 DB14219 | ||
| 0.177 | 0.005 | 0.266 | NMDA receptor agonist | 0.266 0.004 DB14219 | DB14219 | |
| 0.196 | 0.029 | 0.209 | Aldehyde dehydrogenase inhibitor | 0.209 0.026 DB14219 | DB14219 | |
| 0.235 | 0.071 | 0.235 | Cyclic AMP phosphodiesterase inhibitor | 0.19 0.101 DB14219 | ||
| 0.195 | 0.032 | 0.213 | Cell wall synthesis inhibitor | 0.213 0.025 DB14219 | DB14219 | |
| 0.168 | 0.005 | 0.179 | Glycine receptor agonist | 0.179 0.005 DB14219 | DB14219 | |
| 0.165 | 0.003 | 0.165 | Exportin-1 inhibitor | 0.138 0.004 DB14219 | ||
| 0.194 | 0.034 | 0.219 | Mannose-6-phosphate isomerase inhibitor | 0.219 0.021 DB14219 | DB14219 | |
| 0.173 | 0.013 | 0.179 | Electrolyte absorption antagonist | 0.179 0.011 DB14219 | DB14219 | |
| 0.167 | 0.007 | 0.167 | Glutamate release inhibitor | 0.148 0.01 DB14219 | ||
| 0.175 | 0.016 | 0.228 | Porphobilinogen synthase inhibitor | 0.228 0.009 DB14219 | DB14219 | |
| 0.163 | 0.005 | 0.228 | Transcription factor AP-1 inhibitor | 0.228 0.004 DB14219 | DB14219 | |
| 0.254 | 0.097 | 0.259 | Hypoxia-inducible factor 1 alpha inhibitor | 0.259 0.093 DB14219 | DB14219 | |
| 0.162 | 0.008 | 0.162 | Thioredoxin reductase inhibitor | 0.122 0.016 DB14219 | ||
| 0.187 | 0.033 | 0.27 | Protein-tyrosine phosphatase 1B inhibitor | 0.27 0.014 DB14219 | DB14219 | |
| 0.192 | 0.039 | 0.201 | Neurotensin receptor agonist | 0.201 0.034 DB14219 | DB14219 | |
| 0.168 | 0.016 | 0.168 | Prolactin inhibitor | 0.158 0.019 DB14219 | ||
| 0.17 | 0.017 | 0.188 | Caspase 3 inhibitor | 0.188 0.012 DB14219 | DB14219 | |
| 0.156 | 0.007 | 0.176 | GABA aminotransferase inhibitor | 0.176 0.005 DB14219 | DB14219 | |
| 0.288 | 0.139 | 0.288 | 15-Lipoxygenase inhibitor | 0.287 0.14 DB14219 | ||
| 0.158 | 0.01 | 0.207 | Glutathione S-transferase inhibitor | 0.207 0.005 DB14219 | DB14219 | |
| 0.167 | 0.02 | 0.193 | HIV-1 integrase (Overall Integration) inhibitor | 0.193 0.013 DB14219 | DB14219 | |
| 0.178 | 0.033 | 0.178 | Proteasome inhibitor | 0.152 0.045 DB14219 | ||
| 0.152 | 0.007 | 0.152 | ATPase (Vacuolar H+) inhibitor | 0.146 0.009 DB14219 | ||
| 0.177 | 0.033 | 0.246 | Cholesterol synthesis inhibitor | 0.246 0.018 DB14219 | DB14219 | |
| 0.185 | 0.042 | 0.185 | Tubulin antagonist | 0.108 0.093 DB14219 | ||
| 0.151 | 0.009 | 0.166 | Acyl-CoA dehydrogenase inhibitor | 0.166 0.008 DB14219 | DB14219 | |
| 0.153 | 0.011 | 0.189 | Carbamoyl phosphate synthetase inhibitor | 0.189 0.008 DB14219 | DB14219 | |
| 0.148 | 0.012 | 0.188 | Ornithine decarboxylase inhibitor | 0.188 0.005 DB14219 | DB14219 | |
| 0.143 | 0.007 | 0.143 | Protease 3C (Human rhinovirus) inhibitor | 0.106 0.013 DB14219 | ||
| 0.17 | 0.034 | 0.17 | Cyclooxygenase 3 inhibitor | 0.162 0.039 DB14219 | ||
| 0.16 | 0.025 | 0.16 | TRPA1 agonist | 0.139 0.039 DB14219 | ||
| 0.174 | 0.039 | 0.223 | Monophenol monooxygenase inhibitor | 0.223 0.028 DB14219 | DB14219 | |
| 0.144 | 0.01 | 0.179 | Biliverdin reductase inhibitor | 0.179 0.007 DB14219 | DB14219 | |
| 0.172 | 0.04 | 0.172 | Anesthetic local | 0.11 0.075 DB14219 | ||
| 0.138 | 0.007 | 0.138 | Maillard reaction inhibitor | 0.125 0.009 DB14219 | ||
| 0.136 | 0.005 | 0.136 | Estrogen-related receptor beta agonist | 0.129 0.007 DB14219 | ||
| 0.146 | 0.015 | 0.172 | Carbonic anhydrase V inhibitor | 0.172 0.01 DB14219 | DB14219 | |
| 0.175 | 0.046 | 0.175 | Cytokine production inhibitor | 0.164 0.053 DB14219 | ||
| 0.16 | 0.032 | 0.16 | Falcipain 3 inhibitor | 0.121 0.053 DB14219 | ||
| 0.138 | 0.01 | 0.158 | Carbonic anhydrase VB inhibitor | 0.158 0.008 DB14219 | DB14219 | |
| 0.133 | 0.006 | 0.146 | NMDA receptor glycine site agonist | 0.146 0.005 DB14219 | DB14219 | |
| 0.164 | 0.039 | 0.279 | Cell adhesion inhibitor | 0.279 0.012 DB14219 | DB14219 | |
| 0.177 | 0.052 | 0.177 | Hexokinase inhibitor | 0.176 0.052 DB14219 | ||
| 0.144 | 0.02 | 0.144 | NAD(P)H dehydrogenase (quinone) inhibitor | 0.14 0.022 DB14219 | ||
| 0.125 | 0.003 | 0.172 | Glucose-6-phosphate isomerase inhibitor | 0.172 0.002 DB14219 | DB14219 | |
| 0.155 | 0.034 | 0.247 | Chelator | 0.247 0.017 DB14219 | DB14219 | |
| 0.137 | 0.017 | 0.213 | Keratolytic | 0.213 0.007 DB14219 | DB14219 | |
| 0.169 | 0.048 | 0.169 | CF transmembrane conductance regulator agonist | 0.14 0.096 DB14219 | ||
| 0.132 | 0.013 | 0.21 | Aldose reductase inhibitor | 0.21 0.007 DB14219 | DB14219 | |
| 0.134 | 0.014 | 0.155 | Carbonic anhydrase VA inhibitor | 0.155 0.01 DB14219 | DB14219 | |
| 0.13 | 0.014 | 0.14 | Leukotriene synthesis inhibitor | 0.14 0.011 DB14219 | DB14219 | |
| 0.207 | 0.091 | 0.257 | Angiogenesis stimulant | 0.257 0.067 DB14219 | DB14219 | |
| 0.142 | 0.028 | 0.156 | Creatine kinase inhibitor | 0.156 0.021 DB14219 | DB14219 | |
| 0.149 | 0.035 | 0.156 | Xanthine oxidase inhibitor | 0.156 0.032 DB14219 | DB14219 | |
| 0.122 | 0.009 | 0.125 | Caspase 9 inhibitor | 0.125 0.009 DB14219 | DB14219 | |
| 0.118 | 0.005 | 0.118 | Squalene synthetase inhibitor | 0.102 0.006 DB14219 | ||
| 0.172 | 0.061 | 0.172 | Cytidine deaminase inhibitor | |||
| 0.144 | 0.032 | 0.144 | Antineoplastic antibiotic | 0.144 0.032 DB14219 | ||
| 0.137 | 0.026 | 0.137 | Anabolic | 0.132 0.03 DB14219 | ||
| 0.154 | 0.044 | 0.169 | Alkylator | 0.169 0.037 DB14219 | DB14219 | |
| 0.153 | 0.044 | 0.153 | Cathepsin H inhibitor | 0.134 0.059 DB14219 | ||
| 0.206 | 0.096 | 0.206 | Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase inhibitor | 0.153 0.139 DB14219 | ||
| 0.125 | 0.015 | 0.125 | Interferon agonist | 0.12 0.017 DB14219 | ||
| 0.123 | 0.014 | 0.163 | HIV-1 integrase inhibitor | 0.163 0.007 DB14219 | DB14219 | |
| 0.145 | 0.038 | 0.145 | Sphingosine 1-phosphate receptor 4 antagonist | 0.138 0.045 DB14219 | ||
| 0.12 | 0.015 | 0.12 | Caspase 7 inhibitor | 0.101 0.028 DB14219 | ||
| 0.164 | 0.059 | 0.2 | Lipid peroxidase inhibitor | 0.2 0.042 DB14219 | DB14219 | |
| 0.146 | 0.044 | 0.146 | Beta amyloid protein antagonist | 0.097 0.094 DB14219 | ||
| 0.119 | 0.017 | 0.121 | Na+ K+ transporting ATPase inhibitor | 0.121 0.016 DB14219 | DB14219 | |
| 0.121 | 0.02 | 0.223 | Peroxisome proliferator-activated receptor gamma agonist | 0.223 0.005 DB14219 | DB14219 | |
| 0.142 | 0.041 | 0.165 | Aminopeptidase B inhibitor | 0.165 0.032 DB14219 | DB14219 | |
| 0.207 | 0.107 | 0.207 | Neuropeptide Y2 antagonist | 0.181 0.158 DB14219 | ||
| 0.108 | 0.008 | 0.124 | Glutamate (mGluR6) antagonist | 0.124 0.005 DB14219 | DB14219 | |
| 0.136 | 0.037 | 0.136 | Carbonic anhydrase XV inhibitor | 0.116 0.05 DB14219 | ||
| 0.157 | 0.057 | 0.157 | MAO inhibitor | |||
| 0.125 | 0.026 | 0.125 | Glutamate (mGluR7) agonist | 0.111 0.041 DB14219 | ||
| 0.102 | 0.004 | 0.183 | Kynurenine 3 monooxygenase inhibitor | 0.183 0.003 DB14219 | DB14219 | |
| 0.107 | 0.009 | 0.124 | Carbonic anhydrase XIV inhibitor | 0.124 0.006 DB14219 | DB14219 | |
| 0.2 | 0.102 | 0.2 | Aryl hydrocarbon receptor agonist | |||
| 0.271 | 0.173 | 0.271 | Transcription factor inhibitor | |||
| 0.238 | 0.141 | 0.348 | Sodium/bile acid cotransporter inhibitor | 0.348 0.041 DB14219 | DB14219 | |
| 0.121 | 0.023 | 0.121 | Interleukin 5 antagonist | 0.096 0.046 DB14219 | ||
| 0.102 | 0.006 | 0.104 | MDM2 inhibitor | 0.104 0.005 DB14219 | DB14219 | |
| 0.105 | 0.008 | 0.105 | Glutamate (mGluR7) antagonist | 0.103 0.009 DB14219 | ||
| 0.112 | 0.017 | 0.146 | Argininosuccinate synthase inhibitor | 0.146 0.012 DB14219 | DB14219 | |
| 0.112 | 0.017 | 0.112 | MAP3K7 inhibitor | 0.076 0.045 DB14219 | ||
| 0.132 | 0.038 | 0.153 | Mediator release inhibitor | 0.153 0.027 DB14219 | DB14219 | |
| 0.124 | 0.032 | 0.133 | Interleukin 1 beta converting enzyme inhibitor | 0.133 0.026 DB14219 | DB14219 | |
| 0.1 | 0.009 | 0.1 | Potassium channel intermediate-conductance Ca-activated blocker | 0.063 0.036 DB14219 | ||
| 0.102 | 0.012 | 0.102 | Interferon inducer | 0.097 0.014 DB14219 | ||
| 0.205 | 0.115 | 0.213 | Spasmolytic | 0.213 0.109 DB14219 | DB14219 | |
| 0.093 | 0.005 | 0.093 | Ryanodine receptor antagonist | 0.085 0.007 DB14219 | ||
| 0.11 | 0.024 | 0.11 | Glycine receptor antagonist | 0.1 0.032 DB14219 | ||
| 0.179 | 0.093 | 0.179 | Psychostimulant | 0.155 0.112 DB14219 | ||
| 0.132 | 0.047 | 0.132 | MAO A inhibitor | |||
| 0.134 | 0.05 | 0.145 | DNA repair enzyme inhibitor | 0.145 0.036 DB14219 | DB14219 | |
| 0.108 | 0.025 | 0.108 | Vanilloid agonist | 0.091 0.046 DB14219 | ||
| 0.112 | 0.029 | 0.147 | Macrophage migration inhibitory factor inhibitor | 0.147 0.016 DB14219 | DB14219 | |
| 0.137 | 0.054 | 0.137 | Adenylate cyclase inhibitor | 0.136 0.055 DB14219 | ||
| 0.097 | 0.015 | 0.108 | Mannitol-1-phosphate 5-dehydrogenase inhibitor | 0.108 0.013 DB14219 | DB14219 | |
| 0.18 | 0.099 | 0.18 | Histone acetyltransferase inhibitor | |||
| 0.083 | 0.005 | 0.083 | Pregnane X receptor antagonist | 0.077 0.008 DB14219 | ||
| 0.085 | 0.008 | 0.106 | Lysophosphatidic acid 3 receptor antagonist | 0.106 0.004 DB14219 | DB14219 | |
| 0.146 | 0.069 | 0.147 | Sphingosine 1-phosphate receptor 5 antagonist | 0.147 0.066 DB14219 | DB14219 | |
| 0.103 | 0.026 | 0.121 | Aminopeptidase I inhibitor | 0.121 0.019 DB14219 | DB14219 | |
| 0.113 | 0.038 | 0.113 | Lanosterol 14 alpha demethylase inhibitor | 0.102 0.053 DB14219 | ||
| 0.106 | 0.031 | 0.185 | Cell adhesion molecule inhibitor | 0.185 0.011 DB14219 | DB14219 | |
| 0.118 | 0.043 | 0.118 | Sphingomyelinase inhibitor | 0.098 0.062 DB14219 | ||
| 0.106 | 0.031 | 0.133 | Cathepsin G inhibitor | 0.133 0.024 DB14219 | DB14219 | |
| 0.143 | 0.068 | 0.143 | Pregnane X receptor agonist | 0.127 0.109 DB14219 | ||
| 0.219 | 0.145 | 0.219 | Thyroid hormone antagonist | 0.196 0.165 DB14219 | ||
| 0.145 | 0.072 | 0.145 | Neuropeptide Y1 antagonist | |||
| 0.154 | 0.082 | 0.154 | Heat shock protein 90 alpha antagonist | |||
| 0.218 | 0.146 | 0.218 | Prostaglandin dehydrogenase inhibitor | |||
| 0.192 | 0.121 | 0.192 | Calpain inhibitor | |||
| 0.098 | 0.027 | 0.13 | Phenylalanine 4-hydroxylase inhibitor | 0.13 0.015 DB14219 | DB14219 | |
| 0.078 | 0.009 | 0.078 | Adenylate cyclase 1 inhibitor | 0.051 0.025 DB14219 | ||
| 0.134 | 0.065 | 0.134 | Sphingosine 1-phosphate receptor 2 antagonist | 0.131 0.072 DB14219 | ||
| 0.138 | 0.069 | 0.188 | Bone formation stimulant | 0.188 0.039 DB14219 | DB14219 | |
| 0.138 | 0.07 | 0.138 | Calcium channel blocker | |||
| 0.211 | 0.145 | 0.211 | Thyroid hormone beta antagonist | 0.181 0.173 DB14219 | ||
| 0.105 | 0.04 | 0.141 | Aminoacyl-tRNA synthetase inhibitor | 0.141 0.022 DB14219 | DB14219 | |
| 0.084 | 0.019 | 0.084 | Nitric oxide donor | 0.062 0.044 DB14219 | ||
| 0.09 | 0.026 | 0.099 | GABA B receptor agonist | 0.099 0.017 DB14219 | DB14219 | |
| 0.097 | 0.033 | 0.099 | D-Ala-D-Ala ligase inhibitor | 0.099 0.031 DB14219 | DB14219 | |
| 0.084 | 0.02 | 0.106 | Ornithine carbamoyltransferase inhibitor | 0.106 0.015 DB14219 | DB14219 | |
| 0.07 | 0.008 | 0.146 | Prostaglandin agonist | 0.146 0.004 DB14219 | DB14219 | |
| 0.076 | 0.014 | 0.111 | Thromboxane synthase inhibitor | 0.111 0.005 DB14219 | DB14219 | |
| 0.067 | 0.005 | 0.08 | Kainate receptor agonist | 0.08 0.004 DB14219 | DB14219 | |
| 0.088 | 0.025 | 0.088 | S-adenosyl-L-methionine decarboxylase inhibitor | 0.073 0.052 DB14219 | ||
| 0.067 | 0.005 | 0.095 | Glutamate (mGluR8) agonist | 0.095 0.003 DB14219 | DB14219 | |
| 0.132 | 0.07 | 0.132 | Toll-Like receptor antagonist | |||
| 0.067 | 0.006 | 0.067 | Guanylate cyclase inhibitor | 0.067 0.006 DB14219 | ||
| 0.114 | 0.052 | 0.114 | Beta glucuronidase inhibitor | 0.098 0.072 DB14219 | ||
| 0.107 | 0.047 | 0.213 | Uric acid excretion stimulant | 0.213 0.011 DB14219 | DB14219 | |
| 0.07 | 0.01 | 0.106 | Retinoid X receptor agonist | 0.106 0.004 DB14219 | DB14219 | |
| 0.062 | 0.003 | 0.07 | Prostaglandin F2 alpha agonist | 0.07 0.003 DB14219 | DB14219 | |
| 0.097 | 0.039 | 0.097 | Inducible nitric-oxide synthase inhibitor | 0.079 0.063 DB14219 | ||
| 0.086 | 0.028 | 0.134 | Leukotriene antagonist | 0.134 0.013 DB14219 | DB14219 | |
| 0.078 | 0.021 | 0.109 | Thromboxane antagonist | 0.109 0.009 DB14219 | DB14219 | |
| 0.175 | 0.118 | 0.175 | Antiamyloidogenic | 0.168 0.125 DB14219 | ||
| 0.072 | 0.015 | 0.081 | Alpha-mannosidase inhibitor | 0.081 0.011 DB14219 | DB14219 | |
| 0.12 | 0.063 | 0.12 | Interleukin 1b antagonist | 0.103 0.077 DB14219 | ||
| 0.07 | 0.014 | 0.07 | Squalene epoxidase inhibitor | 0.052 0.03 DB14219 | ||
| 0.08 | 0.025 | 0.084 | Purinergic P2X1 antagonist | 0.084 0.023 DB14219 | DB14219 | |
| 0.074 | 0.019 | 0.099 | Thromboxane A2 antagonist | 0.099 0.008 DB14219 | DB14219 | |
| 0.064 | 0.009 | 0.075 | Membrane dipeptidase inhibitor | 0.075 0.006 DB14219 | DB14219 | |
| 0.07 | 0.016 | 0.07 | Glucose-6-phosphate translocase inhibitor | 0.056 0.028 DB14219 | ||
| 0.063 | 0.009 | 0.063 | Farnesoid X receptor agonist | 0.062 0.009 DB14219 | ||
| 0.063 | 0.01 | 0.085 | Nicotinic acid receptor agonist | 0.085 0.005 DB14219 | DB14219 | |
| 0.055 | 0.002 | 0.055 | Carbonic anhydrase X inhibitor | 0.053 0.002 DB14219 | ||
| 0.055 | 0.002 | 0.055 | Carbonic anhydrase VIII inhibitor | 0.053 0.002 DB14219 | ||
| 0.068 | 0.016 | 0.068 | Potassium channel Kv1.3 blocker | 0.041 0.04 DB14219 | ||
| 0.084 | 0.031 | 0.084 | Acetylcholine M5 receptor agonist | |||
| 0.094 | 0.041 | 0.094 | mTOR complex 2 inhibitor | |||
| 0.138 | 0.087 | 0.138 | Heat shock protein 90 antagonist | |||
| 0.113 | 0.063 | 0.122 | GABA receptor agonist | 0.122 0.055 DB14219 | DB14219 | |
| 0.201 | 0.151 | 0.201 | 12-Lipoxygenase inhibitor | |||
| 0.106 | 0.057 | 0.106 | MAO B inhibitor | |||
| 0.07 | 0.022 | 0.117 | Peroxisome proliferator-activated receptor alpha agonist | 0.117 0.009 DB14219 | DB14219 | |
| 0.083 | 0.036 | 0.083 | Calcium channel L-type blocker | |||
| 0.132 | 0.086 | 0.141 | Cyclooxygenase inhibitor | 0.141 0.078 DB14219 | DB14219 | |
| 0.135 | 0.088 | 0.135 | Hemostatic | 0.12 0.115 DB14219 | ||
| 0.063 | 0.018 | 0.063 | Carbonic anhydrase VII inhibitor | 0.063 0.018 DB14219 | ||
| 0.055 | 0.01 | 0.055 | 3-Hydroxyanthranilate 3,4-dioxygenase inhibitor | 0.055 0.01 DB14219 | ||
| 0.067 | 0.022 | 0.105 | Leukotriene B4 antagonist | 0.105 0.009 DB14219 | DB14219 | |
| 0.049 | 0.004 | 0.049 | Calcium-independent phospholipase A2 inhibitor | 0.043 0.008 DB14219 | ||
| 0.072 | 0.029 | 0.075 | 3-Oxoacyl-[acyl-carrier-protein] synthase inhibitor | 0.075 0.028 DB14219 | DB14219 | |
| 0.047 | 0.004 | 0.05 | Lysophosphatidic acid receptor 1 agonist | 0.05 0.004 DB14219 | DB14219 | |
| 0.05 | 0.007 | 0.054 | HMG CoA reductase inhibitor | 0.054 0.005 DB14219 | DB14219 | |
| 0.143 | 0.1 | 0.143 | Interleukin 6 antagonist | 0.138 0.11 DB14219 | ||
| 0.05 | 0.008 | 0.05 | Melatonin receptor 1A agonist | 0.037 0.017 DB14219 | ||
| 0.071 | 0.029 | 0.071 | Transcription factor RelA inhibitor | |||
| 0.081 | 0.04 | 0.081 | Vanilloid 4 agonist | 0.07 0.063 DB14219 | ||
| 0.094 | 0.053 | 0.094 | Phosphodiesterase I inhibitor | |||
| 0.06 | 0.02 | 0.069 | Toll-Like receptor 2 agonist | 0.069 0.018 DB14219 | DB14219 | |
| 0.098 | 0.058 | 0.098 | Breast cancer-resistant protein inhibitor | |||
| 0.058 | 0.018 | 0.067 | Mannosidase inhibitor | 0.067 0.013 DB14219 | DB14219 | |
| 0.097 | 0.057 | 0.101 | Bile acid receptor antagonist | 0.101 0.047 DB14219 | DB14219 | |
| 0.057 | 0.018 | 0.057 | Dopamine beta hydroxylase inhibitor | 0.05 0.031 DB14219 | ||
| 0.048 | 0.009 | 0.064 | Prostaglandin D2 agonist | 0.064 0.005 DB14219 | DB14219 | |
| 0.061 | 0.022 | 0.064 | Heparanase inhibitor | 0.064 0.017 DB14219 | DB14219 | |
| 0.054 | 0.016 | 0.065 | GABA B receptor antagonist | 0.065 0.01 DB14219 | DB14219 | |
| 0.06 | 0.021 | 0.068 | CD45 antagonist | 0.068 0.016 DB14219 | DB14219 | |
| 0.083 | 0.046 | 0.083 | CYP2A6 inhibitor | |||
| 0.057 | 0.019 | 0.057 | Leukocyte elastase inhibitor | 0.047 0.026 DB14219 | ||
| 0.05 | 0.013 | 0.065 | Retinoid X receptor antagonist | 0.065 0.005 DB14219 | DB14219 | |
| 0.052 | 0.015 | 0.052 | Factor XIIIa inhibitor | 0.038 0.025 DB14219 | ||
| 0.091 | 0.054 | 0.091 | Bromodomain-containing protein 2 inhibitor | |||
| 0.056 | 0.018 | 0.056 | Cytokine production stimulant | 0.046 0.04 DB14219 | ||
| 0.059 | 0.022 | 0.062 | Adenosine deaminase inhibitor | 0.062 0.019 DB14219 | DB14219 | |
| 0.076 | 0.039 | 0.087 | Sphingosine 1-phosphate receptor 4 agonist | 0.087 0.032 DB14219 | DB14219 | |
| 0.052 | 0.015 | 0.052 | Dihydropteroate synthase inhibitor | 0.048 0.018 DB14219 | ||
| 0.039 | 0.003 | 0.039 | Lysophosphatidic acid receptor 3 agonist | 0.034 0.003 DB14219 | ||
| 0.09 | 0.054 | 0.09 | Antineoplastic alkaloid | 0.077 0.069 DB14219 | ||
| 0.105 | 0.07 | 0.105 | 5 Hydroxytryptamine 3A agonist | |||
| 0.236 | 0.2 | 0.236 | DNA directed DNA polymerase inhibitor | |||
| 0.036 | 0.002 | 0.036 | Calcineurin inhibitor | 0.027 0.002 DB14219 | ||
| 0.119 | 0.084 | 0.119 | NADPH oxidase inhibitor | |||
| 0.037 | 0.003 | 0.041 | Isoleucine-tRNA ligase inhibitor | 0.041 0.003 DB14219 | DB14219 | |
| 0.075 | 0.042 | 0.075 | Phospholipase D inhibitor | 0.069 0.056 DB14219 | ||
| 0.231 | 0.199 | 0.231 | Alpha-glucosidase inhibitor | |||
| 0.059 | 0.027 | 0.059 | Immunoglobulin Fc receptor antagonist | 0.052 0.05 DB14219 | ||
| 0.071 | 0.039 | 0.074 | Carbonic anhydrase inhibitor | 0.074 0.038 DB14219 | DB14219 | |
| 0.119 | 0.087 | 0.119 | Alkaline phosphatase inhibitor | |||
| 0.043 | 0.011 | 0.056 | Retinoid X alpha receptor antagonist | 0.056 0.004 DB14219 | DB14219 | |
| 0.067 | 0.035 | 0.067 | Calcium channel P-type blocker | |||
| 0.074 | 0.042 | 0.074 | Elastase 1 inhibitor | |||
| 0.06 | 0.029 | 0.064 | Leukotriene C antagonist | 0.064 0.022 DB14219 | DB14219 | |
| 0.042 | 0.011 | 0.07 | Lysophosphatidic acid 2 receptor antagonist | 0.07 0.005 DB14219 | DB14219 | |
| 0.08 | 0.05 | 0.08 | Nicotinic alpha4beta2 receptor antagonist | |||
| 0.096 | 0.066 | 0.096 | Nitric-oxide synthase inhibitor | |||
| 0.046 | 0.016 | 0.094 | Retinoid X alpha receptor agonist | 0.094 0.005 DB14219 | DB14219 | |
| 0.109 | 0.079 | 0.138 | Interleukin 8 antagonist | 0.138 0.042 DB14219 | DB14219 | |
| 0.041 | 0.011 | 0.041 | Methionyl aminopeptidase 1 inhibitor | 0.032 0.021 DB14219 | ||
| 0.065 | 0.035 | 0.091 | Xanthine dehydrogenase inhibitor | 0.091 0.019 DB14219 | DB14219 | |
| 0.052 | 0.023 | 0.052 | Benzodiazepine antagonist | |||
| 0.079 | 0.049 | 0.079 | MAP kinase kinase 7 inhibitor | 0.076 0.058 DB14219 | ||
| 0.047 | 0.018 | 0.05 | GABA uptake inhibitor | 0.05 0.016 DB14219 | DB14219 | |
| 0.082 | 0.053 | 0.082 | Acetylcholine nicotinic antagonist | |||
| 0.065 | 0.036 | 0.069 | Carbonic anhydrase stimulant | 0.069 0.032 DB14219 | DB14219 | |
| 0.064 | 0.035 | 0.064 | Dopamine uptake inhibitor | |||
| 0.059 | 0.031 | 0.059 | Dihydroorotate oxidase inhibitor | 0.058 0.033 DB14219 | ||
| 0.039 | 0.012 | 0.039 | Epoxide hydrolase 1 inhibitor | 0.029 0.025 DB14219 | ||
| 0.075 | 0.048 | 0.075 | Potassium channel (Tandem pore domain) blocker | |||
| 0.047 | 0.02 | 0.047 | Dopamine D5 agonist | 0.037 0.031 DB14219 | ||
| 0.049 | 0.023 | 0.055 | AICAR transformylase inhibitor | 0.055 0.018 DB14219 | DB14219 | |
| 0.057 | 0.031 | 0.057 | Nicotinic alpha3beta2 receptor antagonist | |||
| 0.038 | 0.012 | 0.043 | Glutamate (mGluR3) agonist | 0.043 0.007 DB14219 | DB14219 | |
| 0.038 | 0.013 | 0.038 | Hypoxanthine phosphoribosyltransferase inhibitor | 0.035 0.015 DB14219 | ||
| 0.042 | 0.018 | 0.042 | Vanilloid 3 antagonist | |||
| 0.084 | 0.061 | 0.087 | Transcription factor NF kappa B stimulant | 0.087 0.056 DB14219 | DB14219 | |
| 0.082 | 0.059 | 0.082 | CC chemokine 5 receptor agonist | |||
| 0.072 | 0.049 | 0.091 | Peroxisome proliferator-activated receptor gamma antagonist | 0.091 0.022 DB14219 | DB14219 | |
| 0.032 | 0.01 | 0.032 | Nicotinic acid receptor 2 antagonist | 0.03 0.013 DB14219 | ||
| 0.06 | 0.038 | 0.06 | Botulinum neurotoxin type A inhibitor | 0.056 0.045 DB14219 | ||
| 0.026 | 0.004 | 0.03 | Thromboxane A2 agonist | 0.03 0.003 DB14219 | DB14219 | |
| 0.048 | 0.026 | 0.048 | Dihydroorotase inhibitor | 0.044 0.032 DB14219 | ||
| 0.047 | 0.026 | 0.089 | Glutamate (mGluR group III) agonist | 0.089 0.011 DB14219 | DB14219 | |
| 0.088 | 0.067 | 0.088 | Potassium channel (Ca-activated) activator | 0.085 0.07 DB14219 | ||
| 0.024 | 0.004 | 0.024 | Carbonic anhydrase XI inhibitor | 0.02 0.004 DB14219 | ||
| 0.11 | 0.09 | 0.122 | Cyclooxygenase 1 inhibitor | 0.122 0.078 DB14219 | DB14219 | |
| 0.032 | 0.012 | 0.042 | Prostaglandin H2 antagonist | 0.042 0.005 DB14219 | DB14219 | |
| 0.226 | 0.207 | 0.226 | DNA polymerase beta inhibitor | |||
| 0.039 | 0.02 | 0.041 | Phosphoglycerate kinase inhibitor | 0.041 0.018 DB14219 | DB14219 | |
| 0.11 | 0.091 | 0.11 | Cyclooxygenase 2 inhibitor | 0.106 0.097 DB14219 | ||
| 0.046 | 0.027 | 0.051 | Glutamate (mGluR group III) antagonist | 0.051 0.019 DB14219 | DB14219 | |
| 0.029 | 0.011 | 0.029 | Vanilloid 2 agonist | 0.026 0.016 DB14219 | ||
| 0.04 | 0.022 | 0.05 | Arginase inhibitor | 0.05 0.015 DB14219 | DB14219 | |
| 0.065 | 0.047 | 0.065 | Beta adrenoreceptor antagonist | 0.065 0.046 DB14219 | ||
| 0.03 | 0.012 | 0.03 | Hedgehog signaling activator | 0.028 0.018 DB14219 | ||
| 0.09 | 0.072 | 0.091 | Interleukin 12 antagonist | 0.091 0.07 DB14219 | DB14219 | |
| 0.058 | 0.041 | 0.058 | Cathepsin L inhibitor | |||
| 0.025 | 0.008 | 0.025 | Neuraminidase (Influenza B) inhibitor | 0.024 0.009 DB14219 | ||
| 0.032 | 0.015 | 0.032 | Purinergic P2Y15 antagonist | 0.027 0.023 DB14219 | ||
| 0.024 | 0.008 | 0.024 | Factor XIII inhibitor | |||
| 0.044 | 0.027 | 0.044 | Nerve growth factor antagonist | |||
| 0.03 | 0.014 | 0.03 | Methionyl aminopeptidase 2 inhibitor | 0.026 0.017 DB14219 | ||
| 0.039 | 0.023 | 0.039 | Inosine monophosphate dehydrogenase inhibitor | |||
| 0.049 | 0.034 | 0.049 | HCV NS3/NS4A protease inhibitor | 0.047 0.038 DB14219 | ||
| 0.024 | 0.009 | 0.032 | Retinoid X beta receptor antagonist | 0.032 0.004 DB14219 | DB14219 | |
| 0.038 | 0.023 | 0.048 | Glutamate (mGluR3) antagonist | 0.048 0.014 DB14219 | DB14219 | |
| 0.043 | 0.028 | 0.047 | Angiotensin AT1 receptor antagonist | 0.047 0.021 DB14219 | DB14219 | |
| 0.037 | 0.022 | 0.041 | Tryptophan 5 hydroxylase inhibitor | 0.041 0.013 DB14219 | DB14219 | |
| 0.044 | 0.029 | 0.049 | Glutamate (mGluR4) antagonist | 0.049 0.022 DB14219 | DB14219 | |
| 0.047 | 0.032 | 0.085 | Phosphorylase inhibitor | 0.085 0.015 DB14219 | DB14219 | |
| 0.05 | 0.036 | 0.05 | Prolyl endopeptidase inhibitor | |||
| 0.047 | 0.033 | 0.047 | Aldosterone antagonist | |||
| 0.057 | 0.043 | 0.057 | Lipocortins synthesis agonist | 0.057 0.041 DB14219 | ||
| 0.018 | 0.004 | 0.018 | Immunosuppressant Cyclosporine-like | 0.015 0.005 DB14219 | ||
| 0.032 | 0.018 | 0.032 | Elastase 2B inhibitor | |||
| 0.032 | 0.018 | 0.032 | Elastase 3B inhibitor | |||
| 0.032 | 0.018 | 0.032 | Elastase 3A inhibitor | |||
| 0.031 | 0.017 | 0.032 | Uridine phosphorylase inhibitor | 0.032 0.016 DB14219 | DB14219 | |
| 0.025 | 0.012 | 0.027 | Glutamate (mGluR1a) agonist | 0.027 0.011 DB14219 | DB14219 | |
| 0.017 | 0.004 | 0.017 | 3C-Like protease (MERS coronavirus) inhibitor | 0.012 0.008 DB14219 | ||
| 0.047 | 0.034 | 0.065 | Antimetabolite | 0.065 0.023 DB14219 | DB14219 | |
| 0.045 | 0.031 | 0.045 | Fructose-1,6-bisphosphatase inhibitor | |||
| 0.028 | 0.016 | 0.028 | Glucosylceramidase stimulant | |||
| 0.019 | 0.008 | 0.019 | Telomerase stimulant | 0.019 0.009 DB14219 | ||
| 0.02 | 0.01 | 0.02 | Antibiotic Anthracycline-like | 0.02 0.012 DB14219 | ||
| 0.052 | 0.041 | 0.052 | Carbonic anhydrase IX inhibitor | |||
| 0.034 | 0.024 | 0.048 | Glutamate (mGluR4) agonist | 0.048 0.011 DB14219 | DB14219 | |
| 0.02 | 0.009 | 0.02 | Methylmalonyl-CoA mutase inhibitor | 0.02 0.008 DB14219 | ||
| 0.038 | 0.028 | 0.041 | Leukotriene C4 antagonist | 0.041 0.021 DB14219 | DB14219 | |
| 0.026 | 0.016 | 0.026 | Complement factor 1s inhibitor | |||
| 0.026 | 0.016 | 0.036 | NMDA receptor glycine site antagonist | 0.036 0.009 DB14219 | DB14219 | |
| 0.098 | 0.088 | 0.098 | Calcium channel (voltage-sensitive) blocker | |||
| 0.042 | 0.033 | 0.043 | Geranyltranstransferase inhibitor | 0.043 0.032 DB14219 | DB14219 | |
| 0.021 | 0.012 | 0.021 | Inosine monophosphate dehydrogenase 2 inhibitor | 0.017 0.016 DB14219 | ||
| 0.018 | 0.009 | 0.019 | Vitamin D receptor agonist | 0.019 0.007 DB14219 | DB14219 | |
| 0.052 | 0.043 | 0.052 | Epithelial sodium channel blocker | |||
| 0.072 | 0.063 | 0.078 | Metalloproteinase-2 inhibitor | 0.078 0.054 DB14219 | DB14219 | |
| 0.042 | 0.034 | 0.047 | Purinergic P2Y antagonist | 0.047 0.029 DB14219 | DB14219 | |
| 0.015 | 0.006 | 0.015 | Calcium-dependent phospholipase A2 inhibitor | 0.013 0.008 DB14219 | ||
| 0.014 | 0.006 | 0.026 | Glutamate (mGluR6) agonist | 0.026 0.003 DB14219 | DB14219 | |
| 0.069 | 0.06 | 0.069 | Adenosine A3 receptor antagonist | |||
| 0.114 | 0.106 | 0.114 | Nav1.6 sodium channel blocker | |||
| 0.066 | 0.057 | 0.066 | Benzodiazepine agonist | |||
| 0.02 | 0.012 | 0.023 | Caspase 8 inhibitor | 0.023 0.009 DB14219 | DB14219 | |
| 0.024 | 0.016 | 0.045 | Prostaglandin E2 agonist | 0.045 0.006 DB14219 | DB14219 | |
| 0.037 | 0.029 | 0.037 | Alpha 1d adrenoreceptor agonist | |||
| 0.017 | 0.01 | 0.033 | Prostacyclin agonist | 0.033 0.005 DB14219 | DB14219 | |
| 0.119 | 0.111 | 0.19 | Thrombolytic | 0.19 0.057 DB14219 | DB14219 | |
| 0.021 | 0.015 | 0.029 | Lysophosphatidic acid 1 receptor antagonist | 0.029 0.007 DB14219 | DB14219 | |
| 0.039 | 0.032 | 0.039 | Plasmepsin II inhibitor | 0.038 0.037 DB14219 | ||
| 0.028 | 0.021 | 0.033 | Liver X receptor beta antagonist | 0.033 0.017 DB14219 | DB14219 | |
| 0.023 | 0.016 | 0.105 | Retinoic acid receptor agonist | 0.105 0.004 DB14219 | DB14219 | |
| 0.023 | 0.016 | 0.028 | ICAM 1 antagonist | 0.028 0.008 DB14219 | DB14219 | |
| 0.046 | 0.04 | 0.046 | Bombesin 2 receptor antagonist | 0.045 0.042 DB14219 | ||
| 0.03 | 0.024 | 0.03 | Estradiol 17 beta-dehydrogenase 3 inhibitor | |||
| 0.051 | 0.045 | 0.051 | Beta 1 adrenoreceptor antagonist | 0.049 0.047 DB14219 | ||
| 0.012 | 0.006 | 0.015 | Thromboxane agonist | 0.015 0.005 DB14219 | DB14219 | |
| 0.03 | 0.025 | 0.036 | ATP citrate lysase inhibitor | 0.036 0.017 DB14219 | DB14219 | |
| 0.087 | 0.082 | 0.087 | Urease inhibitor | |||
| 0.013 | 0.009 | 0.013 | 1-Deoxy-D-xylulose-5-phosphate reductoisomerase inhibitor | |||
| 0.021 | 0.017 | 0.045 | Prostaglandin EP2 agonist | 0.045 0.007 DB14219 | DB14219 | |
| 0.026 | 0.021 | 0.055 | NMDA 2D receptor antagonist | 0.055 0.006 DB14219 | DB14219 | |
| 0.065 | 0.061 | 0.065 | Epoxide hydrolase inhibitor | |||
| 0.081 | 0.078 | 0.094 | Alcohol dehydrogenase inhibitor | 0.094 0.06 DB14219 | DB14219 | |
| 0.032 | 0.029 | 0.036 | Angiotensin II receptor antagonist | 0.036 0.021 DB14219 | DB14219 | |
| 0.026 | 0.023 | 0.034 | LFA antagonist | 0.034 0.011 DB14219 | DB14219 | |
| 0.023 | 0.02 | 0.025 | Glutamate (mGluR1) agonist | 0.025 0.016 DB14219 | DB14219 | |
| 0.034 | 0.031 | 0.034 | Diamine oxidase inhibitor | |||
| 0.031 | 0.028 | 0.037 | Free fatty acid receptor 1 antagonist | 0.037 0.019 DB14219 | DB14219 | |
| 0.041 | 0.038 | 0.041 | Heme oxygenase inhibitor | |||
| 0.075 | 0.073 | 0.075 | Histamine N-methyltransferase inhibitor | |||
| 0.025 | 0.022 | 0.08 | Leukotriene B4 receptor 1 antagonist | 0.08 0.004 DB14219 | DB14219 | |
| 0.045 | 0.042 | 0.045 | Topoisomerase II beta inhibitor | |||
| 0.024 | 0.022 | 0.03 | Lysine carboxypeptidase inhibitor | 0.03 0.015 DB14219 | DB14219 | |
| 0.022 | 0.02 | 0.022 | Fructose-1,6-bisphosphatase 1 inhibitor | |||
| 0.04 | 0.039 | 0.04 | Dihydrofolate reductase inhibitor | |||
| 0.037 | 0.035 | 0.047 | Liver X receptor alpha agonist | 0.047 0.022 DB14219 | DB14219 | |
| 0.047 | 0.045 | 0.047 | Carbonic anhydrase I inhibitor | 0.047 0.046 DB14219 | ||
| 0.024 | 0.023 | 0.024 | Calcium-sensing receptor agonist | |||
| 0.027 | 0.026 | 0.027 | Nicotinic alpha3beta4 receptor agonist | |||
| 0.02 | 0.019 | 0.02 | Glutaminyl-peptide cyclotransferase inhibitor | |||
| 0.233 | 0.232 | 0.552 | Cyclophilin D inhibitor | 0.552 0.037 DB14219 | DB14219 | |
| 0.087 | 0.086 | 0.087 | Phosphodiesterase 6D inhibitor | |||
| 0.017 | 0.016 | 0.017 | Estrogen-related receptor gamma agonist | |||
| 0.029 | 0.029 | 0.049 | Peroxisome proliferator-activated receptor delta agonist | 0.049 0.013 DB14219 | DB14219 | |
| 0.05 | 0.051 | 0.274 | Prostaglandin EP2 antagonist | 0.274 0.005 DB14219 | DB14219 | |
| 0.033 | 0.035 | 0.056 | Urate transporter 1 inhibitor | 0.056 0.016 DB14219 | DB14219 | |
| 0.033 | 0.035 | 0.037 | Integrin alpha2 antagonist | 0.037 0.026 DB14219 | DB14219 | |
| 0.01 | 0.014 | 0.037 | Prostaglandin EP4 agonist | 0.037 0.006 DB14219 | DB14219 | |
| 0.023 | 0.027 | 0.031 | Endothelin receptor antagonist | 0.031 0.017 DB14219 | DB14219 | |
| 0.039 | 0.043 | 0.046 | Thymidylate synthase inhibitor | 0.046 0.034 DB14219 | DB14219 | |
| 0.035 | 0.039 | 0.038 | Carbonic anhydrase IV inhibitor | 0.038 0.035 DB14219 | DB14219 | |
| 0.023 | 0.027 | 0.025 | Integrin alpha2beta1 antagonist | 0.025 0.021 DB14219 | DB14219 | |
| 0.029 | 0.034 | 0.034 | Carnitine palmitoyltransferase 1 inhibitor | 0.034 0.023 DB14219 | DB14219 | |
| 0.021 | 0.026 | 0.043 | Prostaglandin EP4 antagonist | 0.043 0.01 DB14219 | DB14219 | |
| 0.024 | 0.029 | 0.059 | Retinoid X gamma receptor antagonist | 0.059 0.002 DB14219 | DB14219 | |
| 0.111 | 0.116 | 0.127 | Diuretic | 0.127 0.097 DB14219 | DB14219 | |
| 0.036 | 0.042 | 0.043 | VCAM-1 antagonist | 0.043 0.018 DB14219 | DB14219 | |
| 0.01 | 0.015 | 0.014 | Angiotensin AT1B receptor antagonist | 0.014 0.009 DB14219 | DB14219 | |
| 0.036 | 0.042 | 0.043 | VCAM antagonist | 0.043 0.018 DB14219 | DB14219 | |
| 0.028 | 0.035 | 0.034 | Carnitine palmitoyltransferase inhibitor | 0.034 0.023 DB14219 | DB14219 | |
| 0.009 | 0.015 | 0.014 | Integrin beta2 antagonist | 0.014 0.007 DB14219 | DB14219 | |
| 0.086 | 0.093 | 0.113 | AMP-activated protein kinase stimulant | 0.113 0.056 DB14219 | DB14219 | |
| 0.043 | 0.049 | 0.047 | Protein 50S ribosomal subunit inhibitor | 0.047 0.043 DB14219 | DB14219 | |
| 0.022 | 0.029 | 0.03 | Thyroid hormone agonist | 0.03 0.013 DB14219 | DB14219 | |
| 0.028 | 0.037 | 0.031 | Carboxypeptidase B inhibitor | 0.031 0.027 DB14219 | DB14219 | |
| 0.039 | 0.052 | 0.235 | Prostaglandin antagonist | 0.235 0.005 DB14219 | DB14219 | |
| 0.078 | 0.092 | 0.314 | ABCA1 expression enhancer | 0.314 0.005 DB14219 | DB14219 | |
| 0.086 | 0.1 | 0.114 | Folate antagonist | 0.114 0.044 DB14219 | DB14219 | |
| 0.023 | 0.04 | 0.033 | Kainate receptor 2 antagonist | 0.033 0.028 DB14219 | DB14219 | |
| 0.048 | 0.065 | 0.065 | NMDA 2C receptor antagonist | 0.065 0.039 DB14219 | DB14219 | |
| 0.046 | 0.063 | 0.079 | DNA helicase inhibitor | 0.079 0.011 DB14219 | DB14219 | |
| 0.065 | 0.084 | 0.073 | Estrogen receptor alpha antagonist | 0.073 0.061 DB14219 | DB14219 | |
| 0.013 | 0.032 | 0.066 | Retinoic acid alpha receptor antagonist | 0.066 0.003 DB14219 | DB14219 | |
| 0.013 | 0.034 | 0.082 | Prostaglandin D2 antagonist | 0.082 0.005 DB14219 | DB14219 | |
| 0.014 | 0.039 | 0.038 | Leukotriene B4 receptor 2 antagonist | 0.038 0.005 DB14219 | DB14219 | |
| 0.008 | 0.033 | 0.02 | Peroxisome proliferator-activated receptor alpha antagonist | 0.02 0.016 DB14219 | DB14219 | |
| 0.013 | 0.038 | 0.178 | Retinoid X beta receptor agonist | 0.178 0.003 DB14219 | DB14219 | |
| 0.016 | 0.043 | 0.047 | Retinoic acid gamma receptor agonist | 0.047 0.004 DB14219 | DB14219 | |
| 0.013 | 0.043 | 0.137 | Retinoid X gamma receptor agonist | 0.137 0.003 DB14219 | DB14219 | |
| 0.124 | 0.154 | 0.18 | Lipocortins synthesis antagonist | 0.18 0.071 DB14219 | DB14219 | |
| 0.031 | 0.063 | 0.042 | Integrin alpha1beta1 antagonist | 0.042 0.016 DB14219 | DB14219 | |
| 0.01 | 0.043 | 0.061 | Retinoic acid receptor antagonist | 0.061 0.004 DB14219 | DB14219 | |
| 0.015 | 0.053 | 0.058 | Prostacyclin antagonist | 0.058 0.01 DB14219 | DB14219 | |
| 0.023 | 0.063 | 0.032 | RNA-directed RNA polymerase inhibitor | 0.032 0.027 DB14219 | DB14219 | |
| 0.027 | 0.068 | 0.09 | Retinoic acid alpha receptor agonist | 0.09 0.004 DB14219 | DB14219 | |
| 0.013 | 0.055 | 0.113 | Prostaglandin EP3 antagonist | 0.113 0.005 DB14219 | DB14219 | |
| 0.007 | 0.05 | 0.021 | Integrin alpha4beta7 antagonist | 0.021 0.014 DB14219 | DB14219 | |
| 0.012 | 0.063 | 0.043 | Retinoic acid beta receptor agonist | 0.043 0.004 DB14219 | DB14219 | |
| 0.125 | 0.179 | 0.152 | Catenin beta inhibitor | 0.152 0.1 DB14219 | DB14219 | |
| 0.041 | 0.101 | 0.066 | Prostaglandin F2 alpha antagonist | 0.066 0.037 DB14219 | DB14219 | |
| 0.087 | 0.159 | 0.114 | Interleukin 1 antagonist | 0.114 0.098 DB14219 | DB14219 | |
| 0.012 | 0.088 | 0.046 | GP IIb/IIIa receptor antagonist | 0.046 0.035 DB14219 | DB14219 | |
| 0.004 | 0.082 | 0.018 | Retinoic acid beta receptor antagonist | 0.018 0.005 DB14219 | DB14219 | |
| 0.029 | 0.107 | 0.078 | Selectin antagonist | 0.078 0.038 DB14219 | DB14219 | |
| 0.005 | 0.084 | 0.016 | Retinoic acid receptor gamma antagonist | 0.016 0.005 DB14219 | DB14219 | |
| 0.023 | 0.105 | 0.042 | Glutamate (mGluR8) antagonist | 0.042 0.014 DB14219 | DB14219 | |
| 0.04 | 0.129 | 0.054 | Adenine nucleotide translocase inhibitor | 0.054 0.043 DB14219 | DB14219 | |
| 0.024 | 0.118 | 0.082 | Plasminogen activator inhibitor antagonist | 0.082 0.014 DB14219 | DB14219 | |
| 0.098 | 0.193 | 0.202 | Interleukin antagonist | 0.202 0.083 DB14219 | DB14219 | |
| 0.034 | 0.144 | 0.067 | CDC25B inhibitor | 0.067 0.042 DB14219 | DB14219 | |
| 0.019 | 0.13 | 0.094 | Prostaglandin E2 antagonist | 0.094 0.016 DB14219 | DB14219 | |
| 0.158 | 0.275 | 0.285 | Interleukin 2 agonist | 0.285 0.085 DB14219 | DB14219 | |
| 0.004 | 0.125 | 0.029 | VLA-4 antagonist | 0.029 0.018 DB14219 | DB14219 | |
| 0.015 | 0.143 | 0.037 | Peroxisome proliferator-activated receptor delta antagonist | 0.037 0.017 DB14219 | DB14219 | |
| 0.124 | 0.289 | 0.208 | Peptidyltransferase inhibitor | 0.208 0.089 DB14219 | DB14219 | |
| 0.005 | 0.173 | 0.018 | Vitronectin receptor antagonist | 0.018 0.017 DB14219 | DB14219 | |
| 0.077 | 0.247 | 0.262 | NOS3 expression enhancer | 0.262 0.024 DB14219 | DB14219 | |
| 0.008 | 0.185 | 0.052 | Integrin antagonist | 0.052 0.026 DB14219 | DB14219 | |
| 0.069 | 0.251 | 0.132 | Farnesoid X receptor antagonist | 0.132 0.079 DB14219 | DB14219 | |
| 0.006 | 0.2 | 0.024 | Integrin beta5 antagonist | 0.024 0.011 DB14219 | DB14219 | |
| 0.027 | 0.237 | 0.068 | CDC25A inhibitor | 0.068 0.061 DB14219 | DB14219 | |
| 0.115 | 0.346 | 0.258 | Toll-Like receptor agonist | 0.258 0.141 DB14219 | DB14219 | |
| 0.115 | 0.348 | 0.257 | Toll-Like receptor 7 agonist | 0.257 0.142 DB14219 | DB14219 | |
| 0.043 | 0.34 | 0.124 | Estrogen antagonist | 0.124 0.049 DB14219 | DB14219 | Ext | Pa | Pi | Pmax | Activity | Other Results | ID Pa_max |