Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.6870.0020.687Neurokinin antagonist

0.686 0.002 DBMET01379

0.617 0.003 DBMET01380

0.6770.0160.719Analgesic

0.658 0.018 DBMET01379

0.719 0.012 DBMET01380

DBMET01380
0.6630.0020.663Neurokinin 1 antagonist

0.662 0.002 DBMET01379

0.59 0.002 DBMET01380

0.5180.0030.518Substance P antagonist

0.515 0.003 DBMET01379

0.445 0.003 DBMET01380

0.4750.0460.505Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.505 0.031 DBMET01379

0.393 0.107 DBMET01380

DBMET01379
0.3440.0030.344Neurokinin 3 antagonist

0.336 0.003 DBMET01379

0.286 0.003 DBMET01380

0.3930.0630.407MAP kinase kinase 6 inhibitor

0.407 0.054 DBMET01379

0.321 0.116 DBMET01380

DBMET01379
0.330.0060.371Vanilloid antagonist

0.325 0.006 DBMET01379

0.371 0.005 DBMET01380

DBMET01380
0.2920.0380.292EphB2 antagonist

0.272 0.046 DBMET01379

0.198 0.089 DBMET01380

0.2520.0570.252Anticonvulsant

0.2 0.083 DBMET01379

0.216 0.072 DBMET01380

0.2030.0090.203Vanilloid 1 antagonist

0.188 0.01 DBMET01379

0.125 0.019 DBMET01380

0.1950.0080.195Interleukin 2 antagonist

0.18 0.01 DBMET01379

0.15 0.018 DBMET01380

0.2960.1130.346Toll-Like receptor 7 agonist

0.317 0.1 DBMET01379

0.346 0.084 DBMET01380

DBMET01380
0.1980.0170.198Calcium channel N-type blocker

0.161 0.031 DBMET01379

0.099 0.097 DBMET01380

0.2860.120.335Toll-Like receptor agonist

0.306 0.107 DBMET01379

0.335 0.09 DBMET01380

DBMET01380
0.2010.0360.212Cytokine production inhibitor

0.212 0.033 DBMET01379

0.111 0.099 DBMET01380

DBMET01379
0.1730.0230.173Ca(v)2.2 blocker

0.165 0.025 DBMET01379

0.111 0.042 DBMET01380

0.1580.020.158Hedgehog signaling inhibitor

0.151 0.023 DBMET01379

0.096 0.071 DBMET01380

0.1680.0450.168Ca2+/calmodulin-dependent protein kinase kinase B inhibitor

0.163 0.052 DBMET01379

0.144 0.085 DBMET01380

0.20.0930.2Potassium channel blocker

0.176 0.11 DBMET01379

0.2180.1190.235Ca2+/calmodulin-dependent kinase IV inhibitor

0.235 0.087 DBMET01379

0.218 0.12 DBMET01380

DBMET01379
0.1220.0350.145Protein kinase C delta inhibitor

0.145 0.024 DBMET01379

DBMET01379
0.1030.0260.105Syk tyrosine kinase inhibitor

0.105 0.026 DBMET01379

0.085 0.037 DBMET01380

DBMET01379
0.140.0710.14Protein-tyrosine kinase Lyn inhibitor

0.13 0.077 DBMET01379

0.1180.0590.118Calcium channel (voltage-sensitive) blocker

0.101 0.082 DBMET01379

0.0990.0420.099Bcr-Abl kinase inhibitor
0.1730.1180.173Potassium channel (Voltage-sensitive) blocker

0.155 0.133 DBMET01379

0.1120.060.112Granulocyte macrophage colony stimulating factor antagonist

0.098 0.074 DBMET01379

0.0880.0410.088Fibroblast growth factor 3 antagonist

0.079 0.052 DBMET01379

0.0640.0170.064Smo receptor antagonist

0.047 0.025 DBMET01379

0.0540.0140.054Nerve growth factor antagonist

0.039 0.037 DBMET01379

0.1190.0830.119Proto-oncogene tyrosine-protein kinase Yes inhibitor

0.116 0.086 DBMET01379

0.1410.1090.141TRKC antagonist

0.127 0.124 DBMET01379

0.0940.0640.098Interleukin 12 antagonist

0.098 0.056 DBMET01379

0.091 0.07 DBMET01380

DBMET01379
0.0570.0280.059Diacylglycerol O-acyltransferase inhibitor

0.059 0.026 DBMET01379

DBMET01379
0.1240.0970.127CC chemokine 6 receptor antagonist

0.127 0.081 DBMET01380

DBMET01380
0.1540.1270.154HERG channel blocker
0.0610.0360.065Protein kinase C theta inhibitor

0.065 0.029 DBMET01379

DBMET01379
0.0320.0070.032Apolipoprotein B inhibitor
0.030.0060.03Apolipoprotein B-100 inhibitor

0.018 0.012 DBMET01379

0.0570.0340.06Protein kinase C epsilon inhibitor

0.06 0.03 DBMET01379

DBMET01379
0.0680.0510.068Glutamate (mGluR group I) antagonist

0.064 0.058 DBMET01379

0.1130.0970.113Toll-Like receptor antagonist
0.0990.0860.099Protein-tyrosine kinase (PTK, not ETK, WZC) inhibitor
0.0990.0860.099Abl kinase inhibitor
0.0350.0230.035Gonadotropin-releasing hormone receptor antagonist

0.035 0.023 DBMET01379

0.030.0190.031Diacylglycerol O-acyltransferase 1 inhibitor

0.031 0.018 DBMET01379

DBMET01379
0.0190.0080.019Microsomal triglyceride transfer protein inhibitor

0.015 0.011 DBMET01379

0.0810.0710.088Protein kinase (Mos, Mil/Raf, MEKK, RIPK, TESK, LIMK, IRAK, ILK, Activin/TGF-beta) inhibitor

0.088 0.064 DBMET01379

DBMET01379
0.0550.0460.055Calcium channel T-type blocker
0.1760.1680.177Neuropeptide Y2 antagonist

0.177 0.166 DBMET01379

DBMET01379
0.060.0520.065 Hydroxytryptamine 1B antagonist
0.1080.1010.108Toll-Like receptor 9 antagonist
0.0780.0710.078Transforming growth factor beta 3 antagonist

0.078 0.073 DBMET01379

0.0560.0490.056TRPA1 antagonist
0.0680.0640.068Glutamate (mGluR) antagonist
0.0630.0610.07Raf kinase inhibitor

0.07 0.055 DBMET01379

DBMET01379
0.060.0610.075Protein kinase C alpha inhibitor

0.075 0.039 DBMET01379

DBMET01379
0.0460.0570.052Raf kinase C inhibitor

0.052 0.05 DBMET01379

DBMET01379
0.1790.1970.185MAP kinase kinase 3 inhibitor

0.185 0.171 DBMET01379

DBMET01379
0.1350.1540.155Focal adhesion kinase 2 inhibitor

0.155 0.122 DBMET01379

DBMET01379
0.0670.0930.091GABA A receptor agonist

0.091 0.046 DBMET01380

DBMET01380
0.0550.0840.068Nav1.8 sodium channel blocker

0.068 0.058 DBMET01379

DBMET01379
0.0870.1180.104Activin receptor-like kinase 4 inhibitor

0.104 0.077 DBMET01379

DBMET01379
0.0780.1110.107GABA receptor agonist

0.107 0.069 DBMET01380

DBMET01380
0.0640.1110.096Protein kinase C mu inhibitor

0.096 0.061 DBMET01379

DBMET01379
0.2040.270.376Cyclophilin D inhibitor

0.235 0.23 DBMET01379

0.376 0.105 DBMET01380

DBMET01380
0.1020.1920.12Death-associated protein kinase 1 inhibitor

0.12 0.114 DBMET01379

DBMET01379
0.0610.1680.106Glutamate receptor antagonist

0.106 0.09 DBMET01380

DBMET01380
0.0940.2210.163Hypolipemic

0.163 0.125 DBMET01380

DBMET01380
0.1490.2770.223Antiobesity

0.223 0.184 DBMET01379

0.223 0.183 DBMET01380

DBMET01380
0.0870.2370.129Interleukin 6 antagonist

0.129 0.127 DBMET01380

DBMET01380
0.0310.1970.069Protein kinase B beta inhibitor

0.069 0.059 DBMET01380

DBMET01380
0.1830.3580.347Antiinflammatory

0.347 0.175 DBMET01380

DBMET01380
0.0080.1890.0495 Hydroxytryptamine 2C agonist

0.049 0.028 DBMET01379

DBMET01379
0.0240.2350.102Androgen antagonist

0.102 0.045 DBMET01380

DBMET01380
0.0770.3570.191Lipocortins synthesis antagonist

0.191 0.062 DBMET01380

DBMET01380
0.0150.2970.061Androgen agonist

0.061 0.04 DBMET01380

DBMET01380
Ext Pa Pi Pmax Activity Other Results ID Pa_max