Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.9280.0010.928Alpha-N-acetylglucosaminidase inhibitor

0.852 0.002 DB03947

0.573 0.004 DBMET02033

0.8610.0020.861Alcohol oxidase inhibitor

0.674 0.003 DB03947

0.154 0.01 DBMET02033

0.8070.0040.807Hypoglycemic

0.495 0.015 DB03947

0.7980.0040.798Aldehyde oxidase inhibitor

0.748 0.005 DB03947

0.45 0.04 DBMET02033

0.7980.0070.839Cyclophilin D inhibitor

0.839 0.005 DB03947

0.574 0.032 DBMET02033

DB03947
0.77100.952Mannitol 2-dehydrogenase inhibitor

0.952 0 DB03947

0.93 0 DBMET02033

DB03947
0.6960.0010.764Triose-phosphate isomerase inhibitor

0.678 0.001 DB03947

0.764 0.001 DBMET02033

DBMET02033
0.6620.0030.662Chelator

0.263 0.015 DB03947

0.151 0.035 DBMET02033

0.6390.0040.639Interleukin 6 antagonist

0.323 0.012 DB03947

0.146 0.095 DBMET02033

0.6330.0070.6335 Hydroxytryptamine release inhibitor

0.547 0.02 DB03947

0.277 0.192 DBMET02033

0.6310.0090.631Immunosuppressant

0.484 0.037 DB03947

0.545 0.022 DBMET02033

0.620.0040.62Amylase inhibitor

0.421 0.008 DB03947

0.231 0.034 DBMET02033

0.6090.0040.609Peroxidase inhibitor

0.512 0.009 DB03947

0.23 0.052 DBMET02033

0.6090.0060.609Hypolipemic

0.446 0.018 DB03947

0.446 0.018 DBMET02033

0.5980.0190.598Cholesterol antagonist

0.514 0.03 DB03947

0.387 0.052 DBMET02033

0.5810.0020.581NADH dehydrogenase inhibitor

0.419 0.004 DB03947

0.533 0.003 DBMET02033

0.5810.0040.581Hematopoietic

0.107 0.029 DB03947

0.11 0.027 DBMET02033

0.5860.0160.5865 Hydroxytryptamine release stimulant

0.5 0.027 DB03947

0.181 0.139 DBMET02033

0.5830.0130.583Immunomodulator
0.60.0360.6Caspase 9 stimulant

0.536 0.048 DB03947

0.442 0.087 DBMET02033

0.5540.0160.554Histamine release inhibitor

0.472 0.039 DB03947

0.5280.0020.528UDP-glucose 4-epimerase inhibitor

0.491 0.003 DB03947

0.518 0.002 DBMET02033

0.5310.0230.531Vasodilator, peripheral

0.453 0.04 DB03947

0.269 0.114 DBMET02033

0.5120.0140.512Vasodilator, coronary

0.401 0.035 DB03947

0.274 0.11 DBMET02033

0.4960.0140.496DNA synthesis inhibitor

0.388 0.023 DB03947

0.479 0.015 DBMET02033

0.4880.0080.85Hepatoprotectant

0.85 0.002 DB03947

0.701 0.004 DBMET02033

DB03947
0.4680.0030.468Phenylalanine 4-hydroxylase inhibitor

0.327 0.004 DB03947

0.097 0.027 DBMET02033

0.4680.0020.568Phosphofructokinase-1 inhibitor

0.369 0.004 DB03947

0.568 0.002 DBMET02033

DBMET02033
0.4420.0170.442Vasodilator

0.217 0.091 DB03947

0.5060.0850.506Antiinflammatory

0.412 0.132 DB03947

0.433 0.12 DBMET02033

0.4120.0030.444Carbamoyl phosphate synthetase inhibitor

0.366 0.004 DB03947

0.444 0.003 DBMET02033

DBMET02033
0.4430.0380.469Immunostimulant

0.394 0.051 DB03947

0.469 0.033 DBMET02033

DBMET02033
0.430.0270.43Interleukin antagonist

0.372 0.035 DB03947

0.4460.0430.446GABA C receptor rho-3 antagonist

0.334 0.095 DB03947

0.4030.0020.403Plasmepsin I inhibitor
0.4030.0040.403Succinate dehydrogenase inhibitor

0.387 0.004 DB03947

0.251 0.022 DBMET02033

0.40.0040.4UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor

0.371 0.004 DB03947

0.365 0.004 DBMET02033

0.3970.0020.397Mannitol-1-phosphate 5-dehydrogenase inhibitor

0.29 0.004 DB03947

0.364 0.002 DBMET02033

0.4230.0310.423Antioxidant

0.214 0.105 DB03947

0.163 0.15 DBMET02033

0.390.0030.39Mannose-6-phosphate isomerase inhibitor

0.272 0.008 DB03947

0.365 0.004 DBMET02033

0.3910.0050.391Growth factor agonist
0.3970.0130.397Diuretic

0.156 0.072 DB03947

0.3950.0280.395Superoxide dismutase inhibitor

0.347 0.037 DB03947

0.430.0640.44Antibacterial

0.363 0.095 DB03947

0.44 0.06 DBMET02033

DBMET02033
0.3680.0050.368Expectorant

0.25 0.013 DB03947

0.211 0.018 DBMET02033

0.360.0020.36Alpha-mannosidase inhibitor

0.184 0.003 DB03947

0.09 0.008 DBMET02033

0.3570.0030.359Biliverdin reductase inhibitor

0.211 0.005 DB03947

0.359 0.002 DBMET02033

DBMET02033
0.360.0060.36GABA C receptor agonist

0.252 0.013 DB03947

0.113 0.055 DBMET02033

0.3510.0060.351Hexokinase inhibitor

0.222 0.025 DB03947

0.302 0.011 DBMET02033

0.3390.0020.339Mannosidase inhibitor

0.176 0.003 DB03947

0.079 0.009 DBMET02033

0.3390.0030.339Neuraminidase (influenza) inhibitor

0.244 0.004 DB03947

0.340.0040.34Mucolytic

0.245 0.007 DB03947

0.201 0.013 DBMET02033

0.3340.0050.419Adenylate kinase inhibitor

0.313 0.006 DB03947

0.419 0.003 DBMET02033

DBMET02033
0.3420.0140.342Peptidyltransferase inhibitor

0.272 0.037 DB03947

0.169 0.149 DBMET02033

0.3370.010.337Alkylator

0.223 0.02 DB03947

0.315 0.012 DBMET02033

0.3470.0240.52Anesthetic general

0.264 0.044 DB03947

0.52 0.007 DBMET02033

DBMET02033
0.3310.0090.331Aldehyde dehydrogenase inhibitor

0.288 0.013 DB03947

0.243 0.019 DBMET02033

0.330.010.33Insulin secretagoues

0.156 0.069 DB03947

0.320.0010.516Glucose-6-phosphate isomerase inhibitor

0.396 0 DB03947

0.516 0 DBMET02033

DBMET02033
0.410.0920.41Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.32 0.187 DB03947

0.3240.0080.404Interleukin 1b antagonist

0.404 0.005 DB03947

0.102 0.079 DBMET02033

DB03947
0.3480.0410.348Sodium/bile acid cotransporter inhibitor

0.264 0.113 DB03947

0.3360.0330.336Interleukin agonist

0.252 0.078 DB03947

0.226 0.098 DBMET02033

0.3490.0460.349Interleukin 2 agonist

0.265 0.103 DB03947

0.3010.0030.301Neuraminidase inhibitor

0.231 0.004 DB03947

0.062 0.041 DBMET02033

0.3160.0260.316Tyrosine 3 hydroxylase inhibitor

0.263 0.057 DB03947

0.3010.0110.301Nitric-oxide synthase stimulant

0.256 0.029 DB03947

0.171 0.15 DBMET02033

0.3480.0650.393Antithrombotic

0.277 0.106 DB03947

0.393 0.051 DBMET02033

DBMET02033
0.2880.0090.288Ferrochelatase inhibitor

0.179 0.028 DB03947

0.2810.0040.281Sphingomyelinase inhibitor

0.191 0.011 DB03947

0.218 0.007 DBMET02033

0.2830.0060.444Selectin antagonist

0.444 0.003 DB03947

0.349 0.004 DBMET02033

DB03947
0.2890.0170.289Hemostatic

0.13 0.096 DB03947

0.3080.0390.308Cyclic AMP phosphodiesterase inhibitor

0.218 0.081 DB03947

0.330.0640.33Calcium channel activator

0.253 0.144 DB03947

0.272 0.122 DBMET02033

0.2960.0320.376RNA-directed DNA polymerase inhibitor

0.221 0.073 DB03947

0.376 0.021 DBMET02033

DBMET02033
0.2830.020.452Phospholipase C inhibitor

0.21 0.038 DB03947

0.452 0.008 DBMET02033

DBMET02033
0.2720.0120.272MAP kinase kinase inhibitor

0.13 0.065 DB03947

0.380.1230.38Alpha-glucosidase inhibitor
0.2670.0130.267Cell wall synthesis inhibitor

0.184 0.038 DB03947

0.165 0.052 DBMET02033

0.2920.0380.299Gastrin inhibitor

0.299 0.034 DB03947

DB03947
0.2550.0070.288Glutamate dehydrogenase inhibitor

0.23 0.008 DB03947

0.288 0.006 DBMET02033

DBMET02033
0.2570.0080.257Catalase inhibitor

0.24 0.009 DB03947

0.168 0.022 DBMET02033

0.2950.0480.2955 Hydroxytryptamine uptake stimulant

0.228 0.106 DB03947

0.2530.0080.253Microtubule formation inhibitor

0.205 0.019 DB03947

0.133 0.048 DBMET02033

0.2470.0040.247Glutamate decarboxylase inhibitor

0.234 0.005 DB03947

0.141 0.015 DBMET02033

0.2830.0410.283MAP kinase kinase 2 inhibitor

0.158 0.114 DB03947

0.2540.0180.309Interleukin 1 antagonist

0.309 0.01 DB03947

DB03947
0.2440.0090.244Histidine decarboxylase inhibitor

0.207 0.012 DB03947

0.217 0.011 DBMET02033

0.2410.0070.241GABA C receptor antagonist

0.157 0.026 DB03947

0.121 0.052 DBMET02033

0.2370.0050.237Keratolytic

0.202 0.008 DB03947

0.186 0.01 DBMET02033

0.2310.0040.247Acyl-CoA dehydrogenase inhibitor

0.203 0.005 DB03947

0.247 0.003 DBMET02033

DBMET02033
0.2310.0050.231Adenylate cyclase stimulant

0.199 0.014 DB03947

0.182 0.024 DBMET02033

0.2490.0270.249Protein kinase stimulant

0.187 0.047 DB03947

0.181 0.049 DBMET02033

0.2590.0390.259Glyceraldehyde-3-phosphate dehydrogenase inhibitor

0.233 0.051 DB03947

0.24 0.047 DBMET02033

0.2310.0110.231MAP kinase kinase 5 inhibitor

0.183 0.057 DB03947

0.2270.0070.227Creatine kinase inhibitor

0.171 0.016 DB03947

0.102 0.057 DBMET02033

0.2290.0120.229Arachidonic acid antagonist

0.22 0.017 DB03947

0.226 0.014 DBMET02033

0.2190.0040.219HIV-1 protease inhibitor

0.041 0.032 DB03947

0.2880.0750.288Spasmolytic

0.167 0.147 DB03947

0.2150.0040.215Maillard reaction inhibitor

0.081 0.024 DB03947

0.2120.0030.212Aconitate hydratase inhibitor

0.195 0.003 DB03947

0.092 0.01 DBMET02033

0.3140.1070.66Antiobesity

0.66 0.014 DB03947

DB03947
0.2470.040.247Neurotrophic factor enhancer

0.216 0.062 DB03947

0.15 0.137 DBMET02033

0.2070.0050.207Interferon agonist

0.128 0.014 DB03947

0.093 0.035 DBMET02033

0.2080.0070.208GABA C receptor rho-1 antagonist

0.141 0.025 DB03947

0.088 0.082 DBMET02033

0.2180.0170.218Aminopeptidase B inhibitor

0.202 0.021 DB03947

0.145 0.04 DBMET02033

0.2410.040.241Insulin sensitizer

0.189 0.085 DB03947

0.2440.0430.244P-glycoprotein inhibitor

0.154 0.111 DB03947

0.149 0.118 DBMET02033

0.2310.0320.231Interferon gamma antagonist

0.175 0.053 DB03947

0.2670.0710.267DNA damaging
0.20.0070.2Aminopeptidase I inhibitor

0.182 0.008 DB03947

0.131 0.016 DBMET02033

0.2630.0730.263Cardiotonic
0.2230.0340.223Melanin inhibitor

0.198 0.042 DB03947

0.158 0.071 DBMET02033

0.2690.080.269Insulysin inhibitor

0.229 0.118 DB03947

0.1920.0040.192Ca2+-transporting ATPase inhibitor

0.174 0.01 DB03947

0.146 0.053 DBMET02033

0.2010.0140.201Mediator release inhibitor

0.118 0.049 DB03947

0.2110.0240.245Cholesterol synthesis inhibitor

0.168 0.036 DB03947

0.245 0.018 DBMET02033

DBMET02033
0.2060.0210.247Toll-Like receptor 2 antagonist

0.167 0.041 DB03947

0.247 0.01 DBMET02033

DBMET02033
0.1910.0070.191Ornithine carbamoyltransferase inhibitor

0.123 0.012 DB03947

0.153 0.009 DBMET02033

0.1860.0060.186MAP kinase kinase 1 inhibitor

0.132 0.025 DB03947

0.1990.0210.199Antineoplastic antibiotic

0.199 0.021 DB03947

0.094 0.049 DBMET02033

0.2070.0320.207ATPase inhibitor

0.171 0.07 DB03947

0.2620.090.262Hypoxia-inducible factor 1 alpha inhibitor
0.1850.0140.202Alcohol dehydrogenase inhibitor

0.202 0.012 DB03947

0.157 0.018 DBMET02033

DB03947
0.1760.0060.176Phosphorylase inhibitor

0.063 0.023 DB03947

0.1 0.013 DBMET02033

0.1710.0020.171Neuraminidase (Influenza A) inhibitor

0.12 0.004 DB03947

0.1770.0120.177Electrolyte absorption antagonist

0.12 0.037 DB03947

0.1690.0040.169Glucosylceramidase inhibitor

0.078 0.017 DB03947

0.1830.0180.183Protease inhibitor

0.163 0.024 DB03947

0.123 0.045 DBMET02033

0.2320.0670.465Pyruvate kinase inhibitor

0.277 0.054 DB03947

0.465 0.012 DBMET02033

DBMET02033
0.210.0470.215 Hydroxytryptamine 3E antagonist

0.179 0.109 DB03947

0.1830.0210.185Sphingosine 1-phosphate receptor 5 antagonist

0.156 0.052 DB03947

0.185 0.02 DBMET02033

DBMET02033
0.1970.0350.197Cyclin-dependent kinase 3 inhibitor

0.139 0.125 DB03947

0.1810.0240.181MAP kinase kinase 4 inhibitor

0.138 0.09 DB03947

0.1840.0280.184Cystathionine beta-synthase inhibitor

0.135 0.048 DB03947

0.1720.0160.198Porphobilinogen synthase inhibitor

0.159 0.019 DB03947

0.198 0.012 DBMET02033

DBMET02033
0.1710.0190.183Sphingosine 1-phosphate receptor 4 antagonist

0.15 0.034 DB03947

0.183 0.014 DBMET02033

DBMET02033
0.1850.0330.278DNA polymerase I inhibitor

0.154 0.047 DB03947

0.278 0.013 DBMET02033

DBMET02033
0.1560.0040.242Sphingosine 1-phosphate receptor 3 agonist

0.072 0.009 DB03947

0.242 0.003 DBMET02033

DBMET02033
0.1880.0360.188GABA C receptor rho-2 antagonist

0.14 0.088 DB03947

0.2290.080.229Angiogenesis stimulant

0.17 0.11 DBMET02033

0.2080.0650.208DNA methyltransferase I inhibitor

0.16 0.094 DB03947

0.1560.0170.176NAD(P)H dehydrogenase (quinone) inhibitor

0.105 0.035 DB03947

0.176 0.013 DBMET02033

DBMET02033
0.1410.0040.163Fumarate hydratase inhibitor

0.119 0.004 DB03947

0.163 0.004 DBMET02033

DBMET02033
0.1990.0670.199Nitric oxide antagonist

0.158 0.089 DB03947

0.1660.0350.166Antibacterial (Helicobacter pylori)
0.140.010.14Sphingosine 1-phosphate receptor 4 agonist

0.087 0.032 DB03947

0.127 0.014 DBMET02033

0.1350.0060.1353(or 17)beta-hydroxysteroid dehydrogenase inhibitor

0.093 0.012 DB03947

0.150.0210.15DOPA decarboxylase inhibitor

0.142 0.026 DB03947

0.146 0.024 DBMET02033

0.1640.0370.164Cyclooxygenase 3 inhibitor

0.124 0.073 DB03947

0.122 0.075 DBMET02033

0.1380.0120.138Histone deacetylase stimulant
0.1380.0120.138Histone deacetylase SIRT1 stimulant
0.2030.0770.203DNA methylase inhibitor

0.152 0.115 DB03947

0.1870.0620.187Tumour necrosis factor antagonist
0.1350.0120.135Toll-Like receptor 2 agonist

0.066 0.019 DB03947

0.1560.0330.165Sphingosine 1-phosphate receptor 2 antagonist

0.128 0.078 DB03947

0.165 0.025 DBMET02033

DBMET02033
0.1260.0040.126Epithelial sodium channel blocker

0.068 0.019 DB03947

0.1430.0220.143Anabolic

0.132 0.029 DB03947

0.143 0.022 DBMET02033

0.160.0390.16Adenylate cyclase inhibitor

0.117 0.07 DB03947

0.137 0.054 DBMET02033

0.130.010.13Glycine receptor agonist

0.093 0.026 DB03947

0.1280.0110.128Cathepsin D inhibitor
0.1420.0250.142Calcium antagonist

0.098 0.049 DB03947

0.1310.0160.131Glutamate release inhibitor

0.116 0.025 DB03947

0.160.0450.16Anesthetic local

0.096 0.087 DB03947

0.1280.0140.155Argininosuccinate synthase inhibitor

0.12 0.015 DB03947

0.155 0.011 DBMET02033

DBMET02033
0.1380.0260.138Androgen antagonist

0.078 0.068 DB03947

0.1550.0430.155Cathepsin H inhibitor

0.139 0.055 DB03947

0.1190.0080.119GABA B receptor agonist

0.104 0.014 DB03947

0.072 0.062 DBMET02033

0.1160.0050.116Sphingosine kinase inhibitor

0.085 0.013 DB03947

0.057 0.045 DBMET02033

0.1290.0180.129Phosphodiesterase 6D inhibitor

0.114 0.031 DB03947

0.1 0.052 DBMET02033

0.1310.0210.131Lanosterol 14 alpha demethylase inhibitor

0.107 0.046 DB03947

0.1130.0050.113Prostaglandin agonist

0.086 0.006 DB03947

0.1890.080.189Non-steroidal antiinflammatory agent

0.147 0.119 DBMET02033

0.1480.0410.192Vanilloid 1 agonist

0.139 0.052 DB03947

0.192 0.014 DBMET02033

DBMET02033
0.1160.0120.116Estrogen-related receptor beta agonist

0.1 0.024 DB03947

0.1340.030.134Prolactin inhibitor

0.086 0.072 DB03947

0.110.0060.132Phosphoglycerate kinase inhibitor

0.082 0.008 DB03947

0.132 0.005 DBMET02033

DBMET02033
0.1080.0050.108Renin inhibitor

0.031 0.03 DB03947

0.2010.10.201Platelet antagonist

0.185 0.113 DBMET02033

0.1180.0170.118Na+ K+ transporting ATPase inhibitor

0.106 0.026 DB03947

0.099 0.032 DBMET02033

0.1640.0630.219Phospholipase A2 inhibitor

0.145 0.079 DB03947

0.219 0.034 DBMET02033

DBMET02033
0.1050.0060.105Sphingosine kinase 2 inhibitor

0.074 0.019 DB03947

0.069 0.023 DBMET02033

0.1070.0080.107Glutamate (mGluR6) antagonist

0.085 0.019 DB03947

0.106 0.008 DBMET02033

0.1310.0330.131HIV-1 integrase (Overall Integration) inhibitor

0.115 0.043 DB03947

0.1370.040.137Photosensitizer

0.123 0.054 DB03947

0.1060.0090.106Prostaglandin F2 alpha antagonist

0.061 0.045 DB03947

0.1210.0250.121Ornithine decarboxylase inhibitor

0.105 0.039 DB03947

0.097 0.048 DBMET02033

0.1460.050.146Nav1.3 sodium channel blocker
0.10.0050.1Sphingosine 1-phosphate receptor agonist

0.055 0.021 DB03947

0.1 0.005 DBMET02033

0.1470.0520.147Heat shock protein 70 antagonist

0.143 0.063 DBMET02033

0.1550.060.155MAP kinase 3 inhibitor
0.1490.0550.149Nav1.6 sodium channel blocker
0.1080.0140.108Purinergic P2X1 antagonist

0.074 0.029 DB03947

0.096 0.018 DBMET02033

0.2040.1120.204Neuropeptide Y2 antagonist
0.1150.0230.115ATPase (Vacuolar H+) inhibitor

0.104 0.035 DB03947

0.1030.0110.103Interferon inducer

0.068 0.037 DB03947

0.150.060.15MAP3K9 inhibitor
0.0930.0050.099Sphingosine 1-phosphate receptor 1 agonist

0.057 0.014 DB03947

0.099 0.004 DBMET02033

DBMET02033
0.1110.0230.111Granulocyte macrophage colony stimulating factor agonist

0.091 0.049 DB03947

0.0980.010.098Exportin-1 inhibitor

0.086 0.019 DB03947

0.0940.0060.094Adenosine deaminase inhibitor

0.075 0.011 DB03947

0.054 0.026 DBMET02033

0.1030.0150.103Vanilloid 4 agonist

0.08 0.041 DB03947

0.1130.0270.113Glutathione S-transferase inhibitor

0.09 0.048 DB03947

0.091 0.047 DBMET02033

0.1010.0140.101Beta 3 adrenoreceptor antagonist

0.068 0.037 DB03947

0.1290.0430.316Sphingosine 1-phosphate receptor 2 agonist

0.316 0.004 DBMET02033

DBMET02033
0.0880.0030.088Prostaglandin EP2 agonist

0.043 0.007 DB03947

0.1030.0190.103Ribonucleoside-diphosphate reductase inhibitor

0.067 0.03 DB03947

0.095 0.02 DBMET02033

0.1040.020.104Ribonucleotide reductase inhibitor

0.069 0.031 DB03947

0.099 0.021 DBMET02033

0.0980.0140.098MAP kinase kinase 7 inhibitor

0.082 0.04 DB03947

0.1890.1060.189Free radical scavenger
0.0860.0050.086Sphingosine kinase 1 inhibitor

0.058 0.01 DB03947

0.039 0.034 DBMET02033

0.0920.010.092MDM2 inhibitor

0.086 0.014 DB03947

0.090.0090.09Calcium channel P-type blocker

0.068 0.032 DB03947

0.1440.0640.284Bone formation stimulant

0.284 0.019 DBMET02033

DBMET02033
0.1520.0720.152CF transmembrane conductance regulator agonist
0.0870.0070.11Lysophosphatidic acid 3 receptor antagonist

0.067 0.016 DB03947

0.11 0.004 DBMET02033

DBMET02033
0.0970.0180.097Beta adrenoreceptor antagonist

0.068 0.042 DB03947

0.0820.0030.082Uridine phosphorylase inhibitor

0.064 0.005 DB03947

0.049 0.008 DBMET02033

0.1030.0250.103GABA aminotransferase inhibitor

0.074 0.055 DB03947

0.120.0430.212Toll-Like receptor 4 antagonist

0.1 0.07 DB03947

0.212 0.005 DBMET02033

DBMET02033
0.1220.0450.122Carbonic anhydrase XV inhibitor

0.1 0.067 DB03947

0.0940.0180.094Phospholipase D inhibitor

0.067 0.061 DB03947

0.1190.0450.119Carbonic anhydrase III inhibitor

0.092 0.072 DB03947

0.0780.0040.078Prostaglandin E2 agonist

0.031 0.01 DB03947

0.0950.0210.095Secretase beta inhibitor

0.067 0.054 DB03947

0.0860.0140.086Beta 1 adrenoreceptor antagonist

0.063 0.032 DB03947

0.1590.0870.1893C-like protease (Human coronavirus) inhibitor

0.189 0.058 DB03947

DB03947
0.1050.0340.105Adrenaline agonist
0.0740.0040.074Guanylate cyclase inhibitor

0.07 0.005 DB03947

0.066 0.007 DBMET02033

0.0750.0050.075Hypoxanthine phosphoribosyltransferase inhibitor

0.054 0.008 DB03947

0.053 0.008 DBMET02033

0.1010.0320.101mTOR complex 2 inhibitor

0.081 0.065 DB03947

0.0910.0220.091Prostaglandin EP2 antagonist
0.1040.0390.104ALK inhibitor
0.0740.010.074Adenylate cyclase 1 inhibitor

0.044 0.035 DB03947

0.0730.010.073Heparanase inhibitor

0.054 0.035 DB03947

0.05 0.044 DBMET02033

0.1230.060.123Monophenol monooxygenase inhibitor

0.1 0.076 DB03947

0.1330.070.133Nav1.2 sodium channel blocker
0.0730.010.073Thymidine kinase inhibitor

0.054 0.016 DB03947

0.058 0.014 DBMET02033

0.1170.0550.117Protein kinase C gamma inhibitor
0.0690.0070.069GABA uptake inhibitor

0.044 0.021 DB03947

0.0990.0380.106Carbonic anhydrase XIII inhibitor

0.077 0.052 DB03947

0.106 0.035 DBMET02033

DBMET02033
0.1650.1040.165Psychostimulant

0.141 0.125 DBMET02033

0.0710.010.071Immunoglobulin Fc receptor antagonist

0.057 0.033 DB03947

0.1160.0560.132Falcipain 3 inhibitor

0.132 0.046 DB03947

DB03947
0.0670.0090.067Dopamine beta hydroxylase inhibitor
0.0720.0150.072Beta 2 adrenoreceptor antagonist

0.05 0.036 DB03947

0.0590.0030.075Lysophosphatidic acid receptor 1 agonist

0.04 0.005 DB03947

0.075 0.002 DBMET02033

DBMET02033
0.0730.0180.073Diacylglycerol O-acyltransferase inhibitor
0.2120.1570.212Transcription factor NF kappa B inhibitor
0.0640.010.064Microtubule stabilization

0.042 0.039 DB03947

0.0930.040.093D-Ala-D-Ala ligase inhibitor

0.079 0.071 DB03947

0.083 0.061 DBMET02033

0.0560.0030.056Ileal bile acid transport inhibitor

0.019 0.01 DB03947

0.1440.0920.144Growth hormone agonist
0.0530.0020.072Lysophosphatidic acid receptor 3 agonist

0.03 0.004 DB03947

0.072 0.002 DBMET02033

DBMET02033
0.0680.0170.068Pregnane X receptor antagonist

0.055 0.046 DB03947

0.0910.0420.091Glycine receptor antagonist
0.0650.0160.065Squalene epoxidase inhibitor

0.046 0.044 DB03947

0.0540.0050.054Methionyl aminopeptidase 1 inhibitor
0.0530.0060.053HMG CoA reductase inhibitor

0.038 0.017 DB03947

0.032 0.029 DBMET02033

0.0520.0040.056Prostaglandin F2 alpha agonist

0.056 0.004 DB03947

0.025 0.012 DBMET02033

DB03947
0.0530.0060.053Sodium/glucose cotransporter 2 inhibitor

0.028 0.015 DB03947

0.0560.0090.056Glutamate (mGluR8) agonist

0.043 0.018 DB03947

0.054 0.009 DBMET02033

0.0520.0060.052Methionyl aminopeptidase 2 inhibitor
0.0770.0310.077Glutamate (mGluR7) antagonist
0.0760.0310.076NMDA receptor glycine site agonist
0.1910.1470.191Transcription factor STAT3 inhibitor

0.191 0.146 DBMET02033

0.070.0260.075Sphingosine 1-phosphate receptor 3 antagonist

0.075 0.021 DBMET02033

DBMET02033
0.0550.010.0553-Hydroxyanthranilate 3,4-dioxygenase inhibitor

0.045 0.021 DB03947

0.0680.0230.068Beta 2 adrenoreceptor agonist
0.0560.0120.056Membrane dipeptidase inhibitor

0.043 0.022 DB03947

0.037 0.03 DBMET02033

0.1330.0890.133Cytidine deaminase inhibitor
0.0780.0330.078Neutrophil collagenase inhibitor
0.0580.0150.058Cytokine production stimulant

0.046 0.042 DB03947

0.0520.0080.094Lysophosphatidic acid 2 receptor antagonist

0.094 0.004 DBMET02033

DBMET02033
0.0530.0110.053Kainate receptor agonist

0.042 0.026 DB03947

0.0940.0520.171Aminoacyl-tRNA synthetase inhibitor

0.171 0.014 DBMET02033

DBMET02033
0.0670.0260.067Protein 50S ribosomal subunit inhibitor

0.048 0.043 DB03947

0.0530.0130.053Arginase inhibitor

0.033 0.029 DB03947

0.1030.0630.103Nav1.1 sodium channel blocker
0.0880.0480.088Carbonic anhydrase VI inhibitor
0.0970.0580.097Potassium channel (Ca-activated) activator
0.1080.0690.108Acetylcholine release stimulant
0.1210.0820.121Sodium channel blocker
0.0780.040.078S-adenosyl-L-methionine decarboxylase inhibitor
0.0550.0170.055Geranyltranstransferase inhibitor

0.05 0.023 DBMET02033

0.1170.0790.117DNA repair enzyme inhibitor
0.0420.0050.042Thymidine kinase (Herpes simplex virus 1) inhibitor

0.032 0.009 DB03947

0.050.0130.05Antibiotic Aminoglycoside-like

0.037 0.024 DB03947

0.050.0140.05Heme oxygenase inhibitor

0.045 0.022 DB03947

0.1110.0750.111Interleukin 8 antagonist
0.0520.0160.052Plasmepsin II inhibitor
0.0790.0430.079Phosphodiesterase VI inhibitor
0.0420.0060.042Sodium/glucose cotransporter inhibitor

0.026 0.018 DB03947

0.0610.0260.061Leukotriene C antagonist

0.055 0.042 DB03947

0.040.0050.04Vitamin D receptor antagonist

0.028 0.008 DB03947

0.040.0050.04Estrogen-related receptor gamma antagonist

0.03 0.016 DB03947

0.0510.0160.051Calcitonin receptor agonist

0.035 0.023 DB03947

0.0440.0090.044Lysine carboxypeptidase inhibitor

0.028 0.017 DB03947

0.0910.0570.091Phosphodiesterase I inhibitor
0.0460.0120.046Vanilloid 3 antagonist

0.041 0.02 DBMET02033

0.0370.0030.037Neuraminidase (Influenza B) inhibitor

0.028 0.005 DB03947

0.0740.040.074Protein kinase C beta inhibitor
0.0730.0390.073Glucagon-like peptide 1 agonist
0.0590.0250.059Bombesin 2 receptor antagonist
0.0440.010.044Cholesterol ester transfer protein antagonist
0.0950.0620.095Bile acid receptor antagonist
0.0640.0310.069Carbonic anhydrase VB inhibitor

0.069 0.028 DBMET02033

DBMET02033
0.0430.0110.043Prostaglandin D2 agonist

0.03 0.023 DB03947

0.0680.0370.068NMDA receptor agonist
0.0490.0190.049Beta adrenoreceptor agonist
0.040.010.04Glutamate (mGluR3) agonist

0.032 0.022 DB03947

0.0360.0060.036Hedgehog signaling activator

0.028 0.018 DB03947

0.0540.0240.054Aldosterone antagonist
0.0580.0290.117Sphingosine 1-phosphate receptor 5 agonist

0.117 0.006 DBMET02033

DBMET02033
0.0380.0080.038Purinergic P2Y15 antagonist

0.028 0.021 DB03947

0.0630.0350.063Heat shock protein 90 beta antagonist
0.0320.0040.032Thymidine kinase (Herpes simplex virus 2) inhibitor

0.026 0.006 DB03947

0.0990.0710.099Topoisomerase I inhibitor
0.0690.0410.069Leukotriene antagonist
0.0590.0310.059Dihydroorotate oxidase inhibitor
0.0420.0140.042Ceramide glucosyltransferase inhibitor
0.0580.0310.058Leukotriene B4 antagonist
0.0320.0050.032Isoleucine-tRNA ligase inhibitor

0.025 0.01 DB03947

0.0590.0320.078Sphingosine 1-phosphate receptor 1 antagonist

0.062 0.026 DB03947

0.078 0.015 DBMET02033

DBMET02033
0.0950.070.095Glutamate (mGluR7) agonist

0.091 0.081 DBMET02033

0.0540.0290.066Antimetabolite

0.066 0.023 DBMET02033

DBMET02033
0.0610.0350.061Ryanodine receptor antagonist

0.056 0.051 DBMET02033

0.0360.0110.036Purinergic P2T antagonist
0.0290.0040.029Thromboxane A2 agonist

0.019 0.006 DB03947

0.0290.0040.029Carbonic anhydrase X inhibitor

0.018 0.01 DB03947

0.0290.0040.029Carbonic anhydrase VIII inhibitor

0.018 0.01 DB03947

0.0390.0140.039ATP citrate lysase inhibitor

0.032 0.022 DB03947

0.0620.0380.062Cathepsin E inhibitor
0.0420.0190.042VCAM-1 antagonist
0.0370.0140.037Estrogen-related receptor beta antagonist
0.0270.0030.027Methylmalonyl-CoA mutase inhibitor

0.022 0.006 DB03947

0.026 0.003 DBMET02033

0.0420.0190.042VCAM antagonist
0.0420.0190.042Glutamate (mGluR3) antagonist
0.0650.0430.065Protease 3C (Human rhinovirus) inhibitor

0.058 0.056 DB03947

0.0970.0750.097AMP-activated protein kinase stimulant
0.0260.0040.026Antibiotic Anthracycline-like

0.023 0.007 DB03947

0.0320.010.032Thymidine phosphorylase inhibitor
0.1280.1060.128Pregnane X receptor agonist
0.1420.1220.142Neurotensin receptor agonist
0.0670.0470.067Acetylcholine M5 receptor agonist
0.1030.0830.103TRPA1 agonist
0.0240.0050.024Vitamin D receptor agonist

0.021 0.006 DB03947

0.0480.0280.079Purinergic P2Y antagonist

0.079 0.013 DBMET02033

DBMET02033
0.0940.0740.094Gastric antisecretory
0.0430.0240.043Dopamine D5 agonist
0.0580.0390.059Lipocortins synthesis agonist

0.055 0.048 DB03947

0.059 0.038 DBMET02033

DBMET02033
0.0510.0320.051Metalloproteinase-3 inhibitor
0.0310.0120.031Calcium-sensing receptor agonist
0.0230.0050.023Telomerase stimulant

0.018 0.011 DB03947

0.0250.0070.025Calcium-sensing receptor antagonist
0.0210.0030.021Purine nucleoside phosphorylase inhibitor

0.013 0.007 DB03947

0.012 0.007 DBMET02033

0.0410.0240.041Vascular adhesion protein 1 inhibitor
0.0480.0310.048Thymidylate synthase inhibitor
0.1030.0860.103Caspase 3 inhibitor
0.0310.0150.031MAP3K8 inhibitor
0.0360.020.036Sirtuin 2 inhibitor
0.0810.0650.081NMDA receptor antagonist
0.0280.0130.028Vanilloid 2 agonist

0.025 0.018 DBMET02033

0.0180.0040.018Thromboxane agonist

0.013 0.005 DB03947

0.0220.0070.022Adenosine A2 receptor agonist
0.0390.0260.039Leukotriene C4 antagonist
0.0540.040.054Neuropeptide agonist
0.0610.0470.061Nitric oxide donor
0.0350.0220.035RNA-directed RNA polymerase inhibitor
0.0570.0450.057Androgen agonist
0.090.0770.09Insulin receptor antagonist
0.0420.030.042GABA B receptor antagonist
0.0860.0740.086Protein kinase C zeta inhibitor
0.0260.0140.026Glutamate (mGluR1) agonist
0.0350.0230.041-Alkyl-2-acetylglycerophosphocholine esterase inhibitor

0.04 0.016 DBMET02033

DBMET02033
0.020.0090.033Prostacyclin agonist

0.033 0.005 DB03947

DB03947
0.0240.0130.024ICAM 1 antagonist
0.0180.0080.018Purinergic P2Y1 agonist

0.018 0.008 DBMET02033

0.0730.0630.096Sphingosine 1-phosphate receptor antagonist

0.077 0.053 DB03947

0.096 0.024 DBMET02033

DBMET02033
0.1140.1040.114Neurotrophic factor
0.020.010.02Cyclin T1 inhibitor
0.0190.0090.019Prostaglandin EP4 agonist
0.0610.0510.061Aryl hydrocarbon receptor antagonist
0.0180.0090.018Adenosine A2a receptor agonist
0.0710.0610.071Potassium channel (Tandem pore domain) blocker
0.0790.0710.087Transcription factor NF kappa B stimulant

0.087 0.055 DBMET02033

DBMET02033
0.0270.020.027LFA antagonist
0.0230.0150.023Glutamate (mGluR1a) agonist
0.0230.0160.023Beta 1 adrenoreceptor agonist
0.0140.0070.014Glutamate (mGluR6) agonist

0.013 0.007 DBMET02033

0.020.0150.02Retinoid X beta receptor antagonist
0.0540.0480.054Cyclin-dependent kinase 6 inhibitor
0.0530.0480.0533-Oxoacyl-[acyl-carrier-protein] synthase inhibitor
0.0380.0340.038Oxytocin agonist
0.0410.0370.041AICAR transformylase inhibitor
0.0620.0570.062Carbonic anhydrase VA inhibitor
0.0220.0180.022Aminopeptidase P inhibitor
0.0450.0410.045Topoisomerase II beta inhibitor
0.0370.0340.037Neurokinin 2 antagonist
0.0310.0280.031Protein kinase (CK2) beta inhibitor
0.0140.0110.014S-adenosyl-L-homocysteine hydrolase inhibitor
0.0350.0320.035Retinoid X receptor antagonist
0.0320.0290.032Retinoid X alpha receptor antagonist
0.0340.0310.034Tryptophan 5 hydroxylase inhibitor
0.0840.0820.084Xanthine oxidase inhibitor
0.0310.0290.031Retinoid X receptor agonist
0.010.0080.01Purinergic P2Y2 agonist

0.01 0.008 DBMET02033

0.0330.0320.0332,3-Oxidosqualene-lanosterol cyclase inhibitor
0.0360.0350.036Glutamate (mGluR1a) antagonist
0.0210.020.021Retinoic acid gamma receptor agonist
0.0330.0320.033Farnesoid X receptor agonist
0.0180.0170.018Hexokinase stimulant
0.0180.0210.025Lysophosphatidic acid 1 receptor antagonist

0.025 0.009 DBMET02033

DBMET02033
0.0560.0590.063Carbonic anhydrase V inhibitor

0.063 0.05 DBMET02033

DBMET02033
0.0920.1020.099Electron transport complex I inhibitor

0.099 0.084 DB03947

DB03947
0.1860.20.473Apoptosis antagonist

0.234 0.143 DB03947

0.473 0.024 DBMET02033

DBMET02033
0.0050.0360.021Purinergic P2Y agonist

0.021 0.005 DBMET02033

DBMET02033
0.0040.0370.028Purinergic P2 agonist

0.028 0.005 DBMET02033

DBMET02033
0.0040.0370.028Purinergic receptor agonist

0.028 0.005 DBMET02033

DBMET02033
0.040.0730.111Purinergic P2X2 antagonist

0.111 0.025 DBMET02033

DBMET02033
0.0240.0590.035p53 inhibitor

0.035 0.026 DB03947

DB03947
0.0110.0560.069Purinergic P2X agonist

0.069 0.005 DBMET02033

DBMET02033
0.2120.2570.508Apoptosis agonist

0.508 0.072 DBMET02033

DBMET02033
0.0270.0730.044Calcium-independent phospholipase A2 inhibitor

0.044 0.007 DB03947

0.032 0.03 DBMET02033

DB03947
0.0190.0720.045Toll-Like receptor 4 agonist

0.045 0.004 DBMET02033

DBMET02033
0.1160.2080.276Tumour necrosis factor alpha release inhibitor

0.276 0.063 DBMET02033

DBMET02033
0.1080.2010.168Lipocortins synthesis antagonist

0.168 0.083 DB03947

DB03947
0.0690.1830.156Folate antagonist

0.156 0.02 DBMET02033

DBMET02033
0.0390.1720.095HIV-1 integrase inhibitor

0.095 0.028 DB03947

0.082 0.036 DBMET02033

DB03947
0.0570.1990.287Vanilloid agonist

0.287 0.005 DBMET02033

DBMET02033
0.0590.2030.3553C-Like protease (SARS coronavirus) inhibitor

0.355 0.003 DB03947

0.257 0.004 DBMET02033

DB03947
0.0050.2210.018Inosine monophosphate dehydrogenase 1 inhibitor

0.018 0.016 DBMET02033

DBMET02033
0.0180.370.112Autotaxin inhibitor

0.112 0.011 DBMET02033

DBMET02033
0.0050.4220.024Urotensin II agonist

0.024 0.023 DBMET02033

DBMET02033
0.010.4880.072Purinergic P2Y2 antagonist

0.072 0.006 DBMET02033

DBMET02033
0.0340.5190.202Platelet adhesion inhibitor

0.202 0.07 DBMET02033

DBMET02033
0.0060.5360.04Growth factor receptor-bound protein 2 antagonist

0.04 0.014 DBMET02033

DBMET02033
0.0060.7410.06Cathepsin B inhibitor

0.06 0.035 DB03947

DB03947
0.0110.8130.056Sodium/calcium exchanger inhibitor

0.056 0.024 DBMET02033

DBMET02033
0.0020.9110.042Purinergic P2Y1 antagonist

0.042 0.004 DBMET02033

DBMET02033
0.0040.9690.114DNA directed RNA polymerase inhibitor

0.114 0.042 DBMET02033

DBMET02033
0.0040.9910.183Falcipain inhibitor

0.183 0.019 DB03947

DB03947
0.0030.9950.167Falcipain 2 inhibitor

0.167 0.022 DB03947

DB03947
Ext Pa Pi Pmax Activity Other Results ID Pa_max