Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.4250.0240.693HERG channel blocker

0.141 0.14 DBMET03658

0.325 0.043 DBMET02204

0.693 0.005 DBMET02205

0.28 0.055 DBMET02213

0.36 0.035 DBMET02214

DBMET02205
0.4220.0230.668Potassium channel (Voltage-sensitive) blocker

0.144 0.142 DBMET03658

0.33 0.041 DBMET02204

0.668 0.005 DBMET02205

0.276 0.057 DBMET02213

0.333 0.04 DBMET02214

DBMET02205
0.3670.0050.449Hedgehog signaling inhibitor

0.216 0.009 DBMET03658

0.275 0.005 DBMET02204

0.449 0.004 DBMET02205

0.249 0.007 DBMET02213

0.164 0.019 DBMET02214

DBMET02205
0.3440.0340.554Potassium channel blocker

0.253 0.065 DBMET02204

0.554 0.008 DBMET02205

0.198 0.094 DBMET02213

0.264 0.06 DBMET02214

DBMET02205
0.3890.110.406Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.373 0.126 DBMET03658

0.286 0.233 DBMET02204

0.406 0.095 DBMET02205

0.295 0.22 DBMET02213

0.3 0.212 DBMET02214

DBMET02205
0.330.1090.33MAP kinase kinase 6 inhibitor

0.302 0.134 DBMET03658

0.329 0.109 DBMET02204

0.312 0.124 DBMET02205

0.326 0.112 DBMET02213

0.278 0.158 DBMET02214

0.2230.0050.223Smo receptor antagonist

0.077 0.013 DBMET03658

0.12 0.006 DBMET02204

0.112 0.007 DBMET02205

0.106 0.007 DBMET02213

0.059 0.019 DBMET02214

0.2640.0640.275Gastrin inhibitor

0.218 0.123 DBMET03658

0.234 0.099 DBMET02204

0.275 0.053 DBMET02205

0.248 0.082 DBMET02213

DBMET02205
0.20.0150.25 Hydroxytryptamine 3A agonist

0.135 0.044 DBMET03658

0.146 0.038 DBMET02204

0.161 0.03 DBMET02205

0.154 0.033 DBMET02213

0.104 0.072 DBMET02214

0.1870.0050.187Melanin-concentrating hormone receptor 1 antagonist

0.048 0.043 DBMET03658

0.163 0.005 DBMET02204

0.128 0.008 DBMET02205

0.086 0.018 DBMET02213

0.2310.0550.275Interleukin-1 receptor-associated protein kinase 1 inhibitor

0.203 0.065 DBMET03658

0.18 0.075 DBMET02204

0.275 0.04 DBMET02205

0.162 0.086 DBMET02213

0.168 0.082 DBMET02214

DBMET02205
0.1860.0170.2Interleukin 8 antagonist

0.12 0.061 DBMET03658

0.2 0.013 DBMET02204

0.17 0.023 DBMET02205

0.135 0.045 DBMET02213

0.105 0.086 DBMET02214

DBMET02204
0.2020.0340.202Cyclin-dependent kinase 8 inhibitor

0.17 0.061 DBMET03658

0.157 0.073 DBMET02204

0.196 0.038 DBMET02205

0.129 0.104 DBMET02213

0.139 0.091 DBMET02214

0.2340.0690.249Ca2+/calmodulin-dependent kinase I alpha inhibitor

0.206 0.086 DBMET03658

0.187 0.101 DBMET02204

0.249 0.061 DBMET02205

0.208 0.085 DBMET02213

0.178 0.11 DBMET02214

DBMET02205
0.1650.0090.194CXC chemokine receptor antagonist

0.146 0.011 DBMET03658

0.126 0.015 DBMET02204

0.194 0.005 DBMET02205

0.121 0.017 DBMET02213

0.091 0.029 DBMET02214

DBMET02205
0.2110.0640.212Proto-oncogene tyrosine-protein kinase Fyn inhibitor

0.156 0.125 DBMET03658

0.212 0.063 DBMET02204

0.205 0.069 DBMET02205

0.211 0.064 DBMET02213

0.15 0.133 DBMET02214

DBMET02204
0.1540.0090.1545 Hydroxytryptamine 3 antagonist

0.08 0.024 DBMET02204

0.06 0.035 DBMET02205

0.103 0.017 DBMET02213

0.107 0.016 DBMET02214

0.2040.0660.212TRKC antagonist

0.181 0.078 DBMET03658

0.168 0.087 DBMET02204

0.212 0.062 DBMET02205

0.143 0.107 DBMET02213

DBMET02205
0.1650.0270.214Check point kinase 2 inhibitor

0.13 0.041 DBMET03658

0.14 0.035 DBMET02204

0.214 0.014 DBMET02205

0.13 0.042 DBMET02213

0.135 0.039 DBMET02214

DBMET02205
0.1890.0520.277Polo-like kinase-3 inhibitor

0.161 0.073 DBMET03658

0.176 0.06 DBMET02204

0.179 0.058 DBMET02205

0.174 0.062 DBMET02213

0.277 0.016 DBMET02214

DBMET02214
0.160.0280.18Chemokine receptor antagonist

0.094 0.07 DBMET03658

0.111 0.054 DBMET02204

0.18 0.022 DBMET02205

0.098 0.065 DBMET02213

DBMET02205
0.1630.0350.313Protein kinase (CK2) alpha inhibitor

0.097 0.079 DBMET03658

0.127 0.058 DBMET02204

0.313 0.01 DBMET02205

0.133 0.053 DBMET02213

DBMET02205
0.2180.0910.231Neuropeptide Y2 antagonist

0.231 0.075 DBMET02205

0.194 0.132 DBMET02213

DBMET02205
0.1410.020.141Acetylcholine nicotinic agonist

0.098 0.039 DBMET02204

0.098 0.039 DBMET02205

0.085 0.051 DBMET02213

0.1260.0090.133Alpha 2 adrenoreceptor agonist

0.082 0.023 DBMET02204

0.133 0.008 DBMET02205

0.074 0.028 DBMET02213

DBMET02205
0.1230.0070.131CC chemokine 3 receptor antagonist

0.056 0.021 DBMET02204

0.131 0.007 DBMET02205

0.051 0.024 DBMET02213

0.076 0.015 DBMET02214

DBMET02205
0.1710.0560.214Protein kinase (CK1) gamma inhibitor

0.149 0.068 DBMET03658

0.132 0.079 DBMET02204

0.214 0.039 DBMET02205

0.117 0.094 DBMET02213

0.118 0.092 DBMET02214

DBMET02205
0.1720.0720.172Sigma receptor agonist

0.153 0.083 DBMET02204

0.1080.0090.108Fatty acid synthase inhibitor

0.059 0.036 DBMET03658

0.084 0.017 DBMET02204

0.085 0.016 DBMET02205

0.056 0.041 DBMET02213

0.063 0.032 DBMET02214

0.2660.1690.498Analgesic

0.291 0.148 DBMET03658

0.255 0.179 DBMET02205

0.498 0.05 DBMET02214

DBMET02214
0.1360.0390.241Protein kinase (CK2) inhibitor

0.114 0.052 DBMET02204

0.241 0.012 DBMET02205

0.1 0.064 DBMET02213

DBMET02205
0.2250.130.245Ca2+/calmodulin-dependent kinase II alpha inhibitor

0.245 0.111 DBMET03658

0.202 0.155 DBMET02204

DBMET03658
0.1440.0510.144TRKB antagonist

0.113 0.082 DBMET03658

0.132 0.06 DBMET02204

0.137 0.056 DBMET02205

0.113 0.083 DBMET02213

0.1530.0610.163Neuropeptide Y1 antagonist

0.163 0.047 DBMET02205

0.13 0.099 DBMET02213

DBMET02205
0.1140.0220.121Tyk2 inhibitor

0.091 0.031 DBMET03658

0.068 0.043 DBMET02204

0.121 0.02 DBMET02205

0.069 0.042 DBMET02213

0.064 0.045 DBMET02214

DBMET02205
0.1540.0620.154Tyrosine-protein kinase receptor antagonist

0.113 0.094 DBMET02204

0.149 0.064 DBMET02205

0.1330.0420.144EphA2 antagonist

0.144 0.034 DBMET02204

0.137 0.038 DBMET02205

0.117 0.058 DBMET02213

DBMET02204
0.1270.0380.127Insulin receptor antagonist

0.089 0.079 DBMET03658

0.104 0.056 DBMET02204

0.103 0.057 DBMET02205

0.104 0.057 DBMET02213

0.1540.0650.164Protein kinase (CK1) gamma 1 inhibitor

0.135 0.082 DBMET03658

0.13 0.087 DBMET02204

0.164 0.059 DBMET02205

0.122 0.095 DBMET02213

DBMET02205
0.0980.0110.098Nicotinic alpha7 receptor agonist

0.056 0.035 DBMET02204

0.053 0.039 DBMET02205

0.059 0.033 DBMET02213

0.0890.0060.089Prolactin release inhibitor

0.063 0.042 DBMET03658

0.083 0.009 DBMET02204

0.069 0.025 DBMET02205

0.084 0.009 DBMET02213

0.0840.0020.084HCV NS5A inhibitor

0.081 0.003 DBMET03658

0.077 0.003 DBMET02204

0.057 0.004 DBMET02205

0.077 0.003 DBMET02213

0.043 0.005 DBMET02214

0.2130.1320.225Ca2+/calmodulin-dependent kinase IV inhibitor

0.225 0.106 DBMET02205

DBMET02205
0.1120.0330.145Neuropeptide Y antagonist

0.145 0.023 DBMET02205

0.076 0.065 DBMET02213

DBMET02205
0.0930.0150.093Nicotinic neuronal receptor agonist

0.065 0.032 DBMET02204

0.069 0.028 DBMET02205

0.054 0.041 DBMET02213

0.180.1030.18EphB2 antagonist

0.163 0.117 DBMET03658

0.154 0.126 DBMET02204

0.178 0.104 DBMET02205

0.155 0.124 DBMET02213

0.1220.0470.122AMP-activated protein kinase stimulant

0.095 0.077 DBMET02204

0.103 0.066 DBMET02205

0.1570.0820.175Protein kinase (CK1) gamma 3 inhibitor

0.146 0.094 DBMET03658

0.137 0.105 DBMET02204

0.175 0.064 DBMET02205

0.128 0.116 DBMET02213

0.127 0.118 DBMET02214

DBMET02205
0.1740.10.212MAP kinase kinase 2 inhibitor

0.139 0.131 DBMET03658

0.212 0.074 DBMET02205

DBMET02205
0.10.0280.1Alpha adrenoreceptor agonist

0.062 0.053 DBMET02204

0.098 0.028 DBMET02205

0.1320.0590.132TRKA antagonist

0.132 0.059 DBMET02205

0.0770.0090.077Histamine H4 receptor antagonist

0.049 0.033 DBMET02204

0.067 0.014 DBMET02205

0.049 0.032 DBMET02213

0.1060.0430.106Acetylcholine agonist
0.2340.1720.412Antiobesity

0.301 0.116 DBMET02205

0.412 0.061 DBMET02214

DBMET02214
0.0980.0360.172Protein kinase (CaMK, MLCK, PhK, SNF, KIN, NIM1, MAPKAP, POLO, CHK, ULK, RSK-2nd domain) inhibitor

0.073 0.057 DBMET03658

0.081 0.049 DBMET02204

0.172 0.016 DBMET02205

0.076 0.053 DBMET02213

0.086 0.045 DBMET02214

DBMET02205
0.120.0650.185Protein kinase (CK1) gamma 2 inhibitor

0.134 0.056 DBMET03658

0.185 0.036 DBMET02205

0.1 0.084 DBMET02214

DBMET02205
0.0810.0260.0815 Hydroxytryptamine 3 agonist

0.061 0.047 DBMET02205

0.0810.030.0815 Hydroxytryptamine 3A antagonist
0.0720.0250.0725 Hydroxytryptamine 5 antagonist
0.0660.020.075Potassium channel (Inward rectifier) blocker

0.075 0.015 DBMET02205

DBMET02205
0.0750.0310.075Janus tyrosine kinase 1 inhibitor

0.073 0.032 DBMET02205

0.1920.1480.2MAP kinase kinase 3 inhibitor

0.2 0.121 DBMET03658

0.199 0.125 DBMET02205

0.187 0.165 DBMET02213

DBMET03658
0.0710.030.0715 Hydroxytryptamine 5A antagonist
0.1110.070.1115 Hydroxytryptamine 2B antagonist
0.0680.0290.068Alpha 1 adrenoreceptor agonist

0.052 0.048 DBMET02204

0.0910.0550.107Interleukin-1 receptor-associated protein kinase 4 inhibitor

0.088 0.059 DBMET03658

0.107 0.04 DBMET02205

DBMET02205
0.0430.0080.047Epoxide hydrolase 2 inhibitor

0.024 0.017 DBMET03658

0.036 0.011 DBMET02204

0.047 0.006 DBMET02205

0.035 0.011 DBMET02213

0.036 0.011 DBMET02214

DBMET02205
0.130.0950.13Acetylcholine M1 receptor antagonist
0.0610.0260.061Chemokine receptor agonist

0.059 0.028 DBMET02205

0.0810.0460.093Vanilloid antagonist

0.093 0.039 DBMET02205

DBMET02205
0.1060.0740.1065 Hydroxytryptamine antagonist
0.0580.0280.058Dipeptidyl peptidase inhibitor
0.0730.0430.073Toll-Like receptor 7 antagonist

0.065 0.05 DBMET02205

0.10.0720.15 Hydroxytryptamine 2 antagonist
0.0390.0120.039Cyclophilin A inhibitor

0.036 0.015 DBMET03658

0.035 0.016 DBMET02204

0.039 0.013 DBMET02205

0.033 0.018 DBMET02213

0.035 0.016 DBMET02214

0.0480.0230.048Dipeptidyl peptidase IV inhibitor
0.0750.0510.076Adenosine A3 receptor antagonist

0.076 0.049 DBMET02205

DBMET02205
0.0830.0590.083Histamine H2 receptor antagonist

0.079 0.067 DBMET02204

0.0840.0610.084Alpha 2 adrenoreceptor antagonist
0.1020.0780.102Tyrosine-protein kinase receptor FLT3 inhibitor

0.09 0.086 DBMET02204

0.1440.1210.155Death-associated protein kinase 2 inhibitor

0.155 0.095 DBMET02205

0.139 0.134 DBMET02214

DBMET02205
0.0880.0650.096Polo-like kinase-1 inhibitor

0.092 0.057 DBMET02213

0.096 0.051 DBMET02214

DBMET02214
0.0630.040.113CXC chemokine 4 receptor antagonist

0.113 0.022 DBMET02205

DBMET02205
0.1410.1190.141Cyclin-dependent kinase 3 inhibitor
0.0610.040.064Cyclin-dependent kinase 6 inhibitor

0.064 0.037 DBMET02205

DBMET02205
0.0810.0610.081CC chemokine 5 receptor agonist

0.078 0.07 DBMET02205

0.0890.070.099DNA directed RNA polymerase inhibitor

0.085 0.077 DBMET03658

0.099 0.058 DBMET02205

DBMET02205
0.1070.0880.132MAP kinase 12 inhibitor

0.102 0.096 DBMET03658

0.132 0.057 DBMET02205

DBMET02205
0.0360.0170.036CXC chemokine 3 receptor antagonist

0.036 0.017 DBMET02205

0.0680.0510.0685 Hydroxytryptamine 1F antagonist
0.0650.0480.075Vanilloid 1 antagonist

0.075 0.04 DBMET02205

DBMET02205
0.1390.1240.139Ca2+/calmodulin-dependent protein kinase inhibitor
0.0390.0250.063DNA gyrase subunit B inhibitor

0.063 0.008 DBMET02205

DBMET02205
0.0650.0510.109Check point kinase 1 inhibitor

0.109 0.025 DBMET02205

DBMET02205
0.1140.10.132Protein kinase C nu inhibitor

0.132 0.082 DBMET02205

DBMET02205
0.0370.0240.0375 Hydroxytryptamine 3B antagonist
0.0680.0570.126MAP kinase 11 inhibitor

0.126 0.024 DBMET02205

DBMET02205
0.1510.140.165Growth factor agonist

0.149 0.144 DBMET03658

0.165 0.111 DBMET02204

0.149 0.143 DBMET02205

DBMET02204
0.060.0490.085DNA gyrase inhibitor

0.057 0.053 DBMET02204

0.085 0.024 DBMET02205

DBMET02205
0.1220.1140.137Ca2+/calmodulin-dependent kinase II gamma inhibitor

0.137 0.098 DBMET03658

DBMET03658
0.0510.0430.051Nicotinic receptor alpha7 subunit antagonist
0.0540.0470.059Raf kinase C inhibitor

0.059 0.043 DBMET02205

DBMET02205
0.0950.0890.118MAP kinase 13 inhibitor

0.118 0.058 DBMET02205

DBMET02205
0.1010.0960.101RET inhibitor
0.0190.0150.144Somatostatin 3 antagonist

0.018 0.016 DBMET03658

0.144 0.003 DBMET02205

DBMET02205
0.0460.0430.046mTOR inhibitor
0.1270.1240.132Ca2+/calmodulin-dependent protein kinase kinase B inhibitor

0.132 0.111 DBMET03658

DBMET03658
0.0750.0730.082Stem cell growth factor agonist

0.076 0.071 DBMET03658

0.082 0.063 DBMET02204

0.074 0.073 DBMET02205

DBMET02204
0.0390.0380.047Purinergic P2Y antagonist

0.047 0.029 DBMET02205

DBMET02205
0.1620.1620.166MAP-kinase-activated kinase 5 inhibitor

0.166 0.156 DBMET02205

DBMET02205
0.1350.1370.154I kappa B kinase epsilon inhibitor

0.138 0.133 DBMET03658

0.139 0.132 DBMET02204

0.154 0.116 DBMET02205

DBMET02205
0.030.0320.031Factor XI inhibitor

0.031 0.029 DBMET02205

DBMET02205
0.0920.0940.258Multidrug resistance-associated protein 1 inhibitor

0.258 0.005 DBMET03658

0.093 0.091 DBMET02213

DBMET03658
0.140.1420.164Ca2+/calmodulin-dependent kinase II beta inhibitor

0.164 0.111 DBMET03658

DBMET03658
0.0470.050.055Lysine-specific demethylase 1A inhibitor

0.055 0.036 DBMET02205

DBMET02205
0.0630.0660.125Rho-associated kinase I inhibitor

0.125 0.02 DBMET02205

DBMET02205
0.1840.1890.35Angiogenesis inhibitor

0.215 0.153 DBMET02204

0.202 0.167 DBMET02213

0.35 0.071 DBMET02214

DBMET02214
0.0260.0330.036Epoxide hydrolase 1 inhibitor

0.036 0.014 DBMET02205

DBMET02205
0.0410.050.045Neuropeptide Y5 antagonist

0.045 0.042 DBMET02205

DBMET02205
0.0530.0630.082I kappa B kinase 2 inhibitor

0.082 0.021 DBMET02205

DBMET02205
0.0680.0810.108I kappa B kinase inhibitor

0.108 0.033 DBMET02205

DBMET02205
0.0590.0730.067Epoxide hydrolase inhibitor

0.067 0.058 DBMET02205

DBMET02205
0.0550.0730.08Raf kinase inhibitor

0.066 0.059 DBMET02205

0.08 0.045 DBMET02214

DBMET02214
0.0180.0370.042Poly(ADP-ribose) polymerase 2 inhibitor

0.042 0.011 DBMET02205

DBMET02205
0.0750.0940.092MAP kinase kinase kinase inhibitor

0.092 0.075 DBMET02205

DBMET02205
0.1220.1420.177Clk dual-specificity kinase inhibitor

0.177 0.093 DBMET02205

DBMET02205
0.1090.1280.173CDC-like kinase 2 inhibitor

0.173 0.081 DBMET02205

DBMET02205
0.0350.0570.053Poly(ADP-ribose) polymerase inhibitor

0.053 0.021 DBMET02205

DBMET02205
0.0660.0890.095Protein kinase (Mos, Mil/Raf, MEKK, RIPK, TESK, LIMK, IRAK, ILK, Activin/TGF-beta) inhibitor

0.08 0.072 DBMET02205

0.095 0.058 DBMET02214

DBMET02214
0.0720.0960.086MAP kinase 9 inhibitor

0.086 0.075 DBMET02205

DBMET02205
0.0880.1140.136Protein-tyrosine kinase Lyn inhibitor

0.136 0.073 DBMET02214

DBMET02214
0.050.0770.095CDC7 inhibitor

0.095 0.026 DBMET02205

DBMET02205
0.150.1810.164ErbB-1 antagonist

0.164 0.146 DBMET02204

DBMET02204
0.0250.0570.038Poly(ADP-ribose) polymerase 1 inhibitor

0.038 0.026 DBMET02205

DBMET02205
0.1860.2210.249Toll-Like receptor 7 agonist

0.249 0.149 DBMET02204

0.229 0.168 DBMET02214

DBMET02204
0.0670.1020.083Vascular endothelial growth factor 1 antagonist

0.083 0.08 DBMET02214

DBMET02214
0.0640.1060.083Platelet activating factor alpha antagonist

0.083 0.077 DBMET02204

DBMET02204
0.0350.080.046Potassium channel (ATP-sensitive) activator

0.046 0.037 DBMET02205

DBMET02205
0.0360.0830.048Potassium channel (Inward rectifier) activator

0.048 0.039 DBMET02205

DBMET02205
0.0660.1150.101Ephrin antagonist

0.101 0.062 DBMET02214

DBMET02214
0.1790.230.241Toll-Like receptor agonist

0.241 0.157 DBMET02204

0.222 0.177 DBMET02214

DBMET02204
0.0810.1330.097Activin receptor-like kinase 4 inhibitor

0.097 0.091 DBMET02205

DBMET02205
0.0310.0870.051Raf kinase B inhibitor

0.051 0.05 DBMET02214

DBMET02214
0.0440.1020.1Rho-associated kinase inhibitor

0.1 0.035 DBMET02205

DBMET02205
0.0810.1410.113Ribosomal protein S6 kinase inhibitor

0.113 0.098 DBMET02205

DBMET02205
0.0980.1660.12NOS3 expression enhancer

0.12 0.115 DBMET02204

DBMET02204
0.060.1630.217Proto-oncogene tyrosine-protein kinase Yes inhibitor

0.217 0.037 DBMET02214

DBMET02214
0.0430.1480.065Heme oxygenase stimulant

0.065 0.033 DBMET02213

DBMET02213
0.040.1450.07MAP-kinase-activated kinase 2 inhibitor

0.07 0.057 DBMET02205

DBMET02205
0.0450.1590.078MAP-kinase-activated kinase inhibitor

0.078 0.065 DBMET02205

DBMET02205
0.0140.140.039Phosphodiesterase 3B inhibitor

0.039 0.038 DBMET02205

DBMET02205
0.0680.2230.175Cholinergic

0.175 0.059 DBMET03658

0.135 0.09 DBMET02214

DBMET03658
0.0260.1820.079CDK2/cyclin E2 inhibitor

0.079 0.039 DBMET02205

DBMET02205
0.0580.2360.116Dual specificity tyrosine-phosphorylation regulated kinase 1B inhibitor

0.116 0.111 DBMET02205

DBMET02205
0.0190.2290.044ATM kinase inhibitor

0.044 0.013 DBMET02204

DBMET02204
0.130.4020.24Cyclophilin D inhibitor

0.24 0.225 DBMET02205

DBMET02205
0.0740.3920.154Death-associated protein kinase 1 inhibitor

0.154 0.034 DBMET02205

DBMET02205
0.0160.4740.123Bronchodilator

0.123 0.043 DBMET02214

DBMET02214
0.0340.5240.204Tumour necrosis factor alpha release inhibitor

0.204 0.106 DBMET02214

DBMET02214
0.0430.7190.144Lipocortins synthesis antagonist

0.144 0.115 DBMET02213

DBMET02213
Ext Pa Pi Pmax Activity Other Results ID Pa_max