Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.880.0040.88Aldehyde oxidase inhibitor

0.236 0.088 DBMET02085

0.8250.0030.825Alcohol oxidase inhibitor

0.126 0.013 DBMET02085

0.7560.0170.781Caspase 9 stimulant

0.781 0.014 DBMET02085

DBMET02085
0.730.0030.811Alpha-N-acetylglucosaminidase inhibitor

0.811 0.002 DBMET02085

DBMET02085
0.6430.0050.643Cardiotonic

0.262 0.074 DBMET02085

0.6360.0120.738Vasodilator, peripheral

0.738 0.005 DBMET02085

DBMET02085
0.5840.0080.584Superoxide dismutase inhibitor
0.5660.0050.667Anesthetic general

0.667 0.004 DBMET02085

DBMET02085
0.5410.0060.541Sigma receptor agonist
0.5520.0190.5525 Hydroxytryptamine release inhibitor

0.482 0.039 DBMET02085

0.5470.0150.547GABA C receptor rho-3 antagonist
0.5350.0070.535Peroxidase inhibitor
0.540.0190.695Spasmolytic

0.695 0.006 DBMET02085

DBMET02085
0.5260.010.605Vasodilator

0.605 0.005 DBMET02085

DBMET02085
0.5120.0140.863Vasodilator, coronary

0.863 0.003 DBMET02085

DBMET02085
0.5190.0230.65Histamine release inhibitor

0.65 0.007 DBMET02085

DBMET02085
0.4950.0040.495GABA C receptor agonist

0.1 0.067 DBMET02085

0.5130.0250.5135 Hydroxytryptamine release stimulant

0.234 0.098 DBMET02085

0.5150.030.766Cholesterol antagonist

0.766 0.005 DBMET02085

DBMET02085
0.4490.0050.449Chelator

0.123 0.051 DBMET02085

0.4420.0050.442Tyrosine 3 hydroxylase inhibitor
0.4240.0040.614NADH dehydrogenase inhibitor

0.614 0.002 DBMET02085

DBMET02085
0.4320.0120.478Cyclic AMP phosphodiesterase inhibitor

0.478 0.008 DBMET02085

DBMET02085
0.4170.0060.476Peptidyltransferase inhibitor

0.476 0.004 DBMET02085

DBMET02085
0.4610.0540.461Ca2+/calmodulin-dependent protein kinase kinase A inhibitor
0.4030.0030.403Creatine kinase inhibitor

0.13 0.034 DBMET02085

0.4190.0180.419Calcium channel activator

0.227 0.176 DBMET02085

0.4030.0080.403Lipocortins synthesis antagonist

0.254 0.032 DBMET02085

0.40.0220.4Psychostimulant

0.334 0.035 DBMET02085

0.3710.0040.371Adenylate kinase inhibitor

0.281 0.008 DBMET02085

0.3710.0040.501Triose-phosphate isomerase inhibitor

0.501 0.002 DBMET02085

DBMET02085
0.3720.0070.487UDP-glucose 4-epimerase inhibitor

0.487 0.003 DBMET02085

DBMET02085
0.3690.0040.369Porphobilinogen synthase inhibitor
0.4080.0470.777Antithrombotic

0.777 0.005 DBMET02085

DBMET02085
0.380.0240.497DNA synthesis inhibitor

0.497 0.014 DBMET02085

DBMET02085
0.3570.0050.357Succinate dehydrogenase inhibitor

0.161 0.094 DBMET02085

0.3610.0120.681Amylase inhibitor

0.681 0.003 DBMET02085

DBMET02085
0.340.0040.34Phenylalanine 4-hydroxylase inhibitor

0.063 0.054 DBMET02085

0.3450.0130.345Glyceraldehyde-3-phosphate dehydrogenase inhibitor

0.293 0.026 DBMET02085

0.3530.0330.353Insulysin inhibitor
0.3450.0270.3455 Hydroxytryptamine uptake stimulant
0.3270.010.327Anesthetic local
0.3270.0110.624Alkylator

0.624 0.003 DBMET02085

DBMET02085
0.3850.070.59Immunosuppressant

0.59 0.014 DBMET02085

DBMET02085
0.3180.0060.318Ferrochelatase inhibitor
0.3220.0120.322Interleukin 6 antagonist

0.285 0.017 DBMET02085

0.3260.0160.326Phospholipase C inhibitor

0.217 0.034 DBMET02085

0.360.0620.632Immunostimulant

0.632 0.013 DBMET02085

DBMET02085
0.3030.0080.303Nav1.1 sodium channel blocker
0.3150.030.315MAP kinase kinase 2 inhibitor
0.290.0130.29Aldehyde dehydrogenase inhibitor

0.18 0.033 DBMET02085

0.2820.0070.2825 Hydroxytryptamine 3E antagonist
0.3140.0420.503Interleukin agonist

0.503 0.009 DBMET02085

DBMET02085
0.2770.0050.277Carbamoyl phosphate synthetase inhibitor

0.129 0.014 DBMET02085

0.2740.0040.274Aminopeptidase I inhibitor

0.105 0.025 DBMET02085

0.3010.0320.301Gastrin inhibitor

0.217 0.123 DBMET02085

0.2810.0160.281Adenylate cyclase inhibitor

0.171 0.034 DBMET02085

0.2680.0040.362Interferon agonist

0.362 0.002 DBMET02085

DBMET02085
0.3230.0590.323Sodium/bile acid cotransporter inhibitor

0.266 0.111 DBMET02085

0.3120.0520.452DNA damaging

0.452 0.019 DBMET02085

DBMET02085
0.2760.0190.276Nitric-oxide synthase stimulant

0.23 0.048 DBMET02085

0.2850.0320.327DNA methyltransferase I inhibitor

0.327 0.018 DBMET02085

DBMET02085
0.3330.0820.684Transcription factor NF kappa B inhibitor

0.684 0.022 DBMET02085

DBMET02085
0.2510.0030.484Alpha-mannosidase inhibitor

0.484 0.001 DBMET02085

DBMET02085
0.2820.0360.282RNA-directed DNA polymerase inhibitor

0.211 0.085 DBMET02085

0.3110.0660.581Interleukin 2 agonist

0.581 0.004 DBMET02085

DBMET02085
0.2530.0070.37Phosphofructokinase-1 inhibitor

0.37 0.004 DBMET02085

DBMET02085
0.2530.0110.253Mannose-6-phosphate isomerase inhibitor

0.253 0.011 DBMET02085

0.2530.0130.253Aminopeptidase B inhibitor

0.082 0.079 DBMET02085

0.2450.0070.245GABA C receptor antagonist
0.2540.0160.254DNA intercalator

0.225 0.02 DBMET02085

0.2740.0370.437DNA methylase inhibitor

0.437 0.009 DBMET02085

DBMET02085
0.2490.0140.294ATPase inhibitor

0.294 0.007 DBMET02085

DBMET02085
0.2490.0160.378Cell wall synthesis inhibitor

0.378 0.007 DBMET02085

DBMET02085
0.2350.0050.235Electrolyte absorption antagonist
0.2470.0180.247Cholesterol synthesis inhibitor

0.202 0.026 DBMET02085

0.2410.0150.241Nav1.3 sodium channel blocker
0.2330.0080.233Glutamate dehydrogenase inhibitor

0.128 0.02 DBMET02085

0.2830.0590.705Hypoglycemic

0.705 0.005 DBMET02085

DBMET02085
0.2490.0250.249Acetylcholine M1 receptor antagonist
0.2260.0060.226Adenylate cyclase stimulant

0.173 0.032 DBMET02085

0.2320.0110.232Arachidonic acid antagonist

0.178 0.056 DBMET02085

0.2320.0120.236UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor

0.236 0.011 DBMET02085

DBMET02085
0.2320.0120.232Nav1.6 sodium channel blocker
0.2350.0150.235GABA C receptor rho-2 antagonist
0.2250.0060.225Mannitol-1-phosphate 5-dehydrogenase inhibitor

0.211 0.006 DBMET02085

0.3010.0820.678Immunomodulator

0.678 0.006 DBMET02085

DBMET02085
0.2210.0030.498Mannosidase inhibitor

0.498 0.001 DBMET02085

DBMET02085
0.240.0270.24Bone formation stimulant

0.146 0.062 DBMET02085

0.2190.0070.219Sphingomyelinase inhibitor

0.193 0.011 DBMET02085

0.2350.0250.235Nav1.2 sodium channel blocker
0.2130.0040.213Acyl-CoA dehydrogenase inhibitor

0.102 0.016 DBMET02085

0.2190.0110.219Calcium antagonist
0.2280.0280.363Topoisomerase II inhibitor

0.363 0.012 DBMET02085

DBMET02085
0.250.0520.25ErbB-1 antagonist
0.2080.0140.208Catalase inhibitor
0.210.0150.435Cyclooxygenase 3 inhibitor

0.435 0.004 DBMET02085

DBMET02085
0.2180.0270.482Hemostatic

0.482 0.005 DBMET02085

DBMET02085
0.1980.0080.198GABA C receptor rho-1 antagonist
0.1970.0070.197Glutamate decarboxylase inhibitor
0.1990.0110.199Sphingosine 1-phosphate receptor 2 agonist
0.190.0040.193Ca2+-transporting ATPase inhibitor

0.193 0.004 DBMET02085

DBMET02085
0.1910.010.191Prolactin inhibitor
0.1870.0060.187Biliverdin reductase inhibitor

0.089 0.022 DBMET02085

0.190.0110.19Hematopoietic
0.1930.0140.193Gastric antisecretory

0.087 0.082 DBMET02085

0.1820.0040.273Interferon inducer

0.273 0.002 DBMET02085

DBMET02085
0.2180.040.218Cytidine deaminase inhibitor
0.2270.050.227P-glycoprotein inhibitor

0.186 0.074 DBMET02085

0.2050.0280.205MAP kinase kinase 5 inhibitor
0.2040.0290.204Catenin beta inhibitor
0.1810.0070.181Interleukin 5 antagonist

0.094 0.049 DBMET02085

0.3170.1430.317Calcium channel L-type activator
0.1880.0160.188Interleukin 8 antagonist
0.2250.0550.225Neurotrophic factor enhancer

0.176 0.103 DBMET02085

0.2080.0380.283Melanin inhibitor

0.283 0.024 DBMET02085

DBMET02085
0.2220.0530.222Insulin sensitizer

0.196 0.078 DBMET02085

0.2370.0690.237Neuropeptide Y2 antagonist
0.2620.0950.262Ca2+/calmodulin-dependent kinase II alpha inhibitor
0.1730.0090.173MAP kinase kinase 1 inhibitor
0.1910.0280.191Toll-Like receptor 2 antagonist
0.170.0080.17Ornithine carbamoyltransferase inhibitor

0.079 0.022 DBMET02085

0.1820.0220.182Sphingosine 1-phosphate receptor 5 antagonist
0.1770.0160.177Sphingosine 1-phosphate receptor 2 antagonist
0.1630.0040.163Estrogen-related receptor beta agonist

0.084 0.056 DBMET02085

0.190.0320.19MAP kinase kinase inhibitor
0.1690.0120.169Keratolytic
0.1850.0280.185Acetylcholine muscarinic antagonist
0.1850.0280.185Cystathionine beta-synthase inhibitor

0.102 0.074 DBMET02085

0.2350.0790.455Platelet antagonist

0.455 0.019 DBMET02085

DBMET02085
0.1820.0280.182Antibacterial (Helicobacter pylori)

0.16 0.039 DBMET02085

0.1630.010.183Acetylcholine release stimulant

0.183 0.005 DBMET02085

DBMET02085
0.170.0180.17Heat shock protein 70 antagonist

0.163 0.024 DBMET02085

0.1570.0070.157Sphingosine 1-phosphate receptor 4 agonist
0.1810.0310.363Topoisomerase I inhibitor

0.363 0.007 DBMET02085

DBMET02085
0.1590.0110.159Histamine N-methyltransferase inhibitor
0.1540.0060.154Glycine receptor agonist

0.129 0.01 DBMET02085

0.150.0030.15Phospholipase D inhibitor

0.092 0.02 DBMET02085

0.1690.0230.169Carbonic anhydrase III inhibitor

0.095 0.067 DBMET02085

0.1690.0230.169Mucolytic

0.154 0.03 DBMET02085

0.1630.0170.163Alcohol dehydrogenase inhibitor

0.108 0.044 DBMET02085

0.1920.0470.192Phospholipase A2 inhibitor

0.163 0.063 DBMET02085

0.1590.0160.159NAD(P)H dehydrogenase (quinone) inhibitor
0.1590.0180.159Histidine decarboxylase inhibitor
0.2220.0810.411Hypolipemic

0.411 0.023 DBMET02085

DBMET02085
0.2050.0660.205I kappa B kinase epsilon inhibitor
0.1780.0390.178Cholinergic antagonist
0.2330.0940.2335 Hydroxytryptamine 1E antagonist
0.2850.1470.644Antibacterial

0.644 0.014 DBMET02085

DBMET02085
0.1560.0180.156DOPA decarboxylase inhibitor
0.1990.0630.199Growth factor agonist

0.184 0.081 DBMET02085

0.1580.0220.284Topoisomerase II alpha inhibitor

0.284 0.008 DBMET02085

DBMET02085
0.1480.0120.148Lanosterol 14 alpha demethylase inhibitor
0.2120.0780.212Interleukin antagonist
0.1510.0170.151Anabolic

0.107 0.054 DBMET02085

0.1620.0280.174Vanilloid 1 agonist

0.174 0.021 DBMET02085

DBMET02085
0.180.0490.215Hexokinase inhibitor

0.215 0.027 DBMET02085

DBMET02085
0.1440.0120.144Myeloperoxidase inhibitor
0.1540.0240.154HIV-1 integrase (Overall Integration) inhibitor
0.1570.0270.216Photosensitizer

0.216 0.01 DBMET02085

DBMET02085
0.170.040.17Acetylcholine antagonist
0.1740.0450.223Alkaline phosphatase inhibitor

0.223 0.026 DBMET02085

DBMET02085
0.1570.0280.157Carbonic anhydrase XV inhibitor
0.1510.0220.151Nitric-oxide synthase inhibitor
0.140.0120.14Argininosuccinate synthase inhibitor

0.066 0.032 DBMET02085

0.1290.0030.167Glucose-6-phosphate isomerase inhibitor

0.167 0.002 DBMET02085

DBMET02085
0.1790.0540.267Diuretic

0.267 0.028 DBMET02085

DBMET02085
0.1760.0530.34Interferon gamma antagonist

0.34 0.015 DBMET02085

DBMET02085
0.2030.080.203Anticonvulsant
0.150.0280.15Potassium channel (Ca-activated) activator
0.1370.0150.137Glutathione S-transferase inhibitor
0.1960.0740.332Non-steroidal antiinflammatory agent

0.332 0.022 DBMET02085

DBMET02085
0.1320.0110.132NMDA receptor agonist
0.1240.0050.124Aconitate hydratase inhibitor
0.1530.0360.217Microtubule formation inhibitor

0.217 0.016 DBMET02085

DBMET02085
0.1620.0440.162MAP3K9 inhibitor
0.1740.0570.174Neurotensin receptor agonist
0.1490.0320.149Protein kinase C gamma inhibitor

0.105 0.068 DBMET02085

0.1210.0050.1215 Hydroxytryptamine 1B agonist
0.120.0040.12Squalene epoxidase inhibitor

0.101 0.005 DBMET02085

0.1190.0050.119Glucosylceramidase inhibitor

0.1 0.008 DBMET02085

0.2060.0920.857Angiogenesis stimulant

0.857 0.003 DBMET02085

DBMET02085
0.1180.0050.118MAP kinase kinase 7 inhibitor
0.1610.0480.161Toll-Like receptor antagonist
0.1620.0490.162Neurotrophic factor

0.134 0.076 DBMET02085

0.1420.0290.557Beta glucuronidase inhibitor

0.557 0.003 DBMET02085

DBMET02085
0.1680.0560.193Protein kinase stimulant

0.193 0.044 DBMET02085

DBMET02085
0.1360.0240.136Carbonic anhydrase VI inhibitor

0.091 0.046 DBMET02085

0.1460.0350.271DNA repair enzyme inhibitor

0.271 0.005 DBMET02085

DBMET02085
0.1390.0290.139Estrogen antagonist

0.106 0.084 DBMET02085

0.1250.0150.145Glycine receptor antagonist

0.145 0.008 DBMET02085

DBMET02085
0.1160.0070.116Gonadotropin-releasing hormone receptor agonist
0.1640.0550.164Toll-Like receptor 9 antagonist
0.1180.010.118Beta 3 adrenoreceptor antagonist
0.1650.0580.341Lipid peroxidase inhibitor

0.341 0.014 DBMET02085

DBMET02085
0.1220.0150.122Granulocyte macrophage colony stimulating factor agonist
0.1440.0380.291Expectorant

0.291 0.009 DBMET02085

DBMET02085
0.1130.0080.113Heat shock protein 90 beta antagonist
0.110.0050.11Epithelial sodium channel blocker
0.110.0050.11Factor XIIIa inhibitor
0.210.1050.21Calpain inhibitor
0.1560.0510.156NADPH oxidase inhibitor
0.1520.0480.152Aurora-C kinase inhibitor
0.2520.1480.252Calpain 2 inhibitor
0.1080.0040.1082,3-Oxidosqualene-lanosterol cyclase inhibitor

0.044 0.016 DBMET02085

0.1140.0090.114GABA B receptor agonist
0.1530.0480.153Pregnane X receptor agonist
0.1290.0260.129Aminoacyl-tRNA synthetase inhibitor
0.2250.1230.225Hypoxia-inducible factor 1 alpha inhibitor

0.195 0.158 DBMET02085

0.1240.0230.124Ornithine decarboxylase inhibitor
0.20.10.2Glucose-6-phosphate dehydrogenase-6-phosphogluconolactonase inhibitor
0.1870.0870.187Proto-oncogene tyrosine-protein kinase Fyn inhibitor
0.1170.0180.135Na+ K+ transporting ATPase inhibitor

0.135 0.01 DBMET02085

DBMET02085
0.1410.0420.141Sphingosine 1-phosphate receptor 4 antagonist
0.1480.050.258DNA polymerase I inhibitor

0.258 0.016 DBMET02085

DBMET02085
0.1040.0070.104Phosphoglycerate kinase inhibitor

0.044 0.016 DBMET02085

0.1240.0290.124Acetylcholine nicotinic antagonist
0.120.0250.12Adrenaline agonist
0.1030.0090.103Glutamate (mGluR6) antagonist
0.1070.0130.107NMDA receptor glycine site agonist
0.1140.0210.114mTOR complex 2 inhibitor
0.1540.0610.154MAP kinase 3 inhibitor
0.1570.0640.157CF transmembrane conductance regulator agonist

0.132 0.114 DBMET02085

0.0970.0040.097GABA uptake inhibitor
0.1350.0430.135TRPA1 agonist
0.110.0180.11I kappa B kinase 1 inhibitor
0.1550.0640.155Thiol protease inhibitor
0.1150.0250.115Glutamate release inhibitor

0.115 0.026 DBMET02085

0.1020.0130.221Phosphorylase inhibitor

0.221 0.004 DBMET02085

DBMET02085
0.0920.0030.092Hypoxanthine phosphoribosyltransferase inhibitor

0.071 0.005 DBMET02085

0.1330.0450.133Falcipain 3 inhibitor
0.1090.0210.109GABA aminotransferase inhibitor

0.109 0.022 DBMET02085

0.0920.0050.092Adenylate cyclase 1 inhibitor
0.1020.0150.102Beta adrenoreceptor antagonist
0.1010.0150.101Potassium channel (ATP-sensitive) blocker
0.1580.0710.158Cyclin-dependent kinase 8 inhibitor
0.0960.010.096Topoisomerase II beta inhibitor

0.047 0.037 DBMET02085

0.1550.0690.155Heat shock protein 90 antagonist
0.090.0050.128Arginase inhibitor

0.128 0.003 DBMET02085

DBMET02085
0.0890.0040.089Geranyltranstransferase inhibitor
0.1070.0220.107Fibroblast growth factor 2 antagonist
0.0980.0150.166Toll-Like receptor 2 agonist

0.166 0.01 DBMET02085

DBMET02085
0.1470.0640.147Cytokine production inhibitor
0.0910.0090.091Potassium channel (Inward rectifier) blocker
0.1160.0340.116Glutamate (mGluR7) agonist
0.1090.0280.109Histamine H2 receptor antagonist
0.0980.0170.098Purinergic P2X1 antagonist
0.1120.0320.112Carbonic anhydrase XIII inhibitor

0.078 0.051 DBMET02085

0.1610.0820.161Antipruritic
0.0960.0170.096Carbonic anhydrase VB inhibitor
0.0920.0130.092Exportin-1 inhibitor
0.1170.0380.117Interleukin 1 beta converting enzyme inhibitor
0.1120.0340.153Phosphodiesterase 6D inhibitor

0.153 0.009 DBMET02085

DBMET02085
0.1020.0240.102Calcium channel L-type blocker
0.0940.0180.094S-adenosyl-L-methionine decarboxylase inhibitor
0.1270.050.1275 Hydroxytryptamine 3A agonist
0.0960.020.096Vanilloid 4 agonist
0.0870.0120.087Sphingosine kinase 2 inhibitor
0.1080.0320.108Bromodomain-containing protein 2 inhibitor
0.0870.0120.087Sphingosine kinase inhibitor
0.1530.0790.353Thrombolytic

0.353 0.016 DBMET02085

DBMET02085
0.0930.0190.0935 Hydroxytryptamine 3 agonist
0.0850.0110.085Calcium channel P-type blocker
0.0810.0080.081Thymidine kinase inhibitor

0.057 0.015 DBMET02085

0.0910.0190.091Protein kinase C beta inhibitor

0.082 0.028 DBMET02085

0.0790.0070.079Fumarate hydratase inhibitor

0.04 0.019 DBMET02085

0.0810.0090.081Adenosine deaminase inhibitor

0.072 0.012 DBMET02085

0.0750.0030.075Estrogen-related receptor beta antagonist
0.0790.0090.079Sphingosine 1-phosphate receptor 3 agonist
0.1290.0590.184Beta amyloid protein antagonist

0.184 0.022 DBMET02085

DBMET02085
0.0910.0210.091Carbonic anhydrase stimulant
0.090.020.09NMDA 2C receptor antagonist
0.1030.0330.103Macrophage migration inhibitory factor inhibitor
0.1590.0890.159LIM domain kinase 1 inhibitor
0.1310.0620.131Cathepsin H inhibitor
0.0710.0020.071Estrogen-related receptor gamma antagonist
0.1180.050.219Mediator release inhibitor

0.219 0.012 DBMET02085

DBMET02085
0.0950.0280.095CC chemokine 5 receptor agonist
0.1610.0950.503Platelet adhesion inhibitor

0.503 0.005 DBMET02085

DBMET02085
0.0870.0210.087Potassium channel (Tandem pore domain) blocker
0.070.0040.07Uridine phosphorylase inhibitor

0.062 0.005 DBMET02085

0.0790.0130.079Nicotinic alpha3beta2 receptor antagonist
0.1010.0350.101CYP2A6 inhibitor
0.070.0050.07Guanylate cyclase inhibitor

0.064 0.008 DBMET02085

0.1570.0920.157Tumour necrosis factor antagonist
0.0950.030.095Estrogen receptor alpha antagonist
0.0820.0180.082MDM2 inhibitor
0.0960.0320.096Acetylcholine M4 receptor antagonist
0.0750.0120.075Beta 2 adrenoreceptor agonist
0.070.0070.079Neuraminidase (Influenza A) inhibitor

0.079 0.005 DBMET02085

DBMET02085
0.0890.0270.089Acetylcholine M5 receptor agonist
0.0740.0130.074Ryanodine receptor antagonist
0.070.010.07CC chemokine 4 receptor antagonist
0.0680.0080.068Membrane dipeptidase inhibitor
0.0750.0150.075H+/K+-transporting ATPase inhibitor
0.0630.0050.063Methionyl aminopeptidase 2 inhibitor
0.1010.0430.101Phosphodiesterase I inhibitor
0.0880.030.093Phosphodiesterase VI inhibitor

0.093 0.025 DBMET02085

DBMET02085
0.0810.0230.081Androgen agonist
0.0770.020.077Beta 1 adrenoreceptor antagonist
0.0660.0090.126Cytokine production stimulant

0.126 0.003 DBMET02085

DBMET02085
0.1320.0750.132Calcium channel blocker
0.0620.0060.062Lysine carboxypeptidase inhibitor
0.070.0140.07Pregnane X receptor antagonist
0.1960.140.196Transcription factor STAT3 inhibitor
0.0830.0280.083Acetylcholine M2 receptor antagonist
0.0740.0190.0743(or 17)beta-hydroxysteroid dehydrogenase inhibitor
0.0870.0320.087Carbonic anhydrase V inhibitor
0.0680.0130.068Immunoglobulin Fc receptor antagonist
0.0760.0210.076Cyclin D1 inhibitor
0.1740.1190.363Antiamyloidogenic

0.363 0.036 DBMET02085

DBMET02085
0.2680.2140.268MAP kinase 1 inhibitor
0.0860.0320.086Carbonic anhydrase VA inhibitor
0.0820.0270.082Cannabinoid CB1 receptor agonist
0.0790.0260.166Neuraminidase (influenza) inhibitor

0.166 0.006 DBMET02085

DBMET02085
0.0660.0130.066Sphingosine 1-phosphate receptor agonist
0.0670.0140.067Sodium/calcium exchanger inhibitor
0.1380.0850.138Neuropeptide Y1 antagonist
0.0930.040.093D-Ala-D-Ala ligase inhibitor
0.0780.0250.078Acetylcholine M5 receptor antagonist
0.0590.0080.0593-Hydroxyanthranilate 3,4-dioxygenase inhibitor
0.1810.1310.668Antioxidant

0.668 0.007 DBMET02085

DBMET02085
0.0620.0120.062Sphingosine 1-phosphate receptor 1 agonist
0.0610.0110.061Dopamine D5 agonist
0.0540.0050.056Ceramide glucosyltransferase inhibitor

0.056 0.005 DBMET02085

DBMET02085
0.0780.0290.078Glutamate (mGluR7) antagonist
0.0590.010.059Sphingosine kinase 1 inhibitor
0.0920.0440.092Vanilloid agonist

0.087 0.052 DBMET02085

0.1150.0670.115Caspase 3 inhibitor
0.0540.0060.054CF transmembrane conductance regulator antagonist
0.0620.0150.062Oxytocin agonist
0.0640.0170.064Carbonic anhydrase IV inhibitor
0.0730.0260.073Phosphodiesterase 1C inhibitor
0.0720.0260.072Acetylcholine muscarinic agonist
0.1150.0690.115Transcription factor STAT6 inhibitor
0.0740.0280.074Prostaglandin F2 alpha antagonist
0.0540.0090.054Glutamate (mGluR8) agonist
0.0640.0190.064Lysophosphatidic acid 3 receptor antagonist
0.0540.010.054Kainate receptor agonist
0.0610.0170.061Thymidylate synthase inhibitor
0.0590.0160.059Dopamine beta hydroxylase inhibitor
0.0690.0260.069Sphingosine 1-phosphate receptor 3 antagonist
0.0530.0110.053Glutamate (mGluR3) antagonist
0.0720.0290.072Cyclin-dependent kinase 6 inhibitor
0.1480.1050.1483C-like protease (Human coronavirus) inhibitor
0.090.0480.09Inducible nitric-oxide synthase inhibitor
0.0510.0090.0511-Alkyl-2-acetylglycerophosphocholine esterase inhibitor
0.0870.0450.087T cell inhibitor
0.0580.0160.058Leukotriene A4 hydrolase inhibitor
0.0970.0560.097Bile acid receptor antagonist
0.0450.0040.045Thymidine kinase (Herpes simplex virus 1) inhibitor

0.029 0.013 DBMET02085

0.0510.0110.051Delayed rectifier potassium channel blocker
0.0720.0320.126Neuraminidase inhibitor

0.126 0.009 DBMET02085

DBMET02085
0.0440.0050.044Lysophosphatidic acid receptor 1 agonist
0.0890.050.089Dual specificity tyrosine-phosphorylation regulated kinase 2 inhibitor
0.070.0310.07Acetylcholine M3 receptor antagonist
0.0670.0290.067Fibroblast growth factor 4 antagonist
0.0440.0070.044Follicle-stimulating hormone agonist
0.0650.0270.065Toll-Like receptor 8 antagonist
0.0540.0170.054Glutamate (mGluR4) antagonist
0.060.0230.06Vanilloid 2 antagonist
0.0440.0070.044Adenosine uptake inhibitor
0.070.0330.093Nitric oxide donor

0.093 0.012 DBMET02085

DBMET02085
0.0420.0060.042Purinergic P2Y15 antagonist
0.0540.0180.054Glutamate (mGluR1a) antagonist
0.0590.0240.059Bombesin 2 receptor antagonist
0.2230.1880.22315-Lipoxygenase inhibitor
0.0570.0230.057Potassium channel Kv1.3 blocker
0.0510.0170.051Plasmepsin II inhibitor
0.0920.0580.092Polo-like kinase-1 inhibitor
0.0510.0170.051Beta adrenoreceptor agonist
0.0370.0030.037Estrogen-related receptor gamma agonist
0.10.0670.1Urease inhibitor
0.0850.0510.085Caspase 7 inhibitor
0.060.0270.06Thromboxane synthase inhibitor
0.1050.0720.283Monophenol monooxygenase inhibitor

0.283 0.02 DBMET02085

DBMET02085
0.0410.0080.041LFA antagonist
0.0890.0550.089NMDA receptor antagonist
0.0370.0030.037Thymidine kinase (Herpes simplex virus 2) inhibitor
0.0580.0260.058Beta 2 adrenoreceptor antagonist
0.0430.0110.043Lysophosphatidic acid 2 receptor antagonist
0.0550.0230.055CC chemokine receptor 2B antagonist
0.0770.0460.077Lipase inhibitor
0.0720.0410.507Selectin antagonist

0.507 0.003 DBMET02085

DBMET02085
0.040.0090.04Glutamate (mGluR3) agonist
0.0350.0050.035ICAM 1 antagonist
0.0720.0430.072Neuronal nicotinic receptor antagonist
0.0370.0080.037Thymidine phosphorylase inhibitor
0.0640.0350.064Potassium channel intermediate-conductance Ca-activated blocker
0.0590.030.059Dihydroorotate oxidase inhibitor
0.0480.0190.048Dihydropteroate synthase inhibitor
0.0680.0410.091Carbonic anhydrase inhibitor

0.091 0.03 DBMET02085

DBMET02085
0.0860.0590.086Acetylcholine agonist
0.0570.030.057Sphingosine 1-phosphate receptor 5 agonist
0.1520.1250.152Ca2+/calmodulin-dependent kinase II beta inhibitor
0.1420.1150.223Amyloid beta aggregation inhibitor

0.223 0.067 DBMET02085

DBMET02085
0.030.0040.066Antibiotic Anthracycline-like

0.066 0.001 DBMET02085

DBMET02085
0.0460.020.046Heme oxygenase inhibitor
0.030.0040.03Lysophosphatidic acid receptor 3 agonist
0.1060.080.106Proteasome inhibitor
0.0850.060.085Androgen antagonist
0.0970.0710.097Estrogen receptor beta antagonist
0.0820.0570.082I kappa B kinase inhibitor
0.0580.0330.058Sphingosine 1-phosphate receptor 1 antagonist
0.1520.1280.152Focal adhesion kinase 2 inhibitor
0.0420.0180.042Retinoid X alpha receptor agonist
0.0290.0050.029Toll-Like receptor 8 agonist
0.0880.0640.088Antiadrenergic
0.0530.0290.053Antimetabolite

0.047 0.034 DBMET02085

0.0440.020.044Diamine oxidase inhibitor
0.0320.0080.032Prostaglandin F2 alpha agonist
0.060.0360.06Ribonucleotide reductase inhibitor
0.1420.1180.576Hepatoprotectant

0.576 0.005 DBMET02085

DBMET02085
0.0380.0140.038Protein kinase (CK2) beta inhibitor
0.0610.0370.061Xanthine dehydrogenase inhibitor
0.0280.0050.051Ileal bile acid transport inhibitor

0.051 0.004 DBMET02085

DBMET02085
0.0320.0090.032Hedgehog signaling activator
0.0590.0360.061Carbonic anhydrase II inhibitor

0.061 0.034 DBMET02085

DBMET02085
0.1170.0930.117Interleukin 1 antagonist
0.0990.0760.099Alpha 2b adrenoreceptor antagonist
0.0340.0110.034Dopamine autoreceptor agonist
0.0420.020.042Retinoid X receptor antagonist
0.0280.0050.028Neuraminidase (Influenza B) inhibitor
0.0470.0250.047Glutamate (mGluR group III) antagonist
0.0890.0670.089Protein kinase C zeta inhibitor
0.0770.0550.077Fibroblast growth factor 3 antagonist
0.0310.0090.036Vanilloid 2 agonist

0.036 0.005 DBMET02085

DBMET02085
0.0830.0610.083Antineoplastic alkaloid
0.1840.1620.184Transcription factor STAT inhibitor
0.0680.0470.068Potassium channel large-conductance Ca-activated activator
0.0570.0360.057Leukotriene C antagonist
0.1960.1750.312Caspase 3 stimulant

0.312 0.073 DBMET02085

DBMET02085
0.0410.020.041Calcitonin receptor agonist
0.0430.0210.043MAP3K5 inhibitor
0.0250.0040.025Methylmalonyl-CoA mutase inhibitor

0.018 0.012 DBMET02085

0.0320.0110.113Sodium/glucose cotransporter 2 inhibitor

0.113 0.002 DBMET02085

DBMET02085
0.0260.0050.026Carbonic anhydrase VIII inhibitor
0.0260.0050.026Carbonic anhydrase X inhibitor
0.0570.0360.057Ribonucleoside-diphosphate reductase inhibitor
0.0960.0760.244AMP-activated protein kinase stimulant

0.244 0.007 DBMET02085

DBMET02085
0.0640.0440.064Protease 3C (Human rhinovirus) inhibitor
0.0380.0180.038Retinoid X alpha receptor antagonist
0.0770.0570.077Viral attachment inhibitor
0.0430.0230.043Alpha 1d adrenoreceptor agonist
0.040.0210.04Vanilloid 3 antagonist
0.0410.0220.041Retinoid X receptor agonist
0.0420.0230.042Vascular adhesion protein 1 inhibitor
0.0420.0230.042AMPA 4 receptor antagonist
0.0360.0180.036Melatonin receptor 1A agonist
0.0380.020.038ATM kinase inhibitor
0.0560.0380.056Carbonic anhydrase I inhibitor
0.0280.010.028Glutamate (mGluR1a) agonist
0.0350.0170.035Peptide deformylase inhibitor
0.0260.0090.026Isoleucine-tRNA ligase inhibitor
0.0230.0050.023Vitamin D receptor agonist

0.02 0.007 DBMET02085

0.0350.0170.035Cholesterol ester transfer protein antagonist
0.050.0330.095Carbonic anhydrase XIV inhibitor

0.095 0.012 DBMET02085

DBMET02085
0.0390.0220.039Kainate receptor 2 antagonist
0.0750.0580.075Sphingosine 1-phosphate receptor antagonist
0.0570.0410.057Adenosine A1 receptor antagonist
0.0690.0530.069Telomerase inhibitor
0.0370.0210.037Tryptophan 5 hydroxylase inhibitor
0.0890.0730.165Xanthine oxidase inhibitor

0.165 0.029 DBMET02085

DBMET02085
0.0240.0080.024Retinoid X beta receptor antagonist
0.0450.0290.045AICAR transformylase inhibitor
0.0510.0360.0515 Hydroxytryptamine 4 antagonist
0.0290.0140.029Calcium-sensing receptor agonist
0.0190.0040.019Cyclin D2 inhibitor
0.0280.0130.028Acid ceramidase inhibitor
0.0280.0130.103Sodium/glucose cotransporter inhibitor

0.103 0.003 DBMET02085

DBMET02085
0.0230.0080.023Cyclin T1 inhibitor
0.0960.0810.096GABA receptor agonist
0.060.0450.06Corticotropin releasing factor 2 receptor antagonist
0.030.0150.03DNA polymerase III inhibitor
0.0590.0440.059Alpha 2 adrenoreceptor agonist
0.020.0050.02Thromboxane A2 agonist
0.040.0260.04Histone deacetylase 9 inhibitor
0.050.0360.05Prolyl endopeptidase inhibitor
0.0330.0190.033Endothelial nitric-oxide synthase inhibitor
0.0390.0250.039Farnesoid X receptor agonist
0.0810.0670.081Adrenaline antagonist
0.0160.0030.016Mannitol 2-dehydrogenase inhibitor
0.0350.0220.035Carnitine palmitoyltransferase 1 inhibitor
0.0470.0340.047Aldosterone antagonist
0.0350.0220.035Carnitine palmitoyltransferase inhibitor
0.0430.030.043Histamine H2 receptor agonist
0.0450.0310.045Purinergic P2Y antagonist
0.020.0070.024Telomerase stimulant

0.024 0.005 DBMET02085

DBMET02085
0.0340.0210.034Carboxypeptidase B inhibitor
0.0170.0050.0171-Deoxy-D-xylulose-5-phosphate reductoisomerase inhibitor
0.0520.040.174Heparanase inhibitor

0.174 0.002 DBMET02085

DBMET02085
0.0420.030.042Acetylcholine M1 receptor agonist
0.1820.1710.18212-Lipoxygenase inhibitor
0.0460.0350.046AMPA receptor antagonist
0.0580.0470.058Phosphodiesterase 1A inhibitor
0.2380.2270.821Cyclophilin D inhibitor

0.821 0.005 DBMET02085

DBMET02085
0.0370.0260.037Integrin alpha2 antagonist
0.0150.0040.015Purine nucleoside phosphorylase inhibitor
0.0810.070.081Interleukin-1 receptor-associated protein kinase 4 inhibitor
0.0790.0690.079Insulin growth factor antagonist
0.0420.0320.042Nerve growth factor antagonist
0.1450.1350.145Platelet aggregation inhibitor
0.0270.0170.027Integrin alpha2beta1 antagonist
0.0290.0190.029Nicotinic alpha4beta2 receptor agonist
0.0360.0270.036Histone deacetylase 7 inhibitor
0.0860.0770.086Phosphodiesterase 7B inhibitor
0.0250.0160.025Glutamate (mGluR1) agonist
0.0270.0190.027Myristoyl transferase inhibitor
0.0170.0090.017Purinergic P2Y1 agonist
0.0590.0510.059Dopamine D1 antagonist
0.0150.0070.015Integrin beta2 antagonist
0.0170.010.017Adenosine A2 receptor agonist
0.0190.0120.019Alpha 2b adrenoreceptor agonist
0.0260.0190.026Nicotinic acid receptor 2 antagonist
0.1490.1410.149Histone acetyltransferase inhibitor
0.0310.0240.031Methionyl aminopeptidase 1 inhibitor
0.0260.0180.026Thyroid hormone agonist
0.0670.060.067Peroxisome proliferator-activated receptor gamma antagonist
0.0280.0210.0285 Hydroxytryptamine 1D agonist
0.0250.0180.025Prostaglandin H2 antagonist
0.0380.0320.038CDK5/p25 inhibitor
0.0910.0850.091Protein kinase (CK2) alpha inhibitor
0.0320.0260.032Free fatty acid receptor 1 antagonist
0.0750.0690.075Insulin like growth factor 1 antagonist
0.0580.0530.058Neutrophil collagenase inhibitor
0.0360.0310.036Glucose-6-phosphate dehydrogenase inhibitor
0.0560.0510.056CDK1/cyclin B inhibitor
0.0750.0710.075Bcr-Abl kinase inhibitor
0.0130.0090.013DNA polymerase III polC-type inhibitor
0.0120.0080.012Glutamate (mGluR6) agonist
0.0260.0220.026Liver X receptor beta antagonist
0.0570.0530.057I kappa B kinase 2 inhibitor
0.0360.0320.036Erythropoietin receptor agonist
0.0670.0630.067Adenosine A3 receptor antagonist
0.0540.0510.074Lipocortins synthesis agonist

0.074 0.018 DBMET02085

DBMET02085
0.0540.0510.054Phosphodiesterase 1B inhibitor
0.0210.0170.021Prostaglandin EP2 agonist
0.0140.010.014Integrin alphaVbeta6 antagonist
0.0060.0020.006Reverse transcriptase (HBV) inhibitor
0.0370.0340.037Leukotriene C4 antagonist
0.0410.0380.041Histamine H1 receptor agonist
0.0160.0130.016CDK2/cyclin A3 inhibitor
0.0280.0250.028Prostaglandin agonist
0.040.0370.04GABA B receptor antagonist
0.120.1170.12Ca2+/calmodulin-dependent kinase II gamma inhibitor
0.0140.0110.014Adenosine A2a receptor agonist
0.0460.0440.046mTOR inhibitor
0.0360.0340.036Retinoic acid alpha receptor agonist
0.1110.1090.111Activin receptor-like kinase 2 inhibitor
0.0270.0250.027MAP3K8 inhibitor
0.0490.0470.049Nicotinic receptor alpha7 subunit antagonist
0.0540.0530.0545 Hydroxytryptamine 2A agonist
0.0180.0170.018Follicle-stimulating hormone antagonist
0.0240.0230.024CXC chemokine 2 receptor antagonist
0.010.0090.01Thromboxane agonist
0.0660.0650.066Metalloproteinase-9 inhibitor
0.0420.0440.106Carbonic anhydrase XII inhibitor

0.106 0.019 DBMET02085

DBMET02085
0.0090.010.011Purinergic P2Y2 agonist

0.011 0.006 DBMET02085

DBMET02085
0.0480.050.049Leukotriene B4 antagonist

0.049 0.046 DBMET02085

DBMET02085
0.020.0230.021Vitamin D receptor antagonist

0.021 0.019 DBMET02085

DBMET02085
0.0310.0350.09Antibiotic Aminoglycoside-like

0.09 0.004 DBMET02085

DBMET02085
0.2310.2360.68Apoptosis agonist

0.68 0.034 DBMET02085

DBMET02085
0.0850.1020.21Toll-Like receptor 4 antagonist

0.21 0.005 DBMET02085

DBMET02085
0.0310.0550.051Estrogen agonist

0.051 0.035 DBMET02085

DBMET02085
0.0130.0370.028Corticosteroid-like

0.028 0.008 DBMET02085

DBMET02085
0.1080.1330.333Insulin secretagoues

0.333 0.009 DBMET02085

DBMET02085
0.0090.0360.014S-adenosyl-L-homocysteine hydrolase inhibitor

0.014 0.012 DBMET02085

DBMET02085
0.0320.0590.065Carbonic anhydrase IX inhibitor

0.065 0.035 DBMET02085

DBMET02085
0.0410.070.049Factor III inhibitor

0.049 0.038 DBMET02085

DBMET02085
0.0770.110.09Interleukin 12 antagonist

0.09 0.072 DBMET02085

DBMET02085
0.1920.2280.484Alpha-glucosidase inhibitor

0.484 0.085 DBMET02085

DBMET02085
0.1310.1750.6Free radical scavenger

0.6 0.008 DBMET02085

DBMET02085
0.030.0790.137Protein 50S ribosomal subunit inhibitor

0.137 0.008 DBMET02085

DBMET02085
0.0350.0850.101Protein kinase C eta inhibitor

0.101 0.017 DBMET02085

DBMET02085
0.0420.1050.089Adenine nucleotide translocase inhibitor

0.089 0.006 DBMET02085

DBMET02085
0.0610.1370.108ATPase (Vacuolar H+) inhibitor

0.108 0.03 DBMET02085

DBMET02085
0.0710.1470.157Multidrug resistance-associated protein 1 inhibitor

0.157 0.022 DBMET02085

DBMET02085
0.0080.0850.048Squalene synthetase inhibitor

0.048 0.015 DBMET02085

DBMET02085
0.0140.1030.0321,3-Beta-glucan synthase inhibitor

0.032 0.011 DBMET02085

DBMET02085
0.0220.1120.04Protein kinase C beta I inhibitor

0.04 0.009 DBMET02085

DBMET02085
0.0020.0980.016Antibiotic Macrolide-like

0.016 0.008 DBMET02085

DBMET02085
0.0280.1350.239Antineoplastic antibiotic

0.239 0.015 DBMET02085

DBMET02085
0.0110.1190.072Protein 30S ribosomal subunit inhibitor

0.072 0.005 DBMET02085

DBMET02085
0.0160.140.05Toll-Like receptor 4 agonist

0.05 0.004 DBMET02085

DBMET02085
0.0480.1830.134Uric acid excretion stimulant

0.134 0.03 DBMET02085

DBMET02085
0.130.270.356Angiogenesis inhibitor

0.356 0.068 DBMET02085

DBMET02085
0.0210.1620.056Microtubule stabilization

0.056 0.02 DBMET02085

DBMET02085
0.0670.2080.399Cell adhesion inhibitor

0.399 0.005 DBMET02085

DBMET02085
0.0530.1990.17Transcription factor NF kappa B stimulant

0.17 0.012 DBMET02085

DBMET02085
0.0620.2360.175Interleukin 4 antagonist

0.175 0.032 DBMET02085

DBMET02085
0.0760.2560.468Nitric oxide antagonist

0.468 0.018 DBMET02085

DBMET02085
0.0230.2260.092Glucose-6-phosphate translocase inhibitor

0.092 0.008 DBMET02085

DBMET02085
0.0550.270.31Anticoagulant

0.31 0.027 DBMET02085

DBMET02085
0.1240.3430.554Apoptosis antagonist

0.554 0.014 DBMET02085

DBMET02085
0.0460.2760.131Protein-tyrosine phosphatase inhibitor

0.131 0.1 DBMET02085

DBMET02085
0.0250.2580.122Protein-tyrosine phosphatase 1B inhibitor

0.122 0.061 DBMET02085

DBMET02085
0.1490.4180.811Antiinflammatory

0.811 0.014 DBMET02085

DBMET02085
0.0660.3380.501Tumour necrosis factor alpha release inhibitor

0.501 0.014 DBMET02085

DBMET02085
0.0210.2940.106Factor IXa inhibitor

0.106 0.009 DBMET02085

DBMET02085
0.0920.3870.227Antiobesity

0.227 0.179 DBMET02085

DBMET02085
0.030.3350.229Cell adhesion molecule inhibitor

0.229 0.008 DBMET02085

DBMET02085
0.0050.380.019O6-alkylguanine-DNA alkyltransferase inhibitor

0.019 0.009 DBMET02085

DBMET02085
0.0270.8090.316NOS3 expression enhancer

0.316 0.016 DBMET02085

DBMET02085
0.0520.8820.141CC chemokine 6 receptor antagonist

0.141 0.038 DBMET02085

DBMET02085
Ext Pa Pi Pmax Activity Other Results ID Pa_max