Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.7680.0020.768Tyrosine 3 hydroxylase inhibitor

0.388 0.009 DBMET03097

0.6710.0020.671Phenylalanine 4-hydroxylase inhibitor

0.436 0.003 DBMET03097

0.6730.0170.673Cyclophilin D inhibitor

0.519 0.045 DBMET03097

0.5830.0030.5835 Hydroxytryptamine uptake stimulant

0.483 0.005 DBMET03097

0.5810.0050.581Peroxidase inhibitor

0.431 0.016 DBMET03097

0.5540.0090.554Superoxide dismutase inhibitor

0.441 0.02 DBMET03097

0.5070.0030.507Histidine decarboxylase inhibitor

0.272 0.008 DBMET03097

0.5030.0010.503DOPA decarboxylase inhibitor

0.273 0.003 DBMET03097

0.510.0260.7075 Hydroxytryptamine release stimulant

0.707 0.007 DBMET03097

DBMET03097
0.4670.0030.467Glutamate decarboxylase inhibitor

0.304 0.004 DBMET03097

0.460.0190.46Hypoglycemic

0.344 0.039 DBMET03097

0.4220.0210.422Interleukin 2 agonist

0.318 0.062 DBMET03097

0.4140.0170.414Interleukin agonist

0.299 0.048 DBMET03097

0.4330.0590.4335 Hydroxytryptamine release inhibitor

0.306 0.158 DBMET03097

0.4180.0460.418Cholesterol antagonist

0.217 0.15 DBMET03097

0.3740.0060.428GABA C receptor agonist

0.428 0.005 DBMET03097

DBMET03097
0.3970.0290.397Antiamyloidogenic

0.283 0.057 DBMET03097

0.3720.0130.372Phospholipase C inhibitor

0.332 0.016 DBMET03097

0.3570.0030.357Glutamate (mGluR group III) agonist

0.042 0.031 DBMET03097

0.3580.0040.358Catalase inhibitor

0.084 0.045 DBMET03097

0.3790.0260.379Psychostimulant

0.237 0.063 DBMET03097

0.3530.0020.353Glutamate (mGluR3) antagonist

0.067 0.007 DBMET03097

0.3520.0050.423Nitric-oxide synthase stimulant

0.423 0.003 DBMET03097

DBMET03097
0.3450.0070.345Cystathionine beta-synthase inhibitor

0.172 0.032 DBMET03097

0.3680.0350.368Free radical scavenger

0.352 0.038 DBMET03097

0.3220.010.322Insulin secretagoues

0.217 0.028 DBMET03097

0.3450.0340.345Angiogenesis stimulant

0.214 0.087 DBMET03097

0.3120.0050.312UDP-N-acetylglucosamine 1-carboxyvinyltransferase inhibitor

0.123 0.038 DBMET03097

0.3370.0390.337Insulysin inhibitor

0.286 0.067 DBMET03097

0.3060.0230.306Thrombolytic

0.157 0.077 DBMET03097

0.4130.1310.413Antiinflammatory

0.329 0.189 DBMET03097

0.2920.0110.292Cell adhesion inhibitor
0.3460.0650.346Immunostimulant

0.182 0.132 DBMET03097

0.3410.0630.341Immunomodulator
0.2750.0080.275NMDA receptor antagonist

0.237 0.01 DBMET03097

0.3440.0790.344Transcription factor NF kappa B inhibitor

0.287 0.102 DBMET03097

0.2740.010.274Aminopeptidase B inhibitor

0.151 0.037 DBMET03097

0.2790.020.279Monophenol monooxygenase inhibitor

0.158 0.044 DBMET03097

0.280.0210.28Insulin sensitizer

0.201 0.072 DBMET03097

0.3150.0560.315Antioxidant

0.293 0.064 DBMET03097

0.2630.0070.263Glutamate dehydrogenase inhibitor

0.098 0.032 DBMET03097

0.2980.0440.298DNA synthesis inhibitor

0.224 0.09 DBMET03097

0.3150.0620.333Aldehyde oxidase inhibitor

0.333 0.058 DBMET03097

DBMET03097
0.2690.0190.294Hemostatic

0.294 0.016 DBMET03097

DBMET03097
0.2610.0140.261Glutamate receptor antagonist

0.111 0.084 DBMET03097

0.2520.0070.252Glutamate receptor agonist

0.069 0.064 DBMET03097

0.2630.0210.263Alpha-N-acetylglucosaminidase inhibitor

0.139 0.062 DBMET03097

0.2770.0370.277Growth hormone agonist

0.14 0.095 DBMET03097

0.3130.0770.313Apoptosis antagonist

0.246 0.131 DBMET03097

0.2860.0510.286Pyruvate kinase inhibitor
0.2360.0060.236Argininosuccinate synthase inhibitor

0.054 0.042 DBMET03097

0.2390.0110.239Toll-Like receptor 2 antagonist

0.208 0.02 DBMET03097

0.2860.0580.286Platelet antagonist
0.2470.0220.247Neurotensin receptor agonist

0.18 0.05 DBMET03097

0.2630.0450.263Anesthetic general

0.215 0.067 DBMET03097

0.2340.0160.234Ferrochelatase inhibitor

0.198 0.023 DBMET03097

0.2460.0290.246Amylase inhibitor

0.154 0.062 DBMET03097

0.2190.0060.219Inducible nitric-oxide synthase inhibitor

0.206 0.008 DBMET03097

0.2120.0040.212AMPA 2 receptor antagonist
0.2340.0280.234Succinate dehydrogenase inhibitor

0.201 0.048 DBMET03097

0.2140.0080.214NMDA 2 receptor antagonist

0.202 0.009 DBMET03097

0.2530.0490.265Peptidyltransferase inhibitor

0.265 0.041 DBMET03097

DBMET03097
0.310.1090.31Immunosuppressant

0.218 0.178 DBMET03097

0.2930.0930.293Antithrombotic
0.3140.1160.314Histamine release inhibitor

0.208 0.193 DBMET03097

0.3130.1260.353Antibacterial

0.353 0.1 DBMET03097

DBMET03097
0.1890.0030.189Glutamate (mGluR6) antagonist

0.076 0.029 DBMET03097

0.1940.0090.194Keratolytic

0.115 0.023 DBMET03097

0.1940.010.194Prolactin inhibitor

0.134 0.029 DBMET03097

0.2370.0540.237Platelet adhesion inhibitor
0.1860.0050.186Glutamate (mGluR7) agonist

0.14 0.016 DBMET03097

0.2010.0210.201Farnesoid X receptor antagonist
0.180.0030.18Glutamate (mGluR1) agonist
0.1880.0110.2Nitric-oxide synthase inhibitor

0.2 0.009 DBMET03097

DBMET03097
0.1870.010.187Cell adhesion molecule inhibitor
0.190.0140.19HIV-1 integrase (Overall Integration) inhibitor

0.172 0.018 DBMET03097

0.1790.0030.179AMPA 3 receptor antagonist

0.037 0.016 DBMET03097

0.3340.1590.446Caspase 9 stimulant

0.446 0.085 DBMET03097

DBMET03097
0.1870.0130.2Creatine kinase inhibitor

0.2 0.01 DBMET03097

DBMET03097
0.190.0160.19Sphingosine 1-phosphate receptor 5 antagonist

0.173 0.031 DBMET03097

0.1910.0180.237Adenylate cyclase stimulant

0.237 0.005 DBMET03097

DBMET03097
0.2250.0520.225Hepatoprotectant

0.142 0.119 DBMET03097

0.2050.0390.205Interferon gamma antagonist

0.143 0.088 DBMET03097

0.1830.0180.183Mucolytic

0.107 0.068 DBMET03097

0.1650.0020.165Glutamate (mGluR8) agonist

0.061 0.007 DBMET03097

0.1690.0090.169Carbonic anhydrase stimulant

0.103 0.018 DBMET03097

0.1680.010.168Aminopeptidase I inhibitor

0.084 0.039 DBMET03097

0.1660.010.166Carbamoyl phosphate synthetase inhibitor

0.068 0.036 DBMET03097

0.1620.0090.345Myeloperoxidase inhibitor

0.345 0.003 DBMET03097

DBMET03097
0.1810.0280.181Chelator

0.145 0.037 DBMET03097

0.1970.0440.197Phospholipase A2 inhibitor

0.153 0.072 DBMET03097

0.2020.0520.202Anticoagulant
0.1680.0210.168Adenylate kinase inhibitor

0.114 0.049 DBMET03097

0.1630.0170.163Alcohol dehydrogenase inhibitor

0.117 0.037 DBMET03097

0.1480.0040.148AMPA 4 receptor antagonist

0.039 0.029 DBMET03097

0.2110.0670.217Neurotrophic factor enhancer

0.217 0.062 DBMET03097

DBMET03097
0.1710.0280.171Expectorant
0.1670.0240.173Sphingosine 1-phosphate receptor 2 antagonist

0.173 0.019 DBMET03097

DBMET03097
0.1570.0170.157Aminoacyl-tRNA synthetase inhibitor

0.082 0.073 DBMET03097

0.1870.0470.187Lipid peroxidase inhibitor

0.117 0.097 DBMET03097

0.1410.0020.141Kainate receptor agonist

0.042 0.027 DBMET03097

0.1460.0080.147GABA aminotransferase inhibitor

0.147 0.008 DBMET03097

DBMET03097
0.1640.0270.164Vanilloid 1 agonist

0.159 0.03 DBMET03097

0.1540.0170.154Phosphofructokinase-1 inhibitor

0.073 0.045 DBMET03097

0.1450.0090.145NMDA receptor agonist

0.063 0.043 DBMET03097

0.1770.0410.177Histone deacetylase SIRT1 inhibitor

0.165 0.05 DBMET03097

0.1490.0140.149Glutamate (mGluR) agonist
0.190.0560.209Antipruritic

0.209 0.043 DBMET03097

DBMET03097
0.1390.0060.2595 Hydroxytryptamine 2A agonist

0.259 0.003 DBMET03097

DBMET03097
0.1430.0110.143Integrin antagonist
0.160.0280.16Interleukin 8 antagonist

0.124 0.056 DBMET03097

0.1330.0020.133Tryptophan hydroxylase 1 inhibitor
0.1820.050.182Melanin inhibitor

0.17 0.059 DBMET03097

0.160.0280.16Heat shock protein 70 antagonist

0.152 0.042 DBMET03097

0.1660.0360.222Adenylate cyclase inhibitor

0.222 0.022 DBMET03097

DBMET03097
0.1730.0450.173Cell wall synthesis inhibitor

0.172 0.045 DBMET03097

0.2310.1030.231Gastrin inhibitor
0.1320.0050.132Kainate receptor antagonist
0.1350.0090.135Glycine transporter 2 inhibitor

0.065 0.023 DBMET03097

0.140.0140.14Ornithine decarboxylase inhibitor

0.115 0.03 DBMET03097

0.1320.0080.132NMDA receptor subunit 3B antagonist
0.180.0560.18Protein-tyrosine phosphatase inhibitor
0.1280.0040.128Glutamate (mGluR group III) antagonist
0.1280.0040.128Glutamate (mGluR7) antagonist

0.066 0.051 DBMET03097

0.1310.0110.131Ornithine carbamoyltransferase inhibitor

0.054 0.036 DBMET03097

0.120.0030.12Glutamate (mGluR1a) agonist

0.022 0.016 DBMET03097

0.1580.0420.158Cyclooxygenase 3 inhibitor

0.129 0.067 DBMET03097

0.20.0840.2Interleukin antagonist

0.163 0.109 DBMET03097

0.1230.0060.123NMDA receptor subunit 3A antagonist
0.1490.0340.149Nav1.4 sodium channel blocker

0.12 0.052 DBMET03097

0.1950.0810.234Amyloid beta aggregation inhibitor

0.234 0.063 DBMET03097

DBMET03097
0.1910.0790.191Non-steroidal antiinflammatory agent

0.175 0.091 DBMET03097

0.1160.0050.116Integrin alpha4 antagonist
0.2170.1070.269Spasmolytic

0.269 0.083 DBMET03097

DBMET03097
0.1140.0040.114Kainate receptor 2 antagonist
0.1420.0320.174Carbonic anhydrase III inhibitor

0.174 0.021 DBMET03097

DBMET03097
0.1180.0080.137GABA B receptor agonist

0.137 0.005 DBMET03097

DBMET03097
0.1440.0350.144Photosensitizer

0.121 0.055 DBMET03097

0.1330.0240.179Porphobilinogen synthase inhibitor

0.179 0.015 DBMET03097

DBMET03097
0.1130.0050.113VLA-4 antagonist
0.1120.0050.112AMPA 1 receptor antagonist
0.1090.0020.109Tryptophan 5 hydroxylase inhibitor

0.039 0.017 DBMET03097

0.2450.140.27Vasodilator, coronary

0.27 0.115 DBMET03097

DBMET03097
0.1350.030.135Toll-Like receptor 4 antagonist

0.134 0.031 DBMET03097

0.1070.0020.107Glutamate (mGluR3) agonist

0.036 0.014 DBMET03097

0.150.0460.15Cathepsin H inhibitor
0.130.0270.13Triose-phosphate isomerase inhibitor

0.107 0.041 DBMET03097

0.270.1660.27Analgesic

0.227 0.206 DBMET03097

0.1080.0050.108Glutamate (mGluR4) antagonist
0.1070.0040.107Dipeptidyl peptidase I inhibitor

0.099 0.004 DBMET03097

0.1050.0040.105Glutamate (mGluR4) agonist
0.2490.1490.249Toll-Like receptor agonist
0.1670.0680.167Arachidonic acid antagonist

0.161 0.075 DBMET03097

0.1170.020.135Vanilloid agonist

0.135 0.013 DBMET03097

DBMET03097
0.1160.0180.116Sphingosine 1-phosphate receptor 4 agonist
0.1590.0620.159Thiol protease inhibitor

0.131 0.094 DBMET03097

0.1120.0150.112Glycine receptor agonist

0.089 0.029 DBMET03097

0.1190.0230.119Glutathione S-transferase inhibitor
0.1110.0150.111Antimetabolite
0.1510.0580.151Bone formation stimulant
0.0960.0030.096AMPA receptor agonist
0.2440.1530.244Toll-Like receptor 7 agonist
0.1110.0190.111HIV-1 integrase inhibitor

0.1 0.025 DBMET03097

0.1420.0520.155Aldehyde dehydrogenase inhibitor

0.155 0.045 DBMET03097

DBMET03097
0.1060.0180.106Ribonucleoside-diphosphate reductase inhibitor
0.0890.0020.089Glutamate (mGluR6) agonist

0.011 0.01 DBMET03097

0.1510.0640.151Mannose-6-phosphate isomerase inhibitor

0.126 0.091 DBMET03097

0.1050.020.105Ribonucleotide reductase inhibitor
0.0880.0030.088Glutamate (mGluR8) antagonist

0.037 0.021 DBMET03097

0.1120.0280.112Bile acid receptor antagonist
0.1120.0270.112Opioid delta receptor antagonist
0.1220.0380.122Folate antagonist
0.0880.0050.088Arginase inhibitor

0.055 0.012 DBMET03097

0.0880.0050.088Glutamate (mGluR group II) antagonist
0.1330.0540.133Protein-tyrosine phosphatase 1B inhibitor
0.1770.0980.303Glyceraldehyde-3-phosphate dehydrogenase inhibitor

0.303 0.023 DBMET03097

DBMET03097
0.0970.0190.125Alcohol oxidase inhibitor

0.125 0.013 DBMET03097

DBMET03097
0.0820.0040.082Kainate receptor 1 antagonist
0.2290.1520.229Sodium/bile acid cotransporter inhibitor
0.0940.0180.094NMDA 2C receptor antagonist

0.077 0.027 DBMET03097

0.0780.0040.0783-Hydroxyanthranilate 3,4-dioxygenase inhibitor

0.076 0.004 DBMET03097

0.1720.0990.172DNA methylase inhibitor
0.1060.0330.188Adrenaline agonist

0.188 0.008 DBMET03097

DBMET03097
0.1930.120.193Calpain inhibitor
0.1030.0320.103Cathepsin G inhibitor
0.1390.0680.139Alkaline phosphatase inhibitor
0.0740.0030.074Thyroid hormone agonist

0.025 0.019 DBMET03097

0.0950.0250.095Glucagon-like peptide 1 agonist
0.1140.0450.114Anabolic

0.108 0.052 DBMET03097

0.2030.1340.253Transcription factor STAT inhibitor

0.253 0.085 DBMET03097

DBMET03097
0.0850.0180.085NMDA 2A receptor antagonist

0.053 0.034 DBMET03097

0.0790.0120.079Alpha-mannosidase inhibitor

0.071 0.016 DBMET03097

0.0820.0160.082Phosphorylase inhibitor
0.0860.0220.086Aminopeptidase microsomal inhibitor
0.1890.1250.189DNA damaging

0.18 0.134 DBMET03097

0.0910.0270.091Sirtuin 1 inhibitor

0.081 0.035 DBMET03097

0.1260.0620.165Beta amyloid protein antagonist

0.165 0.031 DBMET03097

DBMET03097
0.2350.1710.235Antiobesity
0.1210.0580.121Caspase 3 inhibitor
0.080.0170.08Botulinum neurotoxin type A inhibitor

0.08 0.017 DBMET03097

0.1070.0450.167Lanosterol 14 alpha demethylase inhibitor

0.167 0.007 DBMET03097

DBMET03097
0.1170.0550.196GABA C receptor antagonist

0.196 0.014 DBMET03097

DBMET03097
0.1570.0970.157DNA methyltransferase I inhibitor
0.1930.1330.195Neuropeptide Y2 antagonist

0.195 0.128 DBMET03097

DBMET03097
0.1040.0450.104Opioid antagonist
0.110.0510.11Factor V inhibitor
0.1960.1390.209Transcription factor STAT3 inhibitor

0.209 0.122 DBMET03097

DBMET03097
0.1380.0810.139Ca2+-transporting ATPase inhibitor

0.139 0.076 DBMET03097

DBMET03097
0.0990.0430.11Glutamate release inhibitor

0.11 0.03 DBMET03097

DBMET03097
0.0940.0390.158Macrophage migration inhibitory factor inhibitor

0.158 0.013 DBMET03097

DBMET03097
0.0640.0090.064Fumarate hydratase inhibitor
0.0650.010.065Carbonic anhydrase I stimulant

0.048 0.017 DBMET03097

0.1230.0690.33M18 aspartyl aminopeptidase inhibitor

0.33 0.009 DBMET03097

DBMET03097
0.1110.0580.142AMP-activated protein kinase stimulant

0.142 0.034 DBMET03097

DBMET03097
0.1820.1290.203RNA-directed DNA polymerase inhibitor

0.203 0.095 DBMET03097

DBMET03097
0.0610.0090.061Prostacyclin antagonist
0.0650.0140.065Mannosidase inhibitor

0.064 0.014 DBMET03097

0.0680.0170.068Adenine nucleotide translocase inhibitor
0.0630.0130.063AICAR transformylase inhibitor

0.048 0.025 DBMET03097

0.0890.0390.089Analgesic, opioid
0.0670.0180.067Glutamate (mGluR group I) agonist
0.0680.0190.068Aconitate hydratase inhibitor

0.053 0.035 DBMET03097

0.0690.020.092Beta 2 adrenoreceptor agonist

0.092 0.005 DBMET03097

DBMET03097
0.1260.0770.144Interleukin 4 antagonist

0.144 0.055 DBMET03097

DBMET03097
0.0540.0060.054Kainate receptor 4 antagonist
0.1140.0680.114Microtubule formation inhibitor
0.0660.0190.066Complement C3a chemotactic receptor antagonist
0.1670.1210.167Hypolipemic
0.0580.0130.206Dopamine D5 agonist

0.206 0.002 DBMET03097

DBMET03097
0.0840.0380.084Opioid mu receptor antagonist
0.0480.0050.048Integrin alpha4beta7 antagonist
0.0490.0050.049Kainate receptor 5 antagonist
0.1640.1210.243Histone acetyltransferase inhibitor

0.243 0.028 DBMET03097

DBMET03097
0.0780.0350.078HIV-1 integrase (3'-Processing) inhibitor

0.062 0.045 DBMET03097

0.0910.0480.091Hematopoietic
0.0790.0360.079Peroxisome proliferator-activated receptor gamma antagonist
0.0620.020.062Toll-Like receptor 2 agonist
0.0510.0090.051VCAM-1 antagonist
0.0510.0090.051VCAM antagonist
0.1490.1070.149Lipocortins synthesis antagonist
0.050.0090.05Catechol O-methyltransferase inhibitor

0.046 0.01 DBMET03097

0.0640.0230.064Aminopeptidase N inhibitor
0.1150.0740.115Histone deacetylase class III inhibitor
0.0680.0270.068Prolactin release inhibitor
0.0930.0530.095NADH dehydrogenase inhibitor

0.095 0.05 DBMET03097

DBMET03097
0.0620.0240.062AMPA receptor antagonist
0.1130.0750.113Alkylator
0.0630.0250.07Pregnane X receptor antagonist

0.07 0.014 DBMET03097

DBMET03097
0.0770.040.077Secretase beta inhibitor
0.0610.0240.061Dipeptidyl peptidase inhibitor

0.056 0.031 DBMET03097

0.0780.0420.078Peroxisome proliferator-activated receptor gamma agonist
0.1250.0880.179Protein kinase stimulant

0.179 0.051 DBMET03097

DBMET03097
0.0510.0150.051Glutamate (mGluR group II) agonist
0.0860.050.229Carbonic anhydrase VI inhibitor

0.229 0.01 DBMET03097

DBMET03097
0.2060.170.206Vasodilator, peripheral
0.140.1050.141Nitric oxide antagonist

0.141 0.103 DBMET03097

DBMET03097
0.0560.0210.056Thymidylate synthase inhibitor
0.1310.0960.136NOS3 expression enhancer

0.136 0.089 DBMET03097

DBMET03097
0.0680.0340.068Biliverdin reductase inhibitor

0.055 0.047 DBMET03097

0.0620.0280.062Angiotensin-converting enzyme inhibitor
0.110.0760.121DNA polymerase I inhibitor

0.121 0.067 DBMET03097

DBMET03097
0.0510.0190.051Dipeptidyl peptidase IV inhibitor

0.042 0.037 DBMET03097

0.0860.0540.094D-Ala-D-Ala ligase inhibitor

0.094 0.037 DBMET03097

DBMET03097
0.0570.0250.057Opioid mu receptor agonist
0.0410.010.041Lysine carboxypeptidase inhibitor
0.0870.0570.087Granulocyte macrophage colony stimulating factor agonist

0.083 0.066 DBMET03097

0.0350.0050.035Kainate receptor 3 antagonist
0.0630.0330.063Sphingosine 1-phosphate receptor 3 antagonist
0.050.020.05Leukotriene A4 hydrolase inhibitor

0.038 0.026 DBMET03097

0.1380.1090.138Interleukin 6 antagonist
0.0530.0240.134Dopamine beta hydroxylase inhibitor

0.134 0.003 DBMET03097

DBMET03097
0.080.0510.084Somatostatin 1 agonist

0.084 0.047 DBMET03097

DBMET03097
0.0320.0040.032Thyroid hormone alpha agonist
0.0320.0050.032Dipeptidyl peptidase IX inhibitor

0.022 0.008 DBMET03097

0.0520.0270.052Neurotensin receptor antagonist
0.0540.0290.054Lysophosphatidic acid 3 receptor antagonist
0.0410.0150.041Free fatty acid receptor 1 antagonist

0.03 0.029 DBMET03097

0.0550.030.082Beta 2 adrenoreceptor antagonist

0.082 0.011 DBMET03097

DBMET03097
0.0680.0440.068Selectin antagonist
0.0960.0720.289Carbonic anhydrase XV inhibitor

0.289 0.009 DBMET03097

DBMET03097
0.0530.0290.053CD45 antagonist
0.0550.0310.075Vanilloid 2 antagonist

0.075 0.011 DBMET03097

DBMET03097
0.0610.0380.067Sphingosine kinase inhibitor

0.067 0.029 DBMET03097

DBMET03097
0.0380.0150.043Dipeptidyl peptidase II inhibitor

0.043 0.012 DBMET03097

DBMET03097
0.0580.0350.058Leukotriene C antagonist

0.053 0.052 DBMET03097

0.0470.0240.062Beta adrenoreceptor agonist

0.062 0.007 DBMET03097

DBMET03097
0.0830.060.083Factor XII inhibitor
0.030.0090.03Integrin beta7 antagonist
0.0910.070.091Xanthine oxidase inhibitor
0.050.030.05Endothelin-converting enzyme inhibitor
0.0450.0260.045Sphingosine 1-phosphate receptor 1 agonist

0.044 0.026 DBMET03097

0.0470.0280.047Sphingosine 1-phosphate receptor agonist

0.045 0.03 DBMET03097

0.0610.0410.061HIV-1 integrase (Strand Transfer) inhibitor
0.0780.060.078Glycine receptor antagonist
0.0540.0360.054Aldose reductase inhibitor
0.0410.0230.0725 Hydroxytryptamine 2B agonist

0.072 0.005 DBMET03097

DBMET03097
0.0420.0260.042Integrin alpha5beta1 antagonist
0.0280.0120.028Vanilloid 2 agonist

0.028 0.013 DBMET03097

0.1010.0850.111Cholesterol synthesis inhibitor

0.111 0.074 DBMET03097

DBMET03097
0.0520.0360.062Carbonic anhydrase II stimulant

0.062 0.021 DBMET03097

DBMET03097
0.1480.1320.148Anticonvulsant

0.147 0.133 DBMET03097

0.0550.0390.08Sphingosine kinase 2 inhibitor

0.08 0.015 DBMET03097

DBMET03097
0.240.2250.24Apoptosis agonist
0.0410.0260.041Membrane dipeptidase inhibitor
0.060.0450.06NMDA receptor glycine site agonist
0.1060.0910.158Transcription factor STAT6 inhibitor

0.158 0.018 DBMET03097

DBMET03097
0.0410.0280.041Erythropoietin receptor agonist
0.0330.020.033HCV NS5B polymerase inhibitor
0.0350.0220.035Calcitonin receptor agonist
0.060.0470.06Trypsin inhibitor

0.059 0.051 DBMET03097

0.0470.0350.047Glucose-6-phosphate isomerase inhibitor
0.0480.0360.048Bombesin 2 receptor antagonist
0.0190.0070.019Dipeptidyl peptidase VIII inhibitor

0.014 0.012 DBMET03097

0.0380.0260.038Integrin alpha1beta1 antagonist
0.0510.0390.051Opioid agonist
0.0370.0260.112Kinesin-like protein 1 inhibitor

0.112 0.006 DBMET03097

DBMET03097
0.0370.0260.112Kinesin antagonist

0.112 0.006 DBMET03097

DBMET03097
0.030.0190.03Glutamate (mGluR2) antagonist
0.0190.0080.019Thyroid hormone alpha antagonist
0.0150.0040.015Thyroid hormone beta agonist
0.0240.0140.024ICAM 1 antagonist
0.0310.0210.031Endothelial nitric-oxide synthase inhibitor
0.0340.0250.034Opioid delta receptor agonist
0.0190.010.019Nicotinic acid receptor 1 antagonist
0.0610.0530.109Beta adrenoreceptor antagonist

0.109 0.013 DBMET03097

DBMET03097
0.0190.0110.019Aminopeptidase A inhibitor
0.0310.0230.031Glutamate (mGluR2) agonist
0.0270.0190.027NMDA 2D receptor antagonist
0.0330.0250.033RNA-directed RNA polymerase inhibitor
0.050.0430.093(or 17)beta-hydroxysteroid dehydrogenase inhibitor

0.09 0.013 DBMET03097

DBMET03097
0.0790.0720.079Transcription factor NF kappa B stimulant
0.0520.0450.086Epithelial sodium channel blocker

0.086 0.01 DBMET03097

DBMET03097
0.0190.0130.019Integrin alphaVbeta1 antagonist
0.050.0440.057Leukotriene B4 antagonist

0.057 0.031 DBMET03097

DBMET03097
0.0350.0290.035Integrin alpha2 antagonist
0.0850.080.085Protease inhibitor
0.0590.0540.059Protease 3C (Human rhinovirus) inhibitor
0.0260.0210.026Baculoviral IAP repeat-containing protein 4 inhibitor
0.0220.0170.027Prostaglandin F2 alpha agonist

0.027 0.01 DBMET03097

DBMET03097
0.0710.0680.071Chymotrypsin inhibitor
0.0430.0390.043GP IIb/IIIa receptor antagonist
0.0390.0360.039Cathepsin F inhibitor
0.0250.0220.025Integrin alpha2beta1 antagonist
0.0870.0840.133GABA C receptor rho-1 antagonist

0.133 0.03 DBMET03097

DBMET03097
0.0310.0280.031Carboxypeptidase B inhibitor
0.0780.0760.105Estrogen-related receptor beta agonist

0.105 0.019 DBMET03097

DBMET03097
0.0160.0140.016Telomerase stimulant
0.1380.1360.138Catenin beta inhibitor
0.0570.0550.057Caspase 9 inhibitor
0.0240.0230.044Uridine phosphorylase inhibitor

0.044 0.01 DBMET03097

DBMET03097
0.0280.0280.042Sirtuin 2 inhibitor

0.042 0.016 DBMET03097

DBMET03097
0.1730.1730.226Lipoxygenase inhibitor

0.226 0.117 DBMET03097

DBMET03097
0.050.0530.0653-Oxoacyl-[acyl-carrier-protein] synthase inhibitor

0.065 0.035 DBMET03097

DBMET03097
0.1320.1360.143ATPase inhibitor

0.143 0.113 DBMET03097

DBMET03097
0.0360.0410.038Sphingosine kinase 1 inhibitor

0.038 0.035 DBMET03097

DBMET03097
0.0220.0290.029Somatostatin 5 antagonist

0.029 0.024 DBMET03097

DBMET03097
0.0150.0230.027Estrogen-related receptor gamma agonist

0.027 0.005 DBMET03097

DBMET03097
0.0180.0260.049Dopamine D1 agonist

0.049 0.005 DBMET03097

DBMET03097
0.0280.0380.046Somatostatin 5 agonist

0.046 0.014 DBMET03097

DBMET03097
0.0180.0290.026Beta 1 adrenoreceptor agonist

0.026 0.011 DBMET03097

DBMET03097
0.0610.0720.063MDM2 inhibitor

0.063 0.061 DBMET03097

DBMET03097
0.070.0820.09MAP kinase kinase 7 inhibitor

0.09 0.024 DBMET03097

DBMET03097
0.0410.0530.051Topoisomerase II beta inhibitor

0.051 0.031 DBMET03097

DBMET03097
0.0780.0920.084Protein kinase C zeta inhibitor

0.084 0.077 DBMET03097

DBMET03097
0.0890.1030.243MAO inhibitor

0.243 0.029 DBMET03097

DBMET03097
0.0410.0550.051Acyl-CoA dehydrogenase inhibitor

0.051 0.042 DBMET03097

DBMET03097
0.0310.0450.049Oxytocin agonist

0.049 0.024 DBMET03097

DBMET03097
0.0240.0390.047Estradiol 17 beta-dehydrogenase 2 inhibitor

0.047 0.017 DBMET03097

DBMET03097
0.0260.0420.0411-Alkyl-2-acetylglycerophosphocholine esterase inhibitor

0.041 0.015 DBMET03097

DBMET03097
0.0950.1130.123Estrogen antagonist

0.123 0.05 DBMET03097

DBMET03097
0.0550.0730.078Beta 3 adrenoreceptor antagonist

0.078 0.024 DBMET03097

DBMET03097
0.0370.0590.1155 Hydroxytryptamine 2 agonist

0.115 0.007 DBMET03097

DBMET03097
0.0750.0960.1Urease inhibitor

0.1 0.067 DBMET03097

DBMET03097
0.1060.1280.115Papain-like protease (SARS coronavirus) inhibitor

0.115 0.095 DBMET03097

DBMET03097
0.0710.0940.0895-Lipoxygenase inhibitor

0.089 0.073 DBMET03097

DBMET03097
0.0750.0990.094UDP-glucose 4-epimerase inhibitor

0.094 0.067 DBMET03097

DBMET03097
0.0510.0780.127Carbonic anhydrase VA inhibitor

0.127 0.016 DBMET03097

DBMET03097
0.0110.0390.033Estradiol 17 beta-dehydrogenase 1 inhibitor

0.033 0.011 DBMET03097

DBMET03097
0.0970.1280.167Nav1.6 sodium channel blocker

0.167 0.038 DBMET03097

DBMET03097
0.0510.0830.167Carbonic anhydrase XIII inhibitor

0.167 0.019 DBMET03097

DBMET03097
0.0330.0650.064Carbonic anhydrase XIV inhibitor

0.064 0.023 DBMET03097

DBMET03097
0.0230.0580.121Diamine oxidase inhibitor

0.121 0.004 DBMET03097

DBMET03097
0.0440.080.14Carbonic anhydrase V inhibitor

0.14 0.017 DBMET03097

DBMET03097
0.050.0860.096Na+ K+ transporting ATPase inhibitor

0.096 0.035 DBMET03097

DBMET03097
0.0260.0640.037GABA uptake inhibitor

0.037 0.032 DBMET03097

DBMET03097
0.0190.0580.035Cholesterol ester transfer protein antagonist

0.035 0.017 DBMET03097

DBMET03097
0.0360.0750.087Beta 1 adrenoreceptor antagonist

0.087 0.014 DBMET03097

DBMET03097
0.0220.0640.047Estradiol 17 beta-dehydrogenase inhibitor

0.047 0.027 DBMET03097

DBMET03097
0.0560.0990.114Protein kinase A inhibitor

0.114 0.037 DBMET03097

DBMET03097
0.020.0640.031Estrogen-related receptor gamma antagonist

0.031 0.014 DBMET03097

DBMET03097
0.0720.1180.108Estrogen receptor beta antagonist

0.108 0.05 DBMET03097

DBMET03097
0.0260.0780.125Carbonic anhydrase VB inhibitor

0.125 0.012 DBMET03097

DBMET03097
0.0470.10.07NAD(P)H dehydrogenase (quinone) inhibitor

0.07 0.061 DBMET03097

DBMET03097
0.0550.1080.083S-adenosyl-L-methionine decarboxylase inhibitor

0.083 0.033 DBMET03097

DBMET03097
0.0470.1020.067Nav1.8 sodium channel blocker

0.067 0.06 DBMET03097

DBMET03097
0.0950.150.139Acetylcholine M1 receptor antagonist

0.139 0.086 DBMET03097

DBMET03097
0.1530.2140.192Hypoxia-inducible factor 1 alpha inhibitor

0.192 0.161 DBMET03097

DBMET03097
0.0340.0970.068NMDA 2B receptor antagonist

0.068 0.026 DBMET03097

DBMET03097
0.0570.1210.091Estrogen receptor alpha antagonist

0.091 0.034 DBMET03097

DBMET03097
0.1810.2450.309Calcium channel activator

0.309 0.083 DBMET03097

DBMET03097
0.0070.0720.038Alpha 2a adrenoreceptor agonist

0.038 0.004 DBMET03097

DBMET03097
0.2020.270.235Calcium channel L-type activator

0.235 0.222 DBMET03097

DBMET03097
0.0150.0850.043Phosphoglycerate kinase inhibitor

0.043 0.017 DBMET03097

DBMET03097
0.0230.0940.046Geranyltranstransferase inhibitor

0.046 0.027 DBMET03097

DBMET03097
0.0790.1570.161NADPH oxidase inhibitor

0.161 0.048 DBMET03097

DBMET03097
0.0460.1280.063Histone deacetylase SIRT3 inhibitor

0.063 0.04 DBMET03097

DBMET03097
0.0740.1590.108TRPA1 agonist

0.108 0.075 DBMET03097

DBMET03097
0.0640.1510.104MAP kinase kinase 1 inhibitor

0.104 0.051 DBMET03097

DBMET03097
0.0140.1030.063TRPM8 blocker

0.063 0.011 DBMET03097

DBMET03097
0.0370.1280.07Protein kinase C beta inhibitor

0.07 0.048 DBMET03097

DBMET03097
0.0370.1290.056I kappa B kinase 2 inhibitor

0.056 0.055 DBMET03097

DBMET03097
0.0250.1170.084Adenylate cyclase 1 inhibitor

0.084 0.006 DBMET03097

DBMET03097
0.0630.1560.109Acetylcholine muscarinic antagonist

0.109 0.08 DBMET03097

DBMET03097
0.1640.2620.321GABA C receptor rho-3 antagonist

0.321 0.103 DBMET03097

DBMET03097
0.0290.1330.114Dopamine agonist

0.114 0.022 DBMET03097

DBMET03097
0.0720.1790.132Nav1.2 sodium channel blocker

0.132 0.071 DBMET03097

DBMET03097
0.0130.1210.026Purinergic P2Y15 antagonist

0.026 0.025 DBMET03097

DBMET03097
0.0630.1720.081CC chemokine 5 receptor agonist

0.081 0.059 DBMET03097

DBMET03097
0.0230.1340.061Acetylcholine M3 receptor antagonist

0.061 0.04 DBMET03097

DBMET03097
0.0420.1590.131Histamine N-methyltransferase inhibitor

0.131 0.023 DBMET03097

DBMET03097
0.010.1290.0565 Hydroxytryptamine 2C agonist

0.056 0.024 DBMET03097

DBMET03097
0.1040.2250.127MAP kinase kinase 4 inhibitor

0.127 0.125 DBMET03097

DBMET03097
0.040.1670.075I kappa B kinase inhibitor

0.075 0.068 DBMET03097

DBMET03097
0.0240.1640.101Alpha 2 adrenoreceptor agonist

0.101 0.014 DBMET03097

DBMET03097
0.0510.1920.104GABA receptor agonist

0.104 0.072 DBMET03097

DBMET03097
0.0270.170.194MAO B inhibitor

0.194 0.026 DBMET03097

DBMET03097
0.0130.160.057Alpha 1d adrenoreceptor agonist

0.057 0.012 DBMET03097

DBMET03097
0.1360.2920.2525 Hydroxytryptamine 3E antagonist

0.252 0.015 DBMET03097

DBMET03097
0.0180.1840.048Histamine H1 receptor agonist

0.048 0.021 DBMET03097

DBMET03097
0.040.2080.1Sphingomyelinase inhibitor

0.1 0.06 DBMET03097

DBMET03097
0.070.2410.156Protein kinase (CK1) gamma 3 inhibitor

0.156 0.083 DBMET03097

DBMET03097
0.0580.2360.118Nav1.5 sodium channel blocker

0.118 0.058 DBMET03097

DBMET03097
0.0860.2640.132CF transmembrane conductance regulator agonist

0.132 0.114 DBMET03097

DBMET03097
0.0430.2260.2355 Hydroxytryptamine 3A agonist

0.235 0.007 DBMET03097

DBMET03097
0.0150.1970.049Histamine H2 receptor agonist

0.049 0.022 DBMET03097

DBMET03097
0.050.2340.127Sodium channel (voltage-gated) blocker

0.127 0.076 DBMET03097

DBMET03097
0.0790.2770.139Tumour necrosis factor antagonist

0.139 0.115 DBMET03097

DBMET03097
0.0230.230.1285 Hydroxytryptamine 2C antagonist

0.128 0.033 DBMET03097

DBMET03097
0.020.2280.115Alpha adrenoreceptor agonist

0.115 0.023 DBMET03097

DBMET03097
0.0240.2350.109CYP2A6 inhibitor

0.109 0.032 DBMET03097

DBMET03097
0.0110.2240.037Melatonin 1 agonist

0.037 0.018 DBMET03097

DBMET03097
0.0540.2720.173Toll-Like receptor antagonist

0.173 0.042 DBMET03097

DBMET03097
0.020.240.061Dopamine D1 antagonist

0.061 0.049 DBMET03097

DBMET03097
0.0660.2920.161MAP kinase kinase 2 inhibitor

0.161 0.112 DBMET03097

DBMET03097
0.0450.2730.126Sodium channel blocker

0.126 0.078 DBMET03097

DBMET03097
0.0060.2390.051Vascular adhesion protein 1 inhibitor

0.051 0.015 DBMET03097

DBMET03097
0.090.3260.19Death-associated protein kinase 2 inhibitor

0.19 0.043 DBMET03097

DBMET03097
0.1050.3460.25315-Lipoxygenase inhibitor

0.253 0.162 DBMET03097

DBMET03097
0.0070.2630.0295 Hydroxytryptamine 6 agonist

0.029 0.02 DBMET03097

DBMET03097
0.0130.2710.1175 Hydroxytryptamine 2A antagonist

0.117 0.039 DBMET03097

DBMET03097
0.020.2790.0635 Hydroxytryptamine 7 agonist

0.063 0.027 DBMET03097

DBMET03097
0.0330.2930.1135 Hydroxytryptamine 2B antagonist

0.113 0.068 DBMET03097

DBMET03097
0.1720.4450.27Ca2+/calmodulin-dependent protein kinase kinase A inhibitor

0.27 0.256 DBMET03097

DBMET03097
0.0220.3010.1435 Hydroxytryptamine 2 antagonist

0.143 0.047 DBMET03097

DBMET03097
0.010.3040.0875 Hydroxytryptamine 1F antagonist

0.087 0.038 DBMET03097

DBMET03097
0.0080.3070.032Melatonin agonist

0.032 0.024 DBMET03097

DBMET03097
0.0220.3440.0855 Hydroxytryptamine 5A antagonist

0.085 0.021 DBMET03097

DBMET03097
0.0190.3470.0755 Hydroxytryptamine 3 agonist

0.075 0.031 DBMET03097

DBMET03097
0.0050.3470.041Dopamine D2 agonist

0.041 0.033 DBMET03097

DBMET03097
0.010.3620.054Alpha 1 adrenoreceptor agonist

0.054 0.045 DBMET03097

DBMET03097
0.0180.3740.0735 Hydroxytryptamine 5 antagonist

0.073 0.024 DBMET03097

DBMET03097
0.0540.4170.2825 Hydroxytryptamine 1E antagonist

0.282 0.043 DBMET03097

DBMET03097
0.0160.3880.093Alpha 2a adrenoreceptor antagonist

0.093 0.04 DBMET03097

DBMET03097
0.0060.3910.1795 Hydroxytryptamine agonist

0.179 0.017 DBMET03097

DBMET03097
0.0120.4280.083Pim-1 kinase inhibitor

0.083 0.076 DBMET03097

DBMET03097
0.0150.4480.095Alpha 2 adrenoreceptor antagonist

0.095 0.052 DBMET03097

DBMET03097
0.020.4580.081Histamine H2 receptor antagonist

0.081 0.063 DBMET03097

DBMET03097
0.0140.4610.084Adrenaline antagonist

0.084 0.064 DBMET03097

DBMET03097
0.0140.4610.09Antiadrenergic

0.09 0.063 DBMET03097

DBMET03097
0.0360.4910.144Ca2+/calmodulin-dependent protein kinase inhibitor

0.144 0.117 DBMET03097

DBMET03097
0.0160.4820.149Ca2+/calmodulin-dependent kinase II delta inhibitor

0.149 0.066 DBMET03097

DBMET03097
0.0040.7370.0985 Hydroxytryptamine 1 agonist

0.098 0.021 DBMET03097

DBMET03097
0.0070.8410.15 Hydroxytryptamine 1B agonist

0.1 0.007 DBMET03097

DBMET03097
Ext Pa Pi Pmax Activity Other Results ID Pa_max