Min Pa: Min Pa(max): Activity's type:

Ext Pa Pi Pmax Activity Other Results ID Pa_max
0.3750.0040.733Phosphodiesterase IV inhibitor

0.48 0.004 DBMET03249

0.435 0.004 DBMET03250

0.733 0.003 DBMET03251

DBMET03251
0.4060.0630.5Antiobesity

0.387 0.071 DBMET03249

0.482 0.041 DBMET03250

0.5 0.037 DBMET03251

DBMET03251
0.3410.0030.364Lysine-specific demethylase 1A inhibitor

0.168 0.004 DBMET03249

0.364 0.003 DBMET03250

0.09 0.009 DBMET03251

DBMET03250
0.3710.0330.371HERG channel blocker

0.289 0.052 DBMET03249

0.356 0.036 DBMET03250

0.315 0.045 DBMET03251

0.4150.0830.429Cyclophilin D inhibitor

0.387 0.098 DBMET03249

0.429 0.076 DBMET03250

DBMET03250
0.3250.0240.363Interleukin-1 receptor-associated protein kinase 1 inhibitor

0.327 0.024 DBMET03249

0.363 0.016 DBMET03250

0.248 0.049 DBMET03251

DBMET03250
0.3640.0750.451Toll-Like receptor 7 agonist

0.398 0.061 DBMET03249

0.364 0.075 DBMET03250

0.451 0.043 DBMET03251

DBMET03251
0.3640.0750.448Toll-Like receptor agonist

0.397 0.061 DBMET03249

0.363 0.076 DBMET03250

0.448 0.044 DBMET03251

DBMET03251
0.3270.0420.327Potassium channel (Voltage-sensitive) blocker

0.254 0.065 DBMET03249

0.313 0.045 DBMET03250

0.262 0.062 DBMET03251

0.3060.0440.306Potassium channel blocker

0.257 0.063 DBMET03249

0.285 0.052 DBMET03250

0.234 0.074 DBMET03251

0.2790.0170.375Phosphodiesterase inhibitor

0.338 0.011 DBMET03249

0.271 0.019 DBMET03250

0.375 0.008 DBMET03251

DBMET03251
0.2660.0120.266Toll-Like receptor antagonist

0.121 0.082 DBMET03249

0.237 0.019 DBMET03250

0.2550.0050.256Hepatocyte growth factor antagonist

0.239 0.006 DBMET03249

0.256 0.005 DBMET03250

0.215 0.009 DBMET03251

DBMET03250
0.2530.0050.375Phosphodiesterase 4B inhibitor

0.375 0.004 DBMET03249

0.29 0.005 DBMET03250

0.07 0.044 DBMET03251

DBMET03249
0.2090.010.225Phosphodiesterase 4D inhibitor

0.225 0.009 DBMET03249

0.213 0.01 DBMET03250

0.146 0.02 DBMET03251

DBMET03249
0.1810.0130.22Interleukin-1 receptor-associated protein kinase 4 inhibitor

0.186 0.012 DBMET03249

0.22 0.007 DBMET03250

0.099 0.046 DBMET03251

DBMET03250
0.1930.0320.276Sodium channel (voltage-gated) blocker

0.198 0.03 DBMET03249

0.213 0.025 DBMET03250

0.276 0.011 DBMET03251

DBMET03251
0.2240.0680.284Anticonvulsant

0.284 0.045 DBMET03249

0.177 0.101 DBMET03250

DBMET03249
0.1890.0360.255Sodium channel blocker

0.177 0.042 DBMET03249

0.194 0.035 DBMET03250

0.255 0.017 DBMET03251

DBMET03251
0.1870.0510.187Growth factor antagonist

0.139 0.077 DBMET03249

0.168 0.059 DBMET03250

0.148 0.07 DBMET03251

0.2410.1160.271Nootropic

0.271 0.091 DBMET03249

0.211 0.144 DBMET03250

0.226 0.129 DBMET03251

DBMET03249
0.1360.0110.166Phosphodiesterase 4A inhibitor

0.166 0.009 DBMET03249

0.137 0.011 DBMET03250

0.089 0.018 DBMET03251

DBMET03249
0.1950.0750.228I kappa B kinase epsilon inhibitor

0.228 0.05 DBMET03250

DBMET03250
0.1310.0220.131Phosphodiesterase I inhibitor

0.109 0.035 DBMET03249

0.09 0.058 DBMET03250

0.1160.0070.116Phosphodiesterase 1A inhibitor

0.112 0.008 DBMET03249

0.073 0.021 DBMET03250

0.1760.0680.176Antipruritic

0.165 0.079 DBMET03249

0.133 0.118 DBMET03250

0.151 0.093 DBMET03251

0.160.0570.16Toll-Like receptor 9 antagonist

0.106 0.103 DBMET03250

0.160.0570.187Hemostatic

0.143 0.077 DBMET03249

0.187 0.038 DBMET03250

0.149 0.07 DBMET03251

DBMET03250
0.1080.0110.108Melanin-concentrating hormone receptor 1 antagonist

0.05 0.04 DBMET03249

0.074 0.022 DBMET03250

0.1010.0090.103Proto-oncogene tyrosine-protein kinase Met inhibitor

0.092 0.012 DBMET03249

0.103 0.009 DBMET03250

0.07 0.021 DBMET03251

DBMET03250
0.10.0090.109Toll-Like receptor 8 antagonist

0.052 0.038 DBMET03249

0.109 0.007 DBMET03250

DBMET03250
0.1120.0220.124Phosphodiesterase 5A inhibitor

0.124 0.017 DBMET03249

0.099 0.027 DBMET03250

0.113 0.021 DBMET03251

DBMET03249
0.1230.0360.123Uric acid excretion stimulant

0.098 0.055 DBMET03249

0.119 0.039 DBMET03250

0.091 0.064 DBMET03251

0.110.0230.121Phosphodiesterase V inhibitor

0.121 0.018 DBMET03249

0.098 0.028 DBMET03250

0.111 0.023 DBMET03251

DBMET03249
0.090.0070.094Guanylate cyclase stimulant

0.087 0.008 DBMET03249

0.094 0.007 DBMET03250

0.069 0.011 DBMET03251

DBMET03250
0.2110.1350.241Ca2+/calmodulin-dependent kinase IV inhibitor

0.241 0.078 DBMET03250

DBMET03250
0.120.0450.299Bronchodilator

0.126 0.041 DBMET03249

0.118 0.046 DBMET03250

0.299 0.009 DBMET03251

DBMET03251
0.0980.0240.118Nav1.7 sodium channel blocker

0.089 0.028 DBMET03249

0.118 0.017 DBMET03250

0.114 0.018 DBMET03251

DBMET03250
0.0850.020.085Phosphodiesterase 1B inhibitor

0.076 0.025 DBMET03249

0.0910.0280.094Toll-Like receptor 7 antagonist

0.058 0.057 DBMET03249

0.094 0.025 DBMET03250

DBMET03250
0.0710.0130.071Glutamate (mGluR5) agonist

0.065 0.015 DBMET03249

0.046 0.031 DBMET03250

0.0710.0160.071Glutamate (mGluR group I) agonist

0.066 0.018 DBMET03249

0.051 0.03 DBMET03250

0.0860.030.137Phosphodiesterase III inhibitor

0.129 0.013 DBMET03249

0.086 0.03 DBMET03250

0.137 0.012 DBMET03251

DBMET03251
0.0960.040.109Glutamate receptor agonist

0.109 0.031 DBMET03249

DBMET03249
0.1350.080.167Vascular endothelial growth factor 3 antagonist

0.167 0.056 DBMET03250

DBMET03250
0.2440.1880.458Analgesic

0.246 0.186 DBMET03249

0.458 0.062 DBMET03251

DBMET03251
0.0930.0390.158Phosphodiesterase 3A inhibitor

0.158 0.014 DBMET03249

0.086 0.048 DBMET03250

DBMET03249
0.0870.0330.087Amidase inhibitor

0.068 0.052 DBMET03249

0.0830.030.085Orexin receptor 1 antagonist

0.085 0.027 DBMET03249

0.074 0.044 DBMET03250

DBMET03249
0.0620.0140.062Acetyl-CoA carboxylase inhibitor

0.061 0.014 DBMET03249

0.061 0.014 DBMET03250

0.04 0.03 DBMET03251

0.0580.010.058Phosphodiesterase 6C inhibitor

0.056 0.012 DBMET03249

0.052 0.017 DBMET03250

0.049 0.023 DBMET03251

0.0670.020.067Histamine H3 receptor antagonist

0.053 0.025 DBMET03250

0.10.0550.1Antihistaminic

0.091 0.063 DBMET03251

0.1350.090.247Cholinergic

0.118 0.11 DBMET03249

0.247 0.029 DBMET03251

DBMET03251
0.1080.0630.122Granulocyte macrophage colony stimulating factor antagonist

0.099 0.072 DBMET03250

0.122 0.052 DBMET03251

DBMET03251
0.070.0270.079Phosphodiesterase 4C inhibitor

0.079 0.022 DBMET03249

0.07 0.026 DBMET03250

DBMET03249
0.0770.0370.077Cannabinoid receptor agonist
0.0930.0530.093Histamine antagonist

0.084 0.06 DBMET03251

0.0680.0330.068Phosphodiesterase 1C inhibitor

0.067 0.033 DBMET03249

0.2740.240.274Antiinflammatory

0.263 0.253 DBMET03250

0.0720.0380.073Orexin receptor antagonist

0.073 0.036 DBMET03249

0.06 0.058 DBMET03250

DBMET03249
0.0490.0170.049Glutamate (mGluR group II) antagonist

0.042 0.022 DBMET03249

0.04 0.025 DBMET03250

0.0410.0110.041Glutamate (mGluR2) antagonist

0.035 0.015 DBMET03249

0.032 0.017 DBMET03250

0.040.0120.04Phosphodiesterase 6B inhibitor

0.036 0.015 DBMET03249

0.031 0.021 DBMET03250

0.0820.0550.099Acetylcholine nicotinic agonist

0.099 0.038 DBMET03250

DBMET03250
0.0750.0490.075Phosphodiesterase VI inhibitor
0.0430.0180.045Orexin receptor 2 antagonist

0.045 0.016 DBMET03249

0.033 0.029 DBMET03250

DBMET03249
0.1080.0840.114Protein kinase (CK1) delta inhibitor

0.114 0.078 DBMET03250

DBMET03250
0.0370.0130.045Nicotinic alpha3beta4 receptor agonist

0.045 0.008 DBMET03250

DBMET03250
0.1640.140.323Tumour necrosis factor alpha release inhibitor

0.174 0.131 DBMET03250

0.323 0.045 DBMET03251

DBMET03251
0.1190.0970.119Nav1.6 sodium channel blocker
0.0590.0390.059Fibroblast growth factor 4 antagonist
0.030.0120.03Acetyl-CoA carboxylase 2 inhibitor

0.028 0.012 DBMET03249

0.03 0.012 DBMET03250

0.0260.0090.026Guanylate cyclase 1 stimulant

0.024 0.009 DBMET03249

0.026 0.009 DBMET03250

0.019 0.014 DBMET03251

0.0270.0110.027Phosphodiesterase 6G inhibitor

0.025 0.014 DBMET03249

0.022 0.019 DBMET03250

0.0270.0110.027Phosphodiesterase 6H inhibitor

0.025 0.014 DBMET03249

0.022 0.019 DBMET03250

0.1630.1470.163ErbB-1 antagonist
0.0490.0340.058Nicotinic receptor alpha4 subunit antagonist

0.049 0.034 DBMET03249

0.058 0.023 DBMET03250

DBMET03250
0.0570.0420.057Adenosine A1 receptor antagonist
0.0360.0220.036Glucose-dependent insulinotropic receptor agonist
0.0610.0480.061Adenosine A2 receptor antagonist
0.0320.020.032Prostaglandin D2 agonist

0.032 0.019 DBMET03249

0.032 0.019 DBMET03250

0.1190.1090.119Tyrosine kinase inhibitor
0.0240.0150.024Phosphodiesterase 6A inhibitor

0.022 0.02 DBMET03249

0.0570.0480.057Adenosine A2a receptor antagonist
0.0610.0530.0615 Hydroxytryptamine 3A antagonist
0.0410.0350.0895 Hydroxytryptamine 2C agonist

0.089 0.009 DBMET03250

DBMET03250
0.0290.0250.029Potassium channel (Inward rectifier) 1 blocker
0.050.0460.066Nicotinic neuronal receptor agonist

0.066 0.031 DBMET03250

DBMET03250
0.1980.1950.198Ca(v)3.3 blocker
0.0790.0760.089Interleukin 5 antagonist

0.078 0.077 DBMET03249

0.089 0.056 DBMET03250

DBMET03250
0.0330.0320.033G protein-coupled receptor agonist
0.0390.0380.067Phosphodiesterase 3B inhibitor

0.067 0.017 DBMET03249

DBMET03249
0.0650.0660.069Protein kinase B beta inhibitor

0.069 0.058 DBMET03250

DBMET03250
0.0640.0680.11MAP-kinase-activated kinase 2 inhibitor

0.11 0.024 DBMET03250

DBMET03250
0.0710.0760.118MAP-kinase-activated kinase inhibitor

0.118 0.027 DBMET03250

DBMET03250
0.0990.1130.126Cytokine production inhibitor

0.126 0.083 DBMET03250

DBMET03250
0.0970.1110.176Acetylcholinesterase inhibitor

0.176 0.042 DBMET03251

DBMET03251
0.0460.0620.054Glutamate (mGluR) agonist

0.054 0.051 DBMET03249

DBMET03249
0.0950.1210.104Sphingosine 1-phosphate receptor 2 agonist

0.104 0.089 DBMET03250

DBMET03250
0.0530.0790.063Protein kinase B alpha inhibitor

0.063 0.057 DBMET03250

DBMET03250
0.0430.0780.0785 Hydroxytryptamine agonist

0.078 0.043 DBMET03250

DBMET03250
0.0650.1030.086Protein kinase C delta inhibitor

0.086 0.068 DBMET03251

DBMET03251
0.0750.1170.111GABA receptor agonist

0.111 0.065 DBMET03251

DBMET03251
0.1360.1780.176Vasodilator

0.176 0.126 DBMET03249

DBMET03249
0.0640.1080.123Check point kinase 2 inhibitor

0.123 0.047 DBMET03250

DBMET03250
0.1030.150.134CDC-like kinase 4 inhibitor

0.134 0.114 DBMET03250

DBMET03250
0.0710.1290.186MAO inhibitor

0.186 0.045 DBMET03251

DBMET03251
0.0420.1160.078Protein kinase (CaMK, MLCK, PhK, SNF, KIN, NIM1, MAPKAP, POLO, CHK, ULK, RSK-2nd domain) inhibitor

0.078 0.052 DBMET03250

DBMET03250
0.1280.2070.2Cardiotonic

0.2 0.119 DBMET03249

DBMET03249
0.0480.1330.08I kappa B kinase inhibitor

0.08 0.061 DBMET03250

DBMET03250
0.0550.1510.105Polo-like kinase-4 inhibitor

0.105 0.072 DBMET03249

DBMET03249
0.0340.1310.06Check point kinase 1 inhibitor

0.06 0.059 DBMET03250

DBMET03250
0.0220.1310.0445 Hydroxytryptamine 2B agonist

0.044 0.019 DBMET03250

DBMET03250
0.0390.1530.116MAO A inhibitor

0.116 0.055 DBMET03251

DBMET03251
0.0880.2040.194Polo-like kinase-3 inhibitor

0.194 0.048 DBMET03251

DBMET03251
0.0720.2160.137Dual specificity tyrosine-phosphorylation regulated kinase 3 inhibitor

0.137 0.132 DBMET03250

DBMET03250
0.0430.1980.088Ephrin antagonist

0.088 0.075 DBMET03251

DBMET03251
Ext Pa Pi Pmax Activity Other Results ID Pa_max