target_name chembl_id variant Number, propensity Number, indirect IAP, propensity IAP, indirect
1 1,25-dihydroxyvitamin D(3) 24-hydroxylase, mitochondrial CHEMBL4521 NA 55 27 0.9943 0.9987
2 1-acyl-sn-glycerol-3-phosphate acyltransferase beta CHEMBL4772 NA 17 11 0.982 1
3 1-phosphatidylinositol 3-phosphate 5-kinase CHEMBL1938222 NA 43 28 0.9921 0.9903
4 11-beta-hydroxysteroid dehydrogenase 1 CHEMBL4235 NA 2216 1323 0.9907 0.9972
5 11-beta-hydroxysteroid dehydrogenase type 2 CHEMBL3746 NA 145 32 0.9918 0.9991
6 15-hydroxyprostaglandin dehydrogenase [NAD(+)] CHEMBL1293255 NA 221 111 0.9984 1
7 17-beta-hydroxysteroid dehydrogenase 13 CHEMBL5305042 NA 38 24 1 1
8 17-beta-hydroxysteroid dehydrogenase 14 CHEMBL3712868 NA 46 43 1 1
9 17-beta-hydroxysteroid dehydrogenase type 1 CHEMBL3181 NA 501 379 0.9929 0.9976
10 17-beta-hydroxysteroid dehydrogenase type 2 CHEMBL2789 NA 475 341 0.9942 0.9991
11 17-beta-hydroxysteroid dehydrogenase type 3 CHEMBL4234 NA 175 112 0.9944 0.9998
12 2-acylglycerol O-acyltransferase 2 CHEMBL2439944 NA 90 19 0.9998 1
13 2-hydroxyacylsphingosine 1-beta-galactosyltransferase CHEMBL4739855 NA 21 21 1 1
14 26S proteasome CHEMBL2364701 NA 31 26 0.9998 0.9999
15 26S proteasome non-ATPase regulatory subunit 14 CHEMBL2007629 NA 33 11 0.9936 1
16 3',5'-cyclic-AMP phosphodiesterase 4A CHEMBL254 NA 292 34 0.9747 0.9795
17 3',5'-cyclic-AMP phosphodiesterase 4B CHEMBL275 S133D 1291 17 0.9883 1
18 3',5'-cyclic-AMP phosphodiesterase 4B CHEMBL275 NA 1291 187 0.9883 0.9827
19 3',5'-cyclic-AMP phosphodiesterase 4D CHEMBL288 NA 867 168 0.9751 0.9805
20 3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase CHEMBL4931 NA 64 42 0.9597 0.9649
21 3-hydroxy-3-methylglutaryl-coenzyme A reductase CHEMBL402 NA 97 26 0.9949 0.9984
22 3-oxo-5-alpha-steroid 4-dehydrogenase 1 CHEMBL1787 NA 68 38 0.9997 0.9997
23 3-oxo-5-alpha-steroid 4-dehydrogenase 2 CHEMBL1856 NA 160 54 0.9996 0.9994
24 3-phosphoinositide-dependent protein kinase 1 CHEMBL2534 NA 200 44 0.9739 0.9999
25 4-hydroxyphenylpyruvate dioxygenase CHEMBL1861 NA 111 63 0.9999 0.9999
26 5'-nucleotidase CHEMBL5957 NA 360 214 0.9811 0.9985
27 5-hydroxytryptamine receptor 1A CHEMBL214 NA 3638 2399 0.9815 0.9898
28 5-hydroxytryptamine receptor 1B CHEMBL1898 NA 534 281 0.9755 0.9928
29 5-hydroxytryptamine receptor 1D CHEMBL1983 NA 516 251 0.9804 0.9915
30 5-hydroxytryptamine receptor 1F CHEMBL1805 NA 42 18 0.997 0.9999
31 5-hydroxytryptamine receptor 2A CHEMBL224 NA 3335 1916 0.9789 0.9874
32 5-hydroxytryptamine receptor 2A/Metabotropic glutamate receptor 2 CHEMBL4630758 NA 11 11 1 1
33 5-hydroxytryptamine receptor 2B CHEMBL1833 NA 1140 640 0.9681 0.9821
34 5-hydroxytryptamine receptor 2C CHEMBL225 NA 2273 1380 0.9788 0.9852
35 5-hydroxytryptamine receptor 3A CHEMBL1899 NA 393 186 0.9769 0.9875
36 5-hydroxytryptamine receptor 4 CHEMBL1875 NA 499 392 0.9943 0.999
37 5-hydroxytryptamine receptor 5A CHEMBL3426 NA 186 35 0.9523 0.9704
38 5-hydroxytryptamine receptor 6 CHEMBL3371 NA 3356 2443 0.9905 0.996
39 5-hydroxytryptamine receptor 7 CHEMBL3155 NA 2238 1470 0.9845 0.9909
40 6-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 3 CHEMBL2331053 NA 108 37 0.9962 0.9973
41 72 kDa type IV collagenase CHEMBL333 NA 1515 51 0.9801 0.9686
42 A disintegrin and metalloproteinase with thrombospondin motifs 5 CHEMBL2285 NA 273 35 0.9958 0.9954
43 ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1 CHEMBL4660 NA 236 77 0.9996 1
44 ALK tyrosine kinase receptor CHEMBL4247 G1269A 1035 11 0.9875 0.8529
45 ALK tyrosine kinase receptor CHEMBL4247 F1174L 1035 13 0.9875 0.9136
46 ALK tyrosine kinase receptor CHEMBL4247 C1156Y 1035 22 0.9875 0.954
47 ALK tyrosine kinase receptor CHEMBL4247 G1202R 1035 36 0.9875 0.972
48 ALK tyrosine kinase receptor CHEMBL4247 L1196M 1035 156 0.9875 0.9934
49 ALK tyrosine kinase receptor CHEMBL4247 NA 1035 280 0.9875 0.9955
50 AMP-activated protein kinase (AMPK) alpha-1/beta-1/gamma-1 CHEMBL2111345 NA 74 57 0.9452 0.9373
51 AMPK alpha1/beta2/gamma1 CHEMBL3038453 NA 16 14 0.9867 0.9999
52 AMPK alpha2/beta1/gamma1 CHEMBL3038455 NA 76 42 0.9784 0.9673
53 AP2-associated protein kinase 1 CHEMBL3830 NA 278 146 0.9746 0.9863
54 ATP-binding cassette sub-family C member 9 CHEMBL1971 NA 51 27 0.9997 0.9998
55 ATP-dependent Clp protease proteolytic subunit, mitochondrial CHEMBL4523305 NA 132 58 0.9878 0.9927
56 ATP-dependent RNA helicase DDX3X CHEMBL5553 NA 108 24 0.9904 0.9999
57 ATP-dependent translocase ABCB1 CHEMBL4302 NA 1505 658 0.9675 0.9823
58 ATP-sensitive inward rectifier potassium channel 1 CHEMBL1293292 NA 252 218 0.9988 0.9985
59 ATPase family AAA domain-containing protein 2 CHEMBL2150837 NA 193 68 0.9801 0.9791
60 ATR/ATRIP CHEMBL4106138 NA 77 60 0.9957 0.9937
61 Acetyl-CoA carboxylase 1 CHEMBL3351 NA 287 99 0.9934 0.9933
62 Acetyl-CoA carboxylase 2 CHEMBL4829 NA 380 153 0.995 0.9977
63 Acetyl-coenzyme A synthetase, cytoplasmic CHEMBL4523467 NA 23 23 1 1
64 Acetylcholine receptor; alpha1/beta1/delta/gamma CHEMBL1907588 NA 49 26 0.9945 0.9893
65 Acetylcholinesterase CHEMBL220 NA 3626 320 0.9697 0.9945
66 Acid ceramidase CHEMBL5463 NA 151 99 0.9964 0.9963
67 Acid-sensing ion channel 3 CHEMBL5368 NA 24 11 0.995 0.9974
68 Acidic mammalian chitinase CHEMBL1293197 NA 119 77 0.977 1
69 Activated CDC42 kinase 1 CHEMBL4599 NA 225 92 0.9772 0.9887
70 Activin receptor type-1 CHEMBL5903 R206H 322 22 0.9869 0.9909
71 Activin receptor type-1 CHEMBL5903 NA 322 100 0.9869 0.9958
72 Acyl-CoA (8-3)-desaturase CHEMBL5840 NA 45 43 0.9806 0.9918
73 Adenosine kinase CHEMBL3589 NA 195 11 0.9965 0.9651
74 Adenosine receptor A1 CHEMBL226 NA 3887 2528 0.9852 0.9887
75 Adenosine receptor A2a CHEMBL251 NA 4465 3010 0.9853 0.9924
76 Adenosine receptor A2b CHEMBL255 NA 2147 1567 0.993 0.994
77 Adenosine receptor A3 CHEMBL256 NA 3478 2577 0.9886 0.994
78 Adenosylhomocysteinase CHEMBL2664 NA 121 21 0.9932 0.9999
79 Adenylate cyclase type 1 CHEMBL2899 NA 101 52 0.9909 0.9991
80 Adenylate cyclase type 2 CHEMBL3760 NA 40 15 0.968 1
81 Adenylate cyclase type 8 CHEMBL2960 NA 63 31 0.9831 0.9691
82 Alanine--glyoxylate aminotransferase CHEMBL5169121 NA 21 15 0.9997 0.9999
83 Aldehyde dehydrogenase 1A1 CHEMBL3577 NA 288 50 0.9898 0.999
84 Aldo-keto reductase family 1 member A1 CHEMBL2246 NA 68 23 0.999 0.9894
85 Aldo-keto reductase family 1 member B1 CHEMBL1900 NA 399 113 0.9887 0.9974
86 Aldo-keto reductase family 1 member B10 CHEMBL5983 NA 96 36 0.9956 0.9972
87 Aldo-keto reductase family 1 member C1 CHEMBL5905 NA 103 16 0.959 0.9882
88 Aldo-keto reductase family 1 member C2 CHEMBL5847 NA 222 47 0.9853 0.9907
89 Aldo-keto reductase family 1 member C3 CHEMBL4681 NA 556 235 0.9745 0.99
90 Alkaline phosphatase, tissue-nonspecific isozyme CHEMBL5979 NA 133 17 0.9954 0.9995
91 Alpha-1,6-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase CHEMBL2321630 NA 124 75 0.9946 0.9999
92 Alpha-1A adrenergic receptor CHEMBL229 NA 947 569 0.9784 0.9874
93 Alpha-1B adrenergic receptor CHEMBL232 NA 617 377 0.981 0.988
94 Alpha-1D adrenergic receptor CHEMBL223 NA 576 391 0.9873 0.9925
95 Alpha-2A adrenergic receptor CHEMBL1867 NA 549 276 0.9729 0.9899
96 Alpha-2B adrenergic receptor CHEMBL1942 NA 277 125 0.9611 0.9752
97 Alpha-2C adrenergic receptor CHEMBL1916 NA 335 150 0.9714 0.9848
98 Alpha-ketoglutarate-dependent dioxygenase FTO CHEMBL2331065 NA 167 39 0.9702 0.9927
99 Alpha-synuclein CHEMBL6152 NA 208 43 0.9617 0.9653
100 Amine oxidase [copper-containing] 3 CHEMBL3437 NA 185 114 0.9993 0.9994
101 Amine oxidase [flavin-containing] A CHEMBL1951 NA 2033 396 0.9758 0.9929
102 Amine oxidase [flavin-containing] B CHEMBL2039 NA 3526 740 0.9741 0.9939
103 Aminopeptidase N CHEMBL1907 NA 265 70 0.9884 0.9968
104 Amyloid-beta precursor protein CHEMBL2487 NA 1242 383 0.9724 0.9913
105 Androgen receptor CHEMBL1871 F877L 1776 45 0.9893 0.9905
106 Androgen receptor CHEMBL1871 T878A 1776 60 0.9893 0.996
107 Androgen receptor CHEMBL1871 NA 1776 1016 0.9893 0.9924
108 Angiopoietin-1 receptor CHEMBL4128 NA 466 84 0.972 0.9681
109 Angiotensin-converting enzyme CHEMBL1808 NA 126 11 0.987 0.9925
110 Annexin A2/S100-A10 CHEMBL2111435 NA 29 11 1 1
111 Anoctamin-1 CHEMBL2046267 NA 113 31 0.9992 0.9932
112 Apelin receptor CHEMBL1628481 NA 292 251 0.9973 0.9989
113 Apoptosis regulator BAX CHEMBL5318 NA 37 12 0.9667 1
114 Apoptosis regulator Bcl-2 CHEMBL4860 NA 816 92 0.9862 0.9852
115 Arachidonate 5-lipoxygenase-activating protein CHEMBL4550 NA 369 258 0.9955 0.9997
116 Arginase-1 CHEMBL1075097 NA 217 98 0.997 1
117 Arginase-2, mitochondrial CHEMBL1795148 NA 67 22 1 1
118 Aromatase CHEMBL1978 NA 2198 694 0.99 0.9962
119 Aryl hydrocarbon receptor CHEMBL3201 NA 132 76 0.9757 0.9785
120 Aryl hydrocarbon receptor nuclear translocator/Endothelial PAS domain-containing protein 1 CHEMBL3885518 NA 51 29 1 1
121 Aspartyl/asparaginyl beta-hydroxylase CHEMBL4680030 NA 35 19 0.8847 0.9203
122 Atrial natriuretic peptide receptor 1 CHEMBL1988 NA 50 29 0.9977 0.9941
123 Atypical chemokine receptor 3 CHEMBL2010631 NA 313 148 0.9869 0.9901
124 Aurora kinase A CHEMBL4722 NA 1103 296 0.9689 0.9813
125 Aurora kinase A/Targeting protein for Xklp2 CHEMBL3883304 NA 18 10 0.9971 0.9992
126 Aurora kinase B CHEMBL2185 NA 984 286 0.9735 0.9745
127 Aurora kinase B/Inner centromere protein CHEMBL3430907 NA 99 48 0.9842 0.9538
128 Autotaxin CHEMBL3691 NA 724 183 0.9827 0.989
129 B-cell lymphoma 6 protein CHEMBL4105786 C8Q,C67R,C84N 235 31 0.9918 1
130 B-cell lymphoma 6 protein CHEMBL4105786 NA 235 103 0.9918 1
131 B1 bradykinin receptor CHEMBL4308 NA 483 310 0.9988 0.9979
132 B2 bradykinin receptor CHEMBL3157 NA 144 111 0.9951 0.9999
133 BCL-6/NCOR2 CHEMBL4523673 NA 32 19 0.9999 0.9999
134 BCL2/BCL2L11 CHEMBL5169264 NA 31 28 0.9999 0.9999
135 BCL2A1/BID CHEMBL5169268 NA 37 28 0.9509 0.9972
136 BDNF/NT-3 growth factors receptor CHEMBL4898 NA 433 127 0.9696 0.9572
137 BMP-2-inducible protein kinase CHEMBL4522 NA 58 20 0.9342 0.9684
138 Baculoviral IAP repeat-containing protein 2 CHEMBL5462 NA 237 97 0.9995 0.9994
139 Baculoviral IAP repeat-containing protein 3 CHEMBL5335 NA 90 27 0.9993 0.9993
140 Baculoviral IAP repeat-containing protein 7 CHEMBL1075127 NA 13 11 0.9997 0.9996
141 Bcl-2-like protein 1 CHEMBL4625 NA 526 58 0.9907 0.9983
142 Bcl-2-related protein A1 CHEMBL6044 NA 93 15 0.9677 0.9795
143 Bcl-xL/BAK CHEMBL3137283 NA 29 14 0.9852 0.992
144 Bcl-xL/Bcl-2-like protein 11 CHEMBL3883287 NA 36 21 0.9963 0.9975
145 Bcl2-associated agonist of cell death CHEMBL3817 NA 49 14 0.9687 1
146 Bcr/Abl fusion protein CHEMBL2096618 T315I 431 61 0.9887 0.9812
147 Bcr/Abl fusion protein CHEMBL2096618 NA 431 231 0.9887 0.9874
148 Beta-1 adrenergic receptor CHEMBL213 NA 857 628 0.9897 0.9965
149 Beta-2 adrenergic receptor CHEMBL210 NA 1087 760 0.9887 0.9968
150 Beta-3 adrenergic receptor CHEMBL246 NA 826 707 0.9932 0.9978
151 Beta-adrenergic receptor kinase 1 CHEMBL4079 S670A 224 16 0.9783 0.9996
152 Beta-adrenergic receptor kinase 1 CHEMBL4079 NA 224 76 0.9783 0.9862
153 Beta-secretase 1 CHEMBL4822 NA 2980 1389 0.9818 0.9987
154 Beta-secretase 2 CHEMBL2525 NA 276 14 0.9949 0.9721
155 Bifunctional epoxide hydrolase 2 CHEMBL2409 NA 2058 365 0.987 0.992
156 Bifunctional purine biosynthesis protein ATIC CHEMBL2518 NA 64 21 0.9918 0.9998
157 Bile acid receptor CHEMBL2047 NA 1378 630 0.987 0.9966
158 Bile salt export pump CHEMBL6020 NA 30 13 0.6726 0.8413
159 Bombesin receptor subtype-3 CHEMBL4080 NA 165 139 0.9985 0.9992
160 Bone morphogenetic protein 1 CHEMBL3898 NA 99 94 0.9999 1
161 Bone morphogenetic protein receptor type-2 CHEMBL5467 NA 43 19 0.9667 1
162 Branched-chain-amino-acid aminotransferase, cytosolic CHEMBL4679 NA 70 30 0.9842 0.9929
163 Branched-chain-amino-acid aminotransferase, mitochondrial CHEMBL3616354 NA 120 33 0.9937 1
164 Broad substrate specificity ATP-binding cassette transporter ABCG2 CHEMBL5393 NA 1017 562 0.9542 0.9891
165 Bromodomain adjacent to zinc finger domain protein 2B CHEMBL1741220 NA 77 26 0.9723 0.9767
166 Bromodomain testis-specific protein CHEMBL1795185 NA 148 34 0.9516 0.9198
167 Bromodomain-containing protein 1 CHEMBL2176774 NA 82 42 0.9764 0.9946
168 Bromodomain-containing protein 2 CHEMBL1293289 NA 276 58 0.9713 0.9244
169 Bromodomain-containing protein 3 CHEMBL1795186 NA 262 50 0.9771 0.9161
170 Bromodomain-containing protein 4 CHEMBL1163125 Y97A 3824 25 0.9819 0.9997
171 Bromodomain-containing protein 4 CHEMBL1163125 Y390A 3824 115 0.9819 0.9997
172 Bromodomain-containing protein 4 CHEMBL1163125 NA 3824 988 0.9819 0.9892
173 Bromodomain-containing protein 7 CHEMBL3085622 NA 46 17 0.9565 0.9998
174 Bromodomain-containing protein 9 CHEMBL3108640 NA 225 56 0.991 0.9831
175 Butyrophilin subfamily 3 member A1 CHEMBL4105758 NA 51 36 1 0.9999
176 C-C chemokine receptor type 1 CHEMBL2413 NA 409 298 0.9938 0.9988
177 C-C chemokine receptor type 10 CHEMBL2321628 NA 33 26 1 1
178 C-C chemokine receptor type 2 CHEMBL4015 I40L 1391 25 0.9953 1
179 C-C chemokine receptor type 2 CHEMBL4015 NA 1391 840 0.9953 0.9956
180 C-C chemokine receptor type 3 CHEMBL3473 NA 657 499 0.9936 0.9968
181 C-C chemokine receptor type 4 CHEMBL2414 NA 347 251 0.9915 0.9989
182 C-C chemokine receptor type 5 CHEMBL274 NA 1089 771 0.9891 0.9956
183 C-C chemokine receptor type 6 CHEMBL4423 NA 75 58 0.9902 0.9923
184 C-C chemokine receptor type 8 CHEMBL4596 NA 141 112 0.9974 0.9995
185 C-C chemokine receptor type 9 CHEMBL5815 NA 120 70 0.9938 0.9921
186 C-C motif chemokine 2 CHEMBL1649052 NA 47 37 0.9441 0.9612
187 C-X-C chemokine receptor type 1 CHEMBL4029 NA 152 53 0.976 0.9915
188 C-X-C chemokine receptor type 2 CHEMBL2434 NA 711 451 0.9973 0.999
189 C-X-C chemokine receptor type 3 CHEMBL4441 NA 832 610 0.9957 0.998
190 C-X-C chemokine receptor type 4 CHEMBL2107 NA 531 397 0.9865 0.9916
191 C-X-C chemokine receptor type 6 CHEMBL5994 NA 49 28 0.9877 1
192 C3a anaphylatoxin chemotactic receptor CHEMBL4761 NA 152 88 0.9999 0.9999
193 C5a anaphylatoxin chemotactic receptor 1 CHEMBL2373 NA 265 185 0.9953 0.9941
194 CDC7/DBF4 (Cell division cycle 7-related protein kinase/Activator of S phase kinase) CHEMBL2111377 NA 230 190 0.9963 0.996
195 CDGSH iron-sulfur domain-containing protein 1 CHEMBL1795168 NA 73 34 0.9293 0.9737
196 CDGSH iron-sulfur domain-containing protein 2 CHEMBL4523399 NA 35 21 0.9997 1
197 CDK1/Cyclin A CHEMBL3038467 NA 60 39 0.9764 0.9487
198 CDK12/Cyclin K CHEMBL4106169 NA 150 137 0.9631 0.9631
199 CDK2/Cyclin A1 CHEMBL3038470 NA 121 91 0.9819 0.9749
200 CDK2/Cyclin A2 CHEMBL3038469 NA 835 536 0.9829 0.9836
201 CDK3/Cyclin E CHEMBL3038471 NA 30 16 0.8822 0.8191
202 CDK4/Cyclin D3 CHEMBL3038472 NA 143 132 0.9772 0.9799
203 CDK6/cyclin D1 CHEMBL2111455 NA 161 138 0.9867 0.9881
204 CDK6/cyclin D3 CHEMBL2111448 NA 252 219 0.9838 0.983
205 CDK7/Cyclin H/MNAT1 CHEMBL3038473 NA 226 172 0.9666 0.9641
206 CDK8/Cyclin C CHEMBL3038474 NA 500 465 0.9821 0.9845
207 CDK9/Cyclin K CHEMBL3038475 NA 66 44 0.9765 0.9453
208 CDK9/cyclin T1 CHEMBL2111389 NA 951 746 0.9832 0.9859
209 CREB-binding protein CHEMBL5747 NA 491 102 0.9751 0.9848
210 CRY2/PER2 CHEMBL4296116 NA 55 42 1 1
211 CX3C chemokine receptor 1 CHEMBL4843 NA 48 43 0.981 1
212 Calcitonin gene-related peptide 1 CHEMBL5293 NA 65 49 0.9898 0.985
213 Calcitonin gene-related peptide 2 CHEMBL3713541 NA 24 23 1 1
214 Calcitonin gene-related peptide type 1 receptor CHEMBL3798 NA 542 402 0.9982 0.9994
215 Calcitonin-gene-related peptide receptor, CALCRL/RAMP1 CHEMBL2107838 NA 73 67 0.9896 0.9868
216 Calcium/calmodulin-dependent protein kinase kinase 2 CHEMBL5284 NA 107 23 0.9584 0.9751
217 Calcium/calmodulin-dependent protein kinase type 1D CHEMBL5073 NA 27 13 0.9027 1
218 Calcium/calmodulin-dependent protein kinase type II subunit delta CHEMBL2801 NA 57 34 0.9638 0.9992
219 Calpain 1 CHEMBL2111357 NA 16 16 0.9999 0.9999
220 Calpain-1 catalytic subunit CHEMBL3891 NA 246 66 0.993 0.9908
221 Cannabinoid receptor 1 CHEMBL218 NA 3682 2340 0.986 0.9909
222 Cannabinoid receptor 2 CHEMBL253 Q63R 4237 11 0.9897 0.9997
223 Cannabinoid receptor 2 CHEMBL253 NA 4237 2667 0.9897 0.9918
224 Carbonic anhydrase 1 CHEMBL261 NA 5499 328 0.9908 0.9996
225 Carbonic anhydrase 12 CHEMBL3242 NA 4419 304 0.9905 0.9996
226 Carbonic anhydrase 13 CHEMBL3912 NA 364 114 0.9914 0.9999
227 Carbonic anhydrase 14 CHEMBL3510 NA 654 113 0.9902 0.9991
228 Carbonic anhydrase 2 CHEMBL205 N67I 6038 10 0.9903 0.9977
229 Carbonic anhydrase 2 CHEMBL205 NA 6038 380 0.9903 0.9993
230 Carbonic anhydrase 3 CHEMBL2885 NA 180 51 0.9769 0.9998
231 Carbonic anhydrase 4 CHEMBL3729 NA 1319 160 0.9918 0.9956
232 Carbonic anhydrase 5A, mitochondrial CHEMBL4789 NA 570 99 0.9855 0.9997
233 Carbonic anhydrase 5B, mitochondrial CHEMBL3969 NA 490 147 0.9908 0.9999
234 Carbonic anhydrase 6 CHEMBL3025 NA 371 112 0.9861 0.9999
235 Carbonic anhydrase 7 CHEMBL2326 NA 1414 132 0.9931 0.9991
236 Carbonic anhydrase 9 CHEMBL3594 NA 5410 364 0.9903 0.9993
237 Carbonic anhydrase-related protein 11 CHEMBL2420 NA 14 14 0.9994 0.9998
238 Carboxypeptidase B2 CHEMBL3419 NA 185 28 0.9999 0.9995
239 Casein kinase I isoform delta CHEMBL2828 NA 296 75 0.9779 0.9999
240 Casein kinase I isoform epsilon CHEMBL4937 NA 203 65 0.9483 0.962
241 Casein kinase II alpha'/ beta CHEMBL3883328 NA 83 58 0.9999 0.9999
242 Casein kinase II alpha/beta CHEMBL3038477 NA 80 70 0.9826 0.9916
243 Casein kinase II subunit alpha CHEMBL3629 NA 328 109 0.9723 0.995
244 Casein kinase II subunit alpha' CHEMBL4070 NA 158 98 0.9724 0.998
245 Caspase-1 CHEMBL4801 NA 364 70 0.9928 0.9882
246 Caspase-3 CHEMBL2334 NA 713 164 0.9936 0.9973
247 Caspase-4 CHEMBL2226 NA 21 13 0.9759 0.9233
248 Caspase-5 CHEMBL3131 NA 22 16 0.9094 0.9377
249 Caspase-7 CHEMBL3468 NA 317 43 0.9982 1
250 Caspase-8 CHEMBL3776 NA 135 15 0.9895 0.9999
251 Catechol O-methyltransferase CHEMBL2023 NA 131 73 0.9954 0.9992
252 Catenin beta-1 CHEMBL5866 NA 98 27 0.9549 0.9648
253 Cathepsin B CHEMBL4072 NA 915 93 0.9817 0.9995
254 Cathepsin D CHEMBL2581 NA 763 143 0.9901 0.9865
255 Cathepsin K CHEMBL268 NA 1239 72 0.9922 0.9994
256 Cathepsin L2 CHEMBL3272 NA 91 21 0.9897 0.9997
257 Cathepsin S CHEMBL2954 NA 1358 274 0.9969 0.9982
258 Cell division cycle 7-related protein kinase CHEMBL5443 NA 189 45 0.9932 0.9812
259 Cellular tumor antigen p53 CHEMBL4096 NA 45 11 0.9346 0.9226
260 Ceramide glucosyltransferase CHEMBL2063 NA 152 67 0.9981 0.9951
261 Cereblon/Casein kinase I alpha CHEMBL4296102 NA 10 10 1 1
262 Chemerin-like receptor 1 CHEMBL3540 NA 108 74 0.9951 0.9996
263 Chitinase-3-like protein 1 CHEMBL5724768 NA 26 20 0.9993 1
264 Chitotriosidase-1 CHEMBL3080 NA 118 59 0.9953 0.9912
265 Chloride anion exchanger CHEMBL4523223 NA 20 20 1 1
266 Cholecystokinin receptor type A CHEMBL1901 NA 237 151 0.9901 0.995
267 Cholesterol 24-hydroxylase CHEMBL4523510 NA 59 45 0.9994 0.9997
268 Cholesteryl ester transfer protein CHEMBL3572 NA 614 51 0.9985 0.999
269 Cholinesterase CHEMBL1914 NA 2654 179 0.9771 0.9944
270 Chromatin remodeling regulator CECR2 CHEMBL3108639 NA 128 26 0.9885 0.9891
271 Chromobox protein homolog 7 CHEMBL1764946 NA 79 39 0.9934 0.9995
272 Chromodomain Y-like protein CHEMBL3879827 NA 58 22 0.9771 0.9923
273 Chromodomain Y-like protein 2 CHEMBL3879857 NA 79 40 0.9994 0.9968
274 Coagulation factor VII/tissue factor CHEMBL2095194 NA 263 206 0.9949 0.9984
275 Coagulation factor X CHEMBL244 NA 2612 43 0.9942 0.9979
276 Coagulation factor XI CHEMBL2820 NA 704 13 0.9952 0.9237
277 Cocaine esterase CHEMBL3180 NA 229 38 0.9769 0.9969
278 Coiled-coil domain-containing protein 6/Tyrosine-protein kinase receptor RET CHEMBL3430904 NA 23 23 0.9166 0.9101
279 Collagenase 3 CHEMBL280 NA 1309 110 0.986 0.9865
280 Complement factor D CHEMBL2176771 NA 112 25 0.9889 1
281 Cone cGMP-specific 3',5'-cyclic phosphodiesterase subunit alpha' CHEMBL3977 NA 26 16 0.9414 0.9389
282 Corticotropin-releasing factor receptor 1 CHEMBL1800 NA 880 684 0.9999 1
283 Cyclic AMP-dependent transcription factor ATF-4 CHEMBL6067624 NA 39 38 1 1
284 Cyclic GMP-AMP synthase CHEMBL4105728 NA 113 31 0.9759 0.9657
285 Cyclin-C/Cyclin-dependent kinase 19 CHEMBL3883323 NA 102 98 0.9869 0.9886
286 Cyclin-G-associated kinase CHEMBL4355 NA 236 114 0.9641 0.9979
287 Cyclin-dependent kinase 1 CHEMBL308 NA 337 44 0.9653 0.9687
288 Cyclin-dependent kinase 1/cyclin B CHEMBL2094127 NA 121 69 0.9724 0.9504
289 Cyclin-dependent kinase 1/cyclin B1 CHEMBL1907602 NA 347 169 0.9647 0.9464
290 Cyclin-dependent kinase 11A CHEMBL5416 NA 37 17 0.9629 1
291 Cyclin-dependent kinase 13/Cyclin-K CHEMBL4296067 NA 36 31 0.9817 0.979
292 Cyclin-dependent kinase 14/Cyclin-Y CHEMBL4296115 NA 60 57 0.9799 0.9899
293 Cyclin-dependent kinase 2 CHEMBL301 NA 720 54 0.9509 0.9138
294 Cyclin-dependent kinase 2/cyclin A CHEMBL2094128 NA 284 149 0.9758 0.9748
295 Cyclin-dependent kinase 2/cyclin E CHEMBL2094126 NA 115 59 0.9809 0.9689
296 Cyclin-dependent kinase 2/cyclin E1 CHEMBL1907605 NA 796 505 0.9856 0.9824
297 Cyclin-dependent kinase 4 CHEMBL331 NA 217 20 0.9657 0.8928
298 Cyclin-dependent kinase 4/G1/S-specific cyclin-E1 CHEMBL3885554 NA 29 29 0.9995 0.9996
299 Cyclin-dependent kinase 4/cyclin D1 CHEMBL1907601 NA 478 324 0.9745 0.9757
300 Cyclin-dependent kinase 5/CDK5 activator 1 CHEMBL1907600 NA 879 552 0.9798 0.9812
301 Cyclin-dependent kinase 6 CHEMBL2508 NA 148 23 0.9741 1
302 Cyclin-dependent kinase 7 CHEMBL3055 NA 182 11 0.9662 0.823
303 Cyclin-dependent kinase 7/ cyclin H CHEMBL2111288 NA 145 99 0.9821 0.9737
304 Cyclin-dependent kinase 8 CHEMBL5719 NA 385 169 0.9828 0.9925
305 Cyclin-dependent kinase 9 CHEMBL3116 NA 374 91 0.9679 0.9827
306 Cyclin-dependent kinases regulatory subunit 1/S-phase kinase-associated protein 2 CHEMBL3885558 NA 48 24 0.9893 0.9812
307 Cysteinyl leukotriene receptor 1 CHEMBL1798 NA 200 174 0.9942 0.9977
308 Cysteinyl leukotriene receptor 2 CHEMBL4330 NA 81 59 0.9842 0.9999
309 Cystic fibrosis transmembrane conductance regulator CHEMBL4051 G551D 581 13 0.9839 0.9999
310 Cystic fibrosis transmembrane conductance regulator CHEMBL4051 N1303K 581 15 0.9839 0.9569
311 Cystic fibrosis transmembrane conductance regulator CHEMBL4051 NA 581 110 0.9839 0.9893
312 Cystic fibrosis transmembrane conductance regulator CHEMBL4051 F508del 581 216 0.9839 0.9953
313 Cystine/glutamate transporter CHEMBL1075149 NA 26 16 0.9987 1
314 Cytochrome P450 11B1, mitochondrial CHEMBL1908 NA 589 433 0.9989 0.9988
315 Cytochrome P450 11B2, mitochondrial CHEMBL2722 NA 774 727 0.9974 0.9974
316 Cytochrome P450 1A1 CHEMBL2231 NA 70 24 0.9861 0.9981
317 Cytochrome P450 1A2 CHEMBL3356 NA 49 22 0.9528 0.9815
318 Cytochrome P450 1B1 CHEMBL4878 NA 360 118 0.9888 0.9948
319 Cytochrome P450 26A1 CHEMBL5141 NA 132 77 0.9999 1
320 Cytochrome b-245 heavy chain CHEMBL1287627 NA 80 31 0.9539 0.902
321 Cytoplasmic tyrosine-protein kinase BMX CHEMBL3834 NA 205 81 0.9693 0.9846
322 Cytosolic phospholipase A2 CHEMBL3816 NA 201 33 0.9956 0.9695
323 D(1A) dopamine receptor CHEMBL2056 NA 848 460 0.9818 0.9912
324 D(1B) dopamine receptor CHEMBL1850 NA 272 98 0.9878 0.9921
325 D(2) dopamine receptor CHEMBL217 NA 4737 3089 0.985 0.9895
326 D(3) dopamine receptor CHEMBL234 V87F 3262 12 0.9861 0.9999
327 D(3) dopamine receptor CHEMBL234 NA 3262 2319 0.9861 0.9918
328 D(4) dopamine receptor CHEMBL219 NA 1707 1126 0.9847 0.9893
329 D-3-phosphoglycerate dehydrogenase CHEMBL2311243 NA 205 30 0.9905 0.9653
330 D-amino-acid oxidase CHEMBL5485 NA 243 111 0.9993 0.9998
331 DCN1-like protein 1 CHEMBL4105838 NA 229 62 0.9981 0.9752
332 DCN1-like protein 1/NEDD8-conjugating enzyme Ubc12 CHEMBL4523603 NA 106 68 0.9944 0.9926
333 DDB1- and CUL4-associated factor 1 CHEMBL5465521 NA 22 11 1 1
334 DNA (cytosine-5)-methyltransferase 1 CHEMBL1993 NA 193 21 0.9749 0.9199
335 DNA (cytosine-5)-methyltransferase 3B CHEMBL6095 NA 47 12 0.9336 0.9354
336 DNA excision repair protein ERCC-1/DNA repair endonuclease XPF CHEMBL3883316 NA 80 42 0.9991 0.9997
337 DNA polymerase theta CHEMBL6025 NA 116 41 0.9925 0.9999
338 DNA repair protein complementing XP-A cells CHEMBL4105801 NA 23 12 1 1
339 DNA topoisomerase 1 CHEMBL1781 NA 181 10 0.9751 1
340 DNA topoisomerase 2-alpha CHEMBL1806 NA 340 15 0.969 0.934
341 DNA-dependent protein kinase catalytic subunit CHEMBL3142 NA 602 82 0.9846 0.9894
342 DNA-directed RNA polymerase I subunit RPA1 CHEMBL3286067 NA 60 28 0.9947 1
343 Delta(24)-sterol reductase CHEMBL2331059 NA 13 11 0.9276 1
344 Delta-type opioid receptor CHEMBL236 NA 2213 1434 0.9877 0.9925
345 Deoxycytidine kinase CHEMBL2447 NA 99 87 0.9956 1
346 Deoxyhypusine synthase CHEMBL4415 NA 59 14 0.9933 0.9996
347 Deoxyuridine 5'-triphosphate nucleotidohydrolase, mitochondrial CHEMBL5203 NA 84 19 0.9884 1
348 Diacylglycerol O-acyltransferase 1 CHEMBL6009 NA 580 347 0.9967 0.9997
349 Diacylglycerol O-acyltransferase 2 CHEMBL5853 NA 67 54 0.9958 0.9939
350 Diacylglycerol lipase-alpha CHEMBL5545 NA 134 94 0.9993 0.9999
351 Dihydrofolate reductase CHEMBL202 NA 548 36 0.9934 0.9887
352 Dihydroorotate dehydrogenase (quinone), mitochondrial CHEMBL1966 NA 817 183 0.991 0.9907
353 Dipeptidyl peptidase 1 CHEMBL2252 NA 218 107 0.9955 0.9963
354 Dipeptidyl peptidase 2 CHEMBL3976 NA 314 44 0.9959 0.9998
355 Dipeptidyl peptidase 4 CHEMBL284 NA 2780 679 0.9892 0.9972
356 Dipeptidyl peptidase 8 CHEMBL4657 NA 580 61 0.9976 0.9998
357 Dipeptidyl peptidase 9 CHEMBL4793 NA 407 71 0.996 0.9998
358 Discoidin domain-containing receptor 2 CHEMBL5122 T654M 219 19 0.9738 0.9421
359 Discoidin domain-containing receptor 2 CHEMBL5122 NA 219 44 0.9738 0.9765
360 Disintegrin and metalloproteinase domain-containing protein 10 CHEMBL5028 NA 71 25 0.9932 1
361 Disintegrin and metalloproteinase domain-containing protein 17 CHEMBL3706 NA 828 274 0.9976 0.9999
362 Disintegrin and metalloproteinase domain-containing protein 8 CHEMBL5665 NA 17 14 1 1
363 Disks large homolog 4 CHEMBL5666 NA 24 12 1 1
364 Dual 3',5'-cyclic-AMP and -GMP phosphodiesterase 11A CHEMBL2717 NA 95 29 0.9723 0.9835
365 Dual specificity calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1C CHEMBL4619 NA 71 12 0.9831 0.8627
366 Dual specificity mitogen-activated protein kinase kinase 1 CHEMBL3587 S218E,S222E 417 23 0.9726 1
367 Dual specificity mitogen-activated protein kinase kinase 1 CHEMBL3587 NA 417 90 0.9726 0.9796
368 Dual specificity mitogen-activated protein kinase kinase 4 CHEMBL2897 NA 56 19 0.948 1
369 Dual specificity mitogen-activated protein kinase kinase 7 CHEMBL3530 NA 67 11 0.9796 0.9442
370 Dual specificity protein kinase CLK1 CHEMBL4224 NA 653 289 0.9708 0.9757
371 Dual specificity protein kinase CLK2 CHEMBL4225 NA 419 51 0.9528 0.8864
372 Dual specificity protein kinase CLK3 CHEMBL4226 NA 225 99 0.9649 0.9693
373 Dual specificity protein kinase CLK4 CHEMBL4203 NA 420 66 0.964 0.9224
374 Dual specificity protein kinase TTK CHEMBL3983 NA 512 233 0.9909 0.998
375 Dual specificity tyrosine-phosphorylation-regulated kinase 1A CHEMBL2292 NA 1361 417 0.9808 0.981
376 Dual specificity tyrosine-phosphorylation-regulated kinase 1B CHEMBL5543 NA 602 143 0.9768 0.9523
377 Dual specificity tyrosine-phosphorylation-regulated kinase 2 CHEMBL4376 NA 473 134 0.9805 0.9834
378 Dual specificity tyrosine-phosphorylation-regulated kinase 3 CHEMBL4575 NA 287 64 0.969 0.9637
379 E3 SUMO-protein ligase CBX4 CHEMBL3232685 NA 24 14 1 1
380 E3 ubiquitin-protein ligase CBL-B CHEMBL4879459 NA 127 43 0.9986 0.9748
381 E3 ubiquitin-protein ligase Mdm2 CHEMBL5023 NA 968 295 0.988 0.9981
382 E3 ubiquitin-protein ligase XIAP CHEMBL4198 NA 465 159 0.9983 0.9999
383 E3 ubiquitin-protein ligase XIAP/Receptor-interacting serine/threonine-protein kinase 2 CHEMBL4888447 NA 20 20 1 1
384 EML4-ALK CHEMBL3883330 L1152R 39 17 0.986 0.9672
385 EML4-ALK CHEMBL3883330 S1206Y 39 19 0.986 0.991
386 EML4-ALK CHEMBL3883330 C1156Y 39 20 0.986 0.9911
387 EML4-ALK CHEMBL3883330 F1174L 39 20 0.986 0.9911
388 EML4-ALK CHEMBL3883330 G1269A 39 20 0.986 0.9911
389 EML4-ALK CHEMBL3883330 L1196M 39 22 0.986 0.985
390 EML4-ALK CHEMBL3883330 G1202R 39 23 0.986 0.9824
391 EML4-ALK CHEMBL3883330 NA 39 33 0.986 0.9837
392 EZH1/SUZ12/EED/AEBP2/RBBP4 complex CHEMBL3137287 NA 25 24 1 1
393 Early activation antigen CD69 CHEMBL3308911 NA 34 20 0.9718 0.9435
394 Ectonucleotide pyrophosphatase/phosphodiesterase family member 1 CHEMBL5925 NA 275 81 0.9891 0.9856
395 Ectonucleotide pyrophosphatase/phosphodiesterase family member 3 CHEMBL5580 NA 115 27 0.9674 0.9524
396 Egl nine homolog 1 CHEMBL5697 NA 454 83 0.9971 0.9956
397 Endoplasmic reticulum aminopeptidase 1 CHEMBL5939 NA 145 42 0.9844 0.9726
398 Endoplasmic reticulum aminopeptidase 2 CHEMBL5043 NA 154 62 0.9924 0.9994
399 Endothelial PAS domain-containing protein 1 CHEMBL1744522 NA 154 51 0.9892 0.9943
400 Endothelial lipase CHEMBL5080 NA 128 74 0.9922 0.9772
401 Endothelin receptor type B CHEMBL1785 NA 151 77 0.9974 0.9993
402 Endothelin-1 receptor CHEMBL252 NA 270 196 0.9959 0.9948
403 Ephrin type-A receptor 2 CHEMBL2068 NA 97 17 0.9476 0.9256
404 Ephrin type-A receptor 4 CHEMBL3988 NA 62 34 0.9251 0.9532
405 Ephrin type-B receptor 4 CHEMBL5147 NA 180 63 0.9627 0.9917
406 Epidermal growth factor receptor CHEMBL203 T790M,L858M 5377 12 0.9722 1
407 Epidermal growth factor receptor CHEMBL203 C797S,L858R 5377 24 0.9722 1
408 Epidermal growth factor receptor CHEMBL203 L861Q 5377 40 0.9722 0.9687
409 Epidermal growth factor receptor CHEMBL203 L858R,T790M,C797S 5377 111 0.9722 0.987
410 Epidermal growth factor receptor CHEMBL203 T790M 5377 122 0.9722 0.9767
411 Epidermal growth factor receptor CHEMBL203 UNDEFINED MUTATION 5377 186 0.9722 0.9942
412 Epidermal growth factor receptor CHEMBL203 L858R 5377 420 0.9722 0.9893
413 Epidermal growth factor receptor CHEMBL203 L858R,T790M 5377 889 0.9722 0.9938
414 Epidermal growth factor receptor CHEMBL203 NA 5377 1429 0.9722 0.987
415 Epithelial discoidin domain-containing receptor 1 CHEMBL5319 NA 258 93 0.9578 0.9725
416 Equilibrative nucleoside transporter 1 CHEMBL1997 NA 148 110 0.9977 0.9938
417 Estrogen receptor CHEMBL206 S463P 2436 11 0.9882 0.9997
418 Estrogen receptor CHEMBL206 D538G 2436 21 0.9882 0.9995
419 Estrogen receptor CHEMBL206 Y537S 2436 22 0.9882 0.9977
420 Estrogen receptor CHEMBL206 NA 2436 1226 0.9882 0.996
421 Estrogen receptor beta CHEMBL242 NA 1347 523 0.9915 0.9958
422 Estrogen-related receptor gamma CHEMBL4245 NA 206 51 0.9979 0.9999
423 Eukaryotic initiation factor 4A-I CHEMBL2052028 NA 72 31 0.9805 0.9943
424 Eukaryotic initiation factor 4A-III CHEMBL4105832 NA 48 22 0.9553 0.9886
425 Eukaryotic translation initiation factor 2-alpha kinase 3 CHEMBL6030 NA 84 64 0.9993 0.9998
426 Eukaryotic translation initiation factor 4E CHEMBL4848 NA 87 31 0.9715 0.9835
427 Excitatory amino acid transporter 1 CHEMBL3085 NA 113 64 0.9993 0.9999
428 Excitatory amino acid transporter 2 CHEMBL4973 NA 110 42 0.995 0.9995
429 Excitatory amino acid transporter 3 CHEMBL2721 NA 76 37 0.9993 0.9999
430 Exportin-1 CHEMBL5661 NA 65 40 0.9685 0.9991
431 Extracellular calcium-sensing receptor CHEMBL1878 NA 318 216 0.9998 0.9998
432 Farnesyl pyrophosphate synthase CHEMBL1782 NA 199 67 0.9943 0.9998
433 Fatty acid synthase CHEMBL4158 NA 177 18 0.9903 0.9636
434 Fatty acid-binding protein 5 CHEMBL3674 NA 132 20 0.9935 0.9999
435 Fatty acid-binding protein, adipocyte CHEMBL2083 NA 269 46 0.9918 0.998
436 Fatty acid-binding protein, brain CHEMBL3826863 NA 43 11 0.9968 1
437 Fatty-acid amide hydrolase 1 CHEMBL2243 NA 1169 397 0.9911 0.9957
438 Fibroblast growth factor receptor 1 CHEMBL3650 NA 1094 189 0.9825 0.9792
439 Fibroblast growth factor receptor 2 CHEMBL4142 NA 381 125 0.9828 0.9923
440 Fibroblast growth factor receptor 3 CHEMBL2742 K650E 374 14 0.9844 1
441 Fibroblast growth factor receptor 3 CHEMBL2742 NA 374 162 0.9844 0.9936
442 Fibroblast growth factor receptor 4 CHEMBL3973 NA 662 265 0.9908 0.997
443 Focal adhesion kinase 1 CHEMBL2695 NA 801 188 0.9789 0.9823
444 Folate receptor alpha CHEMBL2121 NA 58 58 0.9999 0.9999
445 Folate receptor beta CHEMBL5064 NA 38 38 0.9999 0.9999
446 Follicle-stimulating hormone receptor CHEMBL2024 NA 41 19 0.9788 0.9571
447 Free fatty acid receptor 1 CHEMBL4422 NA 1577 1036 0.9979 0.9983
448 Free fatty acid receptor 2 CHEMBL5493 NA 203 99 0.9979 0.9998
449 Free fatty acid receptor 3 CHEMBL5201 NA 65 25 0.9998 1
450 Free fatty acid receptor 4 CHEMBL5339 NA 432 247 0.999 0.999
451 Fructose-1,6-bisphosphatase 1 CHEMBL3975 NA 570 321 0.9942 0.9971
452 Furin CHEMBL2611 NA 236 67 0.9943 1
453 G protein-coupled receptor 88 CHEMBL3399910 NA 274 214 1 1
454 G protein-coupled receptor kinase 5 CHEMBL5678 NA 164 32 0.9922 0.9988
455 G-protein coupled bile acid receptor 1 CHEMBL5409 NA 659 459 0.9924 0.9943
456 G-protein coupled receptor 183 CHEMBL3259470 NA 93 90 0.9891 0.99
457 G-protein coupled receptor 35 CHEMBL1293267 NA 263 123 0.9945 0.9954
458 G-protein coupled receptor 39 CHEMBL3091266 NA 79 68 0.9699 0.9864
459 G-protein coupled receptor 4 CHEMBL3638324 NA 38 31 1 1
460 G-protein coupled receptor 52 CHEMBL3297639 NA 154 122 0.9941 1
461 G-protein coupled receptor 55 CHEMBL1075322 NA 166 80 0.9965 0.9845
462 G-protein coupled receptor 6 CHEMBL3714130 NA 28 10 0.941 0.8094
463 G-protein coupled receptor 84 CHEMBL3714079 NA 375 270 0.9995 0.9997
464 GABA A receptor alpha-2/beta-2/gamma-2 CHEMBL2111413 NA 87 48 0.9859 0.9835
465 GABA A receptor alpha-3/beta-2/gamma-2 CHEMBL2111339 NA 43 33 0.9912 0.9989
466 GABA A receptor alpha-4/beta-3/gamma-2 CHEMBL2111366 NA 21 17 0.9575 0.9591
467 GABA-A receptor; alpha-1/beta-2/gamma-2 CHEMBL2095172 NA 181 111 0.9854 0.9763
468 GABA-A receptor; alpha-1/beta-3/gamma-2 CHEMBL2094121 NA 224 195 0.9888 0.9934
469 GABA-A receptor; alpha-2/beta-3/gamma-2 CHEMBL2094130 NA 150 136 0.9901 0.9978
470 GABA-A receptor; alpha-3/beta-3/gamma-2 CHEMBL2094120 NA 190 177 0.9906 0.9983
471 GABA-A receptor; alpha-5/beta-3/gamma-2 CHEMBL2094122 NA 248 241 0.992 0.997
472 GABA-A receptor; alpha-6/beta-3/gamma-2 CHEMBL2095190 NA 18 13 0.9503 0.9558
473 GABA-B receptor CHEMBL2111463 NA 40 18 0.9958 0.9884
474 GRIA1/CACNG8 CHEMBL4296110 NA 20 18 0.9626 0.9622
475 GTPase KRas CHEMBL2189121 G13D 473 10 0.9861 1
476 GTPase KRas CHEMBL2189121 NA 473 35 0.9861 0.9957
477 GTPase KRas CHEMBL2189121 G12D 473 53 0.9861 0.9977
478 GTPase KRas CHEMBL2189121 G12C 473 99 0.9861 0.9999
479 Galectin-3 CHEMBL4531 NA 228 22 0.9996 0.9751
480 Galectin-8 CHEMBL5475 NA 78 10 0.9997 1
481 Gamma-aminobutyric acid receptor subunit alpha-4/beta3/delta CHEMBL3430899 NA 40 34 1 1
482 Gamma-aminobutyric acid receptor subunit alpha-5/beta-2/gamma-2 CHEMBL4523641 NA 36 28 0.998 0.9958
483 Gamma-aminobutyric acid receptor subunit beta-3 CHEMBL1847 NA 16 11 0.9997 1
484 Gamma-aminobutyric acid receptor subunit rho-1 CHEMBL3561 NA 36 19 0.9979 0.9994
485 Gamma-secretase CHEMBL2094135 NA 2081 1668 0.9936 0.9984
486 Gastric inhibitory polypeptide receptor CHEMBL4383 NA 70 23 0.9997 0.9998
487 Gastrin/cholecystokinin type B receptor CHEMBL298 NA 227 115 0.9969 0.9993
488 Geranylgeranyl pyrophosphate synthase CHEMBL4769 NA 148 52 0.9998 1
489 Geranylgeranyl transferase type I CHEMBL2095164 NA 157 71 0.9845 0.9922
490 Glucagon receptor CHEMBL1985 NA 545 394 0.9963 0.996
491 Glucagon-like peptide 1 receptor CHEMBL1784 NA 203 133 0.9948 0.9948
492 Glucocorticoid receptor CHEMBL2034 NA 1938 1213 0.995 0.9974
493 Glucokinase/Glucokinase regulatory protein CHEMBL3885579 NA 33 28 1 1
494 Glucose-6-phosphate 1-dehydrogenase CHEMBL5347 NA 27 10 0.9209 0.8607
495 Glucose-dependent insulinotropic receptor CHEMBL5652 NA 1081 873 0.9972 0.9982
496 Glutamate NMDA receptor; GRIN1/GRIN2A CHEMBL1907604 NA 145 83 0.9878 0.9922
497 Glutamate NMDA receptor; GRIN1/GRIN2B CHEMBL1907603 NA 192 161 0.9943 0.9985
498 Glutamate carboxypeptidase 2 CHEMBL1892 NA 273 116 0.9963 0.9999
499 Glutamate receptor 1 CHEMBL2009 NA 32 17 0.9525 0.9983
500 Glutamate receptor 2 CHEMBL4016 NA 248 89 0.9968 0.9936
501 Glutamate receptor 4 CHEMBL3190 NA 56 37 0.9906 0.9988
502 Glutamate receptor ionotropic, NMDA 1 CHEMBL2015 NA 24 24 0.9841 0.9868
503 Glutamate receptor ionotropic, NMDA 2A CHEMBL1972 NA 31 13 0.985 0.9758
504 Glutamate receptor ionotropic, NMDA 2B CHEMBL1904 NA 173 117 0.9787 0.9972
505 Glutamate receptor ionotropic, kainate 1 CHEMBL1918 NA 94 15 0.9949 0.9949
506 Glutamate receptor ionotropic, kainate 2 CHEMBL3683 NA 34 12 0.9704 0.9928
507 Glutaminase kidney isoform, mitochondrial CHEMBL2146302 NA 356 101 0.9947 0.9999
508 Glutaminyl-peptide cyclotransferase CHEMBL4508 NA 629 162 0.9978 0.9963
509 Glutaminyl-peptide cyclotransferase-like protein CHEMBL3638349 NA 79 24 0.9889 0.9554
510 Glutathione S-transferase omega-1 CHEMBL3174 NA 75 19 0.9562 0.9999
511 Glycine receptor (alpha-1/beta) CHEMBL2363052 NA 31 19 0.9988 0.999
512 Glycine receptor subunit alpha-1 CHEMBL5845 NA 61 28 0.931 0.9416
513 Glycogen phosphorylase, liver form CHEMBL2568 NA 373 153 0.9958 0.9998
514 Glycogen synthase kinase-3 alpha CHEMBL2850 NA 254 45 0.9525 0.9976
515 Glycogen synthase kinase-3 beta CHEMBL262 UNDEFINED MUTATION 2228 103 0.9738 0.9958
516 Glycogen synthase kinase-3 beta CHEMBL262 NA 2228 308 0.9738 0.9763
517 Gonadotropin-releasing hormone receptor CHEMBL1855 NA 679 391 0.9945 0.995
518 Group 10 secretory phospholipase A2 CHEMBL4342 NA 99 16 0.9954 0.9755
519 Group IID secretory phospholipase A2 CHEMBL4281 NA 10 10 1 1
520 Growth hormone secretagogue receptor type 1 CHEMBL4616 NA 1003 835 0.9964 0.9982
521 HSP60/HSP10 CHEMBL4106131 NA 109 44 0.9626 0.9753
522 Heat shock factor protein 1 CHEMBL5869 NA 88 44 0.9704 0.9601
523 Heat shock protein HSP 90-alpha CHEMBL3880 NA 913 121 0.9898 0.995
524 Heat shock protein HSP 90-beta CHEMBL4303 NA 466 71 0.9893 0.9775
525 Hematopoietic prostaglandin D synthase CHEMBL5879 NA 247 123 0.9891 0.9915
526 Heparanase CHEMBL3921 NA 201 12 0.9953 0.8956
527 Hepatic sodium/bile acid cotransporter CHEMBL5287 NA 49 20 0.9488 0.9925
528 Hepatic triacylglycerol lipase CHEMBL2127 NA 45 34 0.9808 0.9741
529 Hepatitis A virus cellular receptor 2 CHEMBL4630879 NA 61 28 0.9862 0.9998
530 Hepatocyte growth factor activator CHEMBL3351190 NA 105 14 0.9989 0.9984
531 Hepatocyte growth factor receptor CHEMBL3717 Y1235D 2745 11 0.9829 0.9989
532 Hepatocyte growth factor receptor CHEMBL3717 D1228N 2745 16 0.9829 1
533 Hepatocyte growth factor receptor CHEMBL3717 Y1230H 2745 25 0.9829 0.9975
534 Hepatocyte growth factor receptor CHEMBL3717 NA 2745 537 0.9829 0.9948
535 Hexokinase-1 CHEMBL2688 NA 22 12 0.9852 1
536 Hexokinase-2 CHEMBL2640 NA 30 17 0.9909 1
537 Hexokinase-4 CHEMBL3820 NA 887 187 0.9975 1
538 High affinity 3',5'-cyclic-AMP phosphodiesterase 7A CHEMBL3012 NA 277 49 0.9818 0.9392
539 High affinity cAMP-specific and IBMX-insensitive 3',5'-cyclic phosphodiesterase 8A CHEMBL4640 NA 29 14 0.9486 0.9967
540 High affinity cGMP-specific 3',5'-cyclic phosphodiesterase 9A CHEMBL3535 NA 139 55 0.9658 0.9823
541 High affinity nerve growth factor receptor CHEMBL2815 F589L 1330 11 0.9748 0.95
542 High affinity nerve growth factor receptor CHEMBL2815 G667C 1330 29 0.9748 0.9548
543 High affinity nerve growth factor receptor CHEMBL2815 G595R 1330 36 0.9748 0.9662
544 High affinity nerve growth factor receptor CHEMBL2815 NA 1330 459 0.9748 0.9797
545 Histamine H1 receptor CHEMBL231 NA 941 592 0.9805 0.9934
546 Histamine H2 receptor CHEMBL1941 NA 280 136 0.9745 0.9919
547 Histamine H3 receptor CHEMBL264 NA 2981 2185 0.9916 0.9945
548 Histamine H4 receptor CHEMBL3759 NA 830 466 0.9921 0.9974
549 Histone acetyltransferase KAT2B CHEMBL5500 NA 153 33 0.9865 0.9823
550 Histone acetyltransferase KAT6A CHEMBL3774298 NA 267 174 0.9984 1
551 Histone acetyltransferase p300 CHEMBL3784 NA 416 73 0.9714 0.9514
552 Histone deacetylase 1 CHEMBL325 NA 4485 995 0.9924 0.9959
553 Histone deacetylase 11 CHEMBL3310 NA 345 67 0.9923 0.998
554 Histone deacetylase 2 CHEMBL1937 NA 1666 337 0.9877 0.9922
555 Histone deacetylase 3 CHEMBL1829 NA 1384 278 0.9913 0.9975
556 Histone deacetylase 3/NCoR1 CHEMBL3038484 NA 66 55 0.9965 0.9951
557 Histone deacetylase 3/Nuclear receptor corepressor 2 (HDAC3/NCoR2) CHEMBL2111363 NA 357 266 0.9948 0.9981
558 Histone deacetylase 4 CHEMBL3524 NA 581 130 0.9914 0.9954
559 Histone deacetylase 5 CHEMBL2563 NA 260 53 0.9824 0.9931
560 Histone deacetylase 6 CHEMBL1865 NA 3396 1021 0.9906 0.9965
561 Histone deacetylase 7 CHEMBL2716 NA 338 65 0.9839 0.983
562 Histone deacetylase 8 CHEMBL3192 NA 1772 315 0.991 0.995
563 Histone deacetylase 9 CHEMBL4145 NA 235 22 0.9821 0.9968
564 Histone-arginine methyltransferase CARM1 CHEMBL5406 NA 280 49 0.9873 0.9878
565 Histone-lysine N-methyltransferase 2A/WDR5 CHEMBL3883320 NA 62 40 0.9846 0.9526
566 Histone-lysine N-methyltransferase EHMT1 CHEMBL6031 NA 179 84 0.9828 0.9999
567 Histone-lysine N-methyltransferase EHMT2 CHEMBL6032 NA 525 114 0.9871 0.9927
568 Histone-lysine N-methyltransferase EZH2 CHEMBL2189110 Y641F 638 29 0.9928 1
569 Histone-lysine N-methyltransferase EZH2 CHEMBL2189110 Y641N 638 42 0.9928 0.9998
570 Histone-lysine N-methyltransferase EZH2 CHEMBL2189110 NA 638 119 0.9928 0.9922
571 Histone-lysine N-methyltransferase NSD2 CHEMBL3108645 NA 237 43 0.9688 0.9971
572 Histone-lysine N-methyltransferase NSD3 CHEMBL3108646 NA 52 12 0.8871 0.9789
573 Histone-lysine N-methyltransferase SETD2 CHEMBL3108647 NA 28 20 0.9704 1
574 Histone-lysine N-methyltransferase SMYD3 CHEMBL2321643 NA 124 75 0.9884 1
575 Histone-lysine N-methyltransferase, H3 lysine-79 specific CHEMBL1795117 NA 158 25 0.9869 0.9965
576 Hormone-sensitive lipase CHEMBL3590 NA 64 31 0.9999 1
577 Hydroxycarboxylic acid receptor 1 CHEMBL1075101 NA 37 29 0.9998 1
578 Hydroxycarboxylic acid receptor 2 CHEMBL3785 NA 467 227 0.9976 0.9992
579 Hydroxycarboxylic acid receptor 3 CHEMBL4421 NA 98 48 0.9975 0.9994
580 Hypoxia-inducible factor 1-alpha CHEMBL4261 NA 416 203 0.9816 0.9784
581 IKK epsilon/TBK1 CHEMBL3038486 NA 21 11 1 1
582 Ileal sodium/bile acid cotransporter CHEMBL2778 NA 163 113 0.9999 0.9999
583 Immunoglobulin lambda variable 6-57 CHEMBL4739844 NA 40 23 1 1
584 Indoleamine 2,3-dioxygenase 1 CHEMBL4685 S167A 2114 10 0.9823 0.9458
585 Indoleamine 2,3-dioxygenase 1 CHEMBL4685 NA 2114 859 0.9823 0.992
586 Indoleamine 2,3-dioxygenase 2 CHEMBL3627587 NA 50 11 0.9812 0.9996
587 Induced myeloid leukemia cell differentiation protein Mcl-1 CHEMBL4361 NA 1220 340 0.9898 0.9959
588 Induced myeloid leukemia cell differentiation protein Mcl-1/BH3-interacting domain death agonist CHEMBL3430886 NA 37 14 0.9275 0.9157
589 Induced myeloid leukemia cell differentiation protein Mcl-1/Bcl-2-like protein 11 CHEMBL3430887 NA 72 25 0.9852 0.9765
590 Inhibitor of NF-kappa-B kinase (IKK) CHEMBL2111328 NA 20 13 0.9914 1
591 Inhibitor of nuclear factor kappa-B kinase subunit alpha CHEMBL3476 NA 173 20 0.9789 0.9929
592 Inhibitor of nuclear factor kappa-B kinase subunit beta CHEMBL1991 NA 601 39 0.9744 0.9727
593 Inhibitor of nuclear factor kappa-B kinase subunit epsilon CHEMBL3529 NA 131 37 0.9781 0.9892
594 Inositol hexakisphosphate kinase 1 CHEMBL4523418 NA 157 27 0.9999 0.9801
595 Inositol hexakisphosphate kinase 2 CHEMBL4523488 NA 58 27 0.996 1
596 Inositol hexakisphosphate kinase 3 CHEMBL4523431 NA 48 13 0.9984 1
597 Insulin receptor CHEMBL1981 NA 275 41 0.9635 0.9959
598 Insulin-like growth factor 1 receptor CHEMBL1957 NA 645 257 0.9799 0.991
599 Integrin alpha-2/beta-3 CHEMBL2111461 NA 18 16 0.995 1
600 Integrin alpha-4 CHEMBL278 NA 117 88 0.9999 0.9999
601 Integrin alpha-4/beta-1 CHEMBL1907599 NA 589 456 0.9995 0.9993
602 Integrin alpha-4/beta-7 CHEMBL2095184 NA 201 173 0.9994 0.9994
603 Integrin alpha-5/beta-1 CHEMBL2095226 NA 216 159 0.9912 0.9981
604 Integrin alpha-IIb/beta-3 CHEMBL2093869 NA 971 644 0.9973 0.9979
605 Integrin alpha-L CHEMBL1803 NA 79 32 0.9817 1
606 Integrin alpha-V/beta-1 CHEMBL2111407 NA 110 98 0.9986 0.9985
607 Integrin alpha-V/beta-3 CHEMBL1907598 NA 725 626 0.9924 0.9941
608 Integrin alpha-V/beta-5 CHEMBL2096675 NA 242 202 0.999 0.9986
609 Integrin alpha-V/beta-6 CHEMBL2111416 NA 243 180 0.9994 0.9989
610 Integrin alpha-V/beta-8 CHEMBL3430892 NA 116 93 0.9992 0.9989
611 Integrin alpha2/beta1 CHEMBL3137268 NA 44 40 0.9955 0.9989
612 Intercellular adhesion molecule (ICAM-1), Integrin alpha-L/beta-2 CHEMBL2096661 NA 173 155 0.9962 0.9964
613 Interleukin-1 receptor antagonist protein CHEMBL4523191 NA 63 23 0.9926 0.9994
614 Interleukin-1 receptor-associated kinase 1 CHEMBL3357 NA 63 11 0.9176 0.9239
615 Interleukin-1 receptor-associated kinase 3 CHEMBL5081 NA 31 16 0.8975 0.9041
616 Interleukin-1 receptor-associated kinase 4 CHEMBL3778 NA 907 344 0.9943 0.9983
617 Interleukin-17A CHEMBL3390822 NA 26 18 0.9557 0.9731
618 Interleukin-2 CHEMBL5880 NA 81 43 0.9649 0.9622
619 Intermediate conductance calcium-activated potassium channel protein 4 CHEMBL4305 NA 47 18 0.9995 1
620 Interstitial collagenase CHEMBL332 NA 715 31 0.9873 0.9973
621 Isocitrate dehydrogenase [NADP] cytoplasmic CHEMBL2007625 R132L 722 10 0.991 0.9961
622 Isocitrate dehydrogenase [NADP] cytoplasmic CHEMBL2007625 NA 722 22 0.991 0.9453
623 Isocitrate dehydrogenase [NADP] cytoplasmic CHEMBL2007625 R132C 722 121 0.991 0.9938
624 Isocitrate dehydrogenase [NADP] cytoplasmic CHEMBL2007625 R132H 722 224 0.991 0.9898
625 Isocitrate dehydrogenase [NADP], mitochondrial CHEMBL3991501 R140Q 103 18 0.9968 1
626 JAK1/JAK2/TYK2 CHEMBL3301390 NA 27 25 0.9695 0.9757
627 JAK1/TYK2 CHEMBL3301391 NA 127 106 0.9909 0.9928
628 JAK2/JAK1 CHEMBL3038492 NA 51 30 0.9815 0.9782
629 JAK2/TYK2 CHEMBL3301392 NA 46 33 0.982 0.9884
630 JAK3/JAK1 CHEMBL3038491 NA 185 161 0.9933 0.9909
631 Kallikrein-5 CHEMBL4447 NA 112 45 0.9891 0.9999
632 Kallikrein-6 CHEMBL4448 NA 44 21 0.961 0.9615
633 Kallikrein-7 CHEMBL2443 NA 138 16 0.9762 1
634 Kallikrein-8 CHEMBL4812 NA 21 12 0.9995 0.9996
635 Kappa-type opioid receptor CHEMBL237 NA 2807 2081 0.9829 0.991
636 Keap1/Nrf2 CHEMBL3038498 NA 524 202 0.9864 0.9931
637 Kelch-like ECH-associated protein 1 CHEMBL2069156 NA 358 85 0.9795 0.998
638 Ketohexokinase CHEMBL1275212 NA 76 45 0.9995 1
639 KiSS-1 receptor CHEMBL5413 NA 153 146 0.9973 0.9993
640 Kinesin-1 heavy chain/ Tyrosine-protein kinase receptor RET CHEMBL3430888 NA 82 46 0.9844 0.9733
641 Kinesin-like protein KIF11 CHEMBL4581 NA 716 193 0.9935 0.996
642 Kinesin-like protein KIF18A CHEMBL4523403 NA 41 33 0.9994 0.9986
643 Kir3.1/Kir3.2 CHEMBL3038489 NA 180 95 0.997 0.9973
644 Kir3.1/Kir3.4 CHEMBL3038488 NA 178 77 0.9997 0.9997
645 Kynurenine 3-monooxygenase CHEMBL2145 NA 179 96 0.998 0.9999
646 L-amino-acid oxidase CHEMBL5291590 NA 20 14 1 1
647 L-lactate dehydrogenase A chain CHEMBL4835 NA 520 125 0.9776 0.9884
648 L-lactate dehydrogenase B chain CHEMBL4940 NA 186 21 0.9925 0.9845
649 LIM domain kinase 1 CHEMBL3836 NA 301 48 0.9703 0.9509
650 LIM domain kinase 2 CHEMBL5932 NA 263 85 0.9719 0.9754
651 LSD1/CoREST complex CHEMBL3137262 NA 183 130 0.9937 0.9949
652 Lactoylglutathione lyase CHEMBL2424 NA 146 42 0.9927 0.9996
653 Lanosterol synthase CHEMBL3593 NA 47 24 0.978 0.999
654 Legumain CHEMBL4244 NA 171 31 0.9998 1
655 Leucine-rich repeat serine/threonine-protein kinase 2 CHEMBL1075104 G2019S 984 250 0.9876 0.9916
656 Leucine-rich repeat serine/threonine-protein kinase 2 CHEMBL1075104 NA 984 258 0.9876 0.9956
657 Leucyl-cystinyl aminopeptidase CHEMBL2693 NA 170 56 0.9877 0.9994
658 Leukotriene A-4 hydrolase CHEMBL4618 NA 311 95 0.9961 0.9964
659 Leukotriene B4 receptor 2 CHEMBL3191 NA 68 52 0.9942 0.9944
660 Leukotriene C4 synthase CHEMBL1743183 NA 47 33 0.9907 0.9998
661 Liver carboxylesterase 1 CHEMBL2265 NA 169 72 0.9909 0.9996
662 Long-chain fatty acid transport protein 4 CHEMBL4327 NA 24 10 1 1
663 Low molecular weight phosphotyrosine protein phosphatase CHEMBL4903 NA 158 37 0.9933 0.9999
664 Lutropin-choriogonadotropic hormone receptor CHEMBL1854 NA 51 31 0.964 0.9756
665 Lysine-specific demethylase 2A CHEMBL1938210 NA 100 16 0.9889 0.9674
666 Lysine-specific demethylase 4A CHEMBL5896 NA 182 65 0.978 0.9975
667 Lysine-specific demethylase 4B CHEMBL3313832 NA 103 68 0.9902 0.9977
668 Lysine-specific demethylase 4C CHEMBL6175 NA 226 52 0.9861 0.976
669 Lysine-specific demethylase 4D CHEMBL6138 NA 97 53 0.992 0.9999
670 Lysine-specific demethylase 4E CHEMBL1293226 NA 91 19 0.9839 0.9949
671 Lysine-specific demethylase 5A CHEMBL2424504 NA 219 49 0.9841 0.9884
672 Lysine-specific demethylase 5B CHEMBL3774295 NA 290 42 0.9954 0.9918
673 Lysine-specific histone demethylase 1A CHEMBL6136 NA 1407 382 0.9801 0.9896
674 Lysophosphatidic acid receptor 1 CHEMBL3819 NA 268 163 0.9962 0.9966
675 Lysophosphatidic acid receptor 2 CHEMBL3724 NA 103 40 0.9954 0.9999
676 Lysophosphatidic acid receptor 3 CHEMBL3250 NA 60 36 0.9763 0.9885
677 Lysophosphatidic acid receptor 5 CHEMBL5700 NA 53 38 0.9989 0.9941
678 Lysosomal acid glucosylceramidase CHEMBL2179 NA 277 14 0.9957 0.9354
679 Lysosomal acid glucosylceramidase CHEMBL2179 N409S 277 45 0.9957 0.9943
680 Lysyl oxidase homolog 2 CHEMBL3714029 NA 125 93 0.9939 0.9975
681 Lysyl oxidase homolog 3 CHEMBL4105989 NA 25 13 0.9771 0.9922
682 M-phase inducer phosphatase 1 CHEMBL3775 NA 204 24 0.9907 0.9932
683 M-phase inducer phosphatase 2 CHEMBL4804 NA 309 41 0.987 0.9953
684 M-phase inducer phosphatase 3 CHEMBL2378 NA 89 11 0.9935 0.9972
685 MAP kinase-activated protein kinase 2 CHEMBL2208 NA 547 69 0.9883 0.9872
686 MAP kinase-activated protein kinase 5 CHEMBL3094 NA 27 10 0.8843 0.9832
687 MAP kinase-interacting serine/threonine-protein kinase 1 CHEMBL4718 NA 442 121 0.9808 0.9787
688 MAP kinase-interacting serine/threonine-protein kinase 2 CHEMBL4204 NA 412 150 0.9792 0.9895
689 MAP/microtubule affinity-regulating kinase 3 CHEMBL5600 NA 73 25 0.9722 0.9865
690 MAP/microtubule affinity-regulating kinase 4 CHEMBL5754 NA 71 26 0.9469 0.9745
691 METTL3/METTL14 CHEMBL4106140 NA 34 15 0.9963 0.9847
692 MIF/CD74 (Macrophage migration inhibitory factor and HLA-DR antigens-associated invariant chain) CHEMBL2111430 NA 17 10 0.9731 0.9678
693 MLL1-ASH2L/RbBP5/WDR5/DPY30 CHEMBL4106124 NA 30 28 0.9998 0.9998
694 Macrophage colony-stimulating factor 1 receptor CHEMBL1844 NA 872 245 0.98 0.9832
695 Macrophage metalloelastase CHEMBL4393 UNDEFINED MUTATION 383 13 0.9913 1
696 Macrophage metalloelastase CHEMBL4393 NA 383 48 0.9913 0.9977
697 Macrophage migration inhibitory factor CHEMBL2085 NA 291 70 0.9692 0.9853
698 Macrophage-stimulating protein receptor CHEMBL2689 NA 103 44 0.9722 0.9874
699 Malate dehydrogenase, cytoplasmic CHEMBL3560 NA 22 13 0.9811 1
700 Mas-related G-protein coupled receptor member X1 CHEMBL5850 NA 115 73 0.9947 0.9919
701 Mas-related G-protein coupled receptor member X2 CHEMBL5849 NA 36 14 0.9554 0.889
702 Mast/stem cell growth factor receptor Kit CHEMBL1936 D816H 797 11 0.972 0.88
703 Mast/stem cell growth factor receptor Kit CHEMBL1936 V559D,T670I 797 17 0.972 0.8936
704 Mast/stem cell growth factor receptor Kit CHEMBL1936 UNDEFINED MUTATION 797 25 0.972 0.9559
705 Mast/stem cell growth factor receptor Kit CHEMBL1936 NA 797 127 0.972 0.954
706 Maternal embryonic leucine zipper kinase CHEMBL4578 NA 131 45 0.9411 0.9141
707 Matrix metalloproteinase-14 CHEMBL3869 NA 505 11 0.9894 0.9878
708 Matrix metalloproteinase-9 CHEMBL321 Q279R 1176 14 0.9774 1
709 Matrix metalloproteinase-9 CHEMBL321 NA 1176 40 0.9774 0.9492
710 Melanin-concentrating hormone receptor 1 CHEMBL344 NA 2557 1987 0.9929 0.9952
711 Melanin-concentrating hormone receptor 2 CHEMBL5038 NA 42 32 0.9909 0.9999
712 Melanocortin receptor 3 CHEMBL4644 NA 484 331 0.995 0.9922
713 Melanocortin receptor 4 CHEMBL259 L106P 1704 28 0.9974 0.9999
714 Melanocortin receptor 4 CHEMBL259 NA 1704 1342 0.9974 0.9978
715 Melanocortin receptor 5 CHEMBL4608 NA 330 231 0.9958 0.992
716 Melanocyte-stimulating hormone receptor CHEMBL3795 NA 417 278 0.9963 0.9967
717 Melatonin receptor type 1A CHEMBL1945 NA 625 513 0.9941 0.999
718 Melatonin receptor type 1B CHEMBL1946 NA 675 549 0.9955 0.9979
719 Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase CHEMBL3984 NA 75 49 0.9956 0.9922
720 Membrane-bound transcription factor site-1 protease CHEMBL5916 NA 21 14 0.9999 1
721 Menin CHEMBL1615381 NA 166 45 0.9928 0.9999
722 Menin/Histone-lysine N-methyltransferase MLL CHEMBL2093861 NA 135 96 0.9929 0.9927
723 Meprin A subunit beta CHEMBL4105879 NA 81 45 0.9937 0.9945
724 Metabotropic glutamate receptor 1 CHEMBL3772 NA 436 300 0.9925 0.9968
725 Metabotropic glutamate receptor 2 CHEMBL5137 NA 819 623 0.9962 0.9978
726 Metabotropic glutamate receptor 3 CHEMBL2888 NA 93 80 0.9836 0.9936
727 Metabotropic glutamate receptor 4 CHEMBL2736 NA 500 261 0.9962 0.9993
728 Metabotropic glutamate receptor 5 CHEMBL3227 NA 1445 1053 0.9945 0.9962
729 Metabotropic glutamate receptor 6 CHEMBL4573 NA 30 17 0.9961 0.9995
730 Metabotropic glutamate receptor 7 CHEMBL3777 NA 56 25 0.933 0.9989
731 Metabotropic glutamate receptor 8 CHEMBL3228 NA 67 32 0.9774 0.9953
732 Methionine aminopeptidase 1 CHEMBL2474 NA 145 36 0.9956 0.9987
733 Methionine aminopeptidase 2 CHEMBL3922 NA 411 96 0.9985 0.9909
734 Methylated-DNA--protein-cysteine methyltransferase CHEMBL2864 NA 31 10 0.9963 1
735 Microsomal triglyceride transfer protein large subunit CHEMBL2569 NA 49 40 1 1
736 Microtubule-associated protein tau CHEMBL1293224 NA 232 97 0.9892 0.9922
737 Mineralocorticoid receptor CHEMBL1994 C808S 586 18 0.9971 1
738 Mineralocorticoid receptor CHEMBL1994 NA 586 221 0.9971 0.9969
739 Mitogen-activated protein kinase 1 CHEMBL4040 NA 662 178 0.9688 0.9902
740 Mitogen-activated protein kinase 10 CHEMBL2637 NA 690 66 0.9836 0.9836
741 Mitogen-activated protein kinase 11 CHEMBL3961 NA 143 47 0.9825 0.9945
742 Mitogen-activated protein kinase 14 CHEMBL260 NA 2452 468 0.988 0.9943
743 Mitogen-activated protein kinase 3 CHEMBL3385 NA 129 23 0.9395 0.9964
744 Mitogen-activated protein kinase 7 CHEMBL5332 NA 140 58 0.9819 0.9999
745 Mitogen-activated protein kinase 8 CHEMBL2276 NA 761 74 0.9831 0.9885
746 Mitogen-activated protein kinase 9 CHEMBL4179 NA 409 60 0.9689 0.9876
747 Mitogen-activated protein kinase kinase kinase 11 CHEMBL2708 NA 66 13 0.9658 0.9999
748 Mitogen-activated protein kinase kinase kinase 12 CHEMBL1908389 NA 105 79 0.993 1
749 Mitogen-activated protein kinase kinase kinase 13 CHEMBL1163124 NA 24 21 0.9998 1
750 Mitogen-activated protein kinase kinase kinase 14 CHEMBL5888 S549D 269 11 0.9985 0.9955
751 Mitogen-activated protein kinase kinase kinase 14 CHEMBL5888 NA 269 87 0.9985 0.9992
752 Mitogen-activated protein kinase kinase kinase 20 CHEMBL3886 NA 88 40 0.9408 0.9799
753 Mitogen-activated protein kinase kinase kinase 5 CHEMBL5285 NA 347 128 0.9942 0.9978
754 Mitogen-activated protein kinase kinase kinase 7 CHEMBL5776 NA 204 68 0.9837 0.9758
755 Mitogen-activated protein kinase kinase kinase 8 CHEMBL4899 NA 137 24 0.9896 1
756 Mitogen-activated protein kinase kinase kinase 9 CHEMBL2872 NA 66 16 0.9114 1
757 Mitogen-activated protein kinase kinase kinase kinase 1 CHEMBL5749 NA 480 212 0.9877 0.9973
758 Mitogen-activated protein kinase kinase kinase kinase 4 CHEMBL6166 NA 186 50 0.9606 0.9812
759 Monoacylglycerol lipase ABHD6 CHEMBL2189127 NA 83 35 0.9678 0.9478
760 Monocarboxylate transporter 1 CHEMBL4360 NA 86 50 0.9789 0.9973
761 Monocarboxylate transporter 4 CHEMBL2073663 NA 104 47 0.9836 0.9778
762 Monoglyceride lipase CHEMBL4191 NA 906 236 0.9926 0.9956
763 Motilin receptor CHEMBL2203 NA 184 129 0.9925 0.9922
764 Mu-type opioid receptor CHEMBL233 NA 3321 2512 0.9841 0.9916
765 Mucolipin-2 CHEMBL4879493 NA 27 16 0.9999 1
766 Mucosa-associated lymphoid tissue lymphoma translocation protein 1 CHEMBL3632452 NA 349 109 0.9934 0.9827
767 Multidrug and toxin extrusion protein 1 CHEMBL1743126 NA 41 22 0.7283 0.6676
768 Multidrug and toxin extrusion protein 2 CHEMBL1743127 NA 23 10 0.6669 0.6991
769 Multidrug resistance-associated protein 1 CHEMBL3004 NA 242 135 0.9617 0.9712
770 Muscarinic acetylcholine receptor M1 CHEMBL216 NA 1285 788 0.9811 0.9861
771 Muscarinic acetylcholine receptor M2 CHEMBL211 NA 666 409 0.9714 0.9859
772 Muscarinic acetylcholine receptor M3 CHEMBL245 NA 970 606 0.985 0.9912
773 Muscarinic acetylcholine receptor M4 CHEMBL1821 NA 948 645 0.9881 0.9913
774 Muscarinic acetylcholine receptor M5 CHEMBL2035 NA 562 272 0.9785 0.9846
775 Myc proto-oncogene protein CHEMBL1250348 NA 53 21 0.9756 0.9989
776 Myeloperoxidase CHEMBL2439 NA 303 29 0.9794 1
777 N-acyl-phosphatidylethanolamine-hydrolyzing phospholipase D CHEMBL4630839 NA 98 60 0.9662 0.9991
778 N-acylethanolamine-hydrolyzing acid amidase CHEMBL4349 NA 217 76 0.9965 0.998
779 N-alpha-acetyltransferase 50 CHEMBL4630854 NA 17 10 0.9583 1
780 N-arachidonyl glycine receptor CHEMBL2384898 NA 90 48 0.9867 0.9966
781 N-formyl peptide receptor 2 CHEMBL4227 NA 374 267 0.9961 0.997
782 N-lysine methyltransferase SMYD2 CHEMBL2169716 NA 113 34 0.9973 0.9993
783 N-terminal Xaa-Pro-Lys N-methyltransferase 1 CHEMBL4523442 NA 82 28 0.9972 0.9977
784 N6-adenosine-methyltransferase catalytic subunit CHEMBL4739695 NA 36 16 0.9496 0.9832
785 NACHT, LRR and PYD domains-containing protein 3 CHEMBL1741208 NA 541 265 0.9926 0.9926
786 NAD-dependent protein deacetylase sirtuin-1 CHEMBL4506 NA 566 192 0.9801 0.9872
787 NAD-dependent protein deacetylase sirtuin-2 CHEMBL4462 NA 764 113 0.9818 0.9899
788 NAD-dependent protein deacetylase sirtuin-3, mitochondrial CHEMBL4461 NA 252 86 0.9812 0.9968
789 NAD-dependent protein deacylase sirtuin-5, mitochondrial CHEMBL2163183 NA 284 22 0.9882 1
790 NADPH oxidase 1 CHEMBL1287628 NA 50 24 0.9427 0.9013
791 NADPH oxidase 4 CHEMBL1250375 NA 127 64 0.9746 1
792 NADPH oxidase 5 CHEMBL1926497 NA 32 16 0.9643 0.9999
793 NEDD8 activating enzyme CHEMBL3831283 NA 75 73 0.9974 1
794 NF-kappa-B inhibitor alpha CHEMBL2898 NA 38 13 0.9832 0.956
795 NKGD2-MICA CHEMBL5483005 NA 30 20 1 1
796 NKGD2-ULBP6 CHEMBL5483006 NA 28 11 1 1
797 NPC1-like intracellular cholesterol transporter 1 CHEMBL2027 I1061T 129 10 0.9955 1
798 NPC1-like intracellular cholesterol transporter 1 CHEMBL2027 NA 129 49 0.9955 0.9936
799 NPM/ALK (Nucleophosmin/ALK tyrosine kinase receptor) CHEMBL2111387 NA 59 42 0.9961 0.9994
800 NT-3 growth factor receptor CHEMBL5608 NA 317 91 0.9791 0.9853
801 NUAK family SNF1-like kinase 1 CHEMBL5784 NA 74 23 0.9295 0.946
802 Na(+)/citrate cotransporter CHEMBL3769293 NA 26 22 0.9691 0.9659
803 Natural resistance-associated macrophage protein 2 CHEMBL1932895 NA 43 31 0.9999 0.9973
804 Neprilysin CHEMBL1944 NA 203 32 0.9935 0.9876
805 Neurogenic locus notch homolog protein 1 CHEMBL2146346 NA 44 30 1 1
806 Neurogenic locus notch homolog protein 3 CHEMBL3407319 NA 20 19 1 1
807 Neuromedin-B receptor CHEMBL3636 NA 35 18 0.9736 0.9523
808 Neuromedin-K receptor CHEMBL4429 NA 329 254 0.9956 0.9968
809 Neuromedin-U receptor 1 CHEMBL1075178 NA 48 47 1 0.9999
810 Neuromedin-U receptor 2 CHEMBL1075144 NA 75 63 0.9967 0.9999
811 Neuronal acetylcholine receptor subunit alpha-7 CHEMBL2492 NA 719 319 0.9832 0.992
812 Neuronal acetylcholine receptor; alpha3/beta4 CHEMBL1907594 NA 398 195 0.9943 0.9975
813 Neuronal acetylcholine receptor; alpha4/beta2 CHEMBL1907589 NA 675 414 0.9943 0.9952
814 Neuronal acetylcholine receptor; alpha4/beta4 CHEMBL1907591 NA 41 16 0.9919 0.977
815 Neuropeptide FF receptor 1 CHEMBL5951 NA 135 106 0.9966 0.9964
816 Neuropeptide FF receptor 2 CHEMBL5952 NA 143 91 0.9969 0.9973
817 Neuropeptide S receptor CHEMBL5162 NA 60 45 0.9917 0.9976
818 Neuropeptide Y receptor type 1 CHEMBL4777 NA 256 207 0.9939 0.9972
819 Neuropeptide Y receptor type 2 CHEMBL4018 NA 164 88 0.9827 0.9868
820 Neuropeptide Y receptor type 4 CHEMBL4877 NA 70 48 0.9779 0.9897
821 Neuropeptide Y receptor type 5 CHEMBL4561 NA 449 317 0.9952 0.9968
822 Neuropeptides B/W receptor type 1 CHEMBL1293293 NA 114 60 0.9999 0.9999
823 Neurotensin receptor type 1 CHEMBL4123 NA 180 109 0.9952 0.9984
824 Neurotensin receptor type 2 CHEMBL2514 NA 78 63 0.9991 0.9992
825 Neutrophil collagenase CHEMBL4588 NA 461 36 0.9867 0.9815
826 Neutrophil cytosol factor 1 CHEMBL1613743 NA 97 35 0.9871 1
827 Nicotinamide N-methyltransferase CHEMBL2346486 NA 180 55 0.9951 0.9987
828 Nicotinamide phosphoribosyltransferase CHEMBL1744525 NA 753 230 0.9947 0.9977
829 Nischarin CHEMBL3923 NA 30 19 0.9954 0.9944
830 Nitric oxide synthase 1 CHEMBL3568 NA 413 161 0.9976 0.9999
831 Nitric oxide synthase 3 CHEMBL4803 NA 239 41 0.999 0.9982
832 Nitric oxide synthase, inducible CHEMBL4481 NA 412 146 0.9918 0.9944
833 Nociceptin receptor CHEMBL2014 NA 1098 940 0.9954 0.9968
834 Non-receptor tyrosine-protein kinase TYK2 CHEMBL3553 NA 1108 399 0.9876 0.9906
835 Nuclear factor erythroid 2-related factor 2 CHEMBL1075094 NA 299 109 0.9883 0.98
836 Nuclear receptor ROR-alpha CHEMBL5868 NA 106 21 0.9826 0.9845
837 Nuclear receptor ROR-beta CHEMBL3091268 NA 218 66 0.9971 0.9999
838 Nuclear receptor ROR-gamma CHEMBL1741186 NA 2408 1414 0.9914 0.9949
839 Nuclear receptor subfamily 1 group D member 1 CHEMBL1961783 NA 90 36 0.9937 1
840 Nuclear receptor subfamily 1 group I member 2 CHEMBL3401 NA 402 88 0.9736 0.976
841 Nuclear receptor subfamily 1 group I member 3 CHEMBL5503 NA 160 44 0.9954 0.9951
842 Nuclear receptor subfamily 2 group C member 2/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1 CHEMBL3885612 NA 21 13 0.9725 0.9047
843 Nuclear receptor subfamily 2 group E member 1 CHEMBL1961788 NA 45 20 0.9697 0.9998
844 Nuclear receptor subfamily 4 group A member 2 CHEMBL5002 NA 157 68 0.9878 0.9976
845 Nuclear receptor subfamily 4immunitygroup A member 1 CHEMBL1293229 NA 39 11 0.992 0.9998
846 Nuclear receptor subfamily 5 group A member 2 CHEMBL3544 NA 70 32 0.9898 0.9875
847 Nucleosome-remodeling factor subunit BPTF CHEMBL3085621 NA 68 29 0.9542 0.9883
848 Nucleotide-binding oligomerization domain-containing protein 1 CHEMBL1293222 NA 164 45 0.9966 0.9812
849 Nucleotide-binding oligomerization domain-containing protein 2 CHEMBL1293266 NA 226 100 0.9914 0.9835
850 ORAI1/STIM1 CHEMBL3832644 NA 15 10 0.9874 0.9879
851 Orexin receptor type 2 CHEMBL4792 NA 1120 780 0.993 0.9952
852 Orexin/Hypocretin receptor type 1 CHEMBL5113 NA 960 576 0.9891 0.9976
853 Ovarian cancer G-protein coupled receptor 1 CHEMBL3713916 NA 10 10 1 1
854 Oxidized purine nucleoside triphosphate hydrolase CHEMBL3708265 NA 139 61 0.994 0.9891
855 Oxoeicosanoid receptor 1 CHEMBL1628461 NA 52 26 1 1
856 Oxysterol-binding protein 1 CHEMBL4523203 NA 30 23 0.9998 0.9999
857 Oxysterols receptor LXR-alpha CHEMBL2808 NA 677 210 0.9927 0.9964
858 Oxysterols receptor LXR-beta CHEMBL4093 NA 755 302 0.9912 0.9947
859 Oxytocin receptor CHEMBL2049 NA 572 424 0.9936 0.9943
860 P2X purinoceptor 1 CHEMBL2094 NA 67 26 0.97 0.9985
861 P2X purinoceptor 3 CHEMBL2998 NA 332 194 0.9687 0.9861
862 P2X purinoceptor 4 CHEMBL2104 NA 143 69 0.9976 0.9857
863 P2X purinoceptor 7 CHEMBL4805 NA 1072 827 0.9912 0.9956
864 P2X2/P2X3 heterotrimeric receptor CHEMBL3831281 NA 29 12 0.9496 0.9679
865 P2Y purinoceptor 1 CHEMBL4315 NA 371 238 0.9933 0.9956
866 P2Y purinoceptor 12 CHEMBL2001 NA 961 785 0.9968 0.9986
867 P2Y purinoceptor 14 CHEMBL4518 NA 288 199 0.9956 0.9989
868 P2Y purinoceptor 2 CHEMBL4398 NA 144 73 0.9964 0.9999
869 P2Y purinoceptor 4 CHEMBL2123 NA 91 32 0.9995 0.9999
870 P2Y purinoceptor 6 CHEMBL4714 NA 144 71 0.9986 0.9998
871 PCSK9/LDLR CHEMBL4523996 NA 35 10 0.9917 0.9459
872 PI3-kinase p110-alpha/p85-alpha CHEMBL2111367 H1047R 697 10 0.9917 0.9653
873 PI3-kinase p110-alpha/p85-alpha CHEMBL2111367 NA 697 567 0.9917 0.9917
874 PI3-kinase p110-delta/p85-alpha CHEMBL2111432 NA 773 730 0.9929 0.9955
875 PI3-kinase subunit gamma/Phosphoinositide 3-kinase regulatory subunit 5 CHEMBL3430881 NA 10 10 0.9622 0.9576
876 PI3K p110 beta/p85 alpha CHEMBL3038510 NA 325 264 0.9942 0.9944
877 PRMT5/MEP50 complex CHEMBL3137261 NA 233 135 0.9764 0.9813
878 Palmitoleoyl-protein carboxylesterase NOTUM CHEMBL3714531 C330S 444 117 0.9977 0.9972
879 Palmitoleoyl-protein carboxylesterase NOTUM CHEMBL3714531 NA 444 140 0.9977 0.9994
880 Pantetheinase CHEMBL4739843 NA 32 13 1 1
881 Pantothenate kinase 3 CHEMBL3407328 NA 83 26 0.9866 1
882 Parathyroid hormone/parathyroid hormone-related peptide receptor CHEMBL1793 NA 79 44 1 1
883 Parkinson disease protein 7 CHEMBL5169188 NA 24 14 0.9148 0.9008
884 Peptide deformylase, mitochondrial CHEMBL4647 NA 45 32 1 1
885 Peptidyl-prolyl cis-trans isomerase A CHEMBL1949 NA 134 31 0.9965 0.9846
886 Peptidyl-prolyl cis-trans isomerase FKBP1A CHEMBL1902 NA 306 50 0.9917 1
887 Peptidyl-prolyl cis-trans isomerase FKBP1B CHEMBL2430 NA 30 29 0.9928 0.9995
888 Peptidyl-prolyl cis-trans isomerase FKBP5 CHEMBL2052031 NA 180 39 0.9899 0.9929
889 Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 CHEMBL2288 NA 372 51 0.9869 0.9852
890 Peregrin CHEMBL3132741 NA 204 63 0.9772 0.996
891 Perforin-1 CHEMBL5480 NA 163 82 1 1
892 Period circadian protein homolog 2 CHEMBL3751648 NA 38 31 1 1
893 Peroxisome proliferator-activated receptor alpha CHEMBL239 NA 1996 909 0.993 0.9969
894 Peroxisome proliferator-activated receptor delta CHEMBL3979 NA 1357 649 0.995 0.997
895 Peroxisome proliferator-activated receptor gamma CHEMBL235 NA 2821 1129 0.984 0.9929
896 Phenylethanolamine N-methyltransferase CHEMBL4617 NA 140 32 0.9994 1
897 Phosphatidylcholine:ceramide cholinephosphotransferase 2 CHEMBL3112379 NA 105 25 0.9933 1
898 Phosphatidylinositol 3-kinase catalytic subunit type 3 CHEMBL1075165 NA 174 64 0.9517 0.9837
899 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform CHEMBL4005 H1047R 3027 25 0.9832 0.9987
900 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform CHEMBL4005 NA 3027 507 0.9832 0.9877
901 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform CHEMBL3145 NA 1326 371 0.9829 0.9904
902 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform CHEMBL3130 NA 2459 702 0.9872 0.9961
903 Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform CHEMBL3267 NA 2045 474 0.9821 0.9932
904 Phosphatidylinositol 4-kinase beta CHEMBL3268 NA 235 62 0.9771 0.9832
905 Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta CHEMBL5554 NA 65 20 0.9628 0.9439
906 Phosphatidylinositol 4-phosphate 5-kinase type-1 gamma CHEMBL1908383 NA 83 31 0.9858 0.984
907 Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha CHEMBL1795194 NA 178 73 0.978 0.9999
908 Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma CHEMBL1770034 NA 80 12 0.9937 0.9791
909 Phosphatidylinositol 5-phosphate 4-kinase type-2 gamma CHEMBL1770034 UNDEFINED MUTATION 80 35 0.9937 1
910 Phospholipase A and acyltransferase 2 CHEMBL4630860 NA 33 10 1 1
911 Phospholipase A and acyltransferase 3 CHEMBL3831244 NA 33 16 1 1
912 Phospholipase A and acyltransferase 4 CHEMBL4630864 NA 35 10 1 1
913 Phospholipase A and acyltransferase 5 CHEMBL4630850 NA 35 28 1 1
914 Phospholipase D1 CHEMBL2536 NA 148 105 0.9944 0.9999
915 Phospholipase D2 CHEMBL2734 NA 120 82 0.9937 0.9948
916 Plasma kallikrein CHEMBL2000 NA 440 100 0.98 0.9906
917 Platelet-activating factor acetylhydrolase CHEMBL3514 NA 194 58 0.9965 0.9995
918 Platelet-activating factor receptor CHEMBL250 NA 62 44 0.9702 0.9895
919 Platelet-derived growth factor receptor CHEMBL2095189 NA 114 85 0.9845 0.9881
920 Platelet-derived growth factor receptor alpha CHEMBL2007 V561D 431 37 0.9711 0.9848
921 Platelet-derived growth factor receptor alpha CHEMBL2007 NA 431 63 0.9711 0.958
922 Platelet-derived growth factor receptor beta CHEMBL1913 NA 656 164 0.9747 0.9811
923 Poly [ADP-ribose] polymerase 1 CHEMBL3105 NA 2152 621 0.9907 0.9951
924 Poly [ADP-ribose] polymerase 2 CHEMBL5366 NA 457 107 0.9919 0.9955
925 Poly [ADP-ribose] polymerase tankyrase-1 CHEMBL6164 NA 483 185 0.9897 0.9846
926 Poly [ADP-ribose] polymerase tankyrase-2 CHEMBL6154 NA 512 188 0.9889 0.9922
927 Poly(ADP-ribose) glycohydrolase CHEMBL1795143 NA 110 27 1 1
928 Polyamine deacetylase HDAC10 CHEMBL5103 NA 311 53 0.991 0.9977
929 Polycomb protein EED CHEMBL2189117 NA 318 110 0.9887 0.9812
930 Polyunsaturated fatty acid 5-lipoxygenase CHEMBL215 NA 1405 515 0.9753 0.991
931 Polyunsaturated fatty acid lipoxygenase ALOX12 CHEMBL3687 NA 114 28 0.9816 0.9947
932 Polyunsaturated fatty acid lipoxygenase ALOX15 CHEMBL2903 NA 296 71 0.9728 0.9756
933 Potassium channel subfamily K member 13 CHEMBL4523461 NA 17 14 1 1
934 Potassium channel subfamily K member 3 CHEMBL2321613 NA 71 56 0.9701 0.9919
935 Potassium channel subfamily K member 9 CHEMBL2321614 NA 54 19 0.8926 0.9064
936 Potassium channel subfamily T member 1 CHEMBL4739688 NA 56 15 0.9532 0.9819
937 Potassium voltage-gated channel subfamily A member 3 CHEMBL4633 NA 152 103 0.9952 0.9988
938 Potassium voltage-gated channel subfamily A member 5 CHEMBL4306 NA 521 288 0.9956 0.9957
939 Potassium voltage-gated channel subfamily B member 1 CHEMBL2363000 NA 26 21 0.9996 0.9997
940 Potassium voltage-gated channel subfamily KQT member 1 CHEMBL1866 NA 33 10 0.9522 1
941 Potassium voltage-gated channel subfamily KQT member 2 CHEMBL2476 NA 37 22 0.9845 0.9999
942 Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 1 CHEMBL1795171 NA 25 13 1 1
943 Potassium/sodium hyperpolarization-activated cyclic nucleotide-gated channel 4 CHEMBL1250417 NA 28 15 1 0.9981
944 Presenilin-1 CHEMBL2473 NA 32 17 0.9792 0.9564
945 Probable G-protein coupled receptor 132 CHEMBL3085618 NA 27 11 0.9981 0.9716
946 Probable G-protein coupled receptor 139 CHEMBL3632455 NA 115 111 0.9995 0.9997
947 Probable G-protein coupled receptor 142 CHEMBL2069161 NA 167 136 0.9999 1
948 Probable G-protein coupled receptor 174 CHEMBL3562167 NA 13 10 1 1
949 Probable G-protein coupled receptor 27 CHEMBL4523923 NA 43 25 0.9999 1
950 Probable G-protein coupled receptor 34 CHEMBL3562165 NA 26 17 0.9998 0.9999
951 Probable global transcription activator SNF2L2 CHEMBL2362979 NA 56 14 0.948 0.935
952 Procathepsin L CHEMBL3837 NA 1344 103 0.9877 0.9977
953 Progesterone receptor CHEMBL208 NA 1150 668 0.995 0.9977
954 Programmed cell death 1 ligand 1 CHEMBL3580522 NA 105 17 0.968 0.9802
955 Programmed cell death protein 1/Programmed cell death 1 ligand 1 CHEMBL4523993 NA 1032 861 0.9959 0.9987
956 Prokineticin receptor 1 CHEMBL5649 NA 26 15 0.9979 0.9979
957 Prolyl endopeptidase CHEMBL3202 NA 291 75 0.9925 0.9999
958 Prolyl endopeptidase FAP CHEMBL4683 NA 292 59 0.9994 1
959 Prolyl hydroxylase EGLN2 CHEMBL3028 NA 84 61 0.9962 0.9969
960 Prolyl hydroxylase EGLN3 CHEMBL5705 NA 59 49 0.9932 0.9963
961 Proprotein convertase subtilisin/kexin type 6 CHEMBL2951 NA 50 42 1 1
962 Proprotein convertase subtilisin/kexin type 9 CHEMBL2929 NA 98 47 0.9793 0.9789
963 Prostacyclin receptor CHEMBL1995 NA 191 113 0.996 0.9997
964 Prostaglandin D2 receptor CHEMBL4427 NA 327 238 0.9966 0.9967
965 Prostaglandin D2 receptor 2 CHEMBL5071 NA 1325 1053 0.9991 0.9995
966 Prostaglandin E synthase CHEMBL5658 NA 913 498 0.9864 0.9895
967 Prostaglandin E2 receptor EP1 subtype CHEMBL1811 NA 592 437 0.999 0.9997
968 Prostaglandin E2 receptor EP2 subtype CHEMBL1881 NA 266 130 0.9943 0.9954
969 Prostaglandin E2 receptor EP3 subtype CHEMBL3710 NA 618 233 0.9955 0.9977
970 Prostaglandin E2 receptor EP4 subtype CHEMBL1836 NA 524 368 0.9964 0.9991
971 Prostaglandin F2-alpha receptor CHEMBL1987 NA 73 51 0.9987 0.9872
972 Prostaglandin G/H synthase 1 CHEMBL221 NA 719 136 0.9751 0.9858
973 Prostaglandin G/H synthase 2 CHEMBL230 NA 2406 163 0.974 0.9883
974 Proteasome Macropain subunit CHEMBL3492 NA 201 71 0.9809 0.9998
975 Proteasome Macropain subunit MB1 CHEMBL4662 NA 975 167 0.9902 0.9962
976 Proteasome component C5 CHEMBL4208 NA 166 39 0.9856 0.9804
977 Proteasome subunit beta type-10 CHEMBL3317334 NA 79 33 0.9978 0.9999
978 Proteasome subunit beta type-8 CHEMBL5620 NA 394 95 0.9945 0.9982
979 Proteasome subunit beta type-9 CHEMBL1944495 NA 125 26 0.9993 0.9989
980 Protein ADM2 CHEMBL5267 NA 25 20 1 1
981 Protein AF-9 CHEMBL4295761 NA 52 20 0.9898 0.974
982 Protein ENL CHEMBL4295801 NA 134 36 0.9803 0.9983
983 Protein Mdm4 CHEMBL1255126 NA 202 43 0.9795 0.9895
984 Protein O-GlcNAcase CHEMBL5921 NA 205 35 1 1
985 Protein Wnt-3a CHEMBL1255137 NA 51 27 0.9883 0.9704
986 Protein arginine N-methyltransferase 1 CHEMBL5524 NA 244 26 0.9761 0.9597
987 Protein arginine N-methyltransferase 5 CHEMBL1795116 NA 362 121 0.9858 0.9978
988 Protein arginine N-methyltransferase 6 CHEMBL1275221 NA 158 61 0.9908 0.9995
989 Protein arginine N-methyltransferase 8 CHEMBL3108648 NA 61 20 0.9931 1
990 Protein cereblon CHEMBL3763008 NA 207 50 0.9955 0.9997
991 Protein cereblon-IKZF2 CHEMBL5465554 NA 10 10 1 1
992 Protein cereblon/Aiolos CHEMBL4296167 NA 34 34 1 1
993 Protein cereblon/Bromodomain-containing protein 4 CHEMBL4296138 NA 10 10 1 1
994 Protein cereblon/Cyclin-dependent kinase 12 CHEMBL4879535 NA 10 10 1 1
995 Protein cereblon/DNA damage-binding protein 1 CHEMBL4630734 NA 100 64 0.9998 0.9998
996 Protein cereblon/Estrogen receptor CHEMBL4523681 NA 15 15 0.9993 0.9991
997 Protein cereblon/GSPT1 CHEMBL4296168 NA 17 14 1 1
998 Protein cereblon/IRAK4 CHEMBL4523710 NA 11 11 0.9889 0.9892
999 Protein cereblon/Serine/threonine-protein kinase WEE1 CHEMBL4630732 NA 12 10 1 1
1000 Protein cereblon/Tyrosine-protein kinase BTK CHEMBL4523704 NA 17 15 0.9998 0.9997
1001 Protein cereblon/Tyrosine-protein kinase ITK/TSK CHEMBL5465213 NA 10 10 1 1
1002 Protein disulfide-isomerase CHEMBL5422 NA 159 83 0.9824 0.9961
1003 Protein farnesyltransferase CHEMBL2094108 NA 609 387 0.984 0.9872
1004 Protein kinase C alpha type CHEMBL299 NA 407 75 0.9811 0.9864
1005 Protein kinase C beta type CHEMBL3045 NA 178 16 0.9474 0.9495
1006 Protein kinase C delta type CHEMBL2996 NA 293 29 0.9834 0.9761
1007 Protein kinase C epsilon type CHEMBL3582 NA 197 63 0.9665 0.9862
1008 Protein kinase C iota type CHEMBL2598 NA 75 28 0.9734 0.9768
1009 Protein kinase C theta type CHEMBL3920 NA 462 134 0.9823 0.997
1010 Protein kinase C zeta type CHEMBL3438 NA 157 15 0.9928 0.9251
1011 Protein mono-ADP-ribosyltransferase PARP10 CHEMBL2429708 NA 150 23 0.9929 0.9689
1012 Protein mono-ADP-ribosyltransferase PARP11 CHEMBL2380189 NA 39 18 0.9914 0.941
1013 Protein mono-ADP-ribosyltransferase PARP14 CHEMBL2176777 NA 131 21 0.9771 0.9995
1014 Protein mono-ADP-ribosyltransferase PARP15 CHEMBL2176778 NA 70 13 0.9804 0.9995
1015 Protein mono-ADP-ribosyltransferase TIPARP CHEMBL2380188 NA 84 13 0.9912 0.969
1016 Protein polybromo-1 CHEMBL1795184 NA 92 31 0.9651 0.9787
1017 Protein smoothened CHEMBL5971 V404M 232 10 0.9742 0.7876
1018 Protein smoothened CHEMBL5971 D473H 232 14 0.9742 0.8429
1019 Protein smoothened CHEMBL5971 NA 232 176 0.9742 0.9877
1020 Protein-S-isoprenylcysteine O-methyltransferase CHEMBL4699 NA 109 14 0.9898 0.9995
1021 Protein-arginine deiminase type-4 CHEMBL6111 NA 96 13 0.9915 1
1022 Protein-glutamine gamma-glutamyltransferase CHEMBL2730 NA 350 28 0.9867 0.9693
1023 Protein-lysine 6-oxidase CHEMBL2249 NA 52 20 0.9859 0.9819
1024 Protein-serine O-palmitoleoyltransferase porcupine CHEMBL1255163 NA 58 55 0.9999 0.9995
1025 Protein-tyrosine kinase 2-beta CHEMBL5469 NA 94 27 0.9513 0.9465
1026 Protein-tyrosine kinase 6 CHEMBL4601 NA 100 17 0.9409 0.9136
1027 Proteinase-activated receptor 1 CHEMBL3974 NA 462 259 0.9974 0.9991
1028 Proteinase-activated receptor 2 CHEMBL5963 NA 85 42 0.9834 0.9859
1029 Proteinase-activated receptor 4 CHEMBL4691 NA 171 148 0.9963 0.9995
1030 Prothrombin CHEMBL204 NA 1703 43 0.9881 0.9566
1031 Proto-oncogene Wnt-3 CHEMBL6079 NA 29 29 1 1
1032 Proto-oncogene tyrosine-protein kinase ROS CHEMBL5568 NA 159 49 0.9714 0.9455
1033 Proto-oncogene tyrosine-protein kinase Src CHEMBL267 NA 1185 167 0.9612 0.9694
1034 Proto-oncogene tyrosine-protein kinase receptor Ret CHEMBL2041 V804M 592 20 0.9735 0.9201
1035 Proto-oncogene tyrosine-protein kinase receptor Ret CHEMBL2041 NA 592 168 0.9735 0.9676
1036 Proton-coupled folate transporter CHEMBL1795188 NA 37 34 0.9999 0.9999
1037 Purine nucleoside phosphorylase CHEMBL4338 H257G 163 10 0.9927 1
1038 Purine nucleoside phosphorylase CHEMBL4338 NA 163 40 0.9927 1
1039 Putative P2Y purinoceptor 10 CHEMBL3562166 NA 32 27 1 1
1040 Pyroglutamylated RF-amide peptide receptor CHEMBL5852 NA 86 41 0.9915 0.9873
1041 Pyruvate kinase PKM CHEMBL1075189 NA 187 28 0.9693 0.8875
1042 RAC-alpha serine/threonine-protein kinase CHEMBL4282 NA 1012 372 0.9763 0.9939
1043 RAC-beta serine/threonine-protein kinase CHEMBL2431 NA 286 78 0.9909 0.9896
1044 RAC-gamma serine/threonine-protein kinase CHEMBL4816 NA 217 77 0.9807 0.9888
1045 RAF proto-oncogene serine/threonine-protein kinase CHEMBL1906 Y340E,Y341E 430 12 0.9796 1
1046 RAF proto-oncogene serine/threonine-protein kinase CHEMBL1906 NA 430 49 0.9796 0.9764
1047 RNA demethylase ALKBH5 CHEMBL3621037 NA 72 24 0.9581 0.9804
1048 RXR alpha/PPAR gamma CHEMBL2111394 NA 15 14 0.9353 0.9347
1049 Ras guanyl-releasing protein 3 CHEMBL3638 NA 41 37 0.9993 0.9991
1050 Receptor tyrosine-protein kinase erbB-2 CHEMBL1824 NA 1086 468 0.981 0.9907
1051 Receptor tyrosine-protein kinase erbB-3 CHEMBL5838 L858R 52 23 0.9948 0.9974
1052 Receptor tyrosine-protein kinase erbB-4 CHEMBL3009 NA 196 104 0.981 0.9789
1053 Receptor-interacting serine/threonine-protein kinase 1 CHEMBL5464 NA 535 227 0.985 0.9952
1054 Receptor-interacting serine/threonine-protein kinase 2 CHEMBL5014 NA 335 145 0.9749 0.9888
1055 Receptor-interacting serine/threonine-protein kinase 3 CHEMBL1795199 NA 94 44 0.9505 0.9394
1056 Receptor-type tyrosine-protein kinase FLT3 CHEMBL1974 D835H 2201 10 0.9752 0.9139
1057 Receptor-type tyrosine-protein kinase FLT3 CHEMBL1974 D835Y 2201 163 0.9752 0.9859
1058 Receptor-type tyrosine-protein kinase FLT3 CHEMBL1974 UNDEFINED MUTATION 2201 208 0.9752 0.9776
1059 Receptor-type tyrosine-protein kinase FLT3 CHEMBL1974 NA 2201 443 0.9752 0.9884
1060 Receptor-type tyrosine-protein phosphatase C CHEMBL3243 NA 47 10 0.9821 0.9888
1061 Receptor-type tyrosine-protein phosphatase alpha CHEMBL3918 NA 24 10 0.9379 0.9989
1062 Reduced folate transporter CHEMBL4833 NA 25 24 0.9999 0.9999
1063 Relaxin receptor 1 CHEMBL1293316 NA 113 68 0.9985 0.9992
1064 Relaxin-3 receptor 1 CHEMBL1628472 NA 63 30 1 1
1065 Relaxin-3 receptor 2 CHEMBL1628473 NA 10 10 1 1
1066 Renin CHEMBL286 NA 1287 313 0.9984 0.9997
1067 Retinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit delta CHEMBL3860 NA 147 24 0.993 0.986
1068 Retinaldehyde dehydrogenase 3 CHEMBL3579 NA 99 12 0.9916 0.9431
1069 Retinoblastoma-associated protein CHEMBL5288 NA 20 12 0.9925 0.9875
1070 Retinoic acid receptor RXR-alpha CHEMBL2061 NA 454 173 0.9923 0.9995
1071 Retinoic acid receptor RXR-alpha/gamma CHEMBL3885633 NA 11 11 1 1
1072 Retinoic acid receptor RXR-alpha/oxysterols receptor LXR-alpha CHEMBL3430879 NA 41 34 0.9959 0.9946
1073 Retinoic acid receptor RXR-alpha/oxysterols receptor LXR-beta CHEMBL3430878 NA 53 49 0.9986 0.9992
1074 Retinoic acid receptor RXR-beta CHEMBL1870 NA 216 122 0.9958 0.9997
1075 Retinoic acid receptor RXR-gamma CHEMBL2004 NA 183 100 0.9957 0.9988
1076 Retinoic acid receptor alpha CHEMBL2055 NA 95 41 0.9997 0.9994
1077 Retinoic acid receptor beta CHEMBL2008 NA 115 76 0.9997 0.9996
1078 Retinoic acid receptor gamma CHEMBL2003 NA 137 70 0.9997 0.9995
1079 Retinol-binding protein 4 CHEMBL3100 NA 160 43 0.9999 1
1080 Rho-associated protein kinase 1 CHEMBL3231 NA 568 109 0.9838 0.9935
1081 Rho-associated protein kinase 2 CHEMBL2973 NA 907 236 0.9866 0.9972
1082 Ribosomal protein S6 kinase alpha-3 CHEMBL2345 NA 160 43 0.9593 0.983
1083 Ribosomal protein S6 kinase alpha-5 CHEMBL4237 NA 87 13 0.9565 0.9991
1084 Ribosomal protein S6 kinase beta-1 CHEMBL4501 NA 118 18 0.9577 0.9201
1085 Ribosomal protein S6 kinase beta-1 CHEMBL4501 D18H,T412E 118 22 0.9577 1
1086 Ribosomal protein S6 kinase beta-1 CHEMBL4501 T412E 118 34 0.9577 1
1087 Ribosyldihydronicotinamide dehydrogenase [quinone] CHEMBL3959 NA 231 51 0.9905 0.9883
1088 S-adenosylmethionine synthase isoform type-2 CHEMBL3313835 NA 235 130 0.9986 0.9987
1089 S-methyl-5'-thioadenosine phosphorylase CHEMBL4941 NA 55 13 1 1
1090 SCN8A/SCN1B CHEMBL4523671 NA 25 23 1 1
1091 SKP1-SKP2-CKS1 CHEMBL5482973 NA 37 20 0.9884 1
1092 SOS1-KRAS CHEMBL5465393 NA 126 13 0.9951 0.9998
1093 SOS1-KRAS CHEMBL5465393 G12D 126 15 0.9951 1
1094 SOS1-KRAS CHEMBL5465393 G12C 126 83 0.9951 0.9978
1095 SUMO-activating enzyme CHEMBL2095174 NA 67 56 0.9985 1
1096 Scavenger receptor class B member 1 CHEMBL1914272 NA 49 47 1 1
1097 Secreted frizzled-related protein 1 CHEMBL5517 NA 68 32 0.9882 1
1098 Sentrin-specific protease 1 CHEMBL1909484 NA 105 29 0.9848 0.9809
1099 Sentrin-specific protease 2 CHEMBL2176776 NA 63 16 0.9905 0.9957
1100 Sentrin-specific protease 5 CHEMBL4802012 NA 48 11 1 1
1101 Serine protease hepsin CHEMBL2079849 D161E,R162K 174 16 0.9977 0.9992
1102 Serine protease hepsin CHEMBL2079849 NA 174 38 0.9977 0.9987
1103 Serine-protein kinase ATM CHEMBL3797 NA 427 166 0.9939 0.9993
1104 Serine/threonine-protein kinase 16 CHEMBL3938 NA 42 19 0.9531 0.9865
1105 Serine/threonine-protein kinase 17A CHEMBL4525 NA 96 21 0.9652 0.9546
1106 Serine/threonine-protein kinase 17B CHEMBL3980 NA 127 34 0.9661 0.9667
1107 Serine/threonine-protein kinase 24 CHEMBL5082 NA 49 28 0.975 0.9873
1108 Serine/threonine-protein kinase 26 CHEMBL5941 NA 63 15 0.9666 0.9695
1109 Serine/threonine-protein kinase 3 CHEMBL4708 NA 104 35 0.9668 0.9719
1110 Serine/threonine-protein kinase 4 CHEMBL4598 NA 125 71 0.983 0.9926
1111 Serine/threonine-protein kinase ATR CHEMBL5024 NA 358 106 0.9963 0.9972
1112 Serine/threonine-protein kinase B-raf CHEMBL5145 NA 1950 88 0.9817 0.9851
1113 Serine/threonine-protein kinase B-raf CHEMBL5145 V600E 1950 1039 0.9817 0.9959
1114 Serine/threonine-protein kinase Chk1 CHEMBL4630 NA 1059 316 0.9931 0.9959
1115 Serine/threonine-protein kinase D1 CHEMBL3863 NA 83 14 0.9322 0.9791
1116 Serine/threonine-protein kinase DCLK1 CHEMBL5683 NA 41 31 0.9317 0.9795
1117 Serine/threonine-protein kinase Nek2 CHEMBL3835 NA 123 38 0.9679 0.9958
1118 Serine/threonine-protein kinase PAK 1 CHEMBL4600 NA 293 104 0.9872 0.9868
1119 Serine/threonine-protein kinase PAK 4 CHEMBL4482 NA 246 49 0.9875 0.9673
1120 Serine/threonine-protein kinase PLK1 CHEMBL3024 T210D 792 41 0.9748 1
1121 Serine/threonine-protein kinase PLK1 CHEMBL3024 NA 792 131 0.9748 0.9849
1122 Serine/threonine-protein kinase PLK2 CHEMBL5938 NA 138 75 0.9729 0.9847
1123 Serine/threonine-protein kinase PLK3 CHEMBL4897 NA 104 44 0.937 0.9521
1124 Serine/threonine-protein kinase PLK4 CHEMBL3788 NA 346 53 0.9873 0.9906
1125 Serine/threonine-protein kinase RIO2 CHEMBL6000 NA 37 18 0.9672 0.9542
1126 Serine/threonine-protein kinase SIK1 CHEMBL6082 NA 67 15 0.9623 0.7438
1127 Serine/threonine-protein kinase SIK2 CHEMBL5699 NA 134 29 0.9824 0.9437
1128 Serine/threonine-protein kinase SIK3 CHEMBL6149 NA 88 33 0.9836 0.9467
1129 Serine/threonine-protein kinase SMG1 CHEMBL1795195 NA 23 19 0.9926 1
1130 Serine/threonine-protein kinase Sgk1 CHEMBL2343 NA 151 75 0.9734 0.9996
1131 Serine/threonine-protein kinase TBK1 CHEMBL5408 NA 146 48 0.9767 0.9808
1132 Serine/threonine-protein kinase TNNI3K CHEMBL5260 NA 219 130 0.9875 0.9995
1133 Serine/threonine-protein kinase ULK1 CHEMBL6006 NA 123 90 0.9759 0.9983
1134 Serine/threonine-protein kinase VRK1 CHEMBL1293199 NA 31 30 0.9936 1
1135 Serine/threonine-protein kinase WNK1 CHEMBL1075173 NA 17 10 0.9326 0.9999
1136 Serine/threonine-protein kinase haspin CHEMBL1075163 NA 98 57 0.9654 0.9491
1137 Serine/threonine-protein kinase mTOR CHEMBL2842 NA 1420 372 0.9883 0.9971
1138 Serine/threonine-protein kinase pim-1 CHEMBL2147 NA 1392 190 0.986 0.988
1139 Serine/threonine-protein kinase pim-2 CHEMBL4523 NA 795 60 0.9929 0.9766
1140 Serine/threonine-protein kinase pim-3 CHEMBL5407 NA 474 75 0.9885 0.9944
1141 Serine/threonine-protein kinase/endoribonuclease IRE1 CHEMBL1163101 NA 120 69 0.9846 0.9952
1142 Short transient receptor potential channel 5 CHEMBL1250411 NA 122 71 0.9801 1
1143 Short transient receptor potential channel 6 CHEMBL2417347 NA 33 23 0.9648 1
1144 Sialidase-1 CHEMBL2726 NA 37 16 0.9999 1
1145 Sialidase-3 CHEMBL3046 NA 46 18 1 1
1146 Sialidase-4 CHEMBL4174 NA 37 11 1 1
1147 Sigma intracellular receptor 2 CHEMBL4105907 NA 462 220 0.9733 0.9897
1148 Sigma non-opioid intracellular receptor 1 CHEMBL287 NA 1044 763 0.9816 0.9931
1149 Signal peptide peptidase-like 2A CHEMBL4105833 NA 33 28 0.9993 0.997
1150 Signal transducer and activator of transcription 3 CHEMBL4026 NA 649 201 0.9757 0.9739
1151 Signal transducer and activator of transcription 6 CHEMBL5401 NA 98 47 0.9978 0.9999
1152 Small conductance calcium-activated potassium channel protein 3 CHEMBL3381 NA 13 10 0.9944 0.9959
1153 Sodium channel protein type 1 subunit alpha CHEMBL1845 NA 58 12 0.9623 0.9172
1154 Sodium channel protein type 10 subunit alpha CHEMBL5451 NA 204 134 0.9845 0.9933
1155 Sodium channel protein type 2 subunit alpha CHEMBL4187 NA 97 22 0.9423 0.9005
1156 Sodium channel protein type 3 subunit alpha CHEMBL5163 NA 117 49 0.959 0.9523
1157 Sodium channel protein type 4 subunit alpha CHEMBL2072 NA 70 24 0.961 0.9713
1158 Sodium channel protein type 5 subunit alpha CHEMBL1980 NA 562 246 0.9696 0.9801
1159 Sodium channel protein type 7 subunit alpha CHEMBL3585 NA 77 44 0.9593 0.9363
1160 Sodium channel protein type 8 subunit alpha CHEMBL5202 NA 52 25 0.948 0.8831
1161 Sodium channel protein type 9 subunit alpha CHEMBL4296 NA 2436 943 0.9892 0.9926
1162 Sodium channel protein type 9 subunit alpha/beta-1/beta-2 CHEMBL4630765 NA 33 30 0.9998 0.9997
1163 Sodium- and chloride-dependent GABA transporter 1 CHEMBL1903 NA 59 33 0.9996 1
1164 Sodium- and chloride-dependent glycine transporter 1 CHEMBL2337 NA 672 400 0.9964 0.9984
1165 Sodium- and chloride-dependent glycine transporter 2 CHEMBL3060 NA 154 48 0.9974 0.9886
1166 Sodium-dependent dopamine transporter CHEMBL238 NA 1452 616 0.9868 0.9962
1167 Sodium-dependent neutral amino acid transporter B(0)AT2 CHEMBL3351189 NA 27 11 1 1
1168 Sodium-dependent noradrenaline transporter CHEMBL222 NA 1750 910 0.9915 0.996
1169 Sodium-dependent phosphate transport protein 2B CHEMBL4295685 NA 67 46 0.9929 0.9908
1170 Sodium-dependent proline transporter CHEMBL3317335 NA 49 34 0.9999 1
1171 Sodium-dependent serotonin transporter CHEMBL228 I179C 2911 15 0.9903 1
1172 Sodium-dependent serotonin transporter CHEMBL228 W103A 2911 15 0.9903 1
1173 Sodium-dependent serotonin transporter CHEMBL228 NA 2911 1669 0.9903 0.9944
1174 Sodium/glucose cotransporter 1 CHEMBL4979 NA 395 179 0.9947 0.9988
1175 Sodium/glucose cotransporter 2 CHEMBL3884 NA 941 793 0.9992 0.9999
1176 Sodium/hydrogen exchanger 1 CHEMBL2781 NA 132 89 0.9979 1
1177 Sodium/hydrogen exchanger 3 CHEMBL3273 NA 87 69 1 1
1178 Sodium/nucleoside cotransporter 2 CHEMBL5780 NA 34 15 0.9996 1
1179 Soluble guanylate cyclase alpha1/beta1 complex CHEMBL3137281 NA 29 15 0.9904 1
1180 Solute carrier family 2, facilitated glucose transporter member 1 CHEMBL2535 NA 183 138 0.9779 0.9775
1181 Solute carrier family 2, facilitated glucose transporter member 2 CHEMBL5873 NA 61 30 0.9844 0.9674
1182 Solute carrier family 2, facilitated glucose transporter member 3 CHEMBL5215 NA 147 84 0.9934 0.9887
1183 Solute carrier family 2, facilitated glucose transporter member 4 CHEMBL5874 NA 64 40 0.9728 0.9996
1184 Solute carrier family 22 member 1 CHEMBL5685 NA 95 25 0.9055 0.8644
1185 Solute carrier family 22 member 12 CHEMBL6120 NA 339 105 0.9952 0.9994
1186 Solute carrier family 22 member 2 CHEMBL1743122 NA 47 20 0.8234 0.7696
1187 Somatostatin receptor type 1 CHEMBL1917 NA 137 20 0.9911 0.9749
1188 Somatostatin receptor type 2 CHEMBL1804 NA 280 177 0.992 0.9991
1189 Somatostatin receptor type 3 CHEMBL2028 NA 311 134 0.9978 0.9946
1190 Somatostatin receptor type 4 CHEMBL1853 NA 194 96 0.9932 0.9853
1191 Somatostatin receptor type 5 CHEMBL1792 NA 360 237 0.9963 0.9956
1192 Son of sevenless homolog 1 CHEMBL2079846 NA 265 88 0.9964 0.9999
1193 Sortilin/Progranulin CHEMBL4680051 NA 30 15 1 1
1194 Sphingomyelin phosphodiesterase CHEMBL2760 NA 125 10 0.9688 0.9835
1195 Sphingomyelin phosphodiesterase 3 CHEMBL4523470 NA 123 71 0.9961 1
1196 Sphingosine 1-phosphate receptor 1 CHEMBL4333 NA 1526 1293 0.995 0.9959
1197 Sphingosine 1-phosphate receptor 2 CHEMBL2955 NA 238 113 0.9977 0.9999
1198 Sphingosine 1-phosphate receptor 3 CHEMBL3892 NA 684 328 0.9956 0.9959
1199 Sphingosine 1-phosphate receptor 4 CHEMBL3230 NA 287 173 0.9973 0.9987
1200 Sphingosine 1-phosphate receptor 5 CHEMBL2274 NA 319 245 0.9964 0.9971
1201 Sphingosine kinase 1 CHEMBL4394 NA 212 54 0.9804 0.9986
1202 Sphingosine kinase 2 CHEMBL3023 NA 180 46 0.9961 0.9978
1203 Spindlin-1 CHEMBL4523509 NA 38 23 0.9992 1
1204 Splicing factor 3B subunit 3 CHEMBL1250378 NA 15 10 0.9399 0.9858
1205 Squalene synthase CHEMBL3338 NA 26 16 0.9965 0.9944
1206 Stearoyl-CoA desaturase CHEMBL5555 NA 503 380 0.9985 0.9995
1207 Steroid 17-alpha-hydroxylase/17,20 lyase CHEMBL3522 NA 302 192 0.9994 0.9993
1208 Steroid 21-hydroxylase CHEMBL2759 NA 13 11 1 1
1209 Steroid hormone receptor ERR1 CHEMBL3429 NA 128 31 0.9964 0.95
1210 Steroidogenic factor 1 CHEMBL4666 NA 44 28 0.9719 0.9674
1211 Sterol O-acyltransferase 1 CHEMBL2782 NA 212 78 0.9878 0.9995
1212 Sterol O-acyltransferase 2 CHEMBL4465 NA 128 54 0.9783 0.9961
1213 Sterol regulatory element-binding protein 1 CHEMBL4630818 NA 28 10 0.999 0.8371
1214 Steryl-sulfatase CHEMBL3559 NA 321 190 0.998 0.9934
1215 Stimulator of interferon genes protein CHEMBL4523377 R293Q 440 25 0.9921 0.9999
1216 Stimulator of interferon genes protein CHEMBL4523377 UNDEFINED MUTATION 440 27 0.9921 0.9074
1217 Stimulator of interferon genes protein CHEMBL4523377 G230A,R293Q 440 50 0.9921 0.9998
1218 Stimulator of interferon genes protein CHEMBL4523377 R71H,G230A,R293Q 440 60 0.9921 0.9994
1219 Stimulator of interferon genes protein CHEMBL4523377 NA 440 175 0.9921 0.9899
1220 Stromal cell-derived factor 1 CHEMBL3286074 NA 34 26 0.9471 0.9787
1221 Stromelysin-1 CHEMBL283 NA 613 13 0.9806 0.829
1222 Substance-K receptor CHEMBL2327 NA 357 152 0.9744 0.9983
1223 Substance-P receptor CHEMBL249 NA 844 723 0.9931 0.9996
1224 Succinate dehydrogenase [ubiquinone] iron-sulfur subunit, mitochondrial CHEMBL4105824 NA 35 16 0.9864 1
1225 Succinate receptor 1 CHEMBL2150838 NA 94 72 0.9993 1
1226 Sulfonylurea receptor 1, Kir6.2 CHEMBL2096972 NA 55 33 0.9586 0.996
1227 Sulfonylurea receptor 2, Kir6.2 CHEMBL2095198 NA 72 43 0.9827 0.975
1228 Suppressor of tumorigenicity 14 protein CHEMBL3018 NA 340 88 0.9932 0.9998
1229 Survival motor neuron protein CHEMBL1293232 NA 38 17 0.9999 0.9999
1230 Synaptic vesicular amine transporter CHEMBL1893 NA 22 10 0.8705 0.9994
1231 Syntenin-1/Syndecan-2 CHEMBL4888448 NA 29 13 1 0.9989
1232 T-cell surface glycoprotein CD4 CHEMBL2754 NA 16 10 0.9408 1
1233 TAK1/TAB1 CHEMBL3038499 NA 110 50 0.9791 0.9571
1234 TEL/KDR CHEMBL4630759 NA 20 14 0.9937 0.9876
1235 TGF-beta receptor type-1 CHEMBL4439 T204D 851 21 0.9902 0.9999
1236 TGF-beta receptor type-1 CHEMBL4439 NA 851 423 0.9902 0.9958
1237 TGF-beta receptor type-2 CHEMBL4267 NA 131 22 0.9742 0.9579
1238 TP53-binding protein 1 CHEMBL2424509 NA 53 22 0.9997 1
1239 TRAF2 and NCK-interacting protein kinase CHEMBL4527 NA 175 11 0.954 0.8768
1240 Taste receptor type 2 member 14 CHEMBL3309105 NA 34 25 0.9797 1
1241 Taste receptor type 2 member 8 CHEMBL3988599 NA 44 32 1 1
1242 Tau-tubulin kinase 1 CHEMBL1926492 NA 78 14 0.9998 1
1243 Telomerase reverse transcriptase CHEMBL2916 NA 445 203 0.9806 0.9809
1244 Testis-specific chromodomain protein Y 1 CHEMBL3879864 NA 42 12 0.9783 0.929
1245 Thioredoxin reductase 1, cytoplasmic CHEMBL1927 NA 24 10 0.9408 0.9423
1246 Thrombopoietin receptor CHEMBL1864 NA 167 131 0.9997 0.9999
1247 Thrombospondin-1 CHEMBL4630810 NA 11 11 1 1
1248 Thromboxane A2 receptor CHEMBL2069 NA 368 138 0.9901 0.9963
1249 Thromboxane-A synthase CHEMBL1835 NA 63 22 0.9934 0.9946
1250 Thymidine phosphorylase CHEMBL3106 NA 170 55 0.9986 1
1251 Thyroid hormone receptor CHEMBL2111462 NA 35 33 0.999 0.9998
1252 Thyroid hormone receptor alpha CHEMBL1860 NA 270 90 0.9989 0.9998
1253 Thyroid hormone receptor beta CHEMBL1947 NA 467 137 0.9958 0.9956
1254 Thyrotropin receptor CHEMBL1963 NA 53 41 0.9894 0.9734
1255 Tissue factor CHEMBL4081 NA 140 78 0.9907 0.9897
1256 Tissue factor pathway inhibitor 2 CHEMBL6066240 NA 25 12 0.9992 1
1257 Toll-like receptor 1/2 CHEMBL3885643 NA 106 99 0.9952 0.9976
1258 Toll-like receptor 2 CHEMBL4163 NA 174 73 0.992 0.9835
1259 Toll-like receptor 4 CHEMBL5255 NA 157 79 0.9803 0.985
1260 Toll-like receptor 7 CHEMBL5936 NA 1136 756 0.9933 0.9958
1261 Toll-like receptor 8 CHEMBL5805 NA 509 230 0.9936 0.998
1262 Toll-like receptor 9 CHEMBL5804 NA 243 165 0.9962 0.9955
1263 Trace amine-associated receptor 1 CHEMBL5857 NA 195 129 0.9953 0.9998
1264 Transcription activator BRG1 CHEMBL3085620 NA 59 13 0.9769 0.9718
1265 Transcription factor AP1 CHEMBL2111421 NA 54 26 0.9807 0.9995
1266 Transcription factor Jun CHEMBL4977 NA 68 24 0.9357 0.962
1267 Transcription factor p65 CHEMBL5533 NA 79 19 0.9719 0.9254
1268 Transcription initiation factor TFIID subunit 1 CHEMBL3217390 NA 147 62 0.9897 0.9807
1269 Transcription intermediary factor 1-alpha CHEMBL3108638 NA 104 24 0.9891 0.9899
1270 Transcriptional activator Myb CHEMBL5169115 NA 26 24 1 1
1271 Transcriptional enhancer factor TEF-1 CHEMBL3334416 NA 31 10 0.9678 0.9311
1272 Transcriptional enhancer factor TEF-3 CHEMBL4295828 NA 63 25 0.9798 0.9507
1273 Transforming protein RhoA CHEMBL6052 NA 36 15 0.9971 0.9906
1274 Transient receptor potential cation channel subfamily A member 1 CHEMBL6007 NA 521 219 0.9872 0.9933
1275 Transient receptor potential cation channel subfamily M member 2 CHEMBL1250402 NA 33 10 0.9595 0.904
1276 Transient receptor potential cation channel subfamily M member 5 CHEMBL1628468 NA 73 35 0.9852 1
1277 Transient receptor potential cation channel subfamily M member 8 CHEMBL1075319 NA 430 248 0.9799 0.9866
1278 Transient receptor potential cation channel subfamily V member 1 CHEMBL4794 NA 2160 1639 0.9901 0.9955
1279 Transient receptor potential cation channel subfamily V member 4 CHEMBL3119 NA 297 198 0.9901 0.9986
1280 Transient receptor potential cation channel subfamily V member 6 CHEMBL1628465 NA 45 13 0.9932 1
1281 Transitional endoplasmic reticulum ATPase CHEMBL1075145 NA 326 79 0.9824 0.9956
1282 Transketolase CHEMBL4983 NA 27 11 0.9757 0.9998
1283 Translocator protein CHEMBL5742 UNDEFINED MUTATION 135 21 0.9562 0.999
1284 Translocator protein CHEMBL5742 NA 135 50 0.9562 0.9973
1285 Transmembrane domain-containing protein TMIGD3 CHEMBL3712907 NA 143 99 0.9933 0.9957
1286 Transmembrane protease serine 6 CHEMBL1795139 NA 90 39 0.9997 0.9999
1287 Transthyretin CHEMBL3194 V50M 179 23 0.9879 0.9673
1288 Transthyretin CHEMBL3194 NA 179 64 0.9879 0.9964
1289 Trifunctional purine biosynthetic protein adenosine-3 CHEMBL3972 NA 69 41 0.9826 0.9999
1290 Tryptophan 2,3-dioxygenase CHEMBL2140 NA 497 127 0.9897 0.9989
1291 Tubulin beta-3 chain CHEMBL2597 NA 13 11 0.9214 0.9103
1292 Tumor necrosis factor CHEMBL1825 NA 155 65 0.9741 0.9767
1293 Tumor necrosis factor ligand superfamily member 11 CHEMBL2364162 NA 35 12 0.9742 1
1294 Tumour suppressor p53/oncoprotein Mdm2 CHEMBL1907611 L33E 579 13 0.9827 1
1295 Tumour suppressor p53/oncoprotein Mdm2 CHEMBL1907611 NA 579 327 0.9827 0.9803
1296 Tumour suppressor protein p53/Mdm4 CHEMBL2221344 NA 52 26 0.92 0.8719
1297 Type-1 angiotensin II receptor CHEMBL227 N111G 391 15 0.9932 1
1298 Type-1 angiotensin II receptor CHEMBL227 NA 391 155 0.9932 0.9977
1299 Type-2 angiotensin II receptor CHEMBL4607 NA 137 94 0.9912 1
1300 Tyrosinase CHEMBL1973 NA 196 41 0.989 0.9977
1301 Tyrosine-protein kinase ABL1 CHEMBL1862 NA 1000 129 0.9725 0.9704
1302 Tyrosine-protein kinase ABL1 CHEMBL1862 T315I 1000 232 0.9725 0.9867
1303 Tyrosine-protein kinase BTK CHEMBL5251 C481R 2027 10 0.99 0.9925
1304 Tyrosine-protein kinase BTK CHEMBL5251 T474I 2027 10 0.99 0.9756
1305 Tyrosine-protein kinase BTK CHEMBL5251 C481S 2027 38 0.99 0.985
1306 Tyrosine-protein kinase BTK CHEMBL5251 NA 2027 1034 0.99 0.9943
1307 Tyrosine-protein kinase Blk CHEMBL2250 NA 163 64 0.9643 0.9871
1308 Tyrosine-protein kinase CSK CHEMBL2634 NA 103 10 0.9471 0.8087
1309 Tyrosine-protein kinase Fer CHEMBL3982 NA 52 20 0.932 0.9565
1310 Tyrosine-protein kinase Fyn CHEMBL1841 NA 135 11 0.9419 0.8211
1311 Tyrosine-protein kinase HCK CHEMBL3234 NA 110 12 0.9482 0.8897
1312 Tyrosine-protein kinase ITK/TSK CHEMBL2959 NA 410 90 0.9839 0.9892
1313 Tyrosine-protein kinase JAK1 CHEMBL2835 NA 1557 416 0.9878 0.9928
1314 Tyrosine-protein kinase JAK2 CHEMBL2971 V617F 1936 76 0.9826 0.9743
1315 Tyrosine-protein kinase JAK2 CHEMBL2971 NA 1936 511 0.9826 0.9915
1316 Tyrosine-protein kinase JAK3 CHEMBL2148 NA 1593 482 0.9828 0.9916
1317 Tyrosine-protein kinase Lck CHEMBL258 NA 771 59 0.96 0.9486
1318 Tyrosine-protein kinase Lyn CHEMBL3905 NA 161 10 0.9546 0.856
1319 Tyrosine-protein kinase Mer CHEMBL5331 NA 434 106 0.9806 0.9941
1320 Tyrosine-protein kinase SYK CHEMBL2599 NA 716 296 0.9765 0.9985
1321 Tyrosine-protein kinase Tec CHEMBL4246 NA 125 25 0.9755 0.9791
1322 Tyrosine-protein kinase ZAP-70 CHEMBL2803 NA 99 11 0.9563 0.9621
1323 Tyrosine-protein kinase receptor TYRO3 CHEMBL5314 NA 340 12 0.9816 0.8822
1324 Tyrosine-protein kinase receptor UFO CHEMBL4895 NA 851 111 0.9815 0.9775
1325 Tyrosine-protein phosphatase non-receptor type 1 CHEMBL335 NA 2229 267 0.979 0.9951
1326 Tyrosine-protein phosphatase non-receptor type 11 CHEMBL3864 NA 775 165 0.9797 0.9835
1327 Tyrosine-protein phosphatase non-receptor type 2 CHEMBL3807 NA 488 57 0.9859 0.9775
1328 Tyrosine-protein phosphatase non-receptor type 22 CHEMBL2889 NA 118 32 0.9872 1
1329 Tyrosine-protein phosphatase non-receptor type 5 CHEMBL2007628 NA 203 20 0.9865 0.9967
1330 Tyrosine-protein phosphatase non-receptor type 6 CHEMBL3166 NA 173 19 0.9661 0.9719
1331 Tyrosyl-DNA phosphodiesterase 1 CHEMBL1075138 NA 267 18 0.9868 0.9919
1332 Tyrosyl-DNA phosphodiesterase 2 CHEMBL2169736 NA 231 26 0.9928 0.9997
1333 U5 small nuclear ribonucleoprotein 200 kDa helicase CHEMBL4105972 NA 30 10 0.9817 1
1334 Ubiquitin carboxyl-terminal hydrolase 1/WD repeat-containing protein 48 CHEMBL3430885 NA 98 58 0.9774 0.9999
1335 Ubiquitin carboxyl-terminal hydrolase 2 CHEMBL1293227 NA 39 14 0.9296 0.9849
1336 Ubiquitin carboxyl-terminal hydrolase 5 CHEMBL6158 NA 52 10 0.9616 0.9519
1337 Ubiquitin carboxyl-terminal hydrolase 7 CHEMBL2157850 NA 420 34 0.9925 0.9822
1338 Ubiquitin carboxyl-terminal hydrolase 8 CHEMBL2157854 NA 68 23 0.9959 0.9904
1339 Ubiquitin-like modifier-activating enzyme ATG7 CHEMBL2321621 NA 31 20 1 1
1340 Urokinase-type plasminogen activator CHEMBL3286 NA 395 19 0.9851 0.9997
1341 Urotensin-2 receptor CHEMBL3764 NA 482 378 0.9968 0.9974
1342 Utrophin CHEMBL4523230 NA 58 42 1 1
1343 Vascular endothelial growth factor receptor 1 CHEMBL1868 NA 412 26 0.9603 0.9231
1344 Vascular endothelial growth factor receptor 2 CHEMBL279 NA 4227 1074 0.9653 0.9894
1345 Vascular endothelial growth factor receptor 3 CHEMBL1955 NA 218 22 0.9418 0.8666
1346 Vasopressin V1a receptor CHEMBL1889 NA 783 570 0.9917 0.9964
1347 Vasopressin V1b receptor CHEMBL1921 NA 396 322 0.9954 0.9987
1348 Vasopressin V2 receptor CHEMBL1790 NA 511 344 0.9912 0.9955
1349 Very long chain fatty acid elongase 1 CHEMBL6001 NA 66 56 0.9944 1
1350 Very long chain fatty acid elongase 6 CHEMBL5704 NA 44 30 1 1
1351 Vesicular acetylcholine transporter CHEMBL4767 NA 34 28 0.9998 1
1352 Vitamin D3 receptor CHEMBL1977 NA 377 182 0.9934 0.9967
1353 Vitamin K epoxide reductase complex subunit 1 CHEMBL1930 NA 17 10 0.9988 0.9992
1354 Voltage-dependent L-type calcium channel subunit alpha-1C CHEMBL1940 NA 75 12 0.8779 1
1355 Voltage-dependent N-type calcium channel subunit alpha-1B CHEMBL4478 NA 410 160 0.9937 0.9996
1356 Voltage-dependent T-type calcium channel subunit alpha-1G CHEMBL4641 NA 413 257 0.9935 0.9956
1357 Voltage-dependent T-type calcium channel subunit alpha-1H CHEMBL1859 NA 376 291 0.995 0.9979
1358 Voltage-dependent T-type calcium channel subunit alpha-1I CHEMBL5558 NA 166 153 0.9974 0.9969
1359 Voltage-dependent calcium channel subunit alpha-2/delta-1 CHEMBL1919 NA 169 110 0.9973 0.9975
1360 Voltage-gated inwardly rectifying potassium channel KCNH2 CHEMBL240 NA 7553 2061 0.9255 0.9439
1361 Voltage-gated potassium channel, KQT; KCNQ2(Kv7.2)/KCNQ3(Kv7.3) CHEMBL2221348 NA 67 58 0.9993 0.9992
1362 Von Hippel-Lindau disease tumor suppressor/Elongin B/Elongin C CHEMBL3301400 NA 94 67 0.9982 0.9993
1363 WD repeat-containing protein 5 CHEMBL1075317 NA 368 179 0.9915 0.9975
1364 Wee1-like protein kinase CHEMBL5491 NA 480 81 0.9948 0.9986
1365 Xanthine dehydrogenase/oxidase CHEMBL1929 NA 395 29 0.9852 0.9984
1366 YAP1-TEAD4 CHEMBL5465250 NA 29 14 1 1
1367 YEATS domain-containing protein 4 CHEMBL4296266 NA 15 13 0.999 1
1368 Zinc finger protein Aiolos CHEMBL4739707 NA 14 12 0.9999 0.9998
1369 [Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial CHEMBL4766 NA 178 67 0.9453 0.9616
1370 beta-catenin-B-cell lymphoma 9 protein complex CHEMBL3885525 NA 200 115 0.9942 0.9939
1371 cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A CHEMBL4409 NA 1126 400 0.9891 0.995
1372 cGMP-dependent 3',5'-cyclic phosphodiesterase CHEMBL2652 NA 510 127 0.9856 0.9935
1373 cGMP-dependent protein kinase 1 CHEMBL4273 NA 82 14 0.9582 0.9939
1374 cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A CHEMBL241 NA 268 33 0.9743 0.9992
1375 cGMP-inhibited 3',5'-cyclic phosphodiesterase 3B CHEMBL290 NA 133 15 0.9836 0.949
1376 cGMP-specific 3',5'-cyclic phosphodiesterase CHEMBL1827 NA 903 322 0.9821 0.9985
1377 dCTP pyrophosphatase 1 CHEMBL3769292 NA 173 85 0.9896 1
1378 eIF-2-alpha kinase GCN2 CHEMBL5358 NA 93 46 0.9799 0.9969
1379 fMet-Leu-Phe receptor CHEMBL3359 NA 308 141 0.9956 0.9978
1380 mTORC1 CHEMBL4296661 NA 162 156 0.9864 0.986
1381 mTORC2 CHEMBL4523999 NA 97 91 0.9843 0.9828
1382 von Hippel-Lindau disease tumor suppressor CHEMBL3108660 NA 168 53 0.9988 0.9999
1383 von Hippel-Lindau disease tumor suppressor/Bromodomain-containing protein 4 CHEMBL4296140 NA 14 13 0.9998 0.9999