IC50 | 3019.95 nM | P-glycoprotein 1 | P08183 | |
IC50 | 3235.94 nM | P-glycoprotein 1 | P08183 | |
IC50 | 75857757503 nM | P-glycoprotein 1 | P08183 | |
IC50 | 26302.68 nM | ATP-binding cassette sub-family G member 2 | Q9UNQ0 | |
IC50 | 3235.94 nM | P-glycoprotein 1 | P08183 | |
Others | 37 % | Canalicular multispecific organic anion transporter 1 | Q92887 | |
IC50 | 160000 nM | DNA topoisomerase I | P11387 | |
Potency | 17782.8 nM | Prelamin-A/C | P02545 | |
Potency | 22387.2 nM | Lysine-specific demethylase 4D-like | B2RXH2 | |
Potency | 25118.9 nM | Endoplasmic reticulum-associated amyloid beta-peptide-binding protein | Q99714 | |
Potency | 28183.8 nM | Histone-lysine N-methyltransferase MLL | Q03164 | |
Potency | 7943.3 nM | Caspase-7 | P55210 | |
Potency | 15848.9 nM | Thyroid stimulating hormone receptor | P16473 | |
Potency | 44668.4 nM | Tyrosyl-DNA phosphodiesterase 1 | Q9NUW8 | |
Potency | 56234.1 nM | Tyrosyl-DNA phosphodiesterase 1 | Q9NUW8 | |
Potency | 10000 nM | Tyrosyl-DNA phosphodiesterase 1 | Q9NUW8 | |
Potency | 14125.4 nM | Microtubule-associated protein tau | P10636 | |
Potency | 19952.6 nM | Aldehyde dehydrogenase 1A1 | P00352 | |
Potency | 39810.7 nM | Aldehyde dehydrogenase 1A1 | P00352 | |
Potency | 47754.8 nM | Peripheral myelin protein 22 | Q01453 | |
Potency | 19952.6 nM | Arachidonate 15-lipoxygenase | P16050 | |
Potency | 7943.3 nM | MAP kinase ERK2 | P28482 | |
Potency | 28183.8 nM | Lethal(3)malignant brain tumor-like protein 1 | Q9Y468 | |
Potency | 17782.8 nM | Bloom syndrome protein | P54132 | |
Potency | 15848.9 nM | Thyroid stimulating hormone receptor | P16473 | |
Potency | 31622.8 nM | Thrombopoietin | P40225 | |
Potency | 7943.3 nM | Caspase-1 | P29466 | |
Potency | 31622.8 nM | Hemoglobin beta chain | P68871 | |
Potency | 10000 nM | Neuropeptide S receptor | Q6W5P4 | |
Potency | 17782.8 nM | Bloom syndrome protein | P54132 | |
Potency | 31622.8 nM | DNA polymerase beta | P06746 | |
Potency | 3981.1 nM | Cytochrome P450 3A4 | P08684 | |
Potency | 11220.2 nM | Geminin | O75496 | |
Potency | 31622.8 nM | Thrombopoietin | P40225 | |
Potency | 3981.1 nM | Cytochrome P450 3A4 | P08684 | |
Potency | 56234.1 nM | Lysine-specific demethylase 4A | O75164 | |
Potency | 25929 nM | Nuclear factor erythroid 2-related factor 2 | Q16236 | |
Potency | 7079.5 nM | Histone acetyltransferase GCN5 | Q92830 | |
Potency | 37685.8 nM | M-phase phosphoprotein 8 | Q99549 | |
Potency | 19952.6 nM | M-phase phosphoprotein 8 | Q99549 | |
Potency | 22387.2 nM | Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 | Q96KQ7 | |
Potency | 2511.9 nM | Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 | Q96KQ7 | |
Potency | 17782.8 nM | Histone-lysine N-methyltransferase, H3 lysine-9 specific 3 | Q96KQ7 | |
Potency | 39810.7 nM | Chromobox protein homolog 1 | P83916 | |
Potency | 28183.8 nM | Bromodomain adjacent to zinc finger domain protein 2B | Q9UIF8 | |
Potency | 10000 nM | ATPase family AAA domain-containing protein 5 | Q96QE3 | |
Potency | 23934.1 nM | Peptidyl-prolyl cis-trans isomerase NIMA-interacting 1 | Q13526 | |
Potency | 11577.4 nM | ATPase family AAA domain-containing protein 5 | Q96QE3 | |
Potency | 16360.1 nM | Geminin | O75496 | |
Potency | 29855.4 nM | Geminin | O75496 | |
Potency | 39810.7 nM | Nuclear factor NF-kappa-B p105 subunit | P19838 | |
Potency | 44668.4 nM | Nuclear factor NF-kappa-B p105 subunit | P19838 | |
Potency | 53080.4 nM | Nuclear factor erythroid 2-related factor 2 | Q16236 | |
Potency | 54482.7 nM | Nuclear factor erythroid 2-related factor 2 | Q16236 | |
Potency | 11220.2 nM | Geminin | O75496 | |
Potency | 29855.4 nM | Geminin | O75496 | |
Potency | 28183.8 nM | Glucagon-like peptide 1 receptor | P43220 | |
Potency | 66824.2 nM | Interleukin-8 | P10145 | |
Potency | 37578 nM | Nuclear receptor ROR-gamma | P51449 | |
Others | 72.3 % | Solute carrier organic anion transporter family member 2B1 | O94956 | |
Others | 25.4 % | Solute carrier organic anion transporter family member 1B3 | Q9NPD5 | |
Others | 67.2 % | Solute carrier organic anion transporter family member 1B1 | Q9Y6L6 | |
Others | 29.2 | P-glycoprotein 1 | P08183 | |
Others | 4.4 | P-glycoprotein 1 | P08183 | |